G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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JTE-907
CAS:282089-49-0
JTE-907 是一种具有高度选择性和口服活性的 CB2 受体反向激动剂。JTE-907在体内展现出抗炎活性。
Formula:
C24H26N2O6
Purity:
100%
Color and Shape:
Solid
Molecular weight:
438.47
Ref: TM-T19705
| 1mg | 56.00 € | ||
| 5mg | 126.00 € | ||
| 10mg | 187.00 € | ||
| 25mg | 329.00 € | ||
| 50mg | 490.00 € | ||
| 100mg | 700.00 € | ||
| 1mL*10mM (DMSO) | 150.00 € |
Estimated delivery in United States, on Friday 16 May 2025
Fipamezole
CAS:150586-58-6
Fipamezole is a potent alpha2 adrenergic receptor antagonist that may be useful for studying autonomic …
Formula:
C14H15FN2
Purity:
100% - 99.32%
Color and Shape:
Solid
Molecular weight:
230.28
Ref: TM-T24064
| 1mg | 597.00 € | ||
| 5mg | 1,283.00 € | ||
| 25mg | 1,691.00 € | ||
| 50mg | 2,072.00 € | ||
| 100mg | 2,660.00 € |
Estimated delivery in United States, on Friday 16 May 2025
Landipirdine
CAS:1000308-25-7
Landipirdine (RO-5025181) is a selective 5-HT6R antagonist for the study of central nervous system disorders …
Formula:
C18H19FN2O3S
Purity:
97.50% - 99.33%
Color and Shape:
Solid
Molecular weight:
362.42
Ref: TM-T27795
| 1mg | 235.00 € | ||
| 5mg | 562.00 € | ||
| 10mg | 753.00 € | ||
| 25mg | 1,216.00 € | ||
| 50mg | 1,549.00 € | ||
| 100mg | 2,205.00 € |
Estimated delivery in United States, on Friday 16 May 2025
Faxeladol
CAS:433265-65-7
Faxeladol: adrenergic, serotonin inhibitor & opioid agonist for neurological studies.
Formula:
C15H23NO
Purity:
99.11% - 99.13%
Color and Shape:
Solid
Molecular weight:
233.35
Ref: TM-T31750
| 1mg | 597.00 € | ||
| 5mg | 1,283.00 € | ||
| 25mg | 1,691.00 € | ||
| 50mg | 2,072.00 € | ||
| 100mg | 2,660.00 € |
Estimated delivery in United States, on Friday 16 May 2025
T-0509
CAS:96843-99-1
T-0509 is a selective beta 1 receptor agonist that increases inotropy in canine ventricular muscle …
Formula:
C18H23NO5
Purity:
97.46% - 98.21%
Color and Shape:
Solid
Molecular weight:
333.38
Ref: TM-T28895
| 1mg | 333.00 € | ||
| 5mg | 787.00 € | ||
| 10mg | 1,074.00 € | ||
| 25mg | 1,510.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Friday 16 May 2025
Edonentan
CAS:210891-04-6
Edonentan is A potent endothelin A (ETA) receptor antagonist that can be used to study …
Formula:
C28H32N4O5S
Purity:
98.78% - 99%
Color and Shape:
Solid
Molecular weight:
536.64
Ref: TM-T31605
| 1mg | 939.00 € | ||
| 5mg | 1,882.00 € | ||
| 25mg | 2,403.00 € | ||
| 50mg | 2,832.00 € | ||
| 100mg | 3,800.00 € |
Estimated delivery in United States, on Friday 16 May 2025
BTB09089
CAS:245728-44-3
BTB09089 (GPR65 agonist ) is a T cell death-associated gene 8 (TDAG8/GPR65)-specific agonist.BTB09089 induces TDAG8 …
Formula:
C14H12Cl2N4OS2
Purity:
100%
Color and Shape:
Soild
Molecular weight:
387.31
Ref: TM-T67892
| 1mg | 71.00 € | ||
| 5mg | 124.00 € | ||
| 10mg | 188.00 € | ||
| 25mg | 343.00 € | ||
| 50mg | 522.00 € | ||
| 100mg | 750.00 € | ||
| 500mg | 1,549.00 € |
Estimated delivery in United States, on Friday 16 May 2025
Darbufelone
CAS:139226-28-1
Darbufelone (CI-1004) is a non-competitive dual inhibitor of PGF2α and LTB4.
