G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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SF-22
CAS:824981-55-7
SF-22 is a Y2R antagonist with potential anti-inflammatory activity that can be used to study …
Formula:
C28H26N2O3S
Purity:
99.09%
Color and Shape:
Liquid
Molecular weight:
470.58
Ref: TM-T71749
| 1mg | 36.00 € | ||
| 5mg | 74.00 € | ||
| 10mg | 111.00 € | ||
| 25mg | 233.00 € | ||
| 50mg | 374.00 € | ||
| 100mg | 594.00 € | ||
| 500mg | 1,217.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
Repinotan HCl
CAS:144980-77-8
Repinotan HCl (Bay-x-3702) is a 5-HT1A receptor agonist with potent neuroprotective effects for the study …
Formula:
C21H25ClN2O4S
Purity:
99.57%
Color and Shape:
Solid
Molecular weight:
436.95
Ref: TM-T28518
| 1mg | 380.00 € | ||
| 5mg | 820.00 € | ||
| 10mg | 1,168.00 € | ||
| 25mg | 1,564.00 € | ||
| 50mg | 1,899.00 € | ||
| 100mg | 2,396.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
Irdabisant
CAS:1005402-19-6
Irdabisant (CEP-26401) is an H3R antagonist/inverse agonist, BBB permeable, with cognition-enhancing effects for schizophrenia/cognitive research.
Formula:
C18H23N3O2
Purity:
99.77%
Color and Shape:
Solid
Molecular weight:
313.39
Ref: TM-T32191
| 1mg | 57.00 € | ||
| 5mg | 131.00 € | ||
| 10mg | 184.00 € | ||
| 25mg | 328.00 € | ||
| 50mg | 460.00 € | ||
| 100mg | 647.00 € | ||
| 500mg | 1,291.00 € | ||
| 1mL*10mM (DMSO) | 92.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
(Rac)-WAY-161503
CAS:75704-24-4
(Rac)-WAY-161503 is a selective and high-affinity agonist of the 5-HT2C receptor (Ki: 4 nM; EC50: …
Formula:
C11H11Cl2N3O
Purity:
98.08%
Color and Shape:
Solid
Molecular weight:
272.13
Ref: TM-T13332
| 5mg | 93.00 € | ||
| 10mg | 115.00 € | ||
| 25mg | 179.00 € | ||
| 50mg | 261.00 € | ||
| 100mg | 386.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
Cilansetron
CAS:120635-74-7
Cilansetron is an effective and selective 5-HT3 receptor antagonist that can be used for related …
Formula:
C20H21N3O
Purity:
99.77% - 99.85%
Color and Shape:
Solid
Molecular weight:
319.4
Ref: TM-T27020
| 1mg | 182.00 € | ||
| 5mg | 449.00 € | ||
| 10mg | 643.00 € | ||
| 25mg | 1,003.00 € | ||
| 50mg | 1,384.00 € | ||
| 100mg | 1,830.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
E6801
CAS:528859-04-3
E6801: selective 5-HT6 agonist for research in dementia, Parkinson's, depression, obesity, epilepsy, anxiety, etc.
Formula:
C17H18ClN5O2S2
Purity:
100% - 96.66%
Color and Shape:
Solid
Molecular weight:
423.94
Ref: TM-T31592
| 1mg | 325.00 € | ||
| 5mg | 769.00 € | ||
| 10mg | 1,050.00 € | ||
| 25mg | 1,476.00 € | ||
| 50mg | 1,850.00 € | ||
| 100mg | 2,321.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
CB2R PAM
CAS:2244579-87-9
CB2R PAM, an oral drug, boosts CB2 receptor response to specific agonists, showing potential in …
Formula:
C21H24BrFN2O2
Purity:
98.17%
Color and Shape:
Liquid
Molecular weight:
435.33
Ref: TM-T37075
| 1mg | 55.00 € | ||
| 5mg | 118.00 € | ||
| 10mg | 172.00 € | ||
| 25mg | 274.00 € | ||
| 50mg | 416.00 € | ||
| 100mg | 612.00 € | ||
| 500mg | 1,281.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
N6-Cyclopentyladenosine
CAS:41552-82-3
N6-Cyclopentyladenosine (CPA) is a selective agonist of the adenosine A1 receptor and can be used …
Formula:
C15H21N5O4
Purity:
99.84%
Color and Shape:
Solid
Molecular weight:
335.36
Ref: TM-T16263
| 5mg | 35.00 € | ||
| 10mg | 49.00 € | ||
| 25mg | 71.00 € | ||
| 50mg | 96.00 € | ||
| 100mg | 157.00 € | ||
| 500mg | 369.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
SB-269970
CAS:201038-74-6
SB-269970 is a antagonist of 5-HT7 receptor(pKi of 8.3).
Formula:
C18H28N2O3S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
352.49
Ref: TM-T12842
| 25mg | 1,406.00 € | ||
| 50mg | 1,845.00 € | ||
| 100mg | 2,329.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
GPR4 antagonist 1
CAS:1197879-16-5
GPR4 antagonist 1 is a GPR4 antagonist (IC50: 189 nM).
