G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Clemastine
CAS:15686-51-8
Clemastine (Meclastin) is an antagonist of the H1 receptor and exhibits anti-inflammatory effects.
Formula:
C21H26ClNO
Purity:
99.83%
Color and Shape:
Solid
Molecular weight:
343.89
Ref: TM-T19966
| 10mg | 66.00 € | ||
| 25mg | 95.00 € | ||
| 50mg | 151.00 € | ||
| 100mg | 220.00 € | ||
| 1mL*10mM (DMSO) | 65.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
Selodenoson
CAS:110299-05-3
Selodenoson (RG-14202) is a selective adenosine A1 receptor agonist used to slow the heart rate …
Formula:
C17H24N6O4
Purity:
99.33%
Color and Shape:
Solid
Molecular weight:
376.41
Ref: TM-T28748
| 1mg | 128.00 € | ||
| 5mg | 298.00 € | ||
| 10mg | 439.00 € | ||
| 25mg | 717.00 € | ||
| 50mg | 1,007.00 € | ||
| 100mg | 1,356.00 € | ||
| 500mg | 2,712.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
Isbogrel
CAS:89667-40-3
Isbogrel (CV4151) is a TXA2 synthase inhibitor for researching arrhythmias, ischemic attacks, and thrombosis.
Formula:
C18H19NO2
Purity:
97.06%
Color and Shape:
Solid
Molecular weight:
281.35
Ref: TM-T27630
| 1mg | 327.00 € | ||
| 5mg | 769.00 € | ||
| 10mg | 1,049.00 € | ||
| 25mg | 1,483.00 € | ||
| 50mg | 1,839.00 € | ||
| 100mg | 2,320.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
Rocastine
CAS:91833-49-7
Rocastine (AHR-11325) is a selective and potent non-sedating H1 receptor antagonist.
Formula:
C13H19N3OS
Purity:
98.26%
Color and Shape:
Solid
Molecular weight:
265.37
Ref: TM-T16778
| 1mg | 650.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
Bavisant
CAS:929622-08-2
Bavisant (JNJ-31001074) is a selective and orally active Human H3 receptor antagonist.
Formula:
C19H27N3O2
Purity:
96.06% - 98%
Color and Shape:
Solid
Molecular weight:
329.44
Ref: TM-TQ0046
| 1mg | 42.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 131.00 € | ||
| 25mg | 217.00 € | ||
| 50mg | 320.00 € | ||
| 100mg | 455.00 € | ||
| 500mg | To inquire | ||
| 1mL*10mM (DMSO) | 93.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
MEN11467
CAS:214487-46-4
MEN11467 is a novel, orally available, potent and selective peptidomimetic tachykinin NK 1 receptor antagonist …
Formula:
C38H40N4O3
Purity:
100%
Color and Shape:
Solid
Molecular weight:
600.75
Ref: TM-T12000
| 1mg | 650.00 € | ||
| 5mg | 1,672.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
N-Arachidonyldopamine
CAS:199875-69-9
N-Arachidonyldopamine (NADA) is a selective and potent endogenous CB1 receptor agonist (Ki: 250 nM).N-Arachidonyldopamine is …
Formula:
C28H41NO3
Purity:
97.65%
Color and Shape:
Solid
Molecular weight:
439.63
Ref: TM-T62530
| 1mg | 52.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 143.00 € | ||
| 25mg | 231.00 € | ||
| 50mg | 346.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
VPC 23019
CAS:449173-19-7
VPC 23019 is a competitive antagonist at the S1P1 and S1P3 receptors (pKi= 7.86 and …
Formula:
C17H29N2O5P
Purity:
98%
Color and Shape:
Solid
Molecular weight:
372.4
Ref: TM-T17237
| 25mg | 616.00 € | ||
| 50mg | 804.00 € | ||
| 100mg | 1,202.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
H3 receptor-MO-1
CAS:1240914-03-7
H3 receptor-MO-1 is a potent modulator of the histamine H3 receptor (H3 receptor) and can …
Formula:
C20H27N3O2
Purity:
99.11%
Color and Shape:
Solid
Molecular weight:
341.45
Ref: TM-T10499
| 1mg | 651.00 € | ||
| 5mg | 1,682.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
TC-MCH 7c
CAS:864756-35-4
TC-MCH 7c is an oral, selectable and blood-brain barrier penetrating MCH1R antagonist with IC50 performance …
Formula:
C24H25FN2O3
Purity:
98.8%
Color and Shape:
Solid
Molecular weight:
408.47
Ref: TM-T13101
| 1mg | 92.00 € | ||
| 5mg | 270.00 € | ||
| 10mg | 387.00 € | ||
| 25mg | 593.00 € | ||
| 50mg | 800.00 € | ||
| 100mg | 1,072.00 € | ||
| 500mg | 2,152.00 € | ||
| 1mL*10mM (DMSO) | 247.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
Tulopafant
CAS:116289-53-3
Tulopafant (RP 59227) is a potent platelet-activating factor (PAF) antagonist that increases capillary patency and …
Formula:
C25H19N3O2S
Purity:
99.38%
Color and Shape:
Solid
Molecular weight:
425.5
Ref: TM-T17178
| 1mg | 650.00 € | ||
| 5mg | 1,678.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
Iprindole
CAS:5560-72-5
Iprindole, a tricyclic indole antidepressant, is a dual weak inhibitor of noradrenaline and 5-HT uptake …
Formula:
C19H28N2
Purity:
99.06%
Color and Shape:
Solid
Molecular weight:
284.44
Ref: TM-T37015
| 5mg | 43.00 € | ||
| 10mg | 62.00 € | ||
| 25mg | 113.00 € | ||
| 50mg | 193.00 € | ||
| 100mg | 322.00 € | ||
| 200mg | 460.00 € | ||
| 1mL*10mM (DMSO) | 62.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
NF-56-EJ40
CAS:2380230-73-7
NF-56-EJ40 is an effective and highly selective antagonist of human SUCNR1 with an IC50 of …
Formula:
C27H29N3O3
Purity:
99.51%
Color and Shape:
Solid
Molecular weight:
443.54
Ref: TM-T12216
| 1mg | 89.00 € | ||
| 5mg | 184.00 € | ||
| 10mg | 305.00 € | ||
| 25mg | 521.00 € | ||
| 50mg | 734.00 € | ||
| 100mg | 1,044.00 € | ||
| 500mg | 2,071.00 € | ||
| 1mL*10mM (DMSO) | 214.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
Avosentan
CAS:290815-26-8
Avosentan(Ro 67-0565; SPP-301) is a potent endothelin receptor (ETA) antagonist.Cost-effective and quality-assured.