Formula:
C18H24N2O2S
Purity:
99.77%
Color and Shape:
Solid
Molecular weight:
332.46
Ref: TM-T10960
| 1mg | 44.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 131.00 € | ||
| 25mg | 279.00 € | ||
| 50mg | 408.00 € | ||
| 100mg | 562.00 € | ||
| 500mg | 1,121.00 € | ||
| 1mL*10mM (DMSO) | 110.00 € |
Estimated delivery in United States, on Friday 16 May 2025
ReN-1869
CAS:170149-99-2
ReN-1869 is a novel selective histamine H(1) receptor antagonist with anti-neurogenic pain and anti-inflammatory activity …
Formula:
C24H27NO2
Purity:
99.87% - 99.89%
Color and Shape:
Solid
Molecular weight:
361.48
Ref: TM-T28516
| 1mg | 208.00 € | ||
| 5mg | 520.00 € | ||
| 10mg | 752.00 € | ||
| 25mg | 1,159.00 € | ||
| 50mg | 1,882.00 € |
Estimated delivery in United States, on Friday 16 May 2025
Avosentan
CAS:290815-26-8
Avosentan(Ro 67-0565; SPP-301) is a potent endothelin receptor (ETA) antagonist.Cost-effective and quality-assured.
Formula:
C23H21N5O5S
Purity:
98.25% - 99.47%
Color and Shape:
Solid
Molecular weight:
479.51
Ref: TM-TQ0282
| 1mg | 40.00 € | ||
| 5mg | 85.00 € | ||
| 10mg | 106.00 € | ||
| 25mg | 216.00 € | ||
| 50mg | 376.00 € | ||
| 100mg | 550.00 € | ||
| 1mL*10mM (DMSO) | 88.00 € |
Estimated delivery in United States, on Friday 16 May 2025
SLM6031434 HCl
CAS:1897379-34-8
SLM6031434 HCl (SLM-6031434 HCl) is a SphK2 inhibitor that reduces LPS-induced TNF伪 and IL-1尾 production.
Formula:
C22H31ClF3N5O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
489.96
Ref: TM-T28806
| 1mg | 126.00 € | ||
| 5mg | 398.00 € | ||
| 10mg | 547.00 € |
Estimated delivery in United States, on Friday 16 May 2025
Isbogrel
CAS:89667-40-3
Isbogrel (CV4151) is a TXA2 synthase inhibitor for researching arrhythmias, ischemic attacks, and thrombosis.
Formula:
C18H19NO2
Purity:
97.06%
Color and Shape:
Solid
Molecular weight:
281.35
Ref: TM-T27630
| 1mg | 333.00 € | ||
| 5mg | 787.00 € | ||
| 10mg | 1,074.00 € | ||
| 25mg | 1,510.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Friday 16 May 2025
p-MPPF dihydrochloride
CAS:223699-41-0
p-MPPF dihydrochloride is a 5-HT antagonist that can be used to study neurological diseases.
