G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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SB-215505
CAS:162100-15-4
SB215505: potent 5-HT2B/2C blocker, enhances rat wakefulness/motor activity. (pKi: 5-HT2B - 8.3, 5-HT2C - 7.66, …
Formula:
C19H16ClN3O
Purity:
98.33%
Color and Shape:
Solid
Molecular weight:
337.8
Ref: TM-T28680
| 1mg | 209.00 € | ||
| 5mg | 521.00 € | ||
| 10mg | 726.00 € | ||
| 25mg | 1,081.00 € | ||
| 50mg | 1,493.00 € | ||
| 100mg | 2,005.00 € |
Estimated delivery in United States, on Friday 22 Nov 2024
WAY-260022
CAS:850692-43-2
WAY-260022 is the norepinephrine transporter inhibitor.
Formula:
C21H31F3N2O2
Purity:
98.65% - 99.06%
Color and Shape:
Solid
Molecular weight:
400.48
Ref: TM-T23711
| 1mg | 273.00 € | ||
| 2mg | 407.00 € | ||
| 5mg | 673.00 € | ||
| 10mg | 920.00 € | ||
| 25mg | 1,415.00 € | ||
| 50mg | 1,832.00 € |
Estimated delivery in United States, on Friday 22 Nov 2024
Opigolix
CAS:912587-25-8
Opigolix is a Gonadotropin-releasing hormone receptor antagonist.
Formula:
C25H19F3N4O5S
Purity:
98.07% - 99.54%
Color and Shape:
Solid
Molecular weight:
544.5
Ref: TM-T17301
| 1mg | 273.00 € | ||
| 5mg | 673.00 € | ||
| 10mg | 930.00 € | ||
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,599.00 € |
Estimated delivery in United States, on Friday 22 Nov 2024
MrgprX2 antagonist-8
CAS:2768216-96-0
MrgprX2 antagonist-8 is an MrgprX2 antagonist that can be used to study inflammatory diseases.
Formula:
C24H24ClF3N4O3S
Purity:
98.87%
Color and Shape:
Solid
Molecular weight:
540.99
Ref: TM-T63812
| 1mg | 100.00 € | ||
| 5mg | 240.00 € | ||
| 10mg | 344.00 € | ||
| 25mg | 564.00 € | ||
| 50mg | 745.00 € | ||
| 100mg | 992.00 € |
Estimated delivery in United States, on Friday 22 Nov 2024
LY2881835
CAS:1292290-38-0
LY2881835 is a potent and selective GPR40 agonist.
Formula:
C33H33NO3
Purity:
97.65% - 97.65%
Color and Shape:
Solid
Molecular weight:
491.62
Ref: TM-T27937
| 1mg | 274.00 € | ||
| 5mg | 673.00 € | ||
| 10mg | 920.00 € | ||
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € |
Estimated delivery in United States, on Friday 22 Nov 2024
L 651896
CAS:99134-29-9
L 651896 is an inhibitor of 5-lipoxygenase.
Formula:
C18H18O3
Purity:
95.87% - 99.70%
Color and Shape:
Solid
Molecular weight:
282.33
Ref: TM-T24306
| 1mg | 311.00 € | ||
| 5mg | 747.00 € | ||
| 10mg | 1,059.00 € | ||
| 25mg | 1,549.00 € | ||
| 50mg | 2,127.00 € |
Estimated delivery in United States, on Friday 22 Nov 2024
![N-[(4-Aminophenyl)methyl]adenosine](https://static.cymitquimica.com/products/TM/thumb/T16166.jpg)
N-[(4-Aminophenyl)methyl]adenosine
CAS:95523-13-0
N-[(4-Aminophenyl)methyl]adenosine is an adenosine receptor inhibitor (Ki: 29 nM for Rat ecto-5′-Nucleotidase).
