G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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48740 RP
CAS:93363-11-2
48740 RP (RP 55779) is an antagonist of platelet-activating factor.
Formula:
C12H11N3OS
Purity:
99.4%
Color and Shape:
Solid
Molecular weight:
245.3
Ref: TM-T10159
| 1mg | 356.00 € | ||
| 5mg | 567.00 € | ||
| 10mg | 907.00 € | ||
| 25mg | 1,339.00 € | ||
| 50mg | 1,815.00 € | ||
| 100mg | 2,432.00 € | ||
| 1mL*10mM (DMSO) | 567.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
GRI977143
CAS:325850-81-5
GRI977143: selective LPA2 agonist (EC50=3.3μM), blocks caspases 3/7/8/9, limits DNA fragmentation.
Formula:
C22H17NO4S
Purity:
98.07%
Color and Shape:
Solid
Molecular weight:
391.44
Ref: TM-T22812
| 1mg | 39.00 € | ||
| 5mg | 84.00 € | ||
| 10mg | 131.00 € | ||
| 25mg | 269.00 € | ||
| 50mg | 432.00 € | ||
| 100mg | 638.00 € | ||
| 500mg | 1,359.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
PPTN hydrochloride
CAS:1992047-65-0
PPTN hydrochloride is a potent, high-affinity, competitive, highly selective P2Y14 receptor antagonist (KB: 434 pM), …
Formula:
C29H25ClF3NO2
Purity:
99.94%
Color and Shape:
Liquid
Molecular weight:
511.96
Ref: TM-T63534
| 1mg | 48.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 160.00 € | ||
| 25mg | 305.00 € | ||
| 50mg | 472.00 € | ||
| 100mg | 687.00 € | ||
| 500mg | 1,444.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
UNC0006
CAS:1354030-14-0
UNC0006 is a β-arrestin-biased dopamine D2 ligand.
Formula:
C24H29Cl2N3O2
Purity:
98.48% - 99.83%
Color and Shape:
Solid
Molecular weight:
462.41
Ref: TM-T29061
| 1mg | 279.00 € | ||
| 5mg | 685.00 € | ||
| 10mg | 938.00 € | ||
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
Clemastine
CAS:15686-51-8
Clemastine (Meclastin) is an antagonist of the H1 receptor and exhibits anti-inflammatory effects.
Formula:
C21H26ClNO
Purity:
99.83%
Color and Shape:
Solid
Molecular weight:
343.89
Ref: TM-T19966
| 10mg | 66.00 € | ||
| 25mg | 97.00 € | ||
| 50mg | 155.00 € | ||
| 100mg | 224.00 € | ||
| 1mL*10mM (DMSO) | 65.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
Org41841
CAS:301847-37-0
Org41841 is an agonist of luteinising hormone/chorionic gonadotropin receptor and thyroid stimulating hormone receptor and …
Formula:
C19H22N4O2S2
Purity:
99.46%
Color and Shape:
Solid
Molecular weight:
402.53
Ref: TM-T16403
| 1mg | 190.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
Falintolol
CAS:90581-63-8
Falintolol is a novel beta-adrenergic antagonist with antihypertensive effects and can be used to study …
Formula:
C12H24N2O2
Purity:
100% - 100%
Color and Shape:
Liquid
Molecular weight:
228.33
Ref: TM-T68402
| 1mg | 279.00 € | ||
| 5mg | 685.00 € | ||
| 10mg | 938.00 € | ||
| 25mg | 1,388.00 € | ||
| 50mg | 1,872.00 € | ||
| 100mg | 2,527.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
Bavisant
CAS:929622-08-2
Bavisant (JNJ-31001074) is a selective and orally active Human H3 receptor antagonist.
Formula:
C19H27N3O2
Purity:
96.06% - 98%
Color and Shape:
Solid
Molecular weight:
329.44
Ref: TM-TQ0046
| 1mg | 43.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 134.00 € | ||
| 25mg | 221.00 € | ||
| 50mg | 325.00 € | ||
| 100mg | 465.00 € | ||
| 500mg | To inquire | ||
| 1mL*10mM (DMSO) | 94.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
N-Arachidonyldopamine
CAS:199875-69-9
N-Arachidonyldopamine (NADA) is a selective and potent endogenous CB1 receptor agonist (Ki: 250 nM).N-Arachidonyldopamine is …
Formula:
C28H41NO3
Purity:
97.65%
Color and Shape:
Liquid
Molecular weight:
439.63
Ref: TM-T62530
| 1mg | 52.00 € | ||
| 5mg | 97.00 € | ||
| 10mg | 145.00 € | ||
| 25mg | 236.00 € | ||
| 50mg | 354.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
VPC 23019
CAS:449173-19-7
VPC 23019 is a competitive antagonist at the S1P1 and S1P3 receptors (pKi= 7.86 and …
Formula:
C17H29N2O5P
Purity:
98%
Color and Shape:
Solid
Molecular weight:
372.4
Ref: TM-T17237
| 25mg | 630.00 € | ||
| 50mg | 820.00 € | ||
| 100mg | 1,225.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
TC-MCH 7c
CAS:864756-35-4
TC-MCH 7c is an oral, selectable and blood-brain barrier penetrating MCH1R antagonist with IC50 performance …
