G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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PSNCBAM-1
CAS:877202-74-9
PSNCBAM-1 (PSNCBAM 1) is a CB1 receptor negative allosteric modulator (EC50 = 0.1 μM) with …
Formula:
C22H21ClN4O
Purity:
98.18%
Color and Shape:
Solid
Molecular weight:
392.88
Ref: TM-T28468
| 1mg | 52.00 € | ||
| 5mg | 110.00 € | ||
| 10mg | 168.00 € | ||
| 25mg | 279.00 € | ||
| 50mg | 435.00 € | ||
| 100mg | 612.00 € |
Estimated delivery in United States, on Monday 10 Feb 2025
WAY-607695
CAS:380469-52-3
WAY-607695 is a potential 5-HT1A receptor agonist.
Formula:
C13H12FNO2
Purity:
99.82%
Color and Shape:
Liquid
Molecular weight:
233.24
Ref: TM-T80805
| 5mg | 46.00 € | ||
| 10mg | 69.00 € | ||
| 25mg | 102.00 € | ||
| 50mg | 148.00 € | ||
| 100mg | 214.00 € |
Estimated delivery in United States, on Monday 10 Feb 2025
GW 833972A
CAS:1092502-33-4
GW 833972A: selective CB2 agonist; reduces neural depolarization and citric acid cough in animals.
Formula:
C18H14Cl2F3N5O
Purity:
98%
Color and Shape:
Soild
Molecular weight:
444.24
Ref: TM-T64394
| 1mg | 327.00 € | ||
| 5mg | 774.00 € | ||
| 10mg | 1,056.00 € | ||
| 25mg | 1,476.00 € | ||
| 50mg | 1,838.00 € | ||
| 100mg | 2,321.00 € | ||
| 500mg | 4,568.00 € | ||
| 1mL*10mM (DMSO) | 933.00 € |
Estimated delivery in United States, on Monday 10 Feb 2025
Sigma-1 receptor antagonist 2
CAS:1639220-15-7
Sigma-1 receptor antagonist 2 is a more potent and selective antagonist of sigma 1 receptor …
Formula:
C20H26ClN3O2
Purity:
99.52%
Color and Shape:
Solid
Molecular weight:
375.89
Ref: TM-T12911
| 1mg | 61.00 € | ||
| 5mg | 140.00 € | ||
| 10mg | 226.00 € | ||
| 25mg | 378.00 € | ||
| 50mg | 538.00 € | ||
| 100mg | 726.00 € | ||
| 200mg | 974.00 € | ||
| 1mL*10mM (DMSO) | 154.00 € |
Estimated delivery in United States, on Monday 10 Feb 2025
PSB-603
CAS:1092351-10-4
PSB-603 is a selective antagonist of Adenosine A2B receptor(Ki = 0.553 nM) with anti-inflammatory effects.
Formula:
C24H25ClN6O4S
Purity:
97.13%
Color and Shape:
Solid
Molecular weight:
529.01
Ref: TM-T23203
| 1mg | 37.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 157.00 € | ||
| 25mg | 338.00 € | ||
| 50mg | 550.00 € | ||
| 100mg | 918.00 € | ||
| 200mg | 1,246.00 € | ||
| 1mL*10mM (DMSO) | 111.00 € |
Estimated delivery in United States, on Monday 10 Feb 2025
GS-6201
CAS:752222-83-6
GS-6201 (CVT-6883) is a selective antagonist of adenosine A2B receptor.
Formula:
C21H21F3N6O2
Purity:
98.32% - 99.74%
Color and Shape:
Solid
Molecular weight:
446.43
Ref: TM-T15418
| 1mg | 43.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 151.00 € | ||
| 25mg | 308.00 € | ||
| 50mg | 490.00 € | ||
| 100mg | 712.00 € | ||
| 1mL*10mM (DMSO) | 114.00 € |
Estimated delivery in United States, on Monday 10 Feb 2025
PD 168368
CAS:204066-82-0
PD 168368 is a mixed neuromodulin B receptor (NMB-R) antagonist and potent FPR1/FPR2/FPR3 agonist that …
Formula:
C31H34N6O4
Purity:
98.44%
Color and Shape:
Solid
Molecular weight:
554.64
Ref: TM-T8691
| 1mg | 97.00 € | ||
| 25mg | To inquire |
Estimated delivery in United States, on Monday 10 Feb 2025
SB 258719
CAS:195199-95-2
SB 258719 is a selective antagonist of 5-HT7 receptor with pKi of 7.5.
