G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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2-Iodomelatonin
CAS:93515-00-5
2-Iodomelatonin, Ki 28 pM, is an MT1 agonist, >5x selective over MT2, used to map …
Formula:
C13H15IN2O2
Purity:
100%
Color and Shape:
Solid
Molecular weight:
358.17
Ref: TM-T10073
| 10mg | 45.00 € | ||
| 25mg | 82.00 € | ||
| 50mg | 123.00 € | ||
| 100mg | 185.00 € | ||
| 200mg | 277.00 € | ||
| 500mg | To inquire | ||
| 1mL*10mM (DMSO) | 36.00 € |
Estimated delivery in United States, on Friday 24 Jan 2025
YIL 781
CAS:875258-85-8
YIL 781 is a selective ghrelin receptor antagonist (GHS-R1a) (Ki = 17 nM), showing a …
Formula:
C24H28FN3O2
Purity:
99.3%
Color and Shape:
Solid
Molecular weight:
409.5
Ref: TM-T23543
| 1mg | 52.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 149.00 € | ||
| 25mg | 306.00 € | ||
| 50mg | 461.00 € | ||
| 100mg | 644.00 € | ||
| 1mL*10mM (DMSO) | 123.00 € |
Estimated delivery in United States, on Friday 24 Jan 2025
Terbogrel
CAS:149979-74-8
Terbogrel is an antiplatelet drug, blocking thromboxane A2 receptor/synthase. Helps prevent clots.
Formula:
C23H27N5O2
Purity:
99.65%
Color and Shape:
Solid
Molecular weight:
405.49
Ref: TM-T17039
| 1mg | 183.00 € | ||
| 5mg | 435.00 € | ||
| 10mg | 635.00 € | ||
| 25mg | 1,000.00 € | ||
| 50mg | 1,336.00 € | ||
| 100mg | 1,803.00 € |
Estimated delivery in United States, on Friday 24 Jan 2025
Acifran
CAS:72420-38-3
Acifran (AY 25712) is an HM74A/GPR109A and GPR109B agonist and displays antihyperlipidemic activity.
Formula:
C12H10O4
Purity:
98.65%
Color and Shape:
Solid
Molecular weight:
218.21
Ref: TM-T22547
| 1mg | 47.00 € | ||
| 5mg | 83.00 € | ||
| 10mg | 125.00 € | ||
| 25mg | 245.00 € | ||
| 50mg | 398.00 € | ||
| 100mg | 580.00 € | ||
| 500mg | 1,190.00 € |
Estimated delivery in United States, on Friday 24 Jan 2025
Odapipam
CAS:131796-63-9
Odapipam is a selective and high affinity antagonist of benzazepine dopamine D1 receptor (Kd of …
Formula:
C19H20ClNO2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
329.82
Ref: TM-T12288
| 25mg | 1,132.00 € | ||
| 50mg | 1,476.00 € | ||
| 100mg | 2,270.00 € |
Estimated delivery in United States, on Friday 24 Jan 2025
Tiospirone
CAS:87691-91-6
Tiospirone (BMY 13859-1 free base) is a 5-HT2 receptor antagonist and a dopamine blocker used …
Formula:
C24H32N4O2S
Purity:
99.52%
Color and Shape:
Solid
Molecular weight:
440.6
Ref: TM-T24885
| 1mg | 127.00 € | ||
| 5mg | 303.00 € | ||
| 10mg | 556.00 € | ||
| 25mg | 892.00 € | ||
| 50mg | 1,200.00 € | ||
| 100mg | 1,610.00 € | ||
| 1mL*10mM (DMSO) | 371.00 € |
Estimated delivery in United States, on Friday 24 Jan 2025
GLPG1205
CAS:1445847-37-9
GLPG1205 is a potent, orally active GPR84 (G protein-coupled receptor) antagonist with anti-inflammatory activity.
Formula:
C22H22N2O4
Purity:
95.97% - 99.34%
Color and Shape:
Solid
Molecular weight:
378.42
Ref: TM-T11411
| 1mg | 95.00 € | ||
| 5mg | 203.00 € | ||
| 10mg | 346.00 € | ||
| 25mg | 587.00 € | ||
| 50mg | 836.00 € | ||
| 100mg | 1,132.00 € | ||
| 1mL*10mM (DMSO) | 225.00 € |
Estimated delivery in United States, on Friday 24 Jan 2025
Molindone
CAS:7416-34-4
Molindone: antipsychotic for schizophrenia; blocks dopamine, often paired with serotonin; dosage affects error/response rates.
