G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
Read more
Milveterol HCl
CAS:804518-03-4
Milveterol HCl is a long-acting β(2) -adrenergic receptor agonist for the potential treatment of chronic …
Formula:
C25H30ClN3O4
Purity:
98.2%
Color and Shape:
Solid
Molecular weight:
471.98
Ref: TM-T33386
| 1mg | 129.00 € | ||
| 5mg | 298.00 € | ||
| 10mg | 438.00 € | ||
| 25mg | 722.00 € | ||
| 50mg | 1,009.00 € | ||
| 100mg | 1,364.00 € | ||
| 500mg | 2,728.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
AM-1235
CAS:335161-27-8
AM-1235 is a potent and selective cannabinoid receptor CB1 agonist.
Formula:
C24H21FN2O3
Purity:
99%
Color and Shape:
Solid
Molecular weight:
404.43
Ref: TM-T29930
| 1mg | 325.00 € | ||
| 5mg | 769.00 € | ||
| 10mg | 1,054.00 € | ||
| 25mg | 1,483.00 € | ||
| 50mg | 1,838.00 € | ||
| 100mg | 2,331.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
A-437203
CAS:220519-06-2
A-437203 (Lu201640), selective D3 antagonist with Ki: D2-71nM, D3-1.6nM, D4-6220nM; based on 1H-pyrimidin-2-one scaffold.
Formula:
C20H27F3N6OS
Purity:
98.62%
Color and Shape:
Solid
Molecular weight:
456.53
Ref: TM-T10213
| 1mg | 146.00 € | ||
| 5mg | 325.00 € | ||
| 10mg | 456.00 € | ||
| 25mg | 709.00 € | ||
| 50mg | 919.00 € | ||
| 100mg | 1,275.00 € | ||
| 500mg | 2,578.00 € | ||
| 1mL*10mM (DMSO) | 377.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
FK-453
CAS:121524-18-3
FK-453 is a potent antagonist of non-xanthine adenosine A1 receptor with diuretic and renal vasodilatory …
Formula:
C23H25N3O2
Purity:
99.69%
Color and Shape:
Solid
Molecular weight:
375.46
Ref: TM-T27323
| 1mg | 233.00 € | ||
| 5mg | 580.00 € | ||
| 10mg | 820.00 € | ||
| 25mg | 1,236.00 € | ||
| 50mg | 1,654.00 € | ||
| 100mg | 2,248.00 € | ||
| 500mg | 4,530.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Femoxetine hydrochloride
CAS:56222-04-9
Femoxetine hydrochloride is a selective 5-hydroxytryptamine reuptake inhibitor used in the study of migraine, depression …
Formula:
C20H26ClNO2
Purity:
99.48%
Color and Shape:
Liquid
Molecular weight:
347.88
Ref: TM-T69096
| 1mg | 195.00 € | ||
| 5mg | 493.00 € | ||
| 10mg | 714.00 € | ||
| 25mg | 1,100.00 € | ||
| 50mg | 1,483.00 € | ||
| 100mg | 2,004.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Dabelotine
CAS:118976-38-8
Dabelotine (UNII-6RY56RB98P) is an adrenergic agonist used in the study of dementia.
Formula:
C15H22N2O2
Purity:
98.55%
Color and Shape:
Solid
Molecular weight:
262.35
Ref: TM-T31175
| 1mg | 141.00 € | ||
| 5mg | 327.00 € | ||
| 10mg | 495.00 € | ||
| 25mg | 801.00 € | ||
| 50mg | 1,096.00 € | ||
| 100mg | 1,483.00 € | ||
| 500mg | 2,960.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
R 59-022 hydrochloride
CAS:93076-98-3
R 59-022 hydrochloride is a 5-HT antagonist, PKC activator, DGK inhibitor (IC50: 2.8 µM), and …
Formula:
C27H27ClFN3OS
Purity:
97.7%
Color and Shape:
Liquid
Molecular weight:
496.04
Ref: TM-T72322
| 1mg | 45.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 142.00 € | ||
| 25mg | 276.00 € | ||
| 50mg | 447.00 € | ||
| 100mg | 643.00 € | ||
| 500mg | 1,319.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
DA-6886
CAS:1645260-76-9
DA-6886 is a 5-HT4 agonist, relaxes rat oesophagus, with 1000x selectivity over hERG channels, pIC50: …
Formula:
C19H28Cl2N6O2
Purity:
99% - 99.89%
Color and Shape:
Solid
Molecular weight:
443.37
Ref: TM-T27117
| 1mg | 136.00 € | ||
| 5mg | 316.00 € | ||
| 10mg | 474.00 € | ||
| 25mg | 772.00 € | ||
| 50mg | 1,068.00 € | ||
| 100mg | 1,448.00 € | ||
| 500mg | 2,775.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Selodenoson
CAS:110299-05-3
Selodenoson (RG-14202) is a selective adenosine A1 receptor agonist used to slow the heart rate …
Formula:
C17H24N6O4
Purity:
99.33%
Color and Shape:
Solid
Molecular weight:
376.41
Ref: TM-T28748
| 1mg | 128.00 € | ||
| 5mg | 298.00 € | ||
| 10mg | 439.00 € | ||
| 25mg | 717.00 € | ||
| 50mg | 1,007.00 € | ||
| 100mg | 1,356.00 € | ||
| 500mg | 2,712.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Isbogrel
CAS:89667-40-3
Isbogrel (CV4151) is a TXA2 synthase inhibitor for researching arrhythmias, ischemic attacks, and thrombosis.