Formula:
C23H21N5O5S
Purity:
98.25% - 99.47%
Color and Shape:
Solid
Molecular weight:
479.51
Ref: TM-TQ0282
| 1mg | 40.00 € | ||
| 5mg | 83.00 € | ||
| 10mg | 104.00 € | ||
| 25mg | 212.00 € | ||
| 50mg | 369.00 € | ||
| 100mg | 539.00 € | ||
| 1mL*10mM (DMSO) | 89.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
A2A receptor antagonist 1
CAS:443103-97-7
A2A receptor antagonist 1 (CPI-444 analog) is an antagonist of both adenosine A2A receptor and …
Formula:
C16H12FN5O
Purity:
99.29% - 99.76%
Color and Shape:
Liquid
Molecular weight:
309.3
Ref: TM-T37792
| 1mg | 37.00 € | ||
| 5mg | 63.00 € | ||
| 10mg | 90.00 € | ||
| 25mg | 182.00 € | ||
| 50mg | 278.00 € | ||
| 100mg | 412.00 € | ||
| 500mg | 866.00 € | ||
| 1mL*10mM (DMSO) | 46.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
SCH-336
CAS:447459-51-0
SCH-336: potent, selective CB2 agonist (Ki=1.8 nM, EC50=2 nM), orally active, 100x CB2 vs. CB1 …
Formula:
C23H25NO8S3
Purity:
95.01%
Color and Shape:
Solid
Molecular weight:
539.64
Ref: TM-T24771
| 1mg | 35.00 € | ||
| 5mg | 79.00 € | ||
| 10mg | 114.00 € | ||
| 25mg | 254.00 € | ||
| 50mg | 367.00 € | ||
| 100mg | 532.00 € | ||
| 500mg | To inquire | ||
| 1mL*10mM (DMSO) | 95.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
EP2 receptor antagonist-2
CAS:615273-95-5
CID891729, an EP2 receptor blocker, hinders PGE2 activation and reduces NMDA-induced LDH release.
Formula:
C15H14F3N3O
Purity:
99.59%
Color and Shape:
Solid
Molecular weight:
309.29
Ref: TM-T67946
| 1mg | 49.00 € | ||
| 5mg | 102.00 € | ||
| 10mg | 166.00 € | ||
| 25mg | 276.00 € | ||
| 50mg | 411.00 € | ||
| 100mg | 593.00 € | ||
| 500mg | 1,235.00 € | ||
| 1mL*10mM (DMSO) | 147.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
Amitifadine hydrochloride
CAS:410074-74-7
Amitifadine hydrochloride (EB-1010 hydrochloride) is a triple reuptake inhibitor (TRI) or serotonin-norepinephrine-dopamine reuptake inhibitor (SNDRI).
Formula:
C11H12Cl3N
Purity:
98%
Color and Shape:
Solid
Molecular weight:
264.58
Ref: TM-T2092
| 1mg | 94.00 € | ||
| 5mg | 223.00 € | ||
| 10mg | 368.00 € | ||
| 1mL*10mM (DMSO) | 248.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
Quinupramine
CAS:31721-17-2
Quinupramine: an oral antidepressant targeting the serotonin system; penetrates CNS; doesn’t affect β-adrenergic system.
Formula:
C21H24N2
Purity:
99.76%
Color and Shape:
Solid
Molecular weight:
304.43
Ref: TM-T60707
| 1mg | 431.00 € | ||
| 5mg | 998.00 € | ||
| 25mg | 1,985.00 € | ||
| 50mg | 2,591.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
Octimibate
CAS:89838-96-0
Octimibate: non-prostaglandin antiplatelet, treats cardiovascular disease, aids atherosclerosis/thrombosis research.
Formula:
C29H30N2O3
Purity:
99.49%
Color and Shape:
Solid
Molecular weight:
454.56
Ref: TM-T24567
| 1mg | 138.00 € | ||
| 5mg | 335.00 € | ||
| 10mg | 492.00 € | ||
| 25mg | 798.00 € | ||
| 50mg | 1,096.00 € | ||
| 100mg | 1,483.00 € | ||
| 500mg | 2,960.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