Formula:
C17H20N6O4
Purity:
98.75%
Color and Shape:
Solid
Molecular weight:
372.38
Ref: TM-T16166
| 1mg | 90.00 € | ||
| 1ml | 235.00 € | ||
| 5mg | 184.00 € | ||
| 10mg | 276.00 € | ||
| 25mg | 546.00 € | ||
| 50mg | 865.00 € | ||
| 100mg | 1,395.00 € |
Estimated delivery in United States, on Friday 22 Nov 2024
AMG-009
CAS:1027847-67-1
AMG-009 is a prostaglandin D2 antagonist. For CRTH2 and DP receptors, the IC50s are 3 …
Formula:
C26H26Cl2N2O7S
Purity:
97.88%
Color and Shape:
Solid
Molecular weight:
581.47
Ref: TM-T14211
| 1mg | 48.00 € | ||
| 5mg | 89.00 € | ||
| 10mg | 129.00 € | ||
| 25mg | 208.00 € | ||
| 50mg | 366.00 € | ||
| 100mg | 623.00 € |
Estimated delivery in United States, on Friday 22 Nov 2024
Romifidine
CAS:65896-16-4
Romifidine is used as a sedative in veterinary medicine mainly in large animals such as …
Formula:
C9H9BrFN3
Color and Shape:
Solid
Molecular weight:
258.09
Ref: TM-T26119
| 1mg | 65.00 € | ||
| 5mg | 134.00 € | ||
| 10mg | 184.00 € | ||
| 25mg | 315.00 € | ||
| 50mg | 460.00 € | ||
| 100mg | 674.00 € | ||
| 500mg | 1,372.00 € |
Estimated delivery in United States, on Friday 22 Nov 2024
GRK6-IN-1
CAS:2677786-61-5
GRK6-IN-1 (compound 18) is a potent GRK6 blocker, with an IC50 of 120 nM, showing …
Formula:
C22H23ClN6O2
Purity:
99.37%
Color and Shape:
Solid
Molecular weight:
438.91
Ref: TM-T62518
| 1mg | 56.00 € | ||
| 1ml | 130.00 € | ||
| 5mg | 119.00 € | ||
| 10mg | 184.00 € | ||
| 25mg | 423.00 € | ||
| 50mg | 730.00 € | ||
| 100mg | 1,187.00 € |
Estimated delivery in United States, on Friday 22 Nov 2024
Itriglumide
CAS:201605-51-8
Itriglumide, a CCK2 receptor antagonist, is used potentially for the treatment of peptic ulcers, dyspepsia, …
Formula:
C33H38N2O4
Purity:
99.95%
Color and Shape:
Solid
Molecular weight:
526.67
Ref: TM-T27640
| 1mg | 272.00 € | ||
| 2mg | 405.00 € | ||
| 5mg | 670.00 € | ||
| 10mg | 915.00 € | ||
| 25mg | 1,409.00 € | ||
| 50mg | 1,836.00 € |
Estimated delivery in United States, on Friday 22 Nov 2024
NGD 94-1
CAS:178928-68-2
NGD 94-1 is a D4 receptor antagonist that can be used to study psychiatric disorders …
Formula:
C18H20N6
Purity:
99.84%
Color and Shape:
Solid
Molecular weight:
320.39
Ref: TM-T23066
| 1mg | 93.00 € | ||
| 5mg | 186.00 € | ||
| 10mg | 281.00 € | ||
| 25mg | 555.00 € | ||
| 50mg | 908.00 € | ||
| 100mg | 1,203.00 € |
Estimated delivery in United States, on Friday 22 Nov 2024
SLV-310
CAS:264869-71-8
SLV-310 is a D2 receptor antagonist and 5-HT reuptake receptor inhibitor for the study of …
Formula:
C25H24FN3O2
Purity:
98.91%
Color and Shape:
Solid
Molecular weight:
417.48
Ref: TM-T28809
| 1mg | 278.00 € | ||
| 5mg | 684.00 € | ||
| 10mg | 935.00 € | ||
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Friday 22 Nov 2024
SC 51089
CAS:146033-02-5
SC 51089 is a somatic PGE2 antagonist with anti-injurious activity and may rescue memory loss.
