G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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NPS ALX Compound 4a dihydrochloride
CAS:1781934-44-8
NPS ALX Compound 4a dihydrochloride is a potent and selective antagonist of 5-HT6 receptor (IC50 …
Formula:
C25H27Cl2N3O2S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
504.47
Ref: TM-T12262L
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Friday 24 Jan 2025
Bavisant
CAS:929622-08-2
Bavisant (JNJ-31001074) is a selective and orally active Human H3 receptor antagonist.
Formula:
C19H27N3O2
Purity:
96.06% - 98%
Color and Shape:
Solid
Molecular weight:
329.44
Ref: TM-TQ0046
| 1mg | 42.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 131.00 € | ||
| 25mg | 217.00 € | ||
| 50mg | 320.00 € | ||
| 100mg | 455.00 € | ||
| 500mg | To inquire | ||
| 1mL*10mM (DMSO) | 93.00 € |
Estimated delivery in United States, on Friday 24 Jan 2025
N-Arachidonyldopamine
CAS:199875-69-9
N-Arachidonyldopamine (NADA) is a selective and potent endogenous CB1 receptor agonist (Ki: 250 nM).N-Arachidonyldopamine is …
Formula:
C28H41NO3
Purity:
97.65%
Color and Shape:
Liquid
Molecular weight:
439.63
Ref: TM-T62530
| 1mg | 52.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 143.00 € | ||
| 25mg | 231.00 € | ||
| 50mg | 346.00 € |
Estimated delivery in United States, on Friday 24 Jan 2025
VPC 23019
CAS:449173-19-7
VPC 23019 is a competitive antagonist at the S1P1 and S1P3 receptors (pKi= 7.86 and …
Formula:
C17H29N2O5P
Purity:
98%
Color and Shape:
Solid
Molecular weight:
372.4
Ref: TM-T17237
| 25mg | 616.00 € | ||
| 50mg | 804.00 € | ||
| 100mg | 1,202.00 € |
Estimated delivery in United States, on Friday 24 Jan 2025
TC-MCH 7c
CAS:864756-35-4
TC-MCH 7c is an oral, selectable and blood-brain barrier penetrating MCH1R antagonist with IC50 performance …
Formula:
C24H25FN2O3
Purity:
98.8%
Color and Shape:
Solid
Molecular weight:
408.47
Ref: TM-T13101
| 1mg | 92.00 € | ||
| 5mg | 270.00 € | ||
| 10mg | 387.00 € | ||
| 25mg | 593.00 € | ||
| 50mg | 800.00 € | ||
| 100mg | 1,072.00 € | ||
| 500mg | 2,152.00 € | ||
| 1mL*10mM (DMSO) | 247.00 € |
Estimated delivery in United States, on Friday 24 Jan 2025
Iprindole
CAS:5560-72-5
Iprindole, a tricyclic indole antidepressant, is a dual weak inhibitor of noradrenaline and 5-HT uptake …
Formula:
C19H28N2
Purity:
99.06%
Color and Shape:
Solid
Molecular weight:
284.44
Ref: TM-T37015
| 2mg | 45.00 € | ||
| 5mg | 67.00 € | ||
| 10mg | 96.00 € | ||
| 25mg | 187.00 € | ||
| 50mg | 330.00 € | ||
| 100mg | 549.00 € | ||
| 200mg | 786.00 € | ||
| 500mg | 1,142.00 € | ||
| 1mL*10mM (DMSO) | 96.00 € |
Estimated delivery in United States, on Friday 24 Jan 2025
NF-56-EJ40
CAS:2380230-73-7
NF-56-EJ40 is an effective and highly selective antagonist of human SUCNR1 with an IC50 of …
Formula:
C27H29N3O3
Purity:
99.51%
Color and Shape:
Solid
Molecular weight:
443.54
Ref: TM-T12216
| 1mg | 89.00 € | ||
| 5mg | 184.00 € | ||
| 10mg | 305.00 € | ||
| 25mg | 521.00 € | ||
| 50mg | 734.00 € | ||
| 100mg | 1,044.00 € | ||
| 500mg | 2,071.00 € | ||
| 1mL*10mM (DMSO) | 214.00 € |
Estimated delivery in United States, on Friday 24 Jan 2025
MRE3008F20
CAS:252979-43-4
MRE3008F20 is an AA3R antagonist that inhibits Cl-IB-MECA-induced cAMP production and can be used to …
Formula:
C21H20N8O3
Purity:
97.66%
Color and Shape:
Solid
Molecular weight:
432.44
Ref: TM-T16132
| 1mg | 69.00 € | ||
| 2mg | 91.00 € | ||
| 5mg | 149.00 € | ||
| 10mg | 212.00 € | ||
| 25mg | 360.00 € | ||
| 50mg | 536.00 € |
Estimated delivery in United States, on Friday 24 Jan 2025
MJ 15
CAS:944154-76-1
MJ 15 is a CB1 receptor antagonist with specificity for the study of obesity-induced diseases.
