G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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N6-Cyclopentyladenosine
CAS:41552-82-3
N6-Cyclopentyladenosine (CPA) is a selective agonist of the adenosine A1 receptor and can be used …
Formula:
C15H21N5O4
Purity:
99.84%
Color and Shape:
Solid
Molecular weight:
335.36
Ref: TM-T16263
| 5mg | 35.00 € | ||
| 10mg | 49.00 € | ||
| 25mg | 71.00 € | ||
| 50mg | 96.00 € | ||
| 100mg | 157.00 € | ||
| 500mg | 369.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
Rp-cAMPS sodium
CAS:142439-94-9
Rp-cAMPS sodium is a phosphorothioate analog of cAMP, a PKA inhibitor and cAMP antagonist that …
Formula:
C10H11N5NaO5PS
Purity:
99.71%
Color and Shape:
Solid
Molecular weight:
367.25
Ref: TM-T36679
| 1mg | 275.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
WAY208466 dihydrochloride
CAS:1207064-61-6
WAY208466 dihydrochloride is a 5-HT6 receptor agonist (EC50=7.3 nM) with antidepressant and anxiolytic activity.
Formula:
C17H20Cl2FN3O2S
Purity:
98.43%
Color and Shape:
Solid
Molecular weight:
420.33
Ref: TM-T23527
| 1mg | 64.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
ISAM-140
CAS:932191-62-3
ISAM-140 is a potent and highly selective antagonist of A2B adenosine receptor.
Formula:
C19H19N3O3
Purity:
97.41%
Color and Shape:
Solid
Molecular weight:
337.37
Ref: TM-T27629
| 1mg | 57.00 € | ||
| 5mg | 123.00 € | ||
| 10mg | 172.00 € | ||
| 25mg | 277.00 € | ||
| 50mg | 418.00 € | ||
| 100mg | 592.00 € | ||
| 500mg | 1,163.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
AM6545
CAS:1245626-05-4
AM6545 is a CB1 receptor antagonist used in the study of obesity and diabetes.
Formula:
C26H23Cl2N5O3S
Purity:
97.03%
Color and Shape:
Solid
Molecular weight:
556.46
Ref: TM-T22563
| 1mg | 96.00 € | ||
| 5mg | 201.00 € | ||
| 10mg | 297.00 € | ||
| 25mg | 674.00 € | ||
| 50mg | 920.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
Palonosetron
CAS:135729-61-2
Palonosetron, a 5-HT3 antagonist with Ki of 0.17 nM, is used in the prevention and …
Formula:
C19H24N2O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
296.41
Ref: TM-T22393
| 25mg | 1,406.00 € | ||
| 50mg | 1,852.00 € | ||
| 100mg | 2,338.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
SCH 546738
CAS:906805-42-3
SCH 546738 is an orally available, selective and potent CXCR3 antagonist that attenuates the development …
Formula:
C23H31Cl2N7O
Purity:
98.67%
Color and Shape:
Solid
Molecular weight:
492.45
Ref: TM-T16863
| 2mg | 215.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
GSK1521498
CAS:1426543-84-1
GSK1521498 is a selective antagonist of the μ-opioid receptor (MOR).
Formula:
C24H23F2N4O4P
Purity:
98%
Color and Shape:
Solid
Molecular weight:
500.43
Ref: TM-T11479
| 25mg | 1,410.00 € | ||
| 50mg | 1,845.00 € | ||
| 100mg | 2,329.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
LP44 hydrochloride
CAS:824958-12-5
LP44 hydrochloride is a 5-HT7 agonist with analgesic effects on formalin-induced orofacial pain in mice …
Formula:
C27H38ClN3OS
Purity:
98.06%
Color and Shape:
Solid
Molecular weight:
488.13
Ref: TM-T22931
| 1mg | 38.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
Dicarbine
CAS:17411-19-7
Double carbene blocks dopamine receptors, aiding schizophrenia and alcoholism research; it maintains defense reflexes despite …
Formula:
C13H18N2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
202.3
Ref: TM-T13652
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
LX-2931
CAS:948840-25-3
LX-2931(LX-3305) is a sphingosine-1-phosphate cleavage enzyme (S1P) inhibitor for the treatment of rheumatoid arthritis.
Formula:
C9H15N3O5
Purity:
100% - 99.83%
Color and Shape:
Solid
Molecular weight:
245.23
Ref: TM-T27864
| 1mg | 241.00 € | ||
| 5mg | 596.00 € | ||
| 10mg | 848.00 € | ||
| 25mg | 1,280.00 € | ||
| 50mg | 1,723.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
CRTh2 antagonist 1
CAS:1379445-54-1
CRTh2 antagonist 1 is a CRTh2 antagonist (IC50: 89 nM).