Formula:
C16H24N2O2
Purity:
98% - 99.37%
Color and Shape:
Off-White Solid
Molecular weight:
276.37
Ref: TM-T21432
| 1mg | 325.00 € | ||
| 5mg | 769.00 € | ||
| 10mg | 1,054.00 € | ||
| 25mg | 1,477.00 € | ||
| 50mg | 1,846.00 € | ||
| 100mg | 2,331.00 € | ||
| 500mg | 4,547.00 € |
Estimated delivery in United States, on Friday 24 Jan 2025
SR144528
CAS:192703-06-3
SR144528 is an antagonist of the CB2 receptor (Ki = 0.6 nM) and inhibits microsomal …
Formula:
C29H34ClN3O
Purity:
99.6%
Color and Shape:
Solid
Molecular weight:
476.05
Ref: TM-T16928
| 1mg | 42.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 152.00 € | ||
| 25mg | 332.00 € | ||
| 50mg | 497.00 € | ||
| 100mg | 719.00 € | ||
| 1mL*10mM (DMSO) | 94.00 € |
Estimated delivery in United States, on Friday 24 Jan 2025
Amgen-23
CAS:1448706-15-7
Amgen-23 is a selective and highly potent sphingosine kinase 1 (SPHK1) inhibitor that inhibits SPHK2 …
Formula:
C23H25Cl2N3O2S
Color and Shape:
Liquid
Molecular weight:
478.44
Ref: TM-T63132
| 1mg | 89.00 € | ||
| 5mg | 181.00 € | ||
| 10mg | 309.00 € | ||
| 25mg | 619.00 € | ||
| 50mg | 908.00 € | ||
| 100mg | 1,578.00 € |
Estimated delivery in United States, on Friday 24 Jan 2025
Masupirdine mesylate
CAS:1791396-46-7
Masupirdine mesylate (SUVN-502 mesylate) is a 5-HT6 receptor antagonist.Masupirdine mesylate is used to study neurological …
Formula:
C23H32BrN3O9S3
Purity:
99.48%
Color and Shape:
Solid
Molecular weight:
670.61
Ref: TM-T11949
| 1mg | 46.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 143.00 € | ||
| 25mg | 248.00 € | ||
| 50mg | 373.00 € | ||
| 100mg | 607.00 € | ||
| 1mL*10mM (DMSO) | 129.00 € |
Estimated delivery in United States, on Friday 24 Jan 2025
AM404
CAS:183718-77-6
AM404 is a cannabinoid reuptake inhibitor and a TRPV (1) activator with neuroprotective and anticancer …
Formula:
C26H37NO2
Color and Shape:
Solid
Molecular weight:
395.58
Ref: TM-T39281
| 5mg | 68.00 € | ||
| 10mg | 109.00 € | ||
| 50mg | 434.00 € | ||
| 100mg | 740.00 € |
Estimated delivery in United States, on Friday 24 Jan 2025
Soquinolol
CAS:61563-18-6
Soquinolol (Soquinolol mucate) is a beta-adrenergic receptor antagonist with weak local anesthetic activity.Soquinolol has good …
Formula:
C17H26N2O3
Purity:
98% - 98.49%
Color and Shape:
Solid
Molecular weight:
306.4
Ref: TM-T28829
| 1mg | 141.00 € | ||
| 5mg | 325.00 € | ||
| 10mg | 492.00 € | ||
| 25mg | 803.00 € | ||
| 50mg | 1,095.00 € | ||
| 100mg | 1,483.00 € | ||
| 500mg | 2,974.00 € |
Estimated delivery in United States, on Friday 24 Jan 2025
Felcisetrag
CAS:916075-84-8
Felcisetrag (TD-8954), an oral 5-HT4 agonist with GI prokinetic effects, has a high affinity (pKi …
Formula:
C25H37N5O3
Purity:
100%
Color and Shape:
Solid
Molecular weight:
455.59
Ref: TM-T28934
| 1mg | 151.00 € | ||
| 5mg | 371.00 € | ||
| 10mg | 547.00 € | ||
