G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Org-13011 fumarate
CAS:142494-13-1
Org-13011 fumarate1 is an agonist of the 5-HT1A receptor and can be used to study …
Formula:
C22H29F3N4O5
Purity:
98.61%
Color and Shape:
Solid
Molecular weight:
486.48
Ref: TM-T28258
| 1mg | 277.00 € | ||
| 5mg | 683.00 € | ||
| 10mg | 933.00 € | ||
| 25mg | 1,442.00 € | ||
| 50mg | 1,832.00 € | ||
| 100mg | 2,342.00 € |
Estimated delivery in United States, on Friday 22 Nov 2024
Enciprazine
CAS:68576-86-3
Enciprazine (D-3112) shows anxiolytic activity, is used to treat anxiety disorders, and can be used …
Formula:
C23H32N2O6
Purity:
98.66%
Color and Shape:
Solid
Molecular weight:
432.51
Ref: TM-T27262
| 1mg | 278.00 € | ||
| 5mg | 685.00 € | ||
| 10mg | 936.00 € | ||
| 25mg | 1,442.00 € | ||
| 50mg | 1,878.00 € | ||
| 100mg | 2,371.00 € |
Estimated delivery in United States, on Friday 22 Nov 2024
Adatanserin
CAS:127266-56-2
Adatanserin (WY 50324) is a mixed 5-HT1A receptor partial agonist and a 5-HT2A and 5-HT2C …
Formula:
C21H31N5O
Purity:
99.17%
Color and Shape:
Solid
Molecular weight:
369.5
Ref: TM-T23631
| 1mg | 279.00 € | ||
| 5mg | 686.00 € | ||
| 10mg | 938.00 € | ||
| 25mg | 1,410.00 € | ||
| 50mg | 1,852.00 € | ||
| 100mg | 2,338.00 € |
Estimated delivery in United States, on Friday 22 Nov 2024
E-4177
CAS:135070-05-2
E-4177 is an angiotensin II type 1 receptor (AT1R) antagonist and can be used to …
Formula:
C24H21N3O2
Purity:
98.63% - 99.39%
Color and Shape:
Solid
Molecular weight:
383.44
Ref: TM-T27229
| 25mg | 1,397.00 € | ||
| 50mg | 1,820.00 € | ||
| 100mg | 2,297.00 € |
Estimated delivery in United States, on Friday 22 Nov 2024
Tiospirone
CAS:87691-91-6
Tiospirone (BMY 13859-1 free base) is a 5-HT2 receptor antagonist and a dopamine blocker used …
Formula:
C24H32N4O2S
Purity:
99.52%
Color and Shape:
Solid
Molecular weight:
440.6
Ref: TM-T24885
| 1mg | 127.00 € | ||
| 1ml | 371.00 € | ||
| 5mg | 303.00 € | ||
| 10mg | 556.00 € | ||
| 25mg | 892.00 € | ||
| 50mg | 1,200.00 € | ||
| 100mg | 1,610.00 € |
Estimated delivery in United States, on Friday 22 Nov 2024
Barbadin
CAS:356568-70-2
Barbadin is an inhibitor of β-arrestin/β2-adaptin interaction.Barbadin enhances the effects of lorcaserin on weight loss …
Formula:
C19H15N3OS
Purity:
98.93%
Color and Shape:
Solid
Molecular weight:
333.41
Ref: TM-T14498
| 1mg | 189.00 € |
Estimated delivery in United States, on Friday 22 Nov 2024
RS 56812 hydrochloride
CAS:143339-12-2
5-HT3 partial agonist
Formula:
C18H22ClN3O2
Purity:
97.69%
Color and Shape:
Solid
Molecular weight:
347.84
Ref: TM-T23264
| 1mg | 64.00 € | ||
| 2mg | 90.00 € | ||
| 5mg | 131.00 € | ||
| 10mg | 185.00 € | ||
| 25mg | 431.00 € |
Estimated delivery in United States, on Friday 22 Nov 2024
Tiopinac
CAS:61220-69-7
Tiopinac: tricyclic with anti-inflammatory, analgesic, antipyretic properties; inhibits prostaglandin synthesis; mild anti-platelet effects in humans.
