G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Clemastine
CAS:15686-51-8
Clemastine (Meclastin) is an antagonist of the H1 receptor and exhibits anti-inflammatory effects.
Formula:
C21H26ClNO
Purity:
99.83%
Color and Shape:
Solid
Molecular weight:
343.89
Ref: TM-T19966
| 1ml | 65.00 € | ||
| 10mg | 66.00 € | ||
| 25mg | 95.00 € | ||
| 50mg | 151.00 € | ||
| 100mg | 220.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
PNU-96391
CAS:146798-66-5
PNU-96391 (OSU-6162) is an antagonist of dopamine D2 and a partial agonist of 5-HT2A. PNU-96391 …
Formula:
C15H23NO2S
Purity:
99.76%
Color and Shape:
Solid
Molecular weight:
281.41
Ref: TM-T28435
| 1mg | 183.00 € | ||
| 1ml | 390.00 € | ||
| 5mg | 406.00 € | ||
| 10mg | 600.00 € | ||
| 25mg | 916.00 € | ||
| 50mg | 1,281.00 € | ||
| 100mg | 1,733.00 € | ||
| 500mg | 3,455.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Bavisant
CAS:929622-08-2
Bavisant (JNJ-31001074) is a selective and orally active Human H3 receptor antagonist.
Formula:
C19H27N3O2
Purity:
96.06% - 98%
Color and Shape:
Solid
Molecular weight:
329.44
Ref: TM-TQ0046
| 1mg | 42.00 € | ||
| 1ml | 93.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 131.00 € | ||
| 25mg | 217.00 € | ||
| 50mg | 320.00 € | ||
| 100mg | 455.00 € | ||
| 500mg | To inquire |
Estimated delivery in United States, on Monday 25 Nov 2024
DL-071-IT
CAS:55104-39-7
DL-071-IT (Afurolol Hydrochloride) is a potent non-selective beta-adrenoceptor antagonist.
Formula:
C15H22ClNO4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
315.79
Ref: TM-T5450
| 5mg | 187.00 € | ||
| 10mg | 280.00 € | ||
| 25mg | 504.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
N-Arachidonyldopamine
CAS:199875-69-9
N-Arachidonyldopamine (NADA) is a selective and potent endogenous CB1 receptor agonist (Ki: 250 nM).N-Arachidonyldopamine is …
Formula:
C28H41NO3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
439.63
Ref: TM-T62530
| 1mg | 52.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 143.00 € | ||
| 25mg | 231.00 € | ||
| 50mg | 346.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
VPC 23019
CAS:449173-19-7
VPC 23019 is a competitive antagonist at the S1P1 and S1P3 receptors (pKi= 7.86 and …
Formula:
C17H29N2O5P
Purity:
98%
Color and Shape:
Solid
Molecular weight:
372.4
Ref: TM-T17237
| 25mg | 616.00 € | ||
| 50mg | 804.00 € | ||
| 100mg | 1,202.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Rezatomidine
CAS:847829-38-3
Rezatomidine (AGN203818) is a selective antagonist of α2-adrenergic receptor and can be used in studies …
Formula:
C13H16N2S
Purity:
99.62%
Color and Shape:
Solid
Molecular weight:
232.34
Ref: TM-T34308
| 1mg | 183.00 € | ||
| 2mg | 272.00 € | ||
| 5mg | 416.00 € | ||
| 10mg | 611.00 € | ||
| 25mg | 917.00 € | ||
| 50mg | 1,290.00 € | ||
| 100mg | 1,762.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
TC-MCH 7c
CAS:864756-35-4
TC-MCH 7c is an oral, selectable and blood-brain barrier penetrating MCH1R antagonist with IC50 performance …
Formula:
C24H25FN2O3
Purity:
98.8%
Color and Shape:
Solid
Molecular weight:
408.47
Ref: TM-T13101
| 1mg | 92.00 € | ||
| 1ml | 247.00 € | ||
| 5mg | 270.00 € | ||
| 10mg | 387.00 € | ||
| 25mg | 593.00 € | ||
| 50mg | 800.00 € | ||
| 100mg | 1,072.00 € | ||
| 500mg | 2,152.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
2-Methyl-5-HT hydrochloride
CAS:845861-49-6
2-Methyl-5-HT hydrochloride (2-Methyl-5-hydroxytryptamine) is a potent and selective 5-HT3 receptor agonist with anti-depressive-like effects.
Formula:
C11H15ClN2O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
226.7
Ref: TM-T10075L2
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Iprindole
CAS:5560-72-5
Iprindole, a tricyclic indole antidepressant, is a dual weak inhibitor of noradrenaline and 5-HT uptake …
Formula:
C19H28N2
Purity:
99.06%
Color and Shape:
Solid
Molecular weight:
284.44
Ref: TM-T37015
| 1ml | 95.00 € | ||
| 2mg | 45.00 € | ||
| 5mg | 66.00 € | ||
| 10mg | 94.00 € | ||
| 25mg | 185.00 € | ||
| 50mg | 322.00 € | ||
| 100mg | 537.00 € | ||
| 200mg | 772.00 € | ||
| 500mg | 1,142.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
NF-56-EJ40
CAS:2380230-73-7
NF-56-EJ40 is an effective and highly selective antagonist of human SUCNR1 with an IC50 of …
Formula:
C27H29N3O3
Purity:
99.51%
Color and Shape:
Solid
Molecular weight:
443.54
Ref: TM-T12216
| 1mg | 89.00 € | ||
| 1ml | 214.00 € | ||
| 5mg | 184.00 € | ||
| 10mg | 305.00 € | ||
| 25mg | 521.00 € | ||
| 50mg | 734.00 € | ||
| 100mg | 1,044.00 € | ||
| 500mg | 2,071.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Nedocromil
CAS:69049-73-6
Nedocromil (FPL 59002) inhibits the action or formation of multiple mediators. Which including histamine, leukotriene …
Formula:
C19H17NO7
Purity:
95%
Color and Shape:
Solid
Molecular weight:
371.34
Ref: TM-T16280
| 5mg | 69.00 € | ||
| 10mg | 94.00 € | ||
| 25mg | 198.00 € | ||
| 50mg | 325.00 € | ||
| 100mg | 508.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
ZK-90055 hydrochloride
CAS:84638-81-3
ZK-90055 hydrochloride is a β2 adrenergic receptor agonist used to study asthma.
