G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
Read more
Cenerimod
CAS:1262414-04-9
Cenerimod (ACT-334441) is an S1P1 agonist used in the study of murine experimental autoimmune encephalomyelitis …
Formula:
C25H31N3O5
Purity:
97.43%
Color and Shape:
Solid
Molecular weight:
453.53
Ref: TM-T14924
| 1ml | 68.00 € | ||
| 2mg | 42.00 € | ||
| 5mg | 61.00 € | ||
| 10mg | 93.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
5-HT3-In-1
CAS:186348-68-5
5-HT3-In-1 (compound example 8) exhabits with 5-HT3 inhibition activity.
Formula:
C16H21ClN4O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
352.82
Ref: TM-T10006
| 25mg | 1,827.00 € | ||
| 50mg | 2,404.00 € | ||
| 100mg | 3,168.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
(±)-Prenalterol
CAS:57526-81-5
(±)-Prenalterol (H 80/62) is an agonist of beta-2- and beta-1-adrenergic receptors and is used to …
Formula:
C12H19NO3
Purity:
99.71%
Color and Shape:
Solid
Molecular weight:
225.28
Ref: TM-T25984
| 1mg | 215.00 € | ||
| 2mg | 323.00 € | ||
| 5mg | 537.00 € | ||
| 10mg | 861.00 € | ||
| 25mg | 1,273.00 € | ||
| 50mg | 1,715.00 € | ||
| 100mg | 2,320.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
CY 208-243
CAS:100999-26-6
CY 208-243 is a selective dopamine D1 receptor agonist with anti-Parkinson disease activity.
Formula:
C19H18N2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
274.36
Ref: TM-T10908
| 25mg | 712.00 € | ||
| 50mg | 929.00 € | ||
| 100mg | 1,454.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
AGN 210676
CAS:910562-15-1
AGN 210676 is a selective agonist of prostaglandin EP2(EC50 : 5 nM).
Formula:
C23H29NO5S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
431.55
Ref: TM-T14146
| 25mg | 1,688.00 € | ||
| 50mg | 2,217.00 € | ||
| 100mg | 2,888.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Celiprolol hydrochloride
CAS:57470-78-7
Celiprolol hydrochloride (Selectrol) is a cardioselective beta-1 adrenergic antagonist that has intrinsic sympathomimetic activity.
Formula:
C20H33N3O4·HCl
Color and Shape:
White Crystalline Solid
Molecular weight:
415.96
Ref: TM-T1244
| 1ml | 138.00 € | ||
| 2mg | 77.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Clazosentan
CAS:180384-56-9
Clazosentan (Ro 61-1790) is a selective ET_A receptor antagonist that inhibits ET-1 vasoconstriction and prevents …
Formula:
C25H23N9O6S
Purity:
95.39% - 99.43%
Color and Shape:
Solid
Molecular weight:
577.57
Ref: TM-T64084
| 1mg | 90.00 € | ||
| 5mg | 184.00 € | ||
| 10mg | 322.00 € | ||
| 25mg | 707.00 € | ||
| 50mg | 1,163.00 € | ||
| 100mg | 1,475.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
CGP-20712
CAS:137888-49-4
CGP-20712 is a selective β 1-adrenoceptor antagonist with an IC50 of 0.7 nM.
Formula:
C23H25F3N4O5
Purity:
100% - 99.40%
Color and Shape:
Solid
Molecular weight:
494.46
Ref: TM-T30846
| 1mg | 327.00 € | ||
| 5mg | 774.00 € | ||
| 10mg | 1,056.00 € | ||
| 25mg | 1,481.00 € | ||
| 50mg | 1,838.00 € | ||
| 100mg | 2,322.00 € | ||
| 500mg | 4,577.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
PSB-603
CAS:1092351-10-4
PSB-603 is a selective antagonist of Adenosine A2B receptor(Ki = 0.553 nM) with anti-inflammatory effects.