| 25mg | 878.00 € | ||
| 50mg | 1,188.00 € | ||
| 100mg | 1,616.00 € | ||
| 500mg | 3,226.00 € | ||
| 1mL*10mM (DMSO) | 411.00 € |
Estimated delivery in United States, on Friday 24 Jan 2025
Bevenopran
CAS:676500-67-7
Bevenopran (CB-5945) is a peripheral antagonist of μ-opioid receptor and can be used in studies …
Formula:
C20H26N4O4
Purity:
98.14% - 98.76%
Color and Shape:
Solid
Molecular weight:
386.44
Ref: TM-T14551
| 1mg | 95.00 € | ||
| 5mg | 217.00 € | ||
| 10mg | 323.00 € | ||
| 25mg | 518.00 € | ||
| 50mg | 705.00 € | ||
| 100mg | 920.00 € | ||
| 500mg | 1,845.00 € | ||
| 1mL*10mM (DMSO) | 242.00 € |
Estimated delivery in United States, on Friday 24 Jan 2025
Medifoxamine
CAS:32359-34-5
Medifoxamine (LG 152) is a selective non-monoamine oxidase inhibitor that exhibits antidepressant activity through inhibition …
Formula:
C16H19NO2
Purity:
98.35%
Color and Shape:
Solid
Molecular weight:
257.33
Ref: TM-T24444
| 1mg | 96.00 € | ||
| 5mg | 229.00 € | ||
| 10mg | 344.00 € | ||
| 25mg | 618.00 € | ||
| 50mg | 868.00 € | ||
| 100mg | 1,128.00 € | ||
| 1mL*10mM (DMSO) | 252.00 € |
Estimated delivery in United States, on Friday 24 Jan 2025
Mavorixafor
CAS:558447-26-0
Mavorixafor (AMD-070) is an effective and selective antagonist of CXCR4, with an IC50 value of …
Formula:
C21H27N5
Purity:
98.56%
Color and Shape:
Solid
Molecular weight:
349.47
Ref: TM-TQ0174
| 1mg | 69.00 € | ||
| 2mg | 90.00 € | ||
| 5mg | 150.00 € | ||
| 10mg | 216.00 € | ||
| 25mg | 387.00 € | ||
| 50mg | 575.00 € | ||
| 100mg | 816.00 € | ||
| 1mL*10mM (DMSO) | 248.00 € |
Estimated delivery in United States, on Friday 24 Jan 2025
ROS 234 dioxalate
CAS:1781941-93-2
ROS 234 dioxalate is a potent antagonist of H3(pKB of 9.46 for Guinea-pig ileum H3-receptor)
Formula:
C17H19N5O8
Purity:
98%
Color and Shape:
Solid
Molecular weight:
421.37
Ref: TM-T12756
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Friday 24 Jan 2025
GSK-239512
CAS:720691-69-0
GSK-239512 is an antagonist of H3 receptor and can be used in studies about the …
Formula:
C23H27N3O2
Purity:
98.50% - 99.72%
Color and Shape:
Solid
Molecular weight:
377.48
Ref: TM-T27462
| 1mg | 46.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 111.00 € | ||
| 25mg | 184.00 € | ||
| 50mg | 276.00 € | ||
| 100mg | 416.00 € |
Estimated delivery in United States, on Friday 24 Jan 2025
Impromidine hydrochloride
CAS:65573-02-6
Impromidine hydrochloride is a very potent and specific histamine H2 receptor agonist for conducting cardiovascular …
Formula:
C14H26Cl3N7S
Purity:
99.50%
Color and Shape:
Liquid
Molecular weight:
430.83
Ref: TM-T68921
| 1mg | 240.00 € | ||
| 5mg | 599.00 € | ||
| 10mg | 853.00 € | ||
| 25mg | 1,280.00 € | ||
| 50mg | 1,729.00 € | ||
| 100mg | 2,331.00 € | ||
| 500mg | 4,577.00 € |
Estimated delivery in United States, on Friday 24 Jan 2025
