G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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GI 181771
CAS:305366-98-7
GI 181771 is an agonist of the cholecystokinin 1 receptor. GI 181771 can be used …
Formula:
C34H31N5O6
Purity:
95.63%
Color and Shape:
Solid
Molecular weight:
605.64
Ref: TM-T15382
| 1mg | 182.00 € | ||
| 5mg | 416.00 € | ||
| 50mg | 1,290.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
5-HT2A antagonist 1
CAS:204643-75-4
5-HT2A antagonist 1, from US5728835A & JP 1007727, may treat gastrointestinal and circulatory issues.
Formula:
C26H28N4O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
428.53
Ref: TM-T10498
| 25mg | 1,406.00 € | ||
| 50mg | 1,845.00 € | ||
| 100mg | 2,329.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Bivamelagon hydrochloride
CAS:2641595-55-1
MC-4R Agonist 2 hydrochloride (Example 1) serves as an MC4R agonist, with applications in researching …
Formula:
C35H54Cl2N4O4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
665.73
Ref: TM-T79091
| 25mg | 1,827.00 € | ||
| 50mg | 2,412.00 € | ||
| 100mg | 3,178.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
WLB-89462
CAS:2849471-75-4
WLB-89462 (Compound 20c) is a selective σ2 receptor ligand with a K i of 13 …
Formula:
C21H29N5O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
399.49
Ref: TM-T79666
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 10 Dec 2024
LTB4 antagonist 1
CAS:2929239-84-7
LTB4 Antagonist 1, a carboxamide-acid derivative, potently inhibits Leukotriene B4 (LTB4) activity with an IC50 …
Formula:
C26H23NO6
Purity:
98%
Color and Shape:
Solid
Molecular weight:
445.46
Ref: TM-T72625
| 25mg | 1,827.00 € | ||
| 50mg | 2,412.00 € | ||
| 100mg | 3,178.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
LTB4 antagonist 3
CAS:2929239-87-0
Compound 24e, a leukotriene B4 (LTB4) antagonist, exhibits an inhibitory concentration 50 (IC50) of 477 …
Formula:
C29H27NO6
Purity:
98%
Color and Shape:
Solid
Molecular weight:
485.53
Ref: TM-T78678
| 25mg | 1,827.00 € | ||
| 50mg | 2,412.00 € | ||
| 100mg | 3,178.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
BLT2 antagonist-1
CAS:2069220-61-5
BLT2 antagonist-1 (compound 15b) is a selective inhibitor of the BLT2 receptor, impeding the chemotaxis …
Formula:
C26H26FNO4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
435.49
Ref: TM-T79418
| 25mg | 1,549.00 € | ||
| 50mg | 2,038.00 € | ||
| 100mg | 2,617.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
(±)-N-Methylcoclaurine
CAS:1472-62-4
N-Methylcoclaurine (±) acts as a selective antagonist at the α2-adrenoceptor [1].
Formula:
C18H21NO3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
299.36
Ref: TM-T79641
| 25mg | 1,827.00 € | ||
| 50mg | 2,412.00 € | ||
| 100mg | 3,178.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Bivamelagon
CAS:2641595-54-0
MC-4R Agonist 2 (Example 1), a melanocortin 4 receptor (MC4R) agonist, is employed in the …
Formula:
C35H53ClN4O4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
629.27
Ref: TM-T79090
| 25mg | 1,827.00 € | ||
| 50mg | 2,412.00 € | ||
| 100mg | 3,178.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
LTB4 antagonist 2
CAS:2929239-85-8
LTB4 antagonist 2, a carboxamide-acid compound, serves as an antagonist to leukotriene B4 (LTB4), possessing …
Formula:
C26H23NO6
Purity:
98%
Color and Shape:
Solid
Molecular weight:
445.46
Ref: TM-T78677
| 25mg | 1,827.00 € | ||
| 50mg | 2,412.00 € | ||
| 100mg | 3,178.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
AM841
CAS:871978-21-1
AM841, a high-affinity electrophilic ligand, covalently interacts with a cysteine residue in helix six, thus …
Formula:
C26H39NO3S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
445.66
Ref: TM-T78949
| 5mg | 1,573.00 € | ||
| 50mg | 3,183.00 € | ||
| 100mg | 4,331.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Prostaglandin D3
CAS:71902-47-1
Prostaglandin D3 (PGD3) functions as an inhibitor of platelet aggregation and modulates autonomic neurotransmission in …
Formula:
C20H30O5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
350.45
Ref: TM-T78584
| 25µg | 160.00 € | ||
| 50µg | 233.00 € | ||
| 100µg | 402.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
BLT2 probe 1
CAS:2893803-05-7
BLT2 Probe 1, based on CAY10583, is a fluorescent tool for studying BLT2 pharmacology, aiding …
Formula:
C50H45N3O11S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
895.97
Ref: TM-T74212
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Mu opioid receptor antagonist 7
CAS:2378397-30-7
Compound 24, also known as Mu opioid receptor antagonist 7, is a potent, centrally-acting µ-opioid …
Formula:
C22H27ClN2O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
386.91
Ref: TM-T79431
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
BVFP
CAS:357158-20-4
BVFP exhibits affinity for the PGRN 588-593 peptide through binding with a dissociation constant (Kd) …
Formula:
C13H8BrF3N2O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
345.11
Ref: TM-T79105
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 10 Dec 2024
NK3R-IN-1
CAS:2854331-14-7
NK3R-IN-1 (compound 16x), an orally active imidazolepiperazine derivative, acts as a Neurokinin Receptor NK3R inhibitor …
Formula:
C17H16FN5OS
Purity:
98%
Color and Shape:
Solid
Molecular weight:
357.41
Ref: TM-T78757
| 5mg | 1,290.00 € | ||
| 50mg | 2,618.00 € | ||
| 100mg | 3,484.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
μ opioid receptor agonist 3
CAS:2378397-91-0
Compound 20, identified as μ opioid receptor agonist 3, is a potent µOR agonist that …
Formula:
C22H28N2O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
352.47
Ref: TM-T79430
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
A1/A3 AR antagonist 3
CAS:2665804-57-7
A1/A3 AR Antagonist 3 is a dual A1R/A3R antagonist that demonstrates high affinity within the …
Formula:
C22H19N5O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
401.42
Ref: TM-T79027
| 25mg | 1,688.00 € | ||
| 50mg | 2,225.00 € | ||
| 100mg | 2,897.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
JTE-952
CAS:1255303-54-8
JTE-952: oral, selective Type II CSF-1R inhibitor, IC50 = 13 nM for CSF1R, 261 nM …
Formula:
C30H34N2O6
Purity:
98%
Color and Shape:
Solid
Molecular weight:
518.6
Ref: TM-T11729
| 25mg | 1,559.00 € | ||
| 50mg | 2,040.00 € | ||
| 100mg | 2,888.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
(R)-Monlunabant
CAS:2765579-76-6
(R)-Monlunabant ((R)-MRI-1891) serves as a CB1 receptor antagonist utilized in obesity and metabolic disease research …
Formula:
C26H22ClF3N6O3S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
591
Ref: TM-T83533
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 10 Dec 2024
