G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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EMDT
CAS:263744-72-5
EMDT oxalate is a selective 5-HT6 agonist, and has antidepressant effects.
Formula:
C15H22N2O
Purity:
98.33% - 98.46%
Color and Shape:
Solid
Molecular weight:
246.35
Ref: TM-T11183
| 1mg | 91.00 € | ||
| 2mg | 123.00 € | ||
| 5mg | 168.00 € | ||
| 10mg | 211.00 € | ||
| 25mg | 467.00 € | ||
| 50mg | 680.00 € | ||
| 100mg | 926.00 € | ||
| 500mg | 1,838.00 € | ||
| 1mL*10mM (DMSO) | 167.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Ancarolol
CAS:75748-50-4
Ancarolol is a blocking agent of beta-adrenergic.
Formula:
C18H24N2O4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
332.39
Ref: TM-T14287
| 25mg | 1,410.00 € | ||
| 50mg | 1,845.00 € | ||
| 100mg | 2,329.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
LY 272015 hydrochloride
CAS:172895-15-7
LY 272015 hydrochloride is a 5-HT2B receptor antagonist.
Formula:
C21H25ClN2O2
Purity:
99.47%
Color and Shape:
Solid
Molecular weight:
372.89
Ref: TM-T22948
| 1mg | 50.00 € | ||
| 5mg | 126.00 € | ||
| 10mg | 195.00 € | ||
| 25mg | 418.00 € | ||
| 50mg | 668.00 € | ||
| 100mg | 1,059.00 € | ||
| 200mg | 1,426.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Tecalcet Hydrochloride
CAS:177172-49-5
Tecalcet Hydrochloride, an allosteric CaSR modulator, enhances extracellular Ca2+ sensitivity.
Formula:
C18H23Cl2NO
Purity:
99.44%
Color and Shape:
Solid
Molecular weight:
340.29
Ref: TM-T13918
| 2mg | 35.00 € | ||
| 5mg | 49.00 € | ||
| 10mg | 74.00 € | ||
| 25mg | 151.00 € | ||
| 50mg | 238.00 € | ||
| 100mg | 347.00 € | ||
| 200mg | To inquire | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Lintopride
CAS:107429-63-0
Lintopride is an antagonist of 5HT4. It has moderate 5HT3 antagonist properties.
Formula:
C14H19ClN4O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
310.78
Ref: TM-T15760
| 25mg | 1,410.00 € | ||
| 50mg | 1,838.00 € | ||
| 100mg | 2,322.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Wy 49051
CAS:113418-56-7
Wy 49051 is an orally active antagonist of H1 receptor(IC50 of 44 nM).
Formula:
C28H33N5O3
Purity:
97.9%
Color and Shape:
Solid
Molecular weight:
487.59
Ref: TM-T13352
| 1mg | 144.00 € | ||
| 5mg | 273.00 € | ||
| 10mg | 397.00 € | ||
| 25mg | 621.00 € | ||
| 50mg | 835.00 € | ||
| 100mg | 1,080.00 € | ||
| 200mg | 1,446.00 € | ||
| 1mL*10mM (DMSO) | 362.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Lusaperidone
CAS:214548-46-6
Kaerophyllin ( (-)-Kaerophylin) inhibits hepatic stellate cell activation and inhibits HSC activation to protect against …
Formula:
C22H21N3O2
Purity:
99.64%
Color and Shape:
Solid
Molecular weight:
359.42
Ref: TM-T11894
| 1mg | 131.00 € | ||
| 5mg | 305.00 € | ||
| 10mg | 491.00 € | ||
| 25mg | 1,012.00 € | ||
| 50mg | 1,718.00 € | ||
| 100mg | 2,524.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
ENMD-1068 HCl
CAS:789488-77-3
ENMD-1068 HCl (ENMD 1068) is a PAR-2 antagonist. ENMD-1068 HCl inhibits the development of endometriosis …
Formula:
C15H29N3O2
Purity:
95.79%
Color and Shape:
Solid
Molecular weight:
283.41
Ref: TM-T27267
| 10mg | 54.00 € | ||
| 25mg | 94.00 € | ||
| 50mg | 132.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Thiethylperazine dimaleate
CAS:1179-69-7
Thiethylperazine dimaleate (Thiethylperazine maleate) is an antagonist of the D2 receptor and H1 receptor.