Formula:
C23H17Cl3N4O
Purity:
99.63%
Color and Shape:
Solid
Molecular weight:
471.77
Ref: TM-T22984
| 1mg | 37.00 € | ||
| 5mg | 110.00 € | ||
| 10mg | 171.00 € | ||
| 25mg | 349.00 € | ||
| 50mg | 559.00 € | ||
| 100mg | 900.00 € | ||
| 500mg | 1,801.00 € |
Estimated delivery in United States, on Friday 24 Jan 2025
A2A receptor antagonist 1
CAS:443103-97-7
A2A receptor antagonist 1 (CPI-444 analog) is an antagonist of both adenosine A2A receptor and …
Formula:
C16H12FN5O
Purity:
99.29% - 99.76%
Color and Shape:
Liquid
Molecular weight:
309.3
Ref: TM-T37792
| 1mg | 37.00 € | ||
| 5mg | 63.00 € | ||
| 10mg | 90.00 € | ||
| 25mg | 182.00 € | ||
| 50mg | 278.00 € | ||
| 100mg | 412.00 € | ||
| 500mg | 866.00 € | ||
| 1mL*10mM (DMSO) | 46.00 € |
Estimated delivery in United States, on Friday 24 Jan 2025
SCH-336
CAS:447459-51-0
SCH-336: potent, selective CB2 agonist (Ki=1.8 nM, EC50=2 nM), orally active, 100x CB2 vs. CB1 …
Formula:
C23H25NO8S3
Purity:
95.01%
Color and Shape:
Solid
Molecular weight:
539.64
Ref: TM-T24771
| 1mg | 35.00 € | ||
| 5mg | 79.00 € | ||
| 10mg | 114.00 € | ||
| 25mg | 254.00 € | ||
| 50mg | 367.00 € | ||
| 100mg | 532.00 € | ||
| 500mg | To inquire | ||
| 1mL*10mM (DMSO) | 95.00 € |
Estimated delivery in United States, on Friday 24 Jan 2025
EP2 receptor antagonist-2
CAS:615273-95-5
CID891729, an EP2 receptor blocker, hinders PGE2 activation and reduces NMDA-induced LDH release.
Formula:
C15H14F3N3O
Purity:
99.59%
Color and Shape:
Liquid
Molecular weight:
309.29
Ref: TM-T67946
| 1mg | 49.00 € | ||
| 5mg | 102.00 € | ||
| 10mg | 166.00 € | ||
| 25mg | 276.00 € | ||
| 50mg | 411.00 € | ||
| 100mg | 593.00 € | ||
| 500mg | 1,235.00 € | ||
| 1mL*10mM (DMSO) | 147.00 € |
Estimated delivery in United States, on Friday 24 Jan 2025
Amitifadine hydrochloride
CAS:410074-74-7
Amitifadine hydrochloride (EB-1010 hydrochloride) is a triple reuptake inhibitor (TRI) or serotonin-norepinephrine-dopamine reuptake inhibitor (SNDRI).