Formula:
C24H25FN2O3
Purity:
98.8%
Color and Shape:
Solid
Molecular weight:
408.47
Ref: TM-T13101
| 1mg | 94.00 € | ||
| 5mg | 274.00 € | ||
| 10mg | 394.00 € | ||
| 25mg | 605.00 € | ||
| 50mg | 815.00 € | ||
| 100mg | 1,093.00 € | ||
| 500mg | 2,195.00 € | ||
| 1mL*10mM (DMSO) | 248.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
Iprindole
CAS:5560-72-5
Iprindole, a tricyclic indole antidepressant, is a dual weak inhibitor of noradrenaline and 5-HT uptake …
Formula:
C19H28N2
Purity:
99.06%
Color and Shape:
Solid
Molecular weight:
284.44
Ref: TM-T37015
| 2mg | 37.00 € | ||
| 5mg | 52.00 € | ||
| 10mg | 80.00 € | ||
| 25mg | 154.00 € | ||
| 50mg | 266.00 € | ||
| 100mg | 455.00 € | ||
| 200mg | 652.00 € | ||
| 1mL*10mM (DMSO) | 84.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
NF-56-EJ40
CAS:2380230-73-7
NF-56-EJ40 is an effective and highly selective antagonist of human SUCNR1 with an IC50 of …
Formula:
C27H29N3O3
Purity:
99.51%
Color and Shape:
Solid
Molecular weight:
443.54
Ref: TM-T12216
| 1mg | 90.00 € | ||
| 5mg | 187.00 € | ||
| 10mg | 311.00 € | ||
| 25mg | 530.00 € | ||
| 50mg | 748.00 € | ||
| 100mg | 1,064.00 € | ||
| 500mg | 2,118.00 € | ||
| 1mL*10mM (DMSO) | 215.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
MRE3008F20
CAS:252979-43-4
MRE3008F20 is an AA3R antagonist that inhibits Cl-IB-MECA-induced cAMP production and can be used to …
Formula:
C21H20N8O3
Purity:
97.66%
Color and Shape:
Solid
Molecular weight:
432.44
Ref: TM-T16132
| 1mg | 70.00 € | ||
| 2mg | 92.00 € | ||
| 5mg | 153.00 € | ||
| 10mg | 216.00 € | ||
| 25mg | 369.00 € | ||
| 50mg | 540.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
A2A receptor antagonist 1
CAS:443103-97-7
A2A receptor antagonist 1 (CPI-444 analog) is an antagonist of both adenosine A2A receptor and …
Formula:
C16H12FN5O
Purity:
99.29% - 99.76%
Color and Shape:
Liquid
Molecular weight:
309.3
Ref: TM-T37792
| 1mg | 37.00 € | ||
| 5mg | 64.00 € | ||
| 10mg | 92.00 € | ||
| 25mg | 185.00 € | ||
| 50mg | 284.00 € | ||
| 100mg | 419.00 € | ||
| 500mg | 883.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
SCH-336
CAS:447459-51-0
SCH-336: potent, selective CB2 agonist (Ki=1.8 nM, EC50=2 nM), orally active, 100x CB2 vs. CB1 …
Formula:
C23H25NO8S3
Purity:
95.01%
Color and Shape:
Solid
Molecular weight:
539.64
Ref: TM-T24771
| 5mg | 52.00 € | ||
| 10mg | 78.00 € | ||
| 25mg | 160.00 € | ||
| 50mg | 225.00 € | ||
| 100mg | 325.00 € | ||
| 200mg | 469.00 € | ||
| 1mL*10mM (DMSO) | 64.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
EP2 receptor antagonist-2
CAS:615273-95-5
CID891729, an EP2 receptor blocker, hinders PGE2 activation and reduces NMDA-induced LDH release.
Formula:
C15H14F3N3O
Purity:
99.59%
Color and Shape:
Liquid
Molecular weight:
309.29
Ref: TM-T67946
| 1mg | 49.00 € | ||
| 5mg | 104.00 € | ||
| 10mg | 169.00 € | ||
| 25mg | 283.00 € | ||
| 50mg | 419.00 € | ||
| 100mg | 607.00 € | ||
| 500mg | 1,264.00 € | ||
| 1mL*10mM (DMSO) | 150.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
Amitifadine hydrochloride
CAS:410074-74-7
Amitifadine hydrochloride (EB-1010 hydrochloride) is a triple reuptake inhibitor (TRI) or serotonin-norepinephrine-dopamine reuptake inhibitor (SNDRI).
Formula:
C11H12Cl3N
Purity:
98%
Color and Shape:
Solid
Molecular weight:
264.58
Ref: TM-T2092
| 1mg | 96.00 € | ||
| 5mg | 227.00 € | ||
| 10mg | 376.00 € | ||
| 1mL*10mM (DMSO) | 250.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
Lintopride
CAS:107429-63-0
Lintopride is an antagonist of 5HT4. It has moderate 5HT3 antagonist properties.
Formula:
C14H19ClN4O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
310.78
Ref: TM-T15760
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
MJ 15
CAS:944154-76-1
MJ 15 is a CB1 receptor antagonist with specificity for the study of obesity-induced diseases.
Formula:
C23H17Cl3N4O
Purity:
99.63%
Color and Shape:
Solid
Molecular weight:
471.77
Ref: TM-T22984
| 1mg | 37.00 € | ||
| 5mg | 111.00 € | ||
| 10mg | 167.00 € | ||
| 25mg | 354.00 € | ||
| 50mg | 567.00 € | ||
| 100mg | 912.00 € | ||
| 500mg | 1,825.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
