G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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CGRP antagonist 1
CAS:1123757-49-2
CGRP antagonist 1 is a potent CGRP receptor antagonist with Ki values of 35 nM …
Formula:
C29H26N4O4
Purity:
100%
Color and Shape:
Solid
Molecular weight:
494.54
Ref: TM-T13453
| 1mg | 324.00 € | ||
| 5mg | 787.00 € | ||
| 10mg | 1,093.00 € | ||
| 25mg | 1,596.00 € | ||
| 50mg | 2,175.00 € | ||
| 100mg | 2,822.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
O-1602
CAS:317321-41-8
O-1602 is a novel GPR55 agonist, an atypical cannabinoid associated with the central nervous system …
Formula:
C17H22O2
Purity:
99.4%
Color and Shape:
Solid
Molecular weight:
258.36
Ref: TM-T23097
| 1mg | 48.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 153.00 € | ||
| 25mg | 298.00 € | ||
| 50mg | 469.00 € | ||
| 100mg | 682.00 € | ||
| 1mL*10mM (DMSO) | 105.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
Ampreloxetine
CAS:1227056-84-9
Ampreloxetine (TD-9855) is a norepinephrine reuptake inhibitor used to study neurological diseases.
Formula:
C18H18F3NO
Purity:
98%
Color and Shape:
Solid
Molecular weight:
321.34
Ref: TM-T26622
| 25mg | 1,444.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
NGD 94-1
CAS:178928-68-2
NGD 94-1 is a D4 receptor antagonist that can be used to study psychiatric disorders …
Formula:
C18H20N6
Purity:
99.84%
Color and Shape:
Solid
Molecular weight:
320.39
Ref: TM-T23066
| 1mg | 93.00 € | ||
| 5mg | 187.00 € | ||
| 10mg | 284.00 € | ||
| 25mg | 560.00 € | ||
| 50mg | 918.00 € | ||
| 100mg | 1,216.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
SLV-310
CAS:264869-71-8
SLV-310 is a D2 receptor antagonist and 5-HT reuptake receptor inhibitor for the study of …
Formula:
C25H24FN3O2
Purity:
98.91%
Color and Shape:
Solid
Molecular weight:
417.48
Ref: TM-T28809
| 1mg | 279.00 € | ||
| 5mg | 685.00 € | ||
| 10mg | 938.00 € | ||
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
EP1-antagonist-1
CAS:851204-35-8
EP1-antagonist-1 (EP1 antagonist 1) is an EP1 antagonist (pKi: 7.54; pIC50: 8.5).
Formula:
C19H15BrCl2N2O3
Purity:
98.51%
Color and Shape:
Solid
Molecular weight:
470.14
Ref: TM-T10031
| 1mg | 185.00 € | ||
| 5mg | 376.00 € | ||
| 10mg | 550.00 € | ||
| 25mg | 867.00 € | ||
| 50mg | 1,159.00 € | ||
| 100mg | 1,568.00 € | ||
| 1mL*10mM (DMSO) | 426.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
5HT6-ligand-1
CAS:1038988-11-2
5HT6-ligand-1 is an orally active ligand of 5-HT6 receptor (Ki = 1.43 nM).
Formula:
C20H22BrN3O2S
Purity:
98.48% - 98.95%
Color and Shape:
Solid
Molecular weight:
448.38
Ref: TM-T10053
| 1mg | 116.00 € | ||
| 5mg | 273.00 € | ||
| 10mg | 373.00 € | ||
| 25mg | 563.00 € | ||
| 50mg | 758.00 € | ||
| 100mg | 998.00 € | ||
| 200mg | 1,320.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
Bedoradrine sulfate
CAS:194785-31-4
Bedoradrine sulfate (MN-221 sulfate) is a novel, highly selective β2-adrenoceptor agonist.Cost-effective and quality-assured.
Formula:
C24H32N2O5H2O4S
Purity:
99.31%
Color and Shape:
Solid
Molecular weight:
477.56
Ref: TM-T26760
| 1mg | 723.00 € | ||
| 5mg | 1,510.00 € | ||
| 25mg | 2,555.00 € | ||
| 50mg | 3,212.00 € | ||
| 100mg | 4,370.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
Ecastolol
CAS:77695-52-4
Ecastolol has anti-angina activity and is an adrenergic receptor antagonist.