Formula:
C18H30N2O2S
Purity:
98.59%
Color and Shape:
Solid
Molecular weight:
338.51
Ref: TM-T12855
| 2mg | 35.00 € | ||
| 5mg | 54.00 € | ||
| 10mg | 88.00 € | ||
| 25mg | 159.00 € | ||
| 50mg | 247.00 € | ||
| 100mg | 365.00 € | ||
| 200mg | 514.00 € | ||
| 1mL*10mM (DMSO) | 60.00 € |
Estimated delivery in United States, on Monday 10 Feb 2025
Ubrogepant
CAS:1374248-77-7
Ubrogepant (MK-1602) is an antagonist of calcitonin gene-related peptide receptor that can be used in …
Formula:
C29H26F3N5O3
Purity:
99.79%
Color and Shape:
Solid
Molecular weight:
549.54
Ref: TM-T17194
| 1mg | 150.00 € | ||
| 5mg | 369.00 € | ||
| 10mg | 583.00 € | ||
| 25mg | 914.00 € | ||
| 50mg | 1,198.00 € | ||
| 100mg | 1,643.00 € | ||
| 1mL*10mM (DMSO) | 484.00 € |
Estimated delivery in United States, on Monday 10 Feb 2025
CB 65
CAS:913534-05-1
CB 65 is a high affinity and selective CB2 receptor agonist with Ki values of …
Formula:
C22H28ClN3O3
Purity:
98.39%
Color and Shape:
Solid
Molecular weight:
417.93
Ref: TM-T41230
| 1mg | 63.00 € | ||
| 5mg | 134.00 € | ||
| 10mg | 193.00 € | ||
| 25mg | 328.00 € | ||
| 50mg | 487.00 € | ||
| 100mg | 693.00 € |
Estimated delivery in United States, on Monday 10 Feb 2025
Facinicline hydrochloride
CAS:677305-02-1
Facinicline hydrochloride (RG3487) is both a novel nicotinic alpha-7 receptor (alpha7nAChR) partial agonist (Ki = …
Formula:
C15H19ClN4O
Purity:
99.72%
Color and Shape:
Solid
Molecular weight:
306.79
Ref: TM-T28531
| 1mg | 52.00 € | ||
| 5mg | 113.00 € | ||
| 10mg | 177.00 € | ||
| 25mg | 291.00 € | ||
| 50mg | 404.00 € | ||
| 1mL*10mM (DMSO) | 125.00 € |
Estimated delivery in United States, on Monday 10 Feb 2025
PAOPA
CAS:114200-31-6
dopamine D2 receptor modulator
Formula:
C11H18N4O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
254.29
Ref: TM-T23121
| 25mg | 1,967.00 € | ||
| 50mg | 2,598.00 € | ||
| 100mg | 3,458.00 € |
Estimated delivery in United States, on Monday 10 Feb 2025
S1R agonist 1 hydrochloride
CAS:242487-82-7
S1R Agonist 1 (Compound 6b) hydrochloride is a selective S1R agonist, displaying K i values …
Formula:
C20H26ClNO
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
331.88
Ref: TM-T78086
| 2mg | 52.00 € |
Estimated delivery in United States, on Monday 10 Feb 2025
TASP 0277308
CAS:945725-50-8
TASP 0277308 is an S1P1 inhibitor with immunomodulatory and anticancer activity that inhibits S1P- and …
Formula:
C23H28Cl2N6O3S
Color and Shape:
Solid
Molecular weight:
539.48
Ref: TM-T41145
| 1mg | 256.00 € | ||
| 5mg | 627.00 € |
Estimated delivery in United States, on Monday 10 Feb 2025
CB-25
CAS:869376-63-6
CB-25 is a partial agonist ligand of CB1 cannabinoid receptors, augmenting Forskolin-induced cAMP formation in …
Formula:
C25H41NO3
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
403.6
Ref: TM-T78083
| 2mg | 94.00 € |
Estimated delivery in United States, on Monday 10 Feb 2025
WAY-639889
CAS:432506-24-6
WAY-639889 is a small molecule compound with selective and potent inhibitory effects on neuropeptide Y-5 …
Formula:
C25H27N5O
Purity:
99.73%
Color and Shape:
Liquid
Molecular weight:
413.51
Ref: TM-T77783
| 1mg | 52.00 € | ||
| 5mg | 115.00 € | ||
| 10mg | 173.00 € | ||
| 25mg | 337.00 € | ||
| 50mg | 499.00 € | ||
| 100mg | 711.00 € |
Estimated delivery in United States, on Monday 10 Feb 2025
Lotiglipron
CAS:2401892-75-7
Lotiglipron (PF-07081532) is a GLP-1R agonist that lowers blood glucose and may be used in …
Formula:
C31H31ClN4O5
Purity:
98.3%
Color and Shape:
Liquid
Molecular weight:
575.05
Ref: TM-T77781
| 1mg | 69.00 € | ||
| 5mg | 138.00 € | ||
| 10mg | 203.00 € | ||
| 25mg | 406.00 € | ||
| 50mg | 610.00 € | ||
| 100mg | 915.00 € |
Estimated delivery in United States, on Monday 10 Feb 2025
4-Chloro-L-phenylalanine
CAS:14173-39-8
4-Chloro-L-phenalanine (L-PCPA) is an inhibitor of 5-HT biosynthesis and a non-specific antagonist of tryptophan hydroxylases …
Formula:
C9H10ClNO2
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
199.63
Ref: TM-T78228
| 5g | 51.00 € |
Estimated delivery in United States, on Monday 10 Feb 2025
iso-TRAP-6
CAS:150242-29-8
iso-TRAP-6 (iso-SFLLRN), a hexapeptide made from isoserine instead of serine, is a PAR1 agonist that …
Formula:
C34H56N10O9
Purity:
98.55%
Color and Shape:
Liquid
Molecular weight:
748.87
Ref: TM-T78099
| 5mg | 47.00 € | ||
| 10mg | 64.00 € | ||
| 25mg | 118.00 € |
Estimated delivery in United States, on Monday 10 Feb 2025
Carmoxirole hydrochloride
CAS:115092-85-8
Carmoxirole hydrochloride (EMD 45609 hydrochloride) is a selective dopamine D2 receptor agonist with antihypertensive activity …
Formula:
C24H27ClN2O2
Purity:
97.8% - 98.12%
Color and Shape:
Solid
Molecular weight:
410.94
Ref: TM-T10683
| 1mg | 56.00 € | ||
| 5mg | 113.00 € | ||
| 10mg | 173.00 € | ||
| 25mg | 296.00 € | ||
| 50mg | 436.00 € | ||
| 100mg | 598.00 € | ||
| 200mg | 805.00 € | ||
| 1mL*10mM (DMSO) | 129.00 € |
Estimated delivery in United States, on Monday 10 Feb 2025