Formula:
C22H20Cl2N4O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
459.33
Ref: TM-T23331
| 1mg | 278.00 € | ||
| 5mg | 684.00 € | ||
| 10mg | 935.00 € | ||
| 25mg | 1,410.00 € | ||
| 50mg | 1,845.00 € | ||
| 100mg | 2,329.00 € |
Estimated delivery in United States, on Friday 22 Nov 2024
(Iso)-FK-480
CAS:167820-10-2
(Iso)-FK-480 is a novel orally available cholecystokinin A (CCK-A) antagonist for investigational treatment of chronic …
Formula:
C26H19FN4O2
Purity:
99.68%
Color and Shape:
Solid
Molecular weight:
438.45
Ref: TM-T10055
| 25mg | 1,410.00 € | ||
| 50mg | 1,845.00 € | ||
| 100mg | 2,329.00 € |
Estimated delivery in United States, on Friday 22 Nov 2024
LY377604
CAS:204592-94-9
LY377604 is a human β3-adrenergic receptor agonist (EC50: 2.4 nM) and β1/2-adrenergic receptor antagonist for …
Formula:
C31H32N4O4
Purity:
100% - 99.72%
Color and Shape:
Solid
Molecular weight:
524.61
Ref: TM-T15819
| 1mg | 123.00 € | ||
| 5mg | 298.00 € | ||
| 10mg | 441.00 € | ||
| 25mg | 722.00 € |
Estimated delivery in United States, on Friday 22 Nov 2024
ST1936
CAS:1210-81-7
ST1936 (ST 1936 oxalate) is a 5-HT6 receptor agonist that stimulates cAMP, Ca2+, ERK1/2, and …
Formula:
C13H17ClN2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
236.74
Ref: TM-T23396
| 1mg | 67.00 € | ||
| 1ml | 159.00 € | ||
| 2mg | 96.00 € | ||
| 5mg | 144.00 € | ||
| 10mg | 233.00 € | ||
| 25mg | 484.00 € | ||
| 50mg | 748.00 € | ||
| 100mg | 1,198.00 € |
Estimated delivery in United States, on Friday 22 Nov 2024
SM-2470
CAS:99899-45-3
SM-2470 is an α1-adrenoceptor antagonist with antihypertensive activity and hypocholesterolemic activity that inhibits cholesterol absorption.
Formula:
C23H30ClN5O3
Purity:
99.05%
Color and Shape:
Solid
Molecular weight:
459.97
Ref: TM-T62893
| 1mg | 437.00 € | ||
| 5mg | 1,012.00 € | ||
| 25mg | 2,014.00 € | ||
| 50mg | 2,628.00 € | ||
| 100mg | 3,338.00 € |
Estimated delivery in United States, on Friday 22 Nov 2024
RXFP3/4 agonist 2
CAS:2752378-78-0
RXFP3/4 agonist 2 is a nonpeptide bis-RXFP3/4 agonist used in the study of diseases caused …
Formula:
C22H22N6O2
Purity:
99.82%
Color and Shape:
Solid
Molecular weight:
402.45
Ref: TM-T61964
| 1mg | 278.00 € |
Estimated delivery in United States, on Friday 22 Nov 2024
mPGES-1 Inhibitor-1
CAS:1381846-21-4
mPGES-1 Inhibitor-1 is an mPGES-1 inhibitor with anti-inflammatory and analgesic activity, which can be used …
Formula:
C16H19ClN4O2
Purity:
97.90% - 98.98%
Color and Shape:
Solid
Molecular weight:
334.8
Ref: TM-T28089
| 1mg | 186.00 € | ||
| 5mg | 417.00 € | ||
| 10mg | 682.00 € | ||
| 25mg | 1,025.00 € | ||
| 50mg | 1,413.00 € |
Estimated delivery in United States, on Friday 22 Nov 2024
