G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Rp-cAMPS sodium
CAS:142439-94-9
Rp-cAMPS sodium is a phosphorothioate analog of cAMP, a PKA inhibitor and cAMP antagonist that …
Formula:
C10H11N5NaO5PS
Purity:
99.71%
Color and Shape:
Liquid
Molecular weight:
367.25
Ref: TM-T36679
| 1mg | 275.00 € |
Estimated delivery in United States, on Monday 3 Feb 2025
WAY208466 dihydrochloride
CAS:1207064-61-6
WAY208466 dihydrochloride is a 5-HT6 receptor agonist (EC50=7.3 nM) with antidepressant and anxiolytic activity.
Formula:
C17H20Cl2FN3O2S
Purity:
98.43%
Color and Shape:
Solid
Molecular weight:
420.33
Ref: TM-T23527
| 1mg | 64.00 € |
Estimated delivery in United States, on Monday 3 Feb 2025
AM6545
CAS:1245626-05-4
AM6545 is a CB1 receptor antagonist used in the study of obesity and diabetes.
Formula:
C26H23Cl2N5O3S
Purity:
97.03%
Color and Shape:
Solid
Molecular weight:
556.46
Ref: TM-T22563
| 1mg | 96.00 € | ||
| 5mg | 201.00 € | ||
| 10mg | 297.00 € | ||
| 25mg | 674.00 € | ||
| 50mg | 920.00 € |
Estimated delivery in United States, on Monday 3 Feb 2025
GSK1521498
CAS:1426543-84-1
GSK1521498 is a selective antagonist of the μ-opioid receptor (MOR).
Formula:
C24H23F2N4O4P
Purity:
98%
Color and Shape:
Solid
Molecular weight:
500.43
Ref: TM-T11479
| 25mg | 1,410.00 € | ||
| 50mg | 1,845.00 € | ||
| 100mg | 2,329.00 € |
Estimated delivery in United States, on Monday 3 Feb 2025
LP44 hydrochloride
CAS:824958-12-5
LP44 hydrochloride is a 5-HT7 agonist with analgesic effects on formalin-induced orofacial pain in mice …
Formula:
C27H38ClN3OS
Purity:
98.06%
Color and Shape:
Solid
Molecular weight:
488.13
Ref: TM-T22931
| 1mg | 38.00 € |
Estimated delivery in United States, on Monday 3 Feb 2025
Molindone
CAS:7416-34-4
Molindone: antipsychotic for schizophrenia; blocks dopamine, often paired with serotonin; dosage affects error/response rates.
Formula:
C16H24N2O2
Purity:
98% - 99.37%
Color and Shape:
Off-White Solid
Molecular weight:
276.37
Ref: TM-T21432
| 1mg | 325.00 € | ||
| 5mg | 769.00 € | ||
| 10mg | 1,054.00 € | ||
| 25mg | 1,477.00 € | ||
| 50mg | 1,846.00 € | ||
| 100mg | 2,331.00 € | ||
| 500mg | 4,547.00 € |
Estimated delivery in United States, on Monday 3 Feb 2025
Repinotan
CAS:144980-29-0
Repinotan (BAY x 3702 free base) is a 5-HT1A receptor agonist used in acute ischemic …
Formula:
C21H24N2O4S
Purity:
99%
Color and Shape:
Liquid
Molecular weight:
400.49
Ref: TM-T61934
| 1mg | 273.00 € | ||
| 5mg | 673.00 € | ||
| 10mg | 920.00 € | ||
| 25mg | 1,416.00 € | ||
| 50mg | 1,845.00 € |
Estimated delivery in United States, on Monday 3 Feb 2025
LX-2931
CAS:948840-25-3
LX-2931(LX-3305) is a sphingosine-1-phosphate cleavage enzyme (S1P) inhibitor for the treatment of rheumatoid arthritis.
