G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
Read more
Siponimod fumarate
CAS:1234627-85-0
Siponimod is a synthetic, polymorphic drug that has been developed to treat autoimmune and inflammatory …
Purity:
Min. 95%
Ref: 3D-BS168323
| 1g | 2,067.00 € | ||
| 50mg | 230.00 € | ||
| 100mg | 380.00 € | ||
| 250mg | 715.00 € | ||
| 500mg | 1,173.00 € |
Estimated delivery in United States, on Friday 29 Nov 2024
MOR agonist-1
CAS:2305781-14-8
MOR Agonist-1 is a μ-opioid receptor (MOR) agonist noted for its potent analgesic properties and …
Formula:
C22H26ClFN2O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
404.91
Ref: TM-T79060
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 10 Dec 2024
PF-02575799
CAS:863491-70-7
PF-02575799 is an inhibitor of microsomal triglyceride transfer protein (MTP) (IC50: 0.77±0.29 nM).
Formula:
C42H37FN4O4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
680.77
Ref: TM-T16158
| 25mg | 1,688.00 € | ||
| 50mg | 2,225.00 € | ||
| 100mg | 2,897.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
GPR40 Agonist 2
CAS:1147729-48-3
GPR40 Agonist 2 is a GPR40 agonist. It can be used in the research of …
Formula:
C24H30O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
366.49
Ref: TM-T10507
| 25mg | 1,822.00 € | ||
| 50mg | 2,406.00 € | ||
| 100mg | 3,170.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
S1P1 agonist 6 hemicalcium
CAS:2941310-03-6
Compound I (S1P1 agonist 6 hemicalcium) is an S1P1 agonist that diminishes autoimmune activity by …
Formula:
C25H26F3NO3Ca
Purity:
98%
Color and Shape:
Solid
Molecular weight:
465.51
Ref: TM-T79817
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 10 Dec 2024
5-HT2A receptor agonist-3
CAS:1391499-52-7
5-HT2A receptor agonist-3 represents the highest selectivity for the human 5-HT2A receptor currently identified, exhibiting …
Formula:
C21H26BrNO3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
420.34
Ref: TM-T79155
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 10 Dec 2024
GPR120 Agonist 1
CAS:1628448-77-0
GPR120 Agonist 1 selectively activates human/mouse GPR120 with EC50 of 42/77 nM in HEK293 cells.
Formula:
C20H12ClF6NO3S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
495.82
Ref: TM-T11452
| 25mg | 1,683.00 € | ||
| 50mg | 2,219.00 € | ||
| 100mg | 2,891.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
WAY-607695
CAS:380469-52-3
WAY-607695 is a potential 5-HT1A receptor agonist.
Formula:
C13H12FNO2
Purity:
99.82%
Color and Shape:
Solid
Molecular weight:
233.24
Ref: TM-T80805
| 5mg | 46.00 € | ||
| 10mg | 69.00 € | ||
| 25mg | 102.00 € | ||
| 50mg | 148.00 € | ||
| 100mg | 214.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
GLP-1R agonist 3
CAS:2428640-18-8
GLP-1R agonist 3 is a GLP-1R agonist, an imidazole derivative.GLP-1R agonist 3 can be used …
Formula:
C31H28FN5O4
Purity:
97.19%
Color and Shape:
Solid
Molecular weight:
553.58
Ref: TM-T63909
| 1mg | 126.00 € | ||
| 5mg | 292.00 € | ||
| 10mg | 479.00 € | ||
| 25mg | 921.00 € | ||
| 50mg | 1,548.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
SB 258719
CAS:195199-95-2
SB 258719 is a selective antagonist of 5-HT7 receptor with pKi of 7.5.
Formula:
C18H30N2O2S
Purity:
98.59%
Color and Shape:
Solid
Molecular weight:
338.51
Ref: TM-T12855
| 1mg | 41.00 € | ||
| 1ml | 92.00 € | ||
| 5mg | 90.00 € | ||
| 10mg | 132.00 € | ||
| 25mg | 258.00 € | ||
| 50mg | 414.00 € | ||
| 100mg | 616.00 € | ||
| 500mg | 1,290.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
OMDM-5
CAS:616884-66-3
OMDM-5 is a potent vanilloid receptor type 1 (TRPV1, EC50 = 75 nM) agonist, showing …
Formula:
C26H44N2O3
Purity:
99.72%
Color and Shape:
Solid
Molecular weight:
432.64
Ref: TM-T12306
| 1mg | 94.00 € | ||
| 1ml | 214.00 € | ||
| 5mg | 181.00 € | ||
| 10mg | 273.00 € | ||
| 25mg | 436.00 € | ||
| 50mg | 621.00 € | ||
| 100mg | 835.00 € | ||
| 200mg | 1,089.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Sigma-1 receptor antagonist 1
CAS:1639220-19-1
Sigma-1 receptor antagonist 1 is an effective and selective antagonist of sigma-1 receptor.
