G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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PF-03654746
CAS:935840-31-6
PF-03654746: selective H3 antagonist, boosts cognition in Alzheimer's, may treat allergic rhinitis.
Formula:
C18H24F2N2O
Purity:
98.83% - 99.1%
Color and Shape:
Solid
Molecular weight:
322.39
Ref: TM-T16476
| 1mg | 236.00 € | ||
| 5mg | 590.00 € | ||
| 10mg | 822.00 € | ||
| 25mg | 1,262.00 € | ||
| 50mg | 1,641.00 € | ||
| 100mg | 2,470.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
ICI 199,441 hydrochloride
CAS:115199-84-3
ICI 199,441 hydrochloride is a potent, selective agonist of κ-opioid receptor.
Formula:
C21H25Cl3N2O
Purity:
99.46%
Color and Shape:
Solid
Molecular weight:
427.8
Ref: TM-T22849
| 2mg | 34.00 € | ||
| 5mg | 49.00 € | ||
| 10mg | 78.00 € | ||
| 25mg | 141.00 € | ||
| 50mg | 218.00 € | ||
| 100mg | 320.00 € | ||
| 200mg | 449.00 € | ||
| 1mL*10mM (DMSO) | 60.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
Ecastolol
CAS:77695-52-4
Ecastolol has anti-angina activity and is an adrenergic receptor antagonist.
Formula:
C26H33N3O6
Purity:
98.1%
Color and Shape:
Solid
Molecular weight:
483.56
Ref: TM-T11148
| 1mg | 361.00 € | ||
| 5mg | 721.00 € | ||
| 10mg | 919.00 € | ||
| 25mg | 1,443.00 € | ||
| 50mg | 1,843.00 € | ||
| 100mg | 2,615.00 € | ||
| 1mL*10mM (DMSO) | 923.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
cis-Urocanic acid
CAS:7699-35-6
cis-Urocanic acid ((E)-Urocanic acid) is a 5-HT2A receptor agonist (Kd: 4.6 nM).
Formula:
C6H6N2O2
Purity:
99.78%
Color and Shape:
Solid
Molecular weight:
138.12
Ref: TM-T10824
| 1mg | 204.00 € | ||
| 5mg | 430.00 € | ||
| 10mg | 635.00 € | ||
| 25mg | 1,000.00 € | ||
| 50mg | 1,346.00 € | ||
| 100mg | 1,810.00 € | ||
| 500mg | 3,611.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
RS 56812 hydrochloride
CAS:143339-12-2
5-HT3 partial agonist
Formula:
C18H22ClN3O2
Purity:
97.69%
Color and Shape:
Solid
Molecular weight:
347.84
Ref: TM-T23264
| 1mg | 64.00 € | ||
| 2mg | 90.00 € | ||
| 5mg | 131.00 € | ||
| 10mg | 185.00 € | ||
| 25mg | 431.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
SLF1081851
CAS:2763730-97-6
SLF1081851 is a Spns2 inhibitor. SLF1081851 inhibits S1P release with IC50 of 1.93 μM.
Formula:
C21H33N3O
Purity:
98.57%
Color and Shape:
Solid
Molecular weight:
343.51
Ref: TM-T61112
| 1mg | 55.00 € | ||
| 5mg | 118.00 € | ||
| 10mg | 183.00 € | ||
| 25mg | 392.00 € | ||
| 50mg | 586.00 € | ||
| 100mg | 835.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
Butofilolol
CAS:58930-32-8
Butofilolol is a novel beta-blocker with antihypertensive activity and can be used to study hypertension.
Formula:
C17H26FNO3
Purity:
100% - 99%
Color and Shape:
Solid
Molecular weight:
311.392
Ref: TM-T60773
| 1mg | 276.00 € | ||
| 5mg | 679.00 € | ||
| 10mg | 928.00 € | ||
| 25mg | 1,430.00 € | ||
| 50mg | 1,862.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
GR 89696 fumarate
CAS:126766-32-3
GR 89696 fumarate is a highly selective κ2 opioid receptor agonist (IC50 = 0.04nM) with …
Formula:
C23H29Cl2N3O7
Purity:
99.19%
Color and Shape:
Solid
Molecular weight:
530.4
Ref: TM-T22810
| 5mg | 63.00 € | ||
| 10mg | 94.00 € | ||
| 25mg | 159.00 € | ||
| 50mg | 222.00 € | ||
| 100mg | 328.00 € | ||
| 1mL*10mM (DMSO) | 78.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
Sitaxsentan
CAS:184036-34-8
Sitaxsentan (TBC-11251), a selective ETA receptor antagonist, prevents vasoconstriction by blocking endothelin.
Formula:
C18H15ClN2O6S2
Purity:
97.99% - 99.34%
Color and Shape:
Solid
Molecular weight:
454.9
Ref: TM-T12924
| 1mg | 88.00 € | ||
| 5mg | 198.00 € | ||
| 10mg | 322.00 € | ||
| 25mg | 499.00 € | ||
| 50mg | 678.00 € | ||
| 100mg | 922.00 € | ||
| 500mg | 1,838.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
Tiopinac
CAS:61220-69-7
Tiopinac: tricyclic with anti-inflammatory, analgesic, antipyretic properties; inhibits prostaglandin synthesis; mild anti-platelet effects in humans.