Formula:
C16H12O3S
Purity:
100%
Color and Shape:
Solid
Molecular weight:
284.33
Ref: TM-T17101
| 1mg | 197.00 € | ||
| 5mg | 497.00 € | ||
| 10mg | 707.00 € | ||
| 25mg | 1,059.00 € | ||
| 50mg | 1,437.00 € | ||
| 100mg | 1,872.00 € |
Estimated delivery in United States, on Friday 22 Nov 2024
PF-184298
CAS:813447-40-4
PF-184298 is a serotonin and norepinephrine monoamine reuptake inhibitor (SNRI) that inhibits dopamine reuptake.
Formula:
C15H20Cl2N2O
Purity:
98.30%
Color and Shape:
Solid
Molecular weight:
315.24
Ref: TM-T28380
| 1mg | 276.00 € | ||
| 5mg | 680.00 € | ||
| 10mg | 930.00 € | ||
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € |
Estimated delivery in United States, on Friday 22 Nov 2024
BL-1020 Mesylate
CAS:916898-61-8
BL-1020 Mesylate (CYP-1020 Mesylate) is a GABA A receptor agonist and D2 antagonist used in …
Formula:
C28H45ClN4O11S4
Purity:
100%
Color and Shape:
Solid
Molecular weight:
777.39
Ref: TM-T26834
| 1mg | 276.00 € | ||
| 5mg | 680.00 € | ||
| 10mg | 930.00 € | ||
| 25mg | 1,410.00 € | ||
| 50mg | 1,845.00 € |
Estimated delivery in United States, on Friday 22 Nov 2024
MK-2894
CAS:1006036-87-8
MK-2894 is a highly potent and selective antagonist of second generation EP4 .
Formula:
C25H22F3NO3S
Purity:
≥98%
Color and Shape:
Solid
Molecular weight:
473.51
Ref: TM-T12061
| 1mg | 60.00 € | ||
| 1ml | 134.00 € | ||
| 5mg | 126.00 € | ||
| 10mg | 216.00 € | ||
| 25mg | 522.00 € | ||
| 50mg | 922.00 € | ||
| 100mg | 1,218.00 € | ||
| 500mg | 2,482.00 € |
Estimated delivery in United States, on Friday 22 Nov 2024
A-65186
CAS:119295-94-2
A-65186 is a CCK antagonist used in the study of inflammation and gastrointestinal tract injury.
Formula:
C25H35N3O4
Purity:
98.37% - 99.94%
Color and Shape:
Solid
Molecular weight:
441.56
Ref: TM-T26483
| 1mg | 277.00 € | ||
| 5mg | 682.00 € | ||
| 10mg | 932.00 € | ||
| 25mg | 1,435.00 € | ||
| 50mg | 1,869.00 € |
Estimated delivery in United States, on Friday 22 Nov 2024
PNU-282987 free base
CAS:711085-63-1
PNU-282987 is an α7 nAChR agonist (EC50=154 nM) and a 5-HT3 antagonist (IC50=4541 nM) for …
Formula:
C14H17ClN2O
Purity:
99.64%
Color and Shape:
Solid
Molecular weight:
264.75
Ref: TM-T60437
| 1mg | 55.00 € | ||
| 5mg | 111.00 € | ||
| 10mg | 201.00 € | ||
| 25mg | 392.00 € | ||
| 50mg | 727.00 € | ||
| 100mg | 1,020.00 € | ||
| 500mg | 2,039.00 € |
Estimated delivery in United States, on Friday 22 Nov 2024
UCM-05194
CAS:2411412-36-5
UCM-05194: potent LPA1 agonist, best for neuropathic pain relief (Emax 118%, EC50 0.24 μM, KD …
Formula:
C19H30BrO6P
Purity:
90% - 98%
Color and Shape:
Solid
Molecular weight:
