G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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AZD9898
CAS:2042347-69-1
AZD9898 inhibits leukotriene-C4 synthetase (IC50: 0.28 nM), aids asthma research, and reduces GABA binding, liver …
Formula:
C20H19ClF3N3O4
Purity:
98.27%
Color and Shape:
Solid
Molecular weight:
457.83
Ref: TM-T14387
| 1mg | 205.00 € | ||
| 5mg | 512.00 € | ||
| 10mg | 750.00 € | ||
| 25mg | 1,206.00 € | ||
| 50mg | 1,605.00 € |
Estimated delivery in United States, on Tuesday 6 May 2025
CB 65
CAS:913534-05-1
CB 65 is a high affinity and selective CB2 receptor agonist with Ki values of …
Formula:
C22H28ClN3O3
Purity:
98.39%
Color and Shape:
Solid
Molecular weight:
417.93
Ref: TM-T41230
| 1mg | 64.00 € | ||
| 5mg | 137.00 € | ||
| 10mg | 197.00 € | ||
| 25mg | 335.00 € | ||
| 50mg | 499.00 € | ||
| 100mg | 710.00 € |
Estimated delivery in United States, on Tuesday 6 May 2025
5-HT3-In-1
CAS:186348-68-5
5-HT3-In-1 (compound example 8) exhabits with 5-HT3 inhibition activity.
Formula:
C16H21ClN4O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
352.82
Ref: TM-T10006
| 25mg | 1,872.00 € | ||
| 50mg | 2,452.00 € | ||
| 100mg | 3,230.00 € |
Estimated delivery in United States, on Tuesday 6 May 2025
NK3R-IN-1
CAS:2854331-14-7
NK3R-IN-1 (compound 16x), an orally active imidazolepiperazine derivative, acts as a Neurokinin Receptor NK3R inhibitor …
Formula:
C17H16FN5OS
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
357.41
Ref: TM-T78757
| 5mg | 1,301.00 € | ||
| 50mg | 2,642.00 € | ||
| 100mg | 3,515.00 € |
Estimated delivery in United States, on Tuesday 6 May 2025
Pentixafor
CAS:1341207-62-2
Pentixafor is a peptide that selectively targets the CXCR4 receptor and can be labeled with …
Formula:
C60H80N14O14
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
1221.36
Ref: TM-T79070
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 6 May 2025
DG-041
CAS:861238-35-9
DG-041: EP3 receptor antagonist, high affinity (IC50: 4.6 & 8.1 nM), inhibits PGE2 in platelets, …
Formula:
C23H15Cl4FN2O3S2
Purity:
97.25%
Color and Shape:
Solid
Molecular weight:
592.32
Ref: TM-T15108
| 1mg | 50.00 € | ||
| 2mg | 66.00 € | ||
| 5mg | 97.00 € | ||
| 10mg | 159.00 € | ||
| 25mg | 300.00 € | ||
| 50mg | 540.00 € | ||
| 100mg | 777.00 € | ||
| 500mg | 1,605.00 € | ||
| 1mL*10mM (DMSO) | 110.00 € |
Estimated delivery in United States, on Tuesday 6 May 2025
Fiduxosin
CAS:208993-54-8
Fiduxosin is a selective and potent α1-adrenoceptor antagonist with inhibitory effects on α1a-adrenoceptor, α1b-adrenoceptor and …
Formula:
C30H29N5O4S
Purity:
99.73%
Color and Shape:
Solid
Molecular weight:
555.65
Ref: TM-T11286
| 1mg | 665.00 € | ||
| 5mg | 1,710.00 € |
Estimated delivery in United States, on Tuesday 6 May 2025
Pentiapine
CAS:81382-51-6
Pentiapine (CGS 10746) is a novel inhibitor of dopamine release.
Formula:
C15H17N5S
Purity:
98.93%
Color and Shape:
Solid
Molecular weight:
299.39
Ref: TM-T12405
| 1mg | 487.00 € | ||
| 5mg | 753.00 € | ||
| 10mg | 1,216.00 € | ||
| 25mg | 1,691.00 € | ||
| 50mg | 2,262.00 € | ||
| 100mg | 3,068.00 € | ||
| 1mL*10mM (DMSO) | 938.00 € |
Estimated delivery in United States, on Tuesday 6 May 2025
GLP-1R agonist 3
CAS:2428640-18-8
GLP-1R agonist 3 is a GLP-1R agonist, an imidazole derivative.GLP-1R agonist 3 can be used …
Formula:
C31H28FN5O4
Purity:
97.19%
Color and Shape:
Liquid
Molecular weight:
553.58
Ref: TM-T63909
| 1mg | 126.00 € | ||
| 5mg | 298.00 € | ||
| 10mg | 487.00 € | ||
| 25mg | 938.00 € | ||
| 50mg | 1,578.00 € |
Estimated delivery in United States, on Tuesday 6 May 2025
Dihydrexidine
CAS:123039-93-0
Dihydrexidine is a full efficacy D1-like dopamine receptor (D1/D5) agonist (IC50: 10 nM for D1 …
Formula:
C17H17NO2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
267.32
Ref: TM-T13463L
| 25mg | 1,872.00 € | ||
| 50mg | 2,452.00 € | ||
| 100mg | 3,230.00 € |
Estimated delivery in United States, on Tuesday 6 May 2025
GV150013
CAS:167355-22-8
GV150013 is an antagonist of cholecystokinin-2 (CCK2) receptor.