Formula:
C24H25ClN6O4S
Purity:
97.13%
Color and Shape:
Solid
Molecular weight:
529.01
Ref: TM-T23203
| 1mg | 49.00 € | ||
| 1ml | 111.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 157.00 € | ||
| 25mg | 338.00 € | ||
| 50mg | 550.00 € | ||
| 100mg | 918.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
EP4 receptor antagonist 1
CAS:2287259-07-6
EP4 antagonist 1: inhibits human/mouse EP4 receptors (IC50: 6.1/16.2 nM), selective over EP1-EP3 (>10 …
Formula:
C23H21F3N4O3
Purity:
99.53%
Color and Shape:
Solid
Molecular weight:
458.43
Ref: TM-T11211
| 1mg | 103.00 € | ||
| 5mg | 239.00 € | ||
| 10mg | 384.00 € | ||
| 25mg | To inquire |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Gepirone
CAS:83928-76-1
Gepirone is a 5-HT1A receptor agonist belonging to the buspirone family. Gepirone HCl possesses greater …
Formula:
C19H29N5O2
Purity:
99.35% - 99.77%
Color and Shape:
Solid
Molecular weight:
359.47
Ref: TM-T19917
| 2mg | 45.00 € | ||
| 5mg | 66.00 € | ||
| 10mg | 89.00 € | ||
| 25mg | 137.00 € | ||
| 50mg | 201.00 € | ||
| 100mg | 276.00 € | ||
| 500mg | 684.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Facinicline hydrochloride
CAS:677305-02-1
Facinicline hydrochloride (RG3487) is both a novel nicotinic alpha-7 receptor (alpha7nAChR) partial agonist (Ki = …
Formula:
C15H19ClN4O
Purity:
99.72%
Color and Shape:
Solid
Molecular weight:
306.79
Ref: TM-T28531
| 1mg | 87.00 € | ||
| 1ml | 205.00 € | ||
| 5mg | 184.00 € | ||
| 10mg | 296.00 € | ||
| 25mg | 489.00 € | ||
| 50mg | 677.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
AZD9898
CAS:2042347-69-1
AZD9898 inhibits leukotriene-C4 synthetase (IC50: 0.28 nM), aids asthma research, and reduces GABA binding, liver …
Formula:
C20H19ClF3N3O4
Purity:
98.27%
Color and Shape:
Solid
Molecular weight:
457.83
Ref: TM-T14387
| 1mg | 200.00 € | ||
| 5mg | 500.00 € | ||
| 10mg | 733.00 € | ||
| 25mg | 1,178.00 € | ||
| 50mg | 1,568.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
TG6-129
CAS:1164464-14-5
TG6-129 is an EP2 receptor antagonist, blocking PGE2 effects, reducing inflammatory markers with 1.6 µM …
Formula:
C20H18FN5O3S3
Purity:
98.39%
Color and Shape:
Solid
Molecular weight:
491.58
Ref: TM-T28958
| 1mg | 119.00 € | ||
| 1ml | 337.00 € | ||
| 5mg | 237.00 € | ||
| 10mg | 419.00 € | ||
| 25mg | 686.00 € | ||
| 50mg | 917.00 € | ||
| 100mg | 1,291.00 € | ||
| 500mg | 2,617.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Didesmethyl cariprazine
CAS:839712-25-3
Didesmethyl cariprazine, Cariprazine's active metabolite, treats schizophrenia/bipolar with D3/D2 affinity; half-life 1-3 weeks.
Formula:
C19H28Cl2N4O
Purity:
99.70%
Color and Shape:
Solid
Molecular weight:
399.36
Ref: TM-T15117
| 1mg | 143.00 € | ||
| 5mg | 346.00 € | ||
| 10mg | 513.00 € | ||
| 25mg | 806.00 € | ||
| 50mg | 1,095.00 € | ||
| 100mg | 1,475.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
SB 216641 hydrochloride
CAS:193611-67-5
SB 216641 hydrochloride (SB-216641A) is a 5-HT1B/D receptor antagonist with anxiolytic properties.
Formula:
C28H31ClN4O4
Purity:
98.40%
Color and Shape:
Solid
Molecular weight:
523.02
Ref: TM-T23315
| 1mg | 74.00 € | ||
| 5mg | 164.00 € | ||
| 10mg | 235.00 € | ||
| 25mg | 395.00 € | ||
| 50mg | 577.00 € | ||
| 100mg | 817.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Sigma-1 receptor antagonist 2
CAS:1639220-15-7
Sigma-1 receptor antagonist 2 is a more potent and selective antagonist of sigma 1 receptor …
Formula:
C20H26ClN3O2
Purity:
99.52%
Color and Shape:
Solid
Molecular weight:
375.89
Ref: TM-T12911
| 1mg | 61.00 € | ||
| 1ml | 154.00 € | ||
| 5mg | 140.00 € | ||
| 10mg | 226.00 € | ||
| 25mg | 378.00 € | ||
| 50mg | 538.00 € | ||
| 100mg | 726.00 € | ||
| 200mg | 974.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
OPC-28326
CAS:167626-17-7
OPC-28326: an α2-adrenergic blocker; dilates blood vessels; inhibits α2A/B/C receptors with Ki 2040/285/55 nM.
Formula:
C26H35N3O2
Purity:
98.56%
Color and Shape:
Solid
Molecular weight:
421.58
Ref: TM-T13804
| 1mg | 306.00 € | ||
| 1ml | 939.00 € | ||
| 5mg | 744.00 € | ||
| 10mg | 1,012.00 € | ||
| 25mg | 1,542.00 € | ||
| 50mg | 2,070.00 € | ||
| 100mg | 2,719.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Sonepiprazole
CAS:170858-33-0
Sonepiprazole (PNU-101387G) is a chemical compound known for its selective antagonistic properties toward D4 dopamine …
Formula:
C21H27N3O3S
Purity:
99.31%
Color and Shape:
Solid
Molecular weight:
401.52
Ref: TM-T23380
| 1ml | 69.00 € | ||
| 2mg | 37.00 € | ||
| 5mg | 56.00 € | ||
| 10mg | 91.00 € | ||
| 25mg | 174.00 € | ||
| 50mg | 296.00 € | ||
| 100mg | 427.00 € | ||
| 200mg | 600.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Carmoxirole hydrochloride
CAS:115092-85-8
Carmoxirole hydrochloride (EMD 45609 hydrochloride) is a selective dopamine D2 receptor agonist with antihypertensive activity …
Formula:
C24H27ClN2O2
Purity:
97.8% - 98.12%
Color and Shape:
Solid
Molecular weight:
410.94
Ref: TM-T10683
| 1mg | 56.00 € | ||
| 1ml | 129.00 € | ||
| 5mg | 113.00 € | ||
| 10mg | 173.00 € | ||
| 25mg | 296.00 € | ||
| 50mg | 436.00 € | ||
| 100mg | 598.00 € | ||
| 200mg | 805.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