Formula:
C9H15N3O5
Purity:
100% - 99.83%
Color and Shape:
Solid
Molecular weight:
245.23
Ref: TM-T27864
| 1mg | 241.00 € | ||
| 5mg | 596.00 € | ||
| 10mg | 848.00 € | ||
| 25mg | 1,280.00 € | ||
| 50mg | 1,723.00 € |
Estimated delivery in United States, on Monday 3 Feb 2025
AZ12216052
CAS:1290628-31-7
AZ12216052 is a GRP8 antagonist with anxiolytic and anti-inflammatory activity and can be used to …
Formula:
C19H22BrNOS
Purity:
99.29%
Color and Shape:
Solid
Molecular weight:
392.35
Ref: TM-T26701
| 1mg | 56.00 € | ||
| 5mg | 118.00 € | ||
| 10mg | 183.00 € | ||
| 25mg | 321.00 € | ||
| 50mg | 476.00 € | ||
| 100mg | 678.00 € |
Estimated delivery in United States, on Monday 3 Feb 2025
Levobunolol hydrochloride
CAS:27912-14-7
Levobunolol hydrochloride is a non-selective blocker of β-adrenergic receptor and can be used in studies …
Formula:
C17H26ClNO3
Purity:
100% - 98.49%
Color and Shape:
Solid
Molecular weight:
327.85
Ref: TM-T15742
| 10mg | 64.00 € | ||
| 25mg | 95.00 € | ||
| 1mL*10mM (DMSO) | 70.00 € |
Estimated delivery in United States, on Monday 3 Feb 2025
PNU-282987 free base
CAS:711085-63-1
PNU-282987 is an α7 nAChR agonist (EC50=154 nM) and a 5-HT3 antagonist (IC50=4541 nM) for …
Formula:
C14H17ClN2O
Purity:
99.64%
Color and Shape:
Liquid
Molecular weight:
264.75
Ref: TM-T60437
| 1mg | 55.00 € | ||
| 5mg | 111.00 € | ||
| 10mg | 201.00 € | ||
| 25mg | 392.00 € | ||
| 50mg | 727.00 € | ||
| 100mg | 1,020.00 € | ||
| 500mg | 2,039.00 € |
Estimated delivery in United States, on Monday 3 Feb 2025
ATC 0175 hydrochloride
CAS:510733-97-8
ATC 0175 hydrochloride is an orally active melanocyte concentrating hormone 1 receptor antagonist that is …
Formula:
C23H26ClF2N5O
Purity:
99.84%
Color and Shape:
Solid
Molecular weight:
461.93
Ref: TM-T22591
| 1mg | 78.00 € | ||
| 5mg | 157.00 € | ||
| 10mg | 245.00 € | ||
| 25mg | 502.00 € | ||
| 50mg | 852.00 € | ||
| 100mg | 1,384.00 € | ||
| 500mg | 2,777.00 € |
Estimated delivery in United States, on Monday 3 Feb 2025
Vapitadine dihydrochloride
CAS:279253-83-7
Vapitadine dihydrochloride(R-129160 2HCl) is a novel, potent, selective and non-sedating compound with inhibitory effects on …
Formula:
C17H22Cl2N4O
Purity:
100% - 99.92%
Color and Shape:
Solid
Molecular weight:
369.29
Ref: TM-T29096
| 1mg | 241.00 € | ||
| 5mg | 600.00 € | ||
| 10mg | 852.00 € | ||
| 25mg | 1,280.00 € | ||
| 50mg | 1,718.00 € |
Estimated delivery in United States, on Monday 3 Feb 2025
Aligeron
CAS:70713-45-0
Aligeron is a non-selective prostaglandin (PG) antagonist that inhibits PGF2α- and PGE2-induced decreases in blood …
Formula:
C20H24N2
Purity:
100% - 98.57%
Color and Shape:
Liquid
Molecular weight:
292.42
Ref: TM-T36619
| 1mg | 651.00 € | ||
| 5mg | 1,682.00 € |
Estimated delivery in United States, on Monday 3 Feb 2025
PSB-16133 sodium
CAS:2089035-40-3
PSB-16133 sodium is a selective P2Y purine receptor variant antagonist with an IC of 233 …
Formula:
C28H21N2NaO5S2
Purity:
98.08% - 99.36%
Color and Shape:
Solid
Molecular weight:
552.60
Ref: TM-T28463
| 1mg | 273.00 € | ||
| 2mg | 406.00 € | ||
| 5mg | 673.00 € | ||
| 10mg | 919.00 € | ||
| 25mg | 1,416.00 € | ||
| 50mg | 1,838.00 € |
Estimated delivery in United States, on Monday 3 Feb 2025
Liafensine
CAS:1198790-53-2
Liafensine(BMS-820836): Selective inhibitor for serotonin, norepinephrine, dopamine reuptake; targets major depression, CNS disorders.
