G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Tedalinab
CAS:916591-01-0
Tedalinab is an effective and selective cannabinoid receptor 2 agonist.
Formula:
C19H21F2N3O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
345.39
Ref: TM-T17027
| 25mg | 1,055.00 € | ||
| 50mg | 1,411.00 € | ||
| 100mg | 2,198.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Timiperone
CAS:57648-21-2
Timiperone exhibits a high affinity for cerebral dopamine D2 receptors, demonstrating antipsychotic activity as it …
Formula:
C22H24FN3OS
Purity:
98%
Color and Shape:
Solid
Molecular weight:
397.51
Ref: TM-T78514
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Omidenepag isopropyl
CAS:1187451-19-9
Omidenepag isopropyl (DE-117) is a prostaglandin EP2 receptor agonist used in the study of glaucoma …
Formula:
C26H28N6O4S
Purity:
99.78%
Color and Shape:
Solid
Molecular weight:
520.6
Ref: TM-T16388
| 1g | 8,740.00 € | ||
| 1mg | 56.00 € | ||
| 5mg | 119.00 € | ||
| 10mg | 185.00 € | ||
| 25mg | 425.00 € | ||
| 50mg | 734.00 € | ||
| 100mg | 1,198.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Icalcaprant
CAS:2227384-17-8
Icalcaprant is a kappa-opioid receptor antagonist [1].
Formula:
C23H26N4O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
406.48
Ref: TM-T79848
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 10 Dec 2024
AM-1638
CAS:1142214-62-7
AM-1638 is a full agonist of GPR40/FFA1 (EC50: 0.16 μM).
Formula:
C33H35FO4
Color and Shape:
Solid
Molecular weight:
514.63
Ref: TM-T14200
| 25mg | 829.00 € | ||
| 50mg | 1,086.00 € | ||
| 100mg | 1,629.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
NKP608
CAS:177707-12-9
NKP608 is a NK-1 receptor antagonist with anticancer and anxiolytic activities.
Formula:
C31H24ClF6N3O2
Purity:
99.88% - 99.88%
Color and Shape:
Solid
Molecular weight:
619.99
Ref: TM-TQ0087
| 2mg | 146.00 € | ||
| 5mg | 243.00 € | ||
| 25mg | 711.00 € | ||
| 50mg | 952.00 € | ||
| 100mg | 1,494.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
E6130
CAS:1427058-33-0
E6130 may be effective in the treatment of inflammatory bowel disease and is a highly …
Formula:
C28H37ClF3N3O3
Color and Shape:
Solid
Molecular weight:
556.06
Ref: TM-T11140
| 5mg | 2,919.00 € | ||
| 25mg | 4,096.00 € | ||
| 50mg | 6,139.00 € | ||
| 100mg | 9,200.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
ASP6432
CAS:1282549-08-9
ASP6432 is an antagonist of type 1 lysophosphatidic acid receptor (LPA1). For human LPA1 and …
Formula:
C26H32KN4O6S2
Color and Shape:
Solid
Molecular weight:
599.78
Ref: TM-T14335
| 1ml | 390.00 € | ||
| 5mg | 278.00 € | ||
| 25mg | 916.00 € | ||
| 50mg | 1,273.00 € | ||
| 100mg | 1,741.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
5-HT2A&5-HT2C agonist-1
CAS:1640-02-4
5-HT2A&5-HT2C agonist-1 (Example 2) is a dual-acting agent targeting the 5-HT2A and 5-HT2C receptors with …
Formula:
C14H20N2O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
232.32
Ref: TM-T79806
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 10 Dec 2024
SKF 81297
CAS:71636-61-8
SKF 81297 is a selective and potent agonist for the dopamine D1 receptor [1].
Formula:
C16H16ClNO2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
289.76
Ref: TM-T81152
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 10 Dec 2024
(S)-FTY720-phosphonate
CAS:1142015-10-8
FTY720 (S)-Phosphate, an S1P receptor 1 (S1PR1) agonist, is utilized in studying acute inflammatory diseases, …
Formula:
C20H36NO4P
Purity:
98%
Color and Shape:
Solid
Molecular weight:
385.48
Ref: TM-T78091
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 10 Dec 2024
CaSR antagonist-1
CAS:1219811-83-2
CaSR Antagonist-1 is a potent inhibitor of the calcium-sensing receptor (CaSR) with an inhibitory concentration …
Formula:
C29H24FN3O2S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
497.58
Ref: TM-T79023
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 10 Dec 2024
MK-7246
CAS:1218918-62-7
MK-7246 is a potent and specific CRTH2 antagonist (Ki: 2.5 nM).
Formula:
C21H21FN2O4S
Color and Shape:
Solid
Molecular weight:
416.47
Ref: TM-TQ0051
| 1mg | 210.00 € | ||
| 5mg | 931.00 € | ||
| 10mg | 1,648.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
IIIM-8
CAS:1128053-62-2
IIIM-8 is a melanogenesis inhibitor that suppresses pigment production in both in vitro and in …
Formula:
C14H17NO4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
263.29
Ref: TM-T79378
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Flesinoxan
CAS:98206-10-1
Flesinoxan is a hypotensive agent and is an effective, high affinity, and selective 5-hydroxytryptamine1A receptor …
Formula:
C22H26FN3O4
Color and Shape:
Solid
Molecular weight:
415.46
Ref: TM-T16711
| 1ml | 431.00 € | ||
| 5mg | 349.00 € | ||
| 25mg | 1,113.00 € | ||
| 50mg | 1,470.00 € | ||
| 100mg | 2,209.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
YM348
CAS:372163-84-3
YM348 is an effective and orally active 5-HT2C receptor agonist. YM348 also shows a high …
Formula:
C14H17N3O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
243.3
Ref: TM-T17275
| 25mg | 1,299.00 € | ||
| 50mg | 1,723.00 € | ||
| 100mg | 2,670.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Uridine 5'-diphosphate
CAS:58-98-0
Uridine 5'-diphosphate acts as a P2Y6 receptor agonist, exhibiting an EC50 value of 0.013 μM …
Formula:
C9H14N2O12P2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
404.16
Ref: TM-T78583
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 10 Dec 2024
AEF0117
CAS:1610878-71-1
AEF0117 is a signaling inhibitor of CB1-SSi that inhibits cannabinoid self-administration and can be used …
Formula:
C29H40O3
Purity:
99.58%
Color and Shape:
Solid
Molecular weight:
436.63
Ref: TM-T79909
| 1mg | 35.00 € | ||
| 5mg | 69.00 € | ||
| 10mg | 95.00 € | ||
| 25mg | 185.00 € | ||
| 50mg | 306.00 € | ||
| 100mg | 502.00 € | ||
| 500mg | 1,072.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
GP 1a
CAS:511532-96-0
GP 1a: potent CB2 receptor agonist (EC50=7.1), 30x CB2 over CB1 preference, boosts P-ERK1/2, aids …
Formula:
C23H22Cl2N4O
Purity:
99.44%
Color and Shape:
Solid
Molecular weight:
441.35
Ref: TM-T41231
| 1mg | 55.00 € | ||
| 5mg | 109.00 € | ||
| 10mg | 171.00 € | ||
| 25mg | 334.00 € | ||
| 50mg | 495.00 € | ||
| 100mg | 705.00 € | ||
| 500mg | 1,427.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
S1P1 agonist 6
CAS:2433782-42-2
Compound I (S1P1 agonist 6) is an S1P1 agonist that mitigates autoimmune activity by inhibiting …
Formula:
C25H26F3NO3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
445.47
Ref: TM-T79816
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 10 Dec 2024