Formula:
C11H12Cl3N
Purity:
98%
Color and Shape:
Solid
Molecular weight:
264.58
Ref: TM-T2092
| 1mg | 94.00 € | ||
| 5mg | 223.00 € | ||
| 10mg | 368.00 € | ||
| 1mL*10mM (DMSO) | 248.00 € |
Estimated delivery in United States, on Friday 24 Jan 2025
ML230
CAS:1776055-05-0
ML230 is a selective ATP-binding cassette (ABC) transporter ABCG2 inhibitor.
Formula:
C25H21N5O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
439.47
Ref: TM-T16107
| 5mg | 844.00 € | ||
| 10mg | 1,499.00 € |
Estimated delivery in United States, on Friday 24 Jan 2025
L748337
CAS:244192-94-7
L748337 is a β3-adrenoceptor antagonist that inhibits β3-, β2-, and β1-adrenoceptors and inhibits the protective …
Formula:
C26H31N3O5S
Purity:
99.67% - 99.67%
Color and Shape:
Solid
Molecular weight:
497.61
Ref: TM-T22905
| 1mg | 68.00 € |
Estimated delivery in United States, on Friday 24 Jan 2025
SB-277011
CAS:215803-78-4
SB-277011A: dopamine D3 antagonist, pKi 8.0 (D3), 6.0 (D2), 5.0 (5-HT1D), <5.2 (5-HT1B).
Formula:
C28H30N4O
Purity:
98.61%
Color and Shape:
Solid
Molecular weight:
438.56
Ref: TM-T12861
| 1mg | 46.00 € | ||
| 5mg | 57.00 € | ||
| 10mg | 92.00 € | ||
| 25mg | 154.00 € | ||
| 50mg | 249.00 € | ||
| 100mg | To inquire |
Estimated delivery in United States, on Friday 24 Jan 2025
GW-493838
CAS:253124-46-8
GW-493838 is a potent adenosine A1A receptor agonist for the treatment of dyslipidemia and neuropathic …
Formula:
C21H21ClFN7O4
Purity:
99.70% - 99.76%
Color and Shape:
Solid
Molecular weight:
489.89
Ref: TM-T27509
| 1mg | 148.00 € | ||
| 5mg | 358.00 € | ||
| 10mg | 508.00 € | ||
| 25mg | 763.00 € | ||
| 50mg | 1,031.00 € | ||
| 100mg | 1,393.00 € | ||
| 500mg | 2,730.00 € | ||
| 1mL*10mM (DMSO) | 419.00 € |
Estimated delivery in United States, on Friday 24 Jan 2025
Lavoltidine
CAS:76956-02-0
Lavoltidine, an irreversible oral H2-receptor antagonist, reduces stomach acid and increases gastrin.
Formula:
C19H29N5O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
359.47
Ref: TM-T15722
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Friday 24 Jan 2025
Dimethindene maleate
CAS:3614-69-5
Dimethindene maleate (SU 6518) is a histamine H1 antagonist and can be used in studies …
Formula:
C24H28N2O4
Purity:
99.87%
Color and Shape:
Solid
Molecular weight:
408.49
Ref: TM-T21472
| 1mg | 36.00 € | ||
| 5mg | 74.00 € | ||
| 10mg | 110.00 € | ||
| 25mg | 246.00 € | ||
| 50mg | 325.00 € | ||
| 100mg | 425.00 € | ||
| 500mg | 922.00 € | ||
| 1mL*10mM (DMSO) | 94.00 € |
Estimated delivery in United States, on Friday 24 Jan 2025
Mianserin
CAS:24219-97-4
Mianserin, an H1 receptor reverse agonist, is a psychoactive compound in the tetracyclic antidepressant (TeCA) …
Formula:
C18H20N2
Purity:
99.39%
Color and Shape:
Solid
Molecular weight:
264.36
Ref: TM-T21428
| 1mg | 369.00 € | ||
| 5mg | 900.00 € | ||
| 10mg | 1,198.00 € | ||
| 25mg | 1,811.00 € | ||
| 50mg | 2,448.00 € |
Estimated delivery in United States, on Friday 24 Jan 2025