Formula:
C16H23ClN2O4
Purity:
99.67%
Color and Shape:
Solid
Molecular weight:
342.82
Ref: TM-T13403
| 1mg | 326.00 € | ||
| 5mg | 774.00 € | ||
| 10mg | 1,050.00 € | ||
| 25mg | 1,477.00 € | ||
| 50mg | 1,850.00 € | ||
| 100mg | 2,331.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
A2A receptor antagonist 1
CAS:443103-97-7
A2A receptor antagonist 1 (CPI-444 analog) is an antagonist of both adenosine A2A receptor and …
Formula:
C16H12FN5O
Purity:
99.29% - 99.76%
Color and Shape:
Solid
Molecular weight:
309.3
Ref: TM-T37792
| 1mg | 37.00 € | ||
| 1ml | 46.00 € | ||
| 5mg | 63.00 € | ||
| 10mg | 90.00 € | ||
| 25mg | 182.00 € | ||
| 50mg | 278.00 € | ||
| 100mg | 412.00 € | ||
| 500mg | 866.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
SCH-336
CAS:447459-51-0
SCH-336: potent, selective CB2 agonist (Ki=1.8 nM, EC50=2 nM), orally active, 100x CB2 vs. CB1 …
Formula:
C23H25NO8S3
Purity:
95.01%
Color and Shape:
Solid
Molecular weight:
539.64
Ref: TM-T24771
| 1mg | 35.00 € | ||
| 1ml | 95.00 € | ||
| 5mg | 79.00 € | ||
| 10mg | 114.00 € | ||
| 25mg | 254.00 € | ||
| 50mg | 367.00 € | ||
| 100mg | 532.00 € | ||
| 500mg | To inquire |
Estimated delivery in United States, on Monday 25 Nov 2024
EP2 receptor antagonist-2
CAS:615273-95-5
CID891729, an EP2 receptor blocker, hinders PGE2 activation and reduces NMDA-induced LDH release.
Formula:
C15H14F3N3O
Purity:
99.59%
Color and Shape:
Solid
Molecular weight:
309.29
Ref: TM-T67946
| 1mg | 52.00 € | ||
| 1ml | 134.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 166.00 € | ||
| 25mg | 323.00 € | ||
| 50mg | 523.00 € | ||
| 100mg | 735.00 € | ||
| 500mg | 1,483.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Amitifadine hydrochloride
CAS:410074-74-7
Amitifadine hydrochloride (EB-1010 hydrochloride) is a triple reuptake inhibitor (TRI) or serotonin-norepinephrine-dopamine reuptake inhibitor (SNDRI).
Formula:
C11H12Cl3N
Purity:
98%
Color and Shape:
Solid
Molecular weight:
264.58
Ref: TM-T2092
| 1mg | 94.00 € | ||
| 1ml | 248.00 € | ||
| 5mg | 223.00 € | ||
| 10mg | 368.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Remoxipride hydrochloride
CAS:73220-03-8
Remoxipride hydrochloride (Roxiam) is a selective antagonist of D2 receptor with IC50s of 1.57 μM, …
Formula:
C16H24BrClN2O3
Purity:
99.32%
Color and Shape:
Solid
Molecular weight:
407.73
Ref: TM-T23232
| 1mg | 46.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 134.00 € | ||
| 25mg | 258.00 € | ||
| 50mg | 389.00 € | ||
| 100mg | 574.00 € | ||
| 500mg | 1,187.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
SB-277011
CAS:215803-78-4
SB-277011A: dopamine D3 antagonist, pKi 8.0 (D3), 6.0 (D2), 5.0 (5-HT1D), <5.2 (5-HT1B).
Formula:
C28H30N4O
Purity:
98.61%
Color and Shape:
Solid
Molecular weight:
438.56
Ref: TM-T12861
| 1mg | 46.00 € | ||
| 1ml | 60.00 € | ||
| 5mg | 57.00 € | ||
| 10mg | 92.00 € | ||
| 25mg | 154.00 € | ||
| 50mg | 249.00 € | ||
| 100mg | To inquire |
Estimated delivery in United States, on Monday 25 Nov 2024
GW-493838
CAS:253124-46-8
GW-493838 is a potent adenosine A1A receptor agonist for the treatment of dyslipidemia and neuropathic …
Formula:
C21H21ClFN7O4
Purity:
99.70% - 99.76%
Color and Shape:
Solid
Molecular weight:
489.89
Ref: TM-T27509
| 1mg | 148.00 € | ||
| 1ml | 419.00 € | ||
| 5mg | 358.00 € | ||
| 10mg | 508.00 € | ||
| 25mg | 763.00 € | ||
| 50mg | 1,031.00 € | ||
| 100mg | 1,393.00 € | ||
| 500mg | 2,730.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