Formula:
C19H23Cl2N3O
Purity:
99.81%
Color and Shape:
Solid
Molecular weight:
380.31
Ref: TM-T12910
| 1mg | 62.00 € | ||
| 5mg | 141.00 € | ||
| 10mg | 218.00 € | ||
| 25mg | 365.00 € | ||
| 50mg | 519.00 € | ||
| 100mg | 703.00 € | ||
| 200mg | 903.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Todralazine hydrochloride
CAS:3778-76-5
Todralazine hydrochloride, a β2AR blocker with antioxidant properties, is used in hypertension studies.
Formula:
C11H13ClN4O2
Purity:
98.32%
Color and Shape:
Solid
Molecular weight:
268.7
Ref: TM-T17111
| 1ml | 34.00 € | ||
| 25mg | 41.00 € | ||
| 50mg | 61.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
CB1 inverse agonist 1
CAS:852315-00-5
MRL-650 is an oral, selective CB1 agonist; IC50: CB1=7.5 nM, CB2=4100 nM; anorexigenic effects noted.
Formula:
C25H18Cl3N3O3
Purity:
99.12%
Color and Shape:
Solid
Molecular weight:
514.79
Ref: TM-T10694
| 1mg | 113.00 € | ||
| 1ml | 310.00 € | ||
| 5mg | 250.00 € | ||
| 10mg | 368.00 € | ||
| 25mg | 552.00 € | ||
| 50mg | 772.00 € | ||
| 100mg | 1,053.00 € | ||
| 500mg | 2,115.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Velagliflozin
CAS:946525-65-1
Velagliflozin is an orally available inhibitor of sodium-glucose cotransporter 2.
Formula:
C23H25NO5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
395.45
Ref: TM-T17221
| 25mg | 1,961.00 € | ||
| 50mg | 2,600.00 € | ||
| 100mg | 3,460.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
RBC10
CAS:362503-73-9
RBC10 inhibits the binding of Ral to its effector RALBP1, as well as inhibiting Ral-mediated …
Formula:
C24H25ClN2O2
Purity:
98.38%
Color and Shape:
Solid
Molecular weight:
408.92
Ref: TM-T24706
| 1mg | 34.00 € | ||
| 1ml | 83.00 € | ||
| 2mg | 51.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 112.00 € | ||
| 25mg | 250.00 € | ||
| 50mg | 361.00 € | ||
| 100mg | 525.00 € | ||
| 200mg | 712.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Talibegron hydrochloride
CAS:178600-17-4
Talibegron hydrochloride: β3 adrenoceptor agonist, pD2 3.72, relaxes rat arteries, reduces leptin in mice.
Formula:
C18H22ClNO4
Purity:
99.82%
Color and Shape:
Solid
Molecular weight:
351.83
Ref: TM-T23557
| 1mg | 53.00 € | ||
| 5mg | 105.00 € | ||
| 10mg | 130.00 € | ||
| 25mg | 278.00 € | ||
| 50mg | 403.00 € | ||
| 100mg | 551.00 € | ||
| 500mg | 1,098.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Selvigaltin
CAS:1978336-95-6
Selvigaltin (GB1211) is a Gal-3 inhibitor with potential anticancer activity. Selvigaltin is used in the …
Formula:
C19H16BrF3N4O4S
Purity:
99.97%
Color and Shape:
Solid
Molecular weight:
533.32
Ref: TM-T63751
| 1mg | 269.00 € | ||
| 5mg | 642.00 € | ||
| 10mg | 1,097.00 € | ||
| 25mg | 2,314.00 € | ||
| 50mg | 3,671.00 € | ||
| 100mg | 5,538.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
COR659
CAS:544450-68-2
COR659: suppresses alcohol/chocolate intake in rats; enhances GABAB receptor, blocks CB1 receptor.
Formula:
C16H16ClNO3S
Purity:
99.56%
Color and Shape:
Solid
Molecular weight:
337.82
Ref: TM-T36520
| 1mg | 51.00 € | ||
| 1ml | 124.00 € | ||
| 2mg | 73.00 € | ||
| 5mg | 112.00 € | ||
| 10mg | 173.00 € | ||
| 25mg | 313.00 € | ||
| 50mg | 436.00 € | ||
| 100mg | 598.00 € | ||
| 200mg | 814.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Sigma-1 receptor antagonist 3
CAS:1639220-17-9
Sigma-1 receptor antagonist 3 is a more potent and selective antagonist of Sigma-1 (σ1) receptor …
Formula:
C19H23ClFN3O
Purity:
100%
Color and Shape:
Solid
Molecular weight:
363.86
Ref: TM-T12912
| 1mg | 87.00 € | ||
| 5mg | 183.00 € | ||
| 10mg | 299.00 € | ||
| 25mg | 491.00 € | ||
| 50mg | 666.00 € | ||
| 100mg | 884.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