Formula:
C27H37N5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
431.62
Ref: TM-T11460
| 25mg | 1,410.00 € | ||
| 50mg | 1,845.00 € | ||
| 100mg | 2,329.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
LPA2 antagonist 2
CAS:36840-10-5
LPA2 antagonist 2 is an and LPA2 antagonist (IC50: 28.3 nM) with potential anticancer activity, …
Formula:
C20H16N2O6
Purity:
96.13%
Color and Shape:
Solid
Molecular weight:
380.35
Ref: TM-T11875
| 1mg | 93.00 € | ||
| 5mg | 222.00 € | ||
| 10mg | 350.00 € | ||
| 25mg | 576.00 € | ||
| 50mg | 812.00 € | ||
| 100mg | 1,094.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
Atrasentan hydrochloride
CAS:195733-43-8
Atrasentan hydrochloride (ABT-627 hydrochloride) is an antagonist of the endothelin receptor(IC50 = 55.1 μM for …
Formula:
C29H39ClN2O6
Purity:
98.64%
Color and Shape:
Solid
Molecular weight:
547.08
Ref: TM-TQ0270
| 2mg | 41.00 € | ||
| 5mg | 62.00 € | ||
| 10mg | 88.00 € | ||
| 25mg | 159.00 € | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 74.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
Aganepag
CAS:910562-18-4
Aganepag: Potent EP2 agonist, EC50 0.19 nM, inactive at EP4, used in wound healing and …
Formula:
C24H31NO4S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
429.57
Ref: TM-T14139
| 25mg | 2,106.00 € | ||
| 50mg | 2,785.00 € | ||
| 100mg | 3,739.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
(S)-(+)-Niguldipine hydrochloride
CAS:113145-69-0
(S)-(+)-Niguldipine hydrochloride is a selective α1A-AR antagonist used in the study of depression and epilepsy.
Formula:
C36H40ClN3O6
Purity:
98.06%
Color and Shape:
Solid
Molecular weight:
646.17
Ref: TM-T23301
| 1mg | 82.00 € | ||
| 5mg | 170.00 € | ||
| 10mg | 249.00 € | ||
| 25mg | 586.00 € | ||
| 50mg | 1,021.00 € | ||
| 100mg | 1,371.00 € | ||
| 500mg | 2,732.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
Anpirtoline hydrochloride
CAS:99201-87-3
Anpirtoline hydrochloride (D-16949 hydrochloride) is a 5-HT1B receptor agonist and 5-HT3 receptor antagonist used in …
Formula:
C10H14Cl2N2S
Purity:
100% - 100%
Color and Shape:
Solid
Molecular weight:
265.20
Ref: TM-T22576
| 1mg | 52.00 € | ||
| 5mg | 109.00 € | ||
| 10mg | 172.00 € | ||
| 25mg | 276.00 € | ||
| 50mg | 421.00 € | ||
| 100mg | 606.00 € | ||
| 500mg | 1,253.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
Rilapine
CAS:79781-95-6
Rilapine (Rilapinum) is an antipsychotic compound that shows high affinity for 5-HT6 receptors and can …
Formula:
C22H20ClN3
Purity:
99% - 99.66%
Color and Shape:
Solid
Molecular weight:
361.87
Ref: TM-T26085
| 1mg | 277.00 € | ||
| 5mg | 681.00 € | ||
| 10mg | 931.00 € | ||
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
PSB-CB5
CAS:1627710-30-8
PSB-CB5 (GPR18-IN-32)2 is a GRP18 antagonist with anti-inflammatory activity and can be used to study …
Formula:
C20H17ClN2O2S
Purity:
99.26%
Color and Shape:
Solid
Molecular weight:
384.88
Ref: TM-T27019
| 1mg | 89.00 € | ||
| 5mg | 184.00 € | ||
| 10mg | 308.00 € | ||
| 25mg | 515.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
Pavinetant
CAS:941690-55-7
Pavinetant (MLE-4901) is an orally available neurokinin-3 receptor (NK3R) antagonist used to improve menopausal symptoms.
Formula:
C26H25N3O3S
Purity:
99.60%
Color and Shape:
Solid
Molecular weight:
459.56
Ref: TM-T16114
| 1mg | 80.00 € | ||
| 2mg | 102.00 € | ||
| 5mg | 173.00 € | ||
| 10mg | 257.00 € | ||
| 25mg | 343.00 € | ||
| 50mg | 429.00 € | ||
| 100mg | 618.00 € | ||
| 1mL*10mM (DMSO) | 172.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
CP 316311
CAS:175139-41-0
CP 316311 is a specific CRF1 receptor antagonist with potential antidepressant activity and may be …
Formula:
C21H29NO2
Purity:
99.47% - 99.60%
Color and Shape:
Solid
Molecular weight:
327.46
Ref: TM-T15008
| 1mg | 277.00 € | ||
| 5mg | 497.00 € | ||
| 10mg | 637.00 € | ||
| 25mg | 865.00 € | ||
| 50mg | 1,174.00 € | ||
| 100mg | 1,565.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
CCX777
CAS:1226686-36-7
CCX777 is a partial agonist recruited to ACKR3 by β-arrestin-2 and is used in cancer …
Formula:
C31H43N7O3S
Purity:
98.73%
Color and Shape:
Solid
Molecular weight:
593.78
Ref: TM-T23866
| 1mg | 278.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
