G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Cyclazosin HCl
CAS:146929-33-1
Cyclazosin HCl is an α-adrenergic receptor antagonist that can be used to study non-arteritic ischemic …
Formula:
C23H28ClN5O4
Purity:
99.44%
Color and Shape:
Liquid
Molecular weight:
473.95
Ref: TM-T70585
| 1mg | 279.00 € | ||
| 5mg | 685.00 € | ||
| 10mg | 938.00 € | ||
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € |
Estimated delivery in United States, on Friday 16 May 2025
L-694,247
CAS:137403-12-4
L-694,247 is a 5-HT receptor agonist with affinity for 5-HT1D, 5-HT1A, 5-HT1B, 5-HT1C, and 5-HT1E …
Formula:
C20H21N5O3S
Purity:
98.36%
Color and Shape:
White Solid
Molecular weight:
411.48
Ref: TM-T19701
| 1mg | 82.00 € | ||
| 5mg | 264.00 € | ||
| 10mg | 452.00 € | ||
| 25mg | 740.00 € | ||
| 50mg | 1,035.00 € |
Estimated delivery in United States, on Friday 16 May 2025
Adatanserin
CAS:127266-56-2
Adatanserin (WY 50324) is a mixed 5-HT1A receptor partial agonist and a 5-HT2A and 5-HT2C …
Formula:
C21H31N5O
Purity:
99.17%
Color and Shape:
Solid
Molecular weight:
369.5
Ref: TM-T23631
| 1mg | 279.00 € | ||
| 5mg | 685.00 € | ||
| 10mg | 938.00 € | ||
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Friday 16 May 2025
Endomorphin 1 acetate
CAS:1276123-71-7
Endomorphin 1 acetate is a μ-opioid receptor agonist with antinociceptive and analgesic effects and can …
Formula:
C36H42N6O7
Color and Shape:
Liquid
Molecular weight:
670.75
Ref: TM-T72423
| 2mg | 44.00 € |
Estimated delivery in United States, on Friday 16 May 2025
GPR35 agonist 2
CAS:494191-73-0
GPR35 agonist 2 (TC-G 1001) is a potent GPR35 agonist.The EC50 values of GPR35 agonist …
Formula:
C17H11FN2O3S
Purity:
97.18% - 98.40%
Color and Shape:
Solid
Molecular weight:
342.34
Ref: TM-T23434
| 1mg | 52.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 170.00 € | ||
| 25mg | 378.00 € | ||
| 50mg | 560.00 € | ||
| 100mg | 800.00 € | ||
| 500mg | 1,644.00 € | ||
| 1mL*10mM (DMSO) | 114.00 € |
Estimated delivery in United States, on Friday 16 May 2025
6-Chloromelatonin
CAS:63762-74-3
6-Chloromelatonin: potent, stable melatonin agonist; binds MT2 receptors (pKi=9.77); could help research sleep disorders.
Formula:
C13H15ClN2O2
Purity:
97.90% - 99.36%
Color and Shape:
Solid
Molecular weight:
266.72
Ref: TM-T22530
| 1mg | 333.00 € | ||
| 5mg | 787.00 € | ||
| 10mg | 1,074.00 € | ||
| 25mg | 1,510.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € | ||
| 500mg | 4,655.00 € |
Estimated delivery in United States, on Friday 16 May 2025
E-4177
CAS:135070-05-2
E-4177 is an angiotensin II type 1 receptor (AT1R) antagonist and can be used to …
Formula:
C24H21N3O2
Purity:
98.63% - 99.39%
Color and Shape:
Solid
Molecular weight:
383.44
Ref: TM-T27229
| 1mg | 279.00 € | ||
| 5mg | 685.00 € | ||
| 10mg | 938.00 € | ||
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € |
Estimated delivery in United States, on Friday 16 May 2025
SC 19220
CAS:19395-87-0
SC 19220 is a prostaglandin E2 receptor EP1 antagonist that inhibits RANKL-induced osteoclastogenesis.
Formula:
C16H14ClN3O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
331.75
Ref: TM-T23330
| 1mg | 58.00 € | ||
| 5mg | 219.00 € | ||
| 10mg | 375.00 € | ||
| 25mg | 795.00 € |
Estimated delivery in United States, on Friday 16 May 2025
QS11
CAS:944328-88-5
QS11, a GTPase ARFGAP1, modulates ARF-GTP levels and synergizes with the Wnt/β-catenin signaling pathway to …
Formula:
C36H33N5O2
Purity:
98.39%
Color and Shape:
Solid
Molecular weight:
567.68
Ref: TM-T4022
| 2mg | 35.00 € | ||
| 5mg | 52.00 € | ||
| 10mg | 85.00 € | ||
| 25mg | 156.00 € | ||
| 50mg | 226.00 € | ||
| 100mg | 340.00 € | ||
| 200mg | 465.00 € | ||
| 1mL*10mM (DMSO) | 65.00 € |
Estimated delivery in United States, on Friday 16 May 2025
L 674573
CAS:127481-29-2
L 674573 is an inhibitor of leukotriene biosynthesis.