Formula:
C30H37N3O8S2
Purity:
99.07%
Color and Shape:
Solid
Molecular weight:
631.76
Ref: TM-T17072
| 5mg | 52.00 € | ||
| 10mg | 79.00 € | ||
| 25mg | 128.00 € | ||
| 50mg | 207.00 € | ||
| 100mg | 319.00 € | ||
| 500mg | To inquire |
Estimated delivery in United States, on Monday 27 Jan 2025
PPTN
CAS:1160271-30-6
PPTN is a high-affinity, competitive and highly selective antagonist of P2Y14 receptor(KB value of 434 …
Formula:
C29H24F3NO2
Purity:
100%
Color and Shape:
Solid
Molecular weight:
475.5
Ref: TM-T12530
| 1mg | 113.00 € | ||
| 5mg | 250.00 € | ||
| 10mg | 367.00 € | ||
| 25mg | 550.00 € | ||
| 50mg | 775.00 € | ||
| 100mg | 1,040.00 € | ||
| 500mg | 2,098.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
KP136
CAS:76239-32-2
KP136 is an orally effective antiallergic compound (IC50: 76.1 μg/mL for histamine release and 63 …
Formula:
C16H18N4O3
Purity:
98.16% - 99.86%
Color and Shape:
Solid
Molecular weight:
314.34
Ref: TM-T15666
| 1mg | 275.00 € | ||
| 5mg | 676.00 € | ||
| 10mg | 924.00 € | ||
| 25mg | 1,410.00 € | ||
| 50mg | 1,847.00 € | ||
| 100mg | 2,331.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Zatosetron maleate
CAS:123482-23-5
Zatosetron maleate(LY 277359 maleate) is a potent and selective serotonin 5HT3 receptor antagonist for the …
Formula:
C23H29ClN2O6
Purity:
99.41%
Color and Shape:
Solid
Molecular weight:
464.94
Ref: TM-T17285
| 1mg | 650.00 € | ||
| 5mg | 1,671.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
NNC 63-0532
CAS:250685-44-0
NNC 63-0532 is a potentnociceptin receptor agonist, Ki=7.3 nM, EC50=305 nM.
Formula:
C27H29N3O3
Purity:
98.75%
Color and Shape:
Solid
Molecular weight:
443.54
Ref: TM-T23074
| 1mg | 49.00 € | ||
| 2mg | 63.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 140.00 € | ||
| 25mg | 277.00 € | ||
| 50mg | 439.00 € | ||
| 100mg | 626.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Aminaftone
CAS:14748-94-8
Aminaftone, a derivative of 4-aminobenzoic acid, inhibits endothelin-1 (ET-1) production and can be used to …
Formula:
C18H15NO4
Purity:
96.31% - 99.39%
Color and Shape:
Solid
Molecular weight:
309.32
Ref: TM-T14219
| 1mg | 325.00 € | ||
| 5mg | 901.00 € | ||
| 10mg | 1,114.00 € | ||
| 25mg | 1,476.00 € | ||
| 50mg | 1,839.00 € | ||
| 100mg | 2,322.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
MEDICA16
CAS:87272-20-6
MEDICA16: GPR40 agonist, GPR120 partial agonist, ATP-citrate lyase inhibitor, lowers TG, boosts insulin sensitivity in …
Formula:
C20H38O4
Purity:
99.13% - 99.85%
Color and Shape:
White Solid
Molecular weight:
342.51
Ref: TM-T22967
| 5mg | 63.00 € | ||
| 10mg | 95.00 € | ||
| 25mg | 174.00 € | ||
| 50mg | 300.00 € | ||
| 100mg | 434.00 € | ||
| 500mg | 905.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
SSR126768A
CAS:785048-28-4
SSR126768A is an oxytocin receptor antagonist that inhibits uterine contractions and may be used to …
Formula:
C33H31Cl2N3O4
Purity:
98.40%
Color and Shape:
Solid
Molecular weight:
604.52
Ref: TM-T28855
| 1mg | 325.00 € | ||
| 5mg | 900.00 € | ||
| 10mg | 1,114.00 € | ||
| 25mg | 1,476.00 € | ||
| 50mg | 1,838.00 € | ||
| 100mg | 2,320.00 € | ||
| 500mg | 6,458.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
(R)-(-)-α-Methylhistamine dihydrobromide
CAS:868698-49-1
(R)-(-)-α-Methylhistamine dihydrobromide is a potent and selective agonist of H3 histamine receptor( Kd of 50.3 …
Formula:
C6H13Br2N3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
287
Ref: TM-T12630
| 50mg | 1,783.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Abt-288
CAS:948845-91-8
ABT-288 is a selective and potent H3 antagonist for the treatment of mild to moderate …
Formula:
C23H24N4O
Purity:
98% - 98.84%
Color and Shape:
Solid
Molecular weight:
372.46
Ref: TM-T26526
| 1mg | 183.00 € | ||
| 5mg | 452.00 € | ||
| 10mg | 643.00 € | ||
| 25mg | 1,009.00 € | ||
| 50mg | 1,383.00 € | ||
| 100mg | 1,828.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
RG-12915
CAS:136174-04-4
RG-12915 is a selective antagonist of 5-HT3(IC50 value of 0.16 nM).
Formula:
C20H25ClN2O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
360.88
Ref: TM-T12716
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Nelonicline
CAS:1026134-63-3
Nelonicline is a selective agonist of neuronal nicotinic receptors.
Formula:
C17H19N3OS
Purity:
98%
Color and Shape:
Solid
Molecular weight:
313.42
Ref: TM-T16281
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