Formula:
C33H34N4O3
Purity:
100%
Color and Shape:
Solid
Molecular weight:
534.65
Ref: TM-T27503
| 1mg | 187.00 € | ||
| 5mg | 455.00 € | ||
| 10mg | 620.00 € | ||
| 25mg | 940.00 € | ||
| 50mg | 1,264.00 € | ||
| 100mg | 1,663.00 € | ||
| 200mg | 2,252.00 € | ||
| 1mL*10mM (DMSO) | 645.00 € |
Estimated delivery in United States, on Tuesday 6 May 2025
H4R antagonist 2
CAS:1148115-99-4
H4R Antagonist 2, a potent Furo[3,2-d]pyrimidine derivative, serves as a histamine H4 receptor antagonist and …
Formula:
C13H17N5O
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
259.31
Ref: TM-T79786
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 6 May 2025
4-Chloro-L-phenylalanine
CAS:14173-39-8
4-Chloro-L-phenalanine (L-PCPA) is an inhibitor of 5-HT biosynthesis and a non-specific antagonist of tryptophan hydroxylases …
Formula:
C9H10ClNO2
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
199.63
Ref: TM-T78228
| 5g | 50.00 € |
Estimated delivery in United States, on Tuesday 6 May 2025
CXCR2-IN-1
CAS:1873376-49-8
CXCR2-IN-1 has a pIC50 of 9.3 and is a CXCR2 antagonist of the central nervous …
Formula:
C19H20Cl2FN3O4S
Purity:
99.53%
Color and Shape:
Solid
Molecular weight:
476.35
Ref: TM-T10905
| 1mg | 80.00 € | ||
| 5mg | 169.00 € | ||
| 10mg | 235.00 € | ||
| 25mg | 394.00 € | ||
| 50mg | 562.00 € | ||
| 100mg | 758.00 € | ||
| 500mg | To inquire |
Estimated delivery in United States, on Tuesday 6 May 2025
(R)-Monlunabant
CAS:2765579-76-6
(R)-Monlunabant ((R)-MRI-1891) serves as a CB1 receptor antagonist utilized in obesity and metabolic disease research …
Formula:
C26H22ClF3N6O3S
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
591
Ref: TM-T83533
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 6 May 2025
H3 receptor antagonist 1
CAS:935840-13-4
H3 receptor antagonist 1 is used in the study of neurological diseases, histamine H3 receptor …
Formula:
C20H28F2N2O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
350.45
Ref: TM-T10911
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Tuesday 6 May 2025
5-HT2 agonist-1
CAS:2708279-78-9
Compound 24, a 5-HT2 agonist-1, selectively activates 5-HT2A, 5-HT2B, and 5-HT2C receptors with IC50 values …
Formula:
C19H23ClN2O2
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
346.85
Ref: TM-T79804
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 6 May 2025
E6130
CAS:1427058-33-0
E6130 may be effective in the treatment of inflammatory bowel disease and is a highly …
Formula:
C28H37ClF3N3O3
Color and Shape:
Solid
Molecular weight:
556.06
Ref: TM-T11140
| 5mg | 2,972.00 € | ||
| 25mg | 4,169.00 € | ||
| 50mg | 6,249.00 € | ||
| 100mg | 9,367.00 € |
Estimated delivery in United States, on Tuesday 6 May 2025
Mu opioid receptor antagonist 7
CAS:2378397-30-7
Compound 24, also known as Mu opioid receptor antagonist 7, is a potent, centrally-acting µ-opioid …
Formula:
C22H27ClN2O2
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
386.91
Ref: TM-T79431
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Tuesday 6 May 2025
Calindol hydrochloride
CAS:729610-18-8
Calindol (hydrochloride) is a positive allosteric modulator (PAM) of calcimimetic calcium-sensing receptor (CaSR) with an …
Formula:
C21H21ClN2
Purity:
99.47%
Color and Shape:
Solid
Molecular weight:
336.86
Ref: TM-T21758
| 1mg | 52.00 € | ||
| 5mg | 149.00 € | ||
| 10mg | 246.00 € | ||
| 25mg | 518.00 € | ||
| 50mg | 825.00 € | ||
| 100mg | 1,320.00 € | ||
| 200mg | 1,776.00 € |
Estimated delivery in United States, on Tuesday 6 May 2025