Formula:
C24H22N4
Purity:
99.46%
Color and Shape:
Solid
Molecular weight:
366.46
Ref: TM-T32737
| 1mg | 360.00 € | ||
| 5mg | 858.00 € | ||
| 10mg | 1,175.00 € | ||
| 25mg | 1,737.00 € | ||
| 50mg | 2,354.00 € |
Estimated delivery in United States, on Monday 3 Feb 2025
2-Iodomelatonin
CAS:93515-00-5
2-Iodomelatonin, Ki 28 pM, is an MT1 agonist, >5x selective over MT2, used to map …
Formula:
C13H15IN2O2
Purity:
100%
Color and Shape:
Solid
Molecular weight:
358.17
Ref: TM-T10073
| 10mg | 45.00 € | ||
| 25mg | 82.00 € | ||
| 50mg | 123.00 € | ||
| 100mg | 185.00 € | ||
| 200mg | 277.00 € | ||
| 500mg | To inquire | ||
| 1mL*10mM (DMSO) | 36.00 € |
Estimated delivery in United States, on Monday 3 Feb 2025
YIL 781
CAS:875258-85-8
YIL 781 is a selective ghrelin receptor antagonist (GHS-R1a) (Ki = 17 nM), showing a …
Formula:
C24H28FN3O2
Purity:
99.3%
Color and Shape:
Solid
Molecular weight:
409.5
Ref: TM-T23543
| 1mg | 52.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 149.00 € | ||
| 25mg | 306.00 € | ||
| 50mg | 461.00 € | ||
| 100mg | 644.00 € | ||
| 1mL*10mM (DMSO) | 123.00 € |
Estimated delivery in United States, on Monday 3 Feb 2025
Terbogrel
CAS:149979-74-8
Terbogrel is an antiplatelet drug, blocking thromboxane A2 receptor/synthase. Helps prevent clots.
Formula:
C23H27N5O2
Purity:
99.65%
Color and Shape:
Solid
Molecular weight:
405.49
Ref: TM-T17039
| 1mg | 183.00 € | ||
| 5mg | 435.00 € | ||
| 10mg | 635.00 € | ||
| 25mg | 1,000.00 € | ||
| 50mg | 1,336.00 € | ||
| 100mg | 1,803.00 € |
Estimated delivery in United States, on Monday 3 Feb 2025
Acifran
CAS:72420-38-3
Acifran (AY 25712) is an HM74A/GPR109A and GPR109B agonist and displays antihyperlipidemic activity.
Formula:
C12H10O4
Purity:
98.65%
Color and Shape:
Solid
Molecular weight:
218.21
Ref: TM-T22547
| 1mg | 47.00 € | ||
| 5mg | 83.00 € | ||
| 10mg | 125.00 € | ||
| 25mg | 245.00 € | ||
| 50mg | 398.00 € | ||
| 100mg | 580.00 € | ||
| 500mg | 1,190.00 € |
Estimated delivery in United States, on Monday 3 Feb 2025
