G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
Read more
Compound C108
CAS:15533-09-2
Compound C108 is an inhibitor of GTPase-activating protein SH3 domain-binding protein 2 (G3BP2).
Formula:
C15H14N2O3
Purity:
99.77%
Color and Shape:
Solid
Molecular weight:
270.28
Ref: TM-T38387
| 1mg | 45.00 € | ||
| 1ml | 123.00 € | ||
| 5mg | 88.00 € | ||
| 10mg | 128.00 € | ||
| 25mg | 247.00 € | ||
| 50mg | 393.00 € | ||
| 100mg | 584.00 € | ||
| 500mg | 1,254.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
IPAG
CAS:193527-91-2
IPAG is a potent σ-receptor antagonist (pKi=4.3). IPAG can induce cell apoptosis.
Formula:
C17H22IN3
Purity:
98.8%
Color and Shape:
Solid
Molecular weight:
395.28
Ref: TM-T22870
| 1mg | 45.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 135.00 € | ||
| 25mg | 259.00 € | ||
| 50mg | 447.00 € | ||
| 100mg | 640.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
IT1t dihydrochloride
CAS:1092776-63-0
IT1t dihydrochloride inhibits CXCL12/CXCR4 interaction with IC50 of 2.1 nM. IT1t dihydrochloride is an antagonist …
Formula:
C21H36Cl2N4S2
Purity:
98.03%
Color and Shape:
Solid
Molecular weight:
479.57
Ref: TM-T11693L
| 1ml | 58.00 € | ||
| 2mg | 34.00 € | ||
| 5mg | 51.00 € | ||
| 10mg | 93.00 € | ||
| 25mg | 169.00 € | ||
| 50mg | 295.00 € | ||
| 100mg | 428.00 € | ||
| 200mg | 594.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
BMY-14802 hydrochloride
CAS:105565-55-7
BMY-14802 hydrochloride (BMS 181100 hydrochloride) is a selective antagonist of σ receptor (IC50 = 112 …
Formula:
C18H23ClF2N4O
Purity:
98.64%
Color and Shape:
Solid
Molecular weight:
384.85
Ref: TM-T22612
| 1mg | 35.00 € | ||
| 5mg | 75.00 € | ||
| 10mg | 109.00 € | ||
| 25mg | 226.00 € | ||
| 50mg | 385.00 € | ||
| 100mg | 574.00 € | ||
| 500mg | 1,239.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Glemanserin
CAS:107703-78-6
Glemanserin (MDL11939) is a specific 5-HT2A antagonist with Ki values of 0.54 nM, 2.5 nM …
Formula:
C20H25NO
Purity:
99.52%
Color and Shape:
Solid
Molecular weight:
295.42
Ref: TM-T22964
| 1mg | 40.00 € | ||
| 1ml | 89.00 € | ||
| 5mg | 86.00 € | ||
| 10mg | 123.00 € | ||
| 25mg | 269.00 € | ||
| 50mg | 423.00 € | ||
| 100mg | 625.00 € | ||
| 500mg | 1,327.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
ReN-1869 hydrochloride
CAS:170149-76-5
ReN 1869 hydrochloride is a novel, selective antagonist of histamine H1 receptor.
Formula:
C24H28ClNO2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
397.94
Ref: TM-T12703
| 25mg | 1,410.00 € | ||
| 50mg | 1,845.00 € | ||
| 100mg | 2,329.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
L-365260
CAS:118101-09-0
L-365260 is a nonpeptide gastrin and cerebral cholecystokinin receptor (CCK-B) antagonist used in the study …
Formula:
C24H22N4O2
Purity:
99.75%
Color and Shape:
Solid
Molecular weight:
398.46
Ref: TM-T22895
| 1mg | 186.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Amosulalol
CAS:85320-68-9
Amosulalol is a combined alpha and beta adrenoceptor antagonist.
Formula:
C18H24N2O5S
Purity:
98.91%
Color and Shape:
Solid
Molecular weight:
380.46
Ref: TM-T30027
| 1mg | 182.00 € | ||
| 1ml | 452.00 € | ||
| 2mg | 272.00 € | ||
| 5mg | 416.00 € | ||
| 10mg | 615.00 € | ||
| 25mg | 917.00 € | ||
| 50mg | 1,287.00 € | ||
| 100mg | 1,761.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
OMDM-6
CAS:616884-67-4
OMDM-6 is a dual agonist of TRPV1(EC50 = 75 nM) and CB1 (Ki = 3.2 …
Formula:
C28H42N2O3
Purity:
99.49%
Color and Shape:
Solid
Molecular weight:
454.64
Ref: TM-T12307
| 1mg | 111.00 € | ||
| 1ml | 272.00 € | ||
| 5mg | 246.00 € | ||
| 10mg | 362.00 € | ||
| 25mg | 542.00 € | ||
| 50mg | 758.00 € | ||
| 100mg | 1,034.00 € | ||
| 200mg | 1,391.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
VUF 5574
CAS:280570-45-8
VUF 5574 is a selective antagonist of adenosine A3 receptor with a Ki of 4.03 …
Formula:
C21H17N5O2
Purity:
97.63%
Color and Shape:
Solid
Molecular weight:
371.39
Ref: TM-T23518
| 1mg | 55.00 € | ||
| 2mg | 83.00 € | ||
| 5mg | 109.00 € | ||
| 10mg | 133.00 € | ||
| 25mg | 277.00 € | ||
| 50mg | 402.00 € | ||
| 100mg | 550.00 € | ||
| 500mg | 1,096.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
BW 245C
CAS:72814-32-5
BW 245C is a DP1 agonist with an inhibitory effect on the aggregation response of …
Formula:
C19H32N2O5
Purity:
99.14%
Color and Shape:
Solid
Molecular weight:
368.47
Ref: TM-T14842
| 1mg | 189.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Ro 363
CAS:74513-77-2
RO 363: Potent β1-adrenoceptor agonist, boosts heart contractility, lowers diastolic pressure.