Formula:
C25H29Cl2FN4O2
Purity:
99.78%
Color and Shape:
Liquid
Molecular weight:
507.43
Ref: TM-T69750
| 1mg | 279.00 € | ||
| 5mg | 685.00 € | ||
| 10mg | 938.00 € | ||
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € |
Estimated delivery in United States, on Friday 16 May 2025
Selodenoson
CAS:110299-05-3
Selodenoson (RG-14202) is a selective adenosine A1 receptor agonist used to slow the heart rate …
Formula:
C17H24N6O4
Purity:
99.33%
Color and Shape:
Solid
Molecular weight:
376.41
Ref: TM-T28748
| 1mg | 88.00 € | ||
| 5mg | 182.00 € | ||
| 10mg | 268.00 € | ||
| 25mg | 439.00 € |
Estimated delivery in United States, on Friday 16 May 2025
DA-6886
CAS:1645260-76-9
DA-6886 is a 5-HT4 agonist, relaxes rat oesophagus, with 1000x selectivity over hERG channels, pIC50: …
Formula:
C19H28Cl2N6O2
Purity:
99% - 99.89%
Color and Shape:
Solid
Molecular weight:
443.37
Ref: TM-T27117
| 1mg | 92.00 € | ||
| 5mg | 192.00 € | ||
| 10mg | 290.00 € | ||
| 25mg | 472.00 € |
Estimated delivery in United States, on Friday 16 May 2025
R 59-022 hydrochloride
CAS:93076-98-3
R 59-022 hydrochloride is a 5-HT antagonist, PKC activator, DGK inhibitor (IC50: 2.8 µM), and …
Formula:
C27H27ClFN3OS
Purity:
97.7%
Color and Shape:
Liquid
Molecular weight:
496.04
Ref: TM-T72322
| 1mg | 46.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 144.00 € | ||
| 25mg | 283.00 € | ||
| 50mg | 454.00 € | ||
| 100mg | 653.00 € | ||
| 500mg | 1,349.00 € |
Estimated delivery in United States, on Friday 16 May 2025
Dabelotine
CAS:118976-38-8
Dabelotine (UNII-6RY56RB98P) is an adrenergic agonist used in the study of dementia.
Formula:
C15H22N2O2
Purity:
98.55%
Color and Shape:
Solid
Molecular weight:
262.35
Ref: TM-T31175
| 1mg | 143.00 € | ||
| 5mg | 333.00 € | ||
| 10mg | 504.00 € | ||
| 25mg | 817.00 € | ||
| 50mg | 1,121.00 € | ||
| 100mg | 1,510.00 € | ||
| 500mg | 3,030.00 € |
Estimated delivery in United States, on Friday 16 May 2025
Femoxetine hydrochloride
CAS:56222-04-9
Femoxetine hydrochloride is a selective 5-hydroxytryptamine reuptake inhibitor used in the study of migraine, depression …
Formula:
C20H26ClNO2
Purity:
99.48%
Color and Shape:
Liquid
Molecular weight:
347.88
Ref: TM-T69096
| 1mg | 124.00 € | ||
| 5mg | 303.00 € | ||
| 10mg | 437.00 € | ||
| 25mg | 672.00 € |
Estimated delivery in United States, on Friday 16 May 2025
FK-453
CAS:121524-18-3
FK-453 is a potent antagonist of non-xanthine adenosine A1 receptor with diuretic and renal vasodilatory …
Formula:
C23H25N3O2
Purity:
99.69%
Color and Shape:
Solid
Molecular weight:
375.46
Ref: TM-T27323
| 1mg | 238.00 € | ||
| 5mg | 590.00 € | ||
| 10mg | 837.00 € | ||
| 25mg | 1,264.00 € | ||
| 50mg | 1,691.00 € | ||
| 100mg | 2,300.00 € | ||
| 500mg | 4,618.00 € |
Estimated delivery in United States, on Friday 16 May 2025
A-437203
CAS:220519-06-2
A-437203 (Lu201640), selective D3 antagonist with Ki: D2-71nM, D3-1.6nM, D4-6220nM; based on 1H-pyrimidin-2-one scaffold.
Formula:
C20H27F3N6OS
Purity:
98.62%
Color and Shape:
Solid
Molecular weight:
456.53
Ref: TM-T10213
| 1mg | 89.00 € | ||
| 5mg | 198.00 € | ||
| 10mg | 279.00 € | ||
| 25mg | 434.00 € | ||
| 50mg | 562.00 € | ||
| 100mg | 780.00 € | ||
| 200mg | 1,035.00 € | ||
| 1mL*10mM (DMSO) | 227.00 € |
Estimated delivery in United States, on Friday 16 May 2025