Formula:
C16H12O3S
Purity:
100%
Color and Shape:
Solid
Molecular weight:
284.33
Ref: TM-T17101
| 1mg | 197.00 € | ||
| 5mg | 497.00 € | ||
| 10mg | 707.00 € | ||
| 25mg | 1,059.00 € | ||
| 50mg | 1,437.00 € | ||
| 100mg | 1,872.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
Pirmagrel
CAS:85691-74-3
pirmagrel is a potent thromboxane synthase inhibitor.
Formula:
C13H16N2O2
Purity:
98.83%
Color and Shape:
Solid
Molecular weight:
232.28
Ref: TM-T67958
| 1mg | 81.00 € | ||
| 5mg | 172.00 € | ||
| 10mg | 253.00 € | ||
| 25mg | 470.00 € | ||
| 50mg | 636.00 € | ||
| 100mg | 920.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
Odapipam
CAS:131796-63-9
Odapipam is a selective and high affinity antagonist of benzazepine dopamine D1 receptor (Kd of …
Formula:
C19H20ClNO2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
329.82
Ref: TM-T12288
| 25mg | 1,132.00 € | ||
| 50mg | 1,476.00 € | ||
| 100mg | 2,270.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
SR144528
CAS:192703-06-3
SR144528 is an antagonist of the CB2 receptor (Ki = 0.6 nM) and inhibits microsomal …
Formula:
C29H34ClN3O
Purity:
99.6%
Color and Shape:
Solid
Molecular weight:
476.05
Ref: TM-T16928
| 1mg | 42.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 152.00 € | ||
| 25mg | 332.00 € | ||
| 50mg | 497.00 € | ||
| 100mg | 719.00 € | ||
| 1mL*10mM (DMSO) | 94.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
ICI 204,448
CAS:121264-04-8
ICI 204,448 is a potent κ-opioid agonist with potential analgesic activity for the study of …
Formula:
C23H27Cl3N2O4
Purity:
100%
Color and Shape:
Solid
Molecular weight:
501.83
Ref: TM-T22850
| 1mg | 52.00 € | ||
| 5mg | 109.00 € | ||
| 10mg | 172.00 € | ||
| 25mg | 276.00 € | ||
| 50mg | 421.00 € | ||
| 100mg | 606.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
ORL1 antagonist 1
CAS:1174985-59-1
ORL1 antagonist 1 is an o antagonist of pioid receptor-like 1 (ORL1) (IC50 of 61 …
Formula:
C20H22ClN5
Purity:
97.87%
Color and Shape:
Solid
Molecular weight:
367.88
Ref: TM-T12320
| 1mg | 113.00 € | ||
| 5mg | 251.00 € | ||
| 10mg | 368.00 € | ||
| 25mg | 551.00 € | ||
| 50mg | 776.00 € | ||
| 100mg | 1,043.00 € | ||
| 500mg | 2,103.00 € | ||
| 1mL*10mM (DMSO) | 262.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
(S)-(-)-Propranolol hydrochloride
CAS:4199-10-4
(S)-(-)-Propranolol hydrochloride is an adrenergic receptor antagonist with potential anticancer activity that may improve the …
Formula:
C16H22ClNO2
Purity:
99.02%
Color and Shape:
Solid
Molecular weight:
295.8
Ref: TM-T23302
| 50mg | 39.00 € | ||
| 100mg | 59.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
Befetupitant
CAS:290296-68-3
Befupupitant(Ro67-5930) is a potent and selective tachykinin 1 receptor (NK1R) antagonist for the study of …
Formula:
C29H29F6N3O2
Purity:
98.67%
Color and Shape:
Solid
Molecular weight:
565.55
Ref: TM-T14524
| 1mg | 457.00 € | ||
| 5mg | 994.00 € | ||
| 10mg | 1,212.00 € | ||
| 25mg | 1,602.00 € | ||
| 50mg | 2,024.00 € | ||
| 100mg | 2,600.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
Masupirdine mesylate
CAS:1791396-46-7
Masupirdine mesylate (SUVN-502 mesylate) is a 5-HT6 receptor antagonist.Masupirdine mesylate is used to study neurological …
Formula:
C23H32BrN3O9S3
Purity:
99.48%
Color and Shape:
Solid
Molecular weight:
670.61
Ref: TM-T11949
| 1mg | 46.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 143.00 € | ||
| 25mg | 248.00 € | ||
| 50mg | 373.00 € | ||
| 100mg | 607.00 € | ||
| 1mL*10mM (DMSO) | 129.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
PF-184298
CAS:813447-40-4
PF-184298 is a serotonin and norepinephrine monoamine reuptake inhibitor (SNRI) that inhibits dopamine reuptake.
Formula:
C15H20Cl2N2O
Purity:
98.30%
Color and Shape:
Solid
Molecular weight:
315.24
Ref: TM-T28380
| 1mg | 276.00 € | ||
| 5mg | 680.00 € | ||
| 10mg | 930.00 € | ||
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
Aminaftone
CAS:14748-94-8
Aminaftone, a derivative of 4-aminobenzoic acid, inhibits endothelin-1 (ET-1) production and can be used to …
Formula:
C18H15NO4
Purity:
96.31% - 99.39%
Color and Shape:
Solid
Molecular weight:
309.32
Ref: TM-T14219
| 1mg | 325.00 € | ||
| 5mg | 901.00 € | ||
| 10mg | 1,114.00 € | ||
| 25mg | 1,476.00 € | ||
| 50mg | 1,839.00 € | ||
| 100mg | 2,322.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