Formula:
C18H19NO2
Purity:
97.06%
Color and Shape:
Solid
Molecular weight:
281.35
Ref: TM-T27630
| 1mg | 327.00 € | ||
| 5mg | 769.00 € | ||
| 10mg | 1,049.00 € | ||
| 25mg | 1,483.00 € | ||
| 50mg | 1,839.00 € | ||
| 100mg | 2,320.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Avosentan
CAS:290815-26-8
Avosentan(Ro 67-0565; SPP-301) is a potent endothelin receptor (ETA) antagonist.Cost-effective and quality-assured.
Formula:
C23H21N5O5S
Purity:
98.25% - 99.47%
Color and Shape:
Solid
Molecular weight:
479.51
Ref: TM-TQ0282
| 1mg | 40.00 € | ||
| 5mg | 83.00 € | ||
| 10mg | 104.00 € | ||
| 25mg | 212.00 € | ||
| 50mg | 369.00 € | ||
| 100mg | 539.00 € | ||
| 1mL*10mM (DMSO) | 89.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Darbufelone
CAS:139226-28-1
Darbufelone (CI-1004) is a non-competitive dual inhibitor of PGF2α and LTB4.
Formula:
C18H24N2O2S
Purity:
99.77%
Color and Shape:
Solid
Molecular weight:
332.46
Ref: TM-T10960
| 1mg | 44.00 € | ||
| 5mg | 85.00 € | ||
| 10mg | 128.00 € | ||
| 25mg | 274.00 € | ||
| 50mg | 400.00 € | ||
| 100mg | 551.00 € | ||
| 500mg | 1,098.00 € | ||
| 1mL*10mM (DMSO) | 110.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Edonentan
CAS:210891-04-6
Edonentan is A potent endothelin A (ETA) receptor antagonist that can be used to study …
Formula:
C28H32N4O5S
Purity:
98.78% - 99%
Color and Shape:
Solid
Molecular weight:
536.64
Ref: TM-T31605
| 1mg | 939.00 € | ||
| 5mg | 1,850.00 € | ||
| 25mg | 2,404.00 € | ||
| 50mg | 2,784.00 € | ||
| 100mg | 3,737.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Faxeladol
CAS:433265-65-7
Faxeladol: adrenergic, serotonin inhibitor & opioid agonist for neurological studies.
Formula:
C15H23NO
Purity:
99.11% - 99.13%
Color and Shape:
Solid
Molecular weight:
233.35
Ref: TM-T31750
| 1mg | 597.00 € | ||
| 5mg | 1,258.00 € | ||
| 25mg | 1,692.00 € | ||
| 50mg | 2,023.00 € | ||
| 100mg | 2,610.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Fipamezole
CAS:150586-58-6
Fipamezole is a potent alpha2 adrenergic receptor antagonist that may be useful for studying autonomic …
Formula:
C14H15FN2
Purity:
100% - 99.32%
Color and Shape:
Solid
Molecular weight:
230.28
Ref: TM-T24064
| 1mg | 597.00 € | ||
| 5mg | 1,253.00 € | ||
| 25mg | 1,692.00 € | ||
| 50mg | 2,025.00 € | ||
| 100mg | 2,601.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
CP-226269
CAS:220941-93-5
CP-226269 is a potent dopamine D4 receptor agonist that regulates calcium flux and has an …
Formula:
C18H19FN4
Purity:
99.08%
Color and Shape:
Solid
Molecular weight:
310.37
Ref: TM-T27060
| 1mg | 95.00 € | ||
| 5mg | 229.00 € | ||
| 10mg | 335.00 € | ||
| 25mg | 538.00 € | ||
| 50mg | 765.00 € | ||
| 100mg | 1,040.00 € | ||
| 500mg | 2,070.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
ONO-8713
CAS:459411-08-6
ONO-8713 is a selective prostaglandin E receptor subtype EP1 antagonist that can be used to …
Formula:
C25H24F3NO6S
Purity:
100.00%
Color and Shape:
Liquid
Molecular weight:
523.52
Ref: TM-T63667
| 1mg | 378.00 € | ||
| 5mg | 900.00 € | ||
| 10mg | 1,122.00 € | ||
| 25mg | 1,502.00 € | ||
| 50mg | 1,838.00 € | ||
| 100mg | 2,320.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Opioid receptor modulator 1
CAS:77514-44-4
Opioid receptor modulator 1 is a modulator of opioid receptor.
Formula:
C18H23NO2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
285.38
Ref: TM-T12314
| 25mg | 1,406.00 € | ||
| 50mg | 1,847.00 € | ||
| 100mg | 2,331.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Cinitapride Hydrogen Tartrate
CAS:1207859-16-2
Cinitapride Hydrogen Tartrate is a gastroprokinetic agent that acts as an antagonist of the 5-HT2 …
Formula:
C25H36N4O10
Purity:
98%
Color and Shape:
Solid
Molecular weight:
552.581
Ref: TM-T22294
| 25mg | 1,410.00 € | ||
| 50mg | 1,852.00 € | ||
| 100mg | 2,338.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
BMS 182874
CAS:153042-42-3
BMS 182874: Oral ETA antagonist, IC50=0.150 μM, Ki=0.055 μM, lowers hypertension in rats.
Formula:
C17H19N3O3S
Purity:
98.38%
Color and Shape:
Solid
Molecular weight:
345.42
Ref: TM-T26841
| 1mg | 73.00 € | ||
| 5mg | 157.00 € | ||
| 10mg | 244.00 € | ||
| 25mg | 422.00 € | ||
| 50mg | 601.00 € | ||
| 100mg | 827.00 € | ||
| 500mg | 1,687.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