Formula:
C23H25N3O5S
Purity:
97.39%
Color and Shape:
Solid
Molecular weight:
455.53
Ref: TM-T10084
| 1mg | 113.00 € | ||
| 5mg | 249.00 € | ||
| 10mg | 366.00 € | ||
| 25mg | 550.00 € | ||
| 50mg | 769.00 € | ||
| 100mg | 1,049.00 € | ||
| 500mg | 2,098.00 € | ||
| 1mL*10mM (DMSO) | 281.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
A-65186
CAS:119295-94-2
A-65186 is a CCK antagonist used in the study of inflammation and gastrointestinal tract injury.
Formula:
C25H35N3O4
Purity:
98.37% - 99.94%
Color and Shape:
Solid
Molecular weight:
441.56
Ref: TM-T26483
| 1mg | 277.00 € | ||
| 5mg | 682.00 € | ||
| 10mg | 932.00 € | ||
| 25mg | 1,435.00 € | ||
| 50mg | 1,869.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
Burixafor hydrobromide
CAS:1191450-19-7
Burixafor hydrobromide is an oral CXCR4 blocker with anti-angiogenic properties, potentially treating choroid neovascularization.
Formula:
C27H52BrN8O3P
Purity:
98%
Color and Shape:
Solid
Molecular weight:
647.644
Ref: TM-T10635
| 25mg | To inquire | ||
| 50mg | To inquire | ||
| 100mg | To inquire |
Estimated delivery in United States, on Tuesday 14 Jan 2025
TC LPA5 4
CAS:1393814-38-4
TC LPA5 4 is a LPA5 receptor antagonist.
Formula:
C23H23ClN2O3
Purity:
99.05%
Color and Shape:
Solid
Molecular weight:
410.89
Ref: TM-T23438
| 1mg | 58.00 € | ||
| 5mg | 124.00 € | ||
| 10mg | 183.00 € | ||
| 25mg | 425.00 € | ||
| 50mg | 625.00 € | ||
| 100mg | 891.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
GPR35 agonist 3
CAS:123021-85-2
GPR35 agonist 3 is a synthetic GPR35 agonist used in the study of cancer, type …
Formula:
C12H9NO5S
Purity:
98.79%
Color and Shape:
Solid
Molecular weight:
279.27
Ref: TM-T72755
| 1mg | 49.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 151.00 € | ||
| 25mg | 301.00 € | ||
| 50mg | 482.00 € | ||
| 100mg | 771.00 € | ||
| 500mg | 1,539.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
L-745870
CAS:158985-00-3
L-745870 is a selective dopamine D4 antagonist, brain-penetrant, with lesser affinity for D2/D3 receptors (Ki: …
Formula:
C18H19ClN4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
326.82
Ref: TM-T11799L
| 2mg | 41.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
ATC 0175 hydrochloride
CAS:510733-97-8
ATC 0175 hydrochloride is an orally active melanocyte concentrating hormone 1 receptor antagonist that is …
Formula:
C23H26ClF2N5O
Purity:
99.84%
Color and Shape:
Solid
Molecular weight:
461.93
Ref: TM-T22591
| 1mg | 78.00 € | ||
| 5mg | 157.00 € | ||
| 10mg | 245.00 € | ||
| 25mg | 502.00 € | ||
| 50mg | 852.00 € | ||
| 100mg | 1,384.00 € | ||
| 500mg | 2,777.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
Vapitadine dihydrochloride
CAS:279253-83-7
Vapitadine dihydrochloride(R-129160 2HCl) is a novel, potent, selective and non-sedating compound with inhibitory effects on …
Formula:
C17H22Cl2N4O
Purity:
100% - 99.92%
Color and Shape:
Solid
Molecular weight:
369.29
Ref: TM-T29096
| 1mg | 241.00 € | ||
| 5mg | 600.00 € | ||
| 10mg | 852.00 € | ||
| 25mg | 1,280.00 € | ||
| 50mg | 1,718.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
Aligeron
CAS:70713-45-0
Aligeron is a non-selective prostaglandin (PG) antagonist that inhibits PGF2α- and PGE2-induced decreases in blood …
Formula:
C20H24N2
Purity:
100% - 98.57%
Color and Shape:
Solid
Molecular weight:
292.42
Ref: TM-T36619
| 1mg | 651.00 € | ||
| 5mg | 1,682.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
