G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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BRL 44408 Maleate Salt
CAS:681806-46-2
BRL 44408 Maleate is an α2A-adrenoceptor antagonist with antidepressant and analgesic activity.
Formula:
C17H21N3O4
Color and Shape:
Solid
Molecular weight:
331.37
Ref: TM-T26904
| 1mg | 74.00 € | ||
| 5mg | 162.00 € | ||
| 10mg | 279.00 € | ||
| 25mg | 462.00 € | ||
| 50mg | 673.00 € | ||
| 100mg | 991.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
KUL-7211 racemate
CAS:911196-40-2
KUL 7211, a selective β-adrenoceptor agonist, exists as a racemate, referred to as KUL 7211 …
Formula:
C19H23NO5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
345.39
Ref: TM-T11786
| 25mg | 1,410.00 € | ||
| 50mg | 1,845.00 € | ||
| 100mg | 2,329.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
5-HT2 antagonist 1
CAS:191592-09-3
5-HT2 antagonist 1 is a potent 5-HT2 receptor antagonist, has weak α1 adrenoceptor blocking activity.
Formula:
C22H29FN4O2
Purity:
99.25%
Color and Shape:
Solid
Molecular weight:
400.49
Ref: TM-T12597
| 1mg | 663.00 € | ||
| 5mg | 1,328.00 € | ||
| 10mg | 1,792.00 € | ||
| 25mg | 2,665.00 € | ||
| 50mg | 3,593.00 € | ||
| 100mg | 4,855.00 € | ||
| 1mL*10mM (DMSO) | 1,595.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
AMX12006
CAS:2639775-01-0
AMX12006, a potent and selective EP4 antagonist, exhibits cytotoxic and antitumor activity, demonstrating oral activity …
Formula:
C26H22F3N3O3
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
481.47
Ref: TM-T78710
| 1mg | 141.00 € | ||
| 5mg | 601.00 € | ||
| 10mg | 1,063.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
KSK94
CAS:2566716-07-0
KSK94 is an H3 receptor antagonist that inhibits sigma-2 receptors , with a Ki value …
Formula:
C25H26N4O
Purity:
99.56%
Color and Shape:
Solid
Molecular weight:
398.5
Ref: TM-T79500
| 1mg | 59.00 € | ||
| 5mg | 122.00 € | ||
| 10mg | 173.00 € | ||
| 25mg | 277.00 € | ||
| 50mg | 428.00 € | ||
| 100mg | 623.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
KSK68
CAS:2566715-91-9
KSK68 is a sigma-1 and histamine H3 receptor antagonist with analgesic activity, inhibits H3 receptors …
Formula:
C23H28N2O2
Purity:
97.22%
Color and Shape:
Solid
Molecular weight:
364.48
Ref: TM-T79499
| 1mg | 74.00 € | ||
| 5mg | 159.00 € | ||
| 10mg | 224.00 € | ||
| 25mg | 372.00 € | ||
| 50mg | 558.00 € | ||
| 100mg | 796.00 € | ||
| 500mg | 2,210.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Pancopride
CAS:121650-80-4
Pancopride(LAS 30451) is a novel, orally available, long-acting, selective 5-HT3 receptor antagonist that blocks nitrogen …
Formula:
C18H24ClN3O2
Purity:
93.64%
Color and Shape:
Solid
Molecular weight:
349.86
Ref: TM-T16433
| 1mg | 650.00 € | ||
| 5mg | 1,682.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
SARS-CoV-2-IN-57
CAS:1265624-68-7
SARS-CoV-2-IN-57 (compound (+)-R-26) is a potent inhibitor of SARS-CoV-2 with an IC50 of 80 nM …
Formula:
C23H37N3O
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
371.56
Ref: TM-T79356
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
APNEA
CAS:89705-21-5
APNEA ((2R,3R,4S,5R)-2-[6-[2-(4-aminophenyl)ethylamino]purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol) is a non-selective agonist of adenosine A3 receptor.