Formula:
C26H33N3O6
Purity:
98.1%
Color and Shape:
Solid
Molecular weight:
483.56
Ref: TM-T11148
| 1mg | 369.00 € | ||
| 5mg | 735.00 € | ||
| 10mg | 938.00 € | ||
| 25mg | 1,473.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,670.00 € | ||
| 1mL*10mM (DMSO) | 929.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
RG-12525
CAS:120128-20-3
RG-12525(NID 525) is an orally available, selective and competitive leukotriene D (LTD) antagonist that inhibits …
Formula:
C25H21N5O2
Purity:
96.77%
Color and Shape:
Solid
Molecular weight:
423.47
Ref: TM-T16739
| 2mg | 166.00 € | ||
| 25mg | 868.00 € | ||
| 50mg | 1,320.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
CCK-A receptor inhibitor 1
CAS:137004-80-9
CCK-A receptor inhibitor 1 is a potent inhibitor of the cholecystokinin A (CCK-A) receptor (IC50: …
Formula:
C25H35NO6S
Purity:
99.47%
Color and Shape:
Solid
Molecular weight:
477.61
Ref: TM-T12404
| 1mg | 665.00 € | ||
| 5mg | 1,710.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
Pamatolol
CAS:59110-35-9
Pamatolol is a selective and potent beta-adrenoceptor antagonist that has not shown sympathomimetic activity in …
Formula:
C16H26N2O4
Purity:
100%
Color and Shape:
Solid
Molecular weight:
310.39
Ref: TM-T16431
| 1mg | 665.00 € | ||
| 5mg | 1,710.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
SC 51089
CAS:146033-02-5
SC 51089 is a somatic PGE2 antagonist with anti-injurious activity and may rescue memory loss.
Formula:
C22H20Cl2N4O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
459.33
Ref: TM-T23331
| 1mg | 279.00 € | ||
| 5mg | 685.00 € | ||
| 10mg | 938.00 € | ||
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
(Iso)-FK-480
CAS:167820-10-2
(Iso)-FK-480 is a novel orally available cholecystokinin A (CCK-A) antagonist for investigational treatment of chronic …
Formula:
C26H19FN4O2
Purity:
100% - 99.68%
Color and Shape:
Solid
Molecular weight:
438.45
Ref: TM-T10055
| 1mg | 279.00 € | ||
| 5mg | 685.00 € | ||
| 10mg | 938.00 € | ||
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
LY377604
CAS:204592-94-9
LY377604 is a human β3-adrenergic receptor agonist (EC50: 2.4 nM) and β1/2-adrenergic receptor antagonist for …
Formula:
C31H32N4O4
Purity:
100% - 99.72%
Color and Shape:
Solid
Molecular weight:
524.61
Ref: TM-T15819
| 1mg | 125.00 € | ||
| 5mg | 303.00 € | ||
| 10mg | 449.00 € | ||
| 25mg | 735.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
Butofilolol
CAS:58930-32-8
Butofilolol is a novel beta-blocker with antihypertensive activity and can be used to study hypertension.
Formula:
C17H26FNO3
Purity:
100% - 99%
Color and Shape:
Liquid
Molecular weight:
311.392
Ref: TM-T60773
| 1mg | 279.00 € | ||
| 5mg | 685.00 € | ||
| 10mg | 938.00 € | ||
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
QF0301B
CAS:149247-12-1
QF0301B is a potent α1-adrenergic receptor antagonist with inhibitory effects on α2-adrenergic receptors, 5-HT2A and …
Formula:
C23H28N2O2
Purity:
99.16%
Color and Shape:
Solid
Molecular weight:
364.48
Ref: TM-T10100
| 1mg | 665.00 € | ||
| 5mg | 1,710.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
Rocastine
CAS:91833-49-7
Rocastine (AHR-11325) is a selective and potent non-sedating H1 receptor antagonist.
Formula:
C13H19N3OS
Purity:
98.26%
Color and Shape:
Solid
Molecular weight:
265.37
Ref: TM-T16778
| 1mg | 665.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
MEN11467
CAS:214487-46-4
MEN11467 is a novel, orally available, potent and selective peptidomimetic tachykinin NK 1 receptor antagonist …
Formula:
C38H40N4O3
Purity:
100%
Color and Shape:
Solid
Molecular weight:
600.75
Ref: TM-T12000
| 1mg | 650.00 € | ||
| 5mg | 1,672.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
H3 receptor-MO-1
CAS:1240914-03-7
H3 receptor-MO-1 is a potent modulator of the histamine H3 receptor (H3 receptor) and can …
Formula:
C20H27N3O2
Purity:
99.11%
Color and Shape:
Solid
Molecular weight:
341.45
Ref: TM-T10499
| 1mg | 665.00 € | ||
| 5mg | 1,710.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