Formula:
C28H27NO3S
Purity:
99.22%
Color and Shape:
Solid
Molecular weight:
457.58
Ref: TM-T24327
| 5mg | 55.00 € | ||
| 10mg | 82.00 € | ||
| 25mg | 126.00 € | ||
| 50mg | 182.00 € | ||
| 100mg | 273.00 € | ||
| 1mL*10mM (DMSO) | 82.00 € |
Estimated delivery in United States, on Friday 16 May 2025
JNJ 10191584 maleate
CAS:869497-75-6
JNJ 10191584 maleate (VUF6002 maleate) is an orally active and selective antagonist of H4 receptor …
Formula:
C17H19ClN4O5
Purity:
99.82%
Color and Shape:
Solid
Molecular weight:
394.81
Ref: TM-T22879
| 1mg | 54.00 € | ||
| 2mg | 82.00 € | ||
| 5mg | 107.00 € | ||
| 10mg | 133.00 € | ||
| 25mg | 284.00 € | ||
| 50mg | 411.00 € | ||
| 100mg | To inquire |
Estimated delivery in United States, on Friday 16 May 2025
Torbafylline
CAS:105102-21-4
Torbafylline is a xanthine-based PDE inhibitor reducing protein breakdown via PDE4/cAMP/EPAC/PI3K/Akt in rats with burns, …
Formula:
C16H26N4O4
Purity:
98% - 99%
Color and Shape:
Soild
Molecular weight:
338.4
Ref: TM-T67965
| 1mg | 128.00 € | ||
| 5mg | 304.00 € | ||
| 10mg | 457.00 € | ||
| 25mg | 747.00 € | ||
| 50mg | 1,026.00 € | ||
| 100mg | 1,406.00 € | ||
| 500mg | 2,812.00 € | ||
| 1mL*10mM (DMSO) | 314.00 € |
Estimated delivery in United States, on Friday 16 May 2025
CAY10786
CAS:1239987-91-7
CAY10786 (GPR52 antagonist-1) is an antagonist of G protein-coupled receptor 52 (GPR52, IC50 = 0.63 …
Formula:
C15H14OS
Purity:
99.84%
Color and Shape:
Solid
Molecular weight:
242.34
Ref: TM-T36036
| 2mg | 40.00 € | ||
| 5mg | 60.00 € | ||
| 10mg | 87.00 € | ||
| 25mg | 187.00 € | ||
| 50mg | 298.00 € | ||
| 100mg | 469.00 € | ||
| 1mL*10mM (DMSO) | 66.00 € |
Estimated delivery in United States, on Friday 16 May 2025
Clonidine
CAS:4205-90-7
Clonidine (Kapvay): central alpha-adrenergic agonist, antihypertensive, often combined, not tied to liver issues.
Formula:
C9H9Cl2N3
Purity:
99.44% - 99.88%
Color and Shape:
Crystals Solid
Molecular weight:
230.09
Ref: TM-T7045
| 50mg | 89.00 € | ||
| 100mg | 130.00 € |
Estimated delivery in United States, on Friday 16 May 2025
Viloxazine
CAS:46817-91-8
Viloxazine (Viloxazin) (Viloxazin) is a dual-action compound that functions as a norepinephrine reuptake inhibitor and …
Formula:
C13H19NO3
Purity:
99.8%
Color and Shape:
Liquid
Molecular weight:
237.29
Ref: TM-T60325
| 5mg | 40.00 € | ||
| 10mg | 52.00 € | ||
| 25mg | 97.00 € | ||
| 50mg | 154.00 € | ||
| 100mg | 235.00 € | ||
| 200mg | 349.00 € |
Estimated delivery in United States, on Friday 16 May 2025
SPD-473 citrate
CAS:161190-26-7
SPD-473 citrate is an inhibitior of serotonin/dopamine/norepinephrine reuptake.
Formula:
C23H31Cl2NO8S
Purity:
99.37%
Color and Shape:
Solid
Molecular weight:
552.47
Ref: TM-T13898
| 1mg | 235.00 € | ||
| 5mg | 588.00 € | ||
| 10mg | 825.00 € | ||
| 25mg | 1,320.00 € | ||
| 50mg | 1,776.00 € | ||
| 100mg | 2,403.00 € |
Estimated delivery in United States, on Friday 16 May 2025
A 61603
CAS:107756-30-9
Cixutumumab (IMC-A12) is a humanized IgG monoclonal antibody targeting the IGF1R with anticancer activity.
Formula:
C14H20BrN3O3S
Color and Shape:
Solid
Molecular weight:
390.3
Ref: TM-T21927
| 1mg | 86.00 € | ||
| 5mg | 238.00 € | ||
| 10mg | 330.00 € |
Estimated delivery in United States, on Friday 16 May 2025
ML192
CAS:460331-61-7
ML192 (CID1434953) is a selective GPR55 ligand antagonist.
Formula:
C20H22N4O2S
Purity:
99.79%
Color and Shape:
Solid
Molecular weight:
382.48
Ref: TM-T33452
| 1mg | 35.00 € | ||
| 5mg | 74.00 € | ||
| 10mg | 110.00 € | ||
| 25mg | 182.00 € | ||
| 50mg | 263.00 € | ||
| 100mg | 369.00 € | ||
| 200mg | 507.00 € | ||
| 1mL*10mM (DMSO) | 96.00 € |
Estimated delivery in United States, on Friday 16 May 2025
GSK1521498 free base (hydrochloride)
CAS:1007578-24-6
GSK1521498 free base (hydrochloride) is a selective antagonist of the μ-opioid receptor (MOR).
Formula:
C24H21ClF2N4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
438.9
Ref: TM-T11478
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Friday 16 May 2025
GW438014A
CAS:469861-49-2
GW438014A 是一种有效且具有选择性的 NPY-Y5 受体拮抗剂。GW438014A 对食物摄入并减少肥胖啮齿动物的体重增加具有抑制作用。
Formula:
C23H23N3O4S
Purity:
100%
Color and Shape:
Solid
Molecular weight:
437.51
Ref: TM-T24121
| 2mg | 35.00 € | ||
| 5mg | 52.00 € | ||
| 10mg | 85.00 € | ||
| 25mg | 156.00 € | ||
| 50mg | 235.00 € | ||
| 100mg | 335.00 € | ||
| 200mg | 467.00 € |
Estimated delivery in United States, on Friday 16 May 2025