Formula:
C19H25NO6
Purity:
98%
Color and Shape:
Solid
Molecular weight:
363.4
Ref: TM-T16769
| 25mg | 1,410.00 € | ||
| 50mg | 1,845.00 € | ||
| 100mg | 2,329.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
ML 10302 hydrochloride
CAS:186826-17-5
ML 10302 hydrochloride is a specific agonist 5-HT4 and binds 5-HT receptors with Kis of …
Formula:
C15H22Cl2N2O3
Purity:
100%
Color and Shape:
Solid
Molecular weight:
349.25
Ref: TM-T22992
| 1mg | 52.00 € | ||
| 5mg | 93.00 € | ||
| 10mg | 115.00 € | ||
| 25mg | 239.00 € | ||
| 50mg | 441.00 € | ||
| 100mg | 542.00 € | ||
| 500mg | 1,184.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
48740 RP
CAS:93363-11-2
48740 RP (RP 55779) is an antagonist of platelet-activating factor.
Formula:
C12H11N3OS
Purity:
99.4%
Color and Shape:
Solid
Molecular weight:
245.3
Ref: TM-T10159
| 1mg | 349.00 € | ||
| 1ml | 564.00 € | ||
| 5mg | 556.00 € | ||
| 10mg | 888.00 € | ||
| 25mg | 1,312.00 € | ||
| 50mg | 1,778.00 € | ||
| 100mg | 2,382.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
GRI977143
CAS:325850-81-5
GRI977143: selective LPA2 agonist (EC50=3.3μM), blocks caspases 3/7/8/9, limits DNA fragmentation.
Formula:
C22H17NO4S
Purity:
98.07%
Color and Shape:
Solid
Molecular weight:
391.44
Ref: TM-T22812
| 1mg | 39.00 € | ||
| 5mg | 82.00 € | ||
| 10mg | 129.00 € | ||
| 25mg | 264.00 € | ||
| 50mg | 423.00 € | ||
| 100mg | 625.00 € | ||
| 500mg | 1,333.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
PPTN hydrochloride
CAS:1992047-65-0
PPTN hydrochloride is a potent, high-affinity, competitive, highly selective P2Y14 receptor antagonist (KB: 434 pM), …
Formula:
C29H25ClF3NO2
Purity:
99.94%
Color and Shape:
Solid
Molecular weight:
511.96
Ref: TM-T63534
| 1mg | 48.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 157.00 € | ||
| 25mg | 300.00 € | ||
| 50mg | 462.00 € | ||
| 100mg | 671.00 € | ||
| 500mg | 1,412.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Laropiprant
CAS:571170-77-9
Laropiprant (MK-0524) is a potent and selective antagonist of prostaglandin D2 (PGD2) receptor (DP) such …
Formula:
C21H19ClFNO4S
Purity:
98.24% - 99.97%
Color and Shape:
Solid
Molecular weight:
435.9
Ref: TM-T15712
| 1mg | 59.00 € | ||
| 1ml | 142.00 € | ||
| 2mg | 84.00 € | ||
| 5mg | 128.00 € | ||
| 10mg | 179.00 € | ||
| 25mg | 358.00 € | ||
| 50mg | 552.00 € | ||
| 100mg | 785.00 € | ||
| 500mg | 1,568.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
KUL-7211 racemate
CAS:911196-40-2
KUL 7211, a selective β-adrenoceptor agonist, exists as a racemate, referred to as KUL 7211 …
Formula:
C19H23NO5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
345.39
Ref: TM-T11786
| 25mg | 1,410.00 € | ||
| 50mg | 1,845.00 € | ||
| 100mg | 2,329.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
UNC9975
CAS:1354030-19-5
UNC9975 is a D(2) receptor agonist with antipsychotic activity used in the study of neurologic …
Formula:
C23H28Cl2N4O2
Purity:
99.02% - 99.02%
Color and Shape:
Solid
Molecular weight:
463.4
Ref: TM-T29064
| 1mg | 277.00 € | ||
| 5mg | 682.00 € | ||
| 10mg | 932.00 € | ||
| 25mg | 1,435.00 € | ||
| 50mg | 1,869.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
CP 96021
CAS:139401-43-7
"CP 96021 is an antagonist of 5-HT1/2 receptors, with anti-inflammatory and anti-ulcer effects for treating …
Formula:
C29H21FN4OS
Purity:
97.81% - 99.11%
Color and Shape:
Soild
Molecular weight:
492.57
Ref: TM-T10872L
| 1mg | 181.00 € | ||
| 1ml | 509.00 € | ||
| 5mg | 416.00 € | ||
| 10mg | 614.00 € | ||
| 25mg | 922.00 € | ||
| 50mg | 1,281.00 € | ||
| 100mg | 1,756.00 € | ||
| 500mg | 3,531.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