465.32
Ref: TM-T69647
| 1mg | 315.00 € | ||
| 5mg | 746.00 € | ||
| 10mg | 1,057.00 € | ||
| 25mg | 1,576.00 € | ||
| 50mg | 2,057.00 € | ||
| 100mg | 2,732.00 € |
Estimated delivery in United States, on Friday 22 Nov 2024
UNC9975
CAS:1354030-19-5
UNC9975 is a D(2) receptor agonist with antipsychotic activity used in the study of neurologic …
Formula:
C23H28Cl2N4O2
Purity:
99.02% - 99.02%
Color and Shape:
Solid
Molecular weight:
463.4
Ref: TM-T29064
| 1mg | 277.00 € | ||
| 5mg | 682.00 € | ||
| 10mg | 932.00 € | ||
| 25mg | 1,435.00 € | ||
| 50mg | 1,869.00 € |
Estimated delivery in United States, on Friday 22 Nov 2024
UNC0006
CAS:1354030-14-0
UNC0006 is a β-arrestin-biased dopamine D2 ligand.
Formula:
C24H29Cl2N3O2
Purity:
98.48% - 99.83%
Color and Shape:
Solid
Molecular weight:
462.41
Ref: TM-T29061
| 1mg | 277.00 € | ||
| 5mg | 682.00 € | ||
| 10mg | 932.00 € | ||
| 25mg | 1,435.00 € | ||
| 50mg | 1,846.00 € |
Estimated delivery in United States, on Friday 22 Nov 2024
Falintolol
CAS:90581-63-8
Falintolol is a novel beta-adrenergic antagonist with antihypertensive effects and can be used to study …
Formula:
C12H24N2O2
Purity:
100% - 100%
Color and Shape:
Solid
Molecular weight:
228.33
Ref: TM-T68402
| 1mg | 277.00 € | ||
| 5mg | 682.00 € | ||
| 10mg | 932.00 € | ||
| 25mg | 1,351.00 € | ||
| 50mg | 1,823.00 € | ||
| 100mg | 2,462.00 € |
Estimated delivery in United States, on Friday 22 Nov 2024
TASP0390325
CAS:1642187-96-9
TASP0390325, a potent and orally active V1B receptor antagonist, has antidepressant and anxiolytic activities in …
Formula:
C25H30Cl2FN5O4
Purity:
98.62%
Color and Shape:
Solid
Molecular weight:
554.44
Ref: TM-T28926
| 1mg | 57.00 € | ||
| 5mg | 121.00 € | ||
| 10mg | 187.00 € | ||
| 25mg | 430.00 € | ||
| 50mg | 743.00 € | ||
| 100mg | 1,208.00 € |
Estimated delivery in United States, on Friday 22 Nov 2024
Ubrogepant
CAS:1374248-77-7
Ubrogepant is a small-molecule drug that is used to treat migraine. It inhibits the activity …
Formula:
C29H26F3N5O3
Purity:
Min. 95%
Molecular weight:
549.54 g/mol
Ref: 3D-FU165699
| 1mg | 693.00 € | ||
| 2mg | 880.00 € | ||
| 5mg | 1,138.00 € | ||
| 10mg | 1,897.00 € |
Estimated delivery in United States, on Friday 29 Nov 2024
PAF (C16)
CAS:74389-68-7
PAF, short for Platelet-activating factor, is a mediator of platelet aggregation and a ligand for …
Formula:
C26H54NO7P
Purity:
Min. 95%
Molecular weight:
523.68 g/mol
Ref: 3D-ZCA38968
| 1mg | 230.00 € | ||
| 2mg | 346.00 € | ||
| 5mg | 500.00 € | ||
| 10mg | 733.00 € | ||
| 25mg | 1,035.00 € |
Estimated delivery in United States, on Friday 29 Nov 2024