Formula:
C18H22N6O4
Purity:
99.58%
Color and Shape:
Solid
Molecular weight:
386.41
Ref: TM-T12159
| 25mg | 50.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
PNU-96391
CAS:146798-66-5
PNU-96391 (OSU-6162) is an antagonist of dopamine D2 and a partial agonist of 5-HT2A. PNU-96391 …
Formula:
C15H23NO2S
Purity:
99.76%
Color and Shape:
Solid
Molecular weight:
281.41
Ref: TM-T28435
| 1mg | 112.00 € | ||
| 5mg | 242.00 € | ||
| 10mg | 359.00 € | ||
| 25mg | 547.00 € | ||
| 50mg | 765.00 € | ||
| 100mg | 1,026.00 € | ||
| 200mg | 1,367.00 € | ||
| 1mL*10mM (DMSO) | 230.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Moprolol
CAS:5741-22-0
Moprolol ((±)-Moprolol) is a beta-adrenergic receptor antagonist utilized in research pertaining to essential hypertension [1] …
Formula:
C13H21NO3
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
239.31
Ref: TM-T78567
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
CXCR4-IN-1
CAS:2304750-48-7
CXCR4-IN-1 (Example C5), with an IC50 of 20 nM, is a potent inhibitor of CXCR4, …
Formula:
C23H32N6
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
392.54
Ref: TM-T79059
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
YL-365
YL-365 is a highly potent and selective GPR34 antagonist that exhibits excellent activity in neuropathic …
Ref: TM-T80753
| 1mg | 75.00 € | ||
| 5mg | 167.00 € | ||
| 10mg | 261.00 € | ||
| 25mg | 527.00 € | ||
| 50mg | 838.00 € | ||
| 100mg | 1,332.00 € | ||
| 200mg | 1,801.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
A-77636
CAS:778546-51-3
A-77636 is a potent, selective, and long-acting oral dopamine D1 receptor agonist with an effective …
Formula:
C20H27NO3
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
329.43
Ref: TM-T78644
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
CAY10786
CAS:1239987-91-7
CAY10786 (GPR52 antagonist-1) is an antagonist of G protein-coupled receptor 52 (GPR52, IC50 = 0.63 …
Formula:
C15H14OS
Purity:
99.84%
Color and Shape:
Solid
Molecular weight:
242.34
Ref: TM-T36036
| 2mg | 40.00 € | ||
| 5mg | 60.00 € | ||
| 10mg | 96.00 € | ||
| 25mg | 184.00 € | ||
| 50mg | 291.00 € | ||
| 100mg | 458.00 € | ||
| 1mL*10mM (DMSO) | 67.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
DL-071-IT
CAS:55104-39-7
DL-071-IT (Afurolol Hydrochloride) is a potent non-selective beta-adrenoceptor antagonist.
Formula:
C15H22ClNO4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
315.79
Ref: TM-T5450
| 5mg | 187.00 € | ||
| 10mg | 280.00 € | ||
| 25mg | 504.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Rezatomidine
CAS:847829-38-3
Rezatomidine (AGN203818) is a selective antagonist of α2-adrenergic receptor and can be used in studies …
Formula:
C13H16N2S
Purity:
99.62%
Color and Shape:
Solid
Molecular weight:
232.34
Ref: TM-T34308
| 1mg | 183.00 € | ||
| 2mg | 272.00 € | ||
| 5mg | 416.00 € | ||
| 10mg | 611.00 € | ||
| 25mg | 917.00 € | ||
| 50mg | 1,290.00 € | ||
| 100mg | 1,762.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
2-Methyl-5-HT hydrochloride
CAS:845861-49-6
2-Methyl-5-HT hydrochloride (2-Methyl-5-hydroxytryptamine) is a potent and selective 5-HT3 receptor agonist with anti-depressive-like effects.
Formula:
C11H15ClN2O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
226.7
Ref: TM-T10075L2
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Remoxipride hydrochloride
CAS:73220-03-8
Remoxipride hydrochloride (Roxiam) is a selective antagonist of D2 receptor with IC50s of 1.57 μM, …
Formula:
C16H24BrClN2O3
Purity:
99.32%
Color and Shape:
Solid
Molecular weight:
407.73
Ref: TM-T23232
| 1mg | 46.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 134.00 € | ||
| 25mg | 258.00 € | ||
| 50mg | 389.00 € | ||
| 100mg | 574.00 € | ||
| 500mg | 1,187.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
5-HT3 antagonist 3
CAS:120635-47-4
5-HT3 antagonist 3 (Compound 15b) is a high-affinity 5-HT3 receptor antagonist. It binds to 5-HT3 …
Formula:
C20H21N3O
Purity:
99.69%
Color and Shape:
Solid
Molecular weight:
319.4
Ref: TM-T10162
| 1mg | 113.00 € | ||
| 2mg | 169.00 € | ||
| 5mg | 250.00 € | ||
| 10mg | 367.00 € | ||
| 25mg | 550.00 € | ||
| 50mg | 775.00 € | ||
| 100mg | 1,040.00 € | ||
| 500mg | To inquire |
Estimated delivery in United States, on Monday 27 Jan 2025
