G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Enerisant
CAS:1152747-82-4
Enerisant (TS-091) is a histamine H3 receptor antagonist that promotes pro-cognitive effects and reverses scopolamine-induced …
Formula:
C22H30N4O3
Purity:
99.7%
Color and Shape:
Soild
Molecular weight:
398.50
Ref: TM-T67828
| 1mg | 95.00 € | ||
| 1ml | 187.00 € | ||
| 5mg | 212.00 € | ||
| 10mg | 340.00 € | ||
| 25mg | 717.00 € | ||
| 50mg | 1,146.00 € | ||
| 100mg | 1,836.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Xanthine amine congener
CAS:96865-92-8
Xanthine amine congener is an Adenosine receptor antagonist.
Formula:
C21H28N6O4
Purity:
99.7%
Color and Shape:
Solid
Molecular weight:
428.48
Ref: TM-T23535
| 10mg | 361.00 € | ||
| 50mg | 1,499.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
INT-777
CAS:1199796-29-6
INT-777 (S-EMCA) is a potent TGR5 agonist with an EC50 of 0.82 μM.
Formula:
C27H46O5
Purity:
99.89%
Color and Shape:
Solid
Molecular weight:
450.65
Ref: TM-T11662L
| 1mg | 134.00 € | ||
| 1ml | 361.00 € | ||
| 2mg | 185.00 € | ||
| 5mg | 322.00 € | ||
| 10mg | 463.00 € | ||
| 25mg | 781.00 € | ||
| 50mg | 1,078.00 € | ||
| 100mg | 1,449.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
GPR120 Agonist 3
CAS:1599477-75-4
GPR120 Agonist 3 (GPR120-IN-1) is a selective agonist of Gpr120 ( logEC50: -7.62).
Formula:
C19H23ClF3NO3
Purity:
99.29%
Color and Shape:
Solid
Molecular weight:
405.84
Ref: TM-T15413
| 1mg | 42.00 € | ||
| 1ml | 87.00 € | ||
| 2mg | 55.00 € | ||
| 5mg | 89.00 € | ||
| 10mg | 144.00 € | ||
| 25mg | 273.00 € | ||
| 50mg | 390.00 € | ||
| 100mg | 584.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
KFM19
CAS:133058-72-7
KFM19 is a potent and selective adenosine receptor (A1-receptor) antagonist (IC50 : 50 nM) for …
Formula:
C16H22N4O3
Purity:
99.18%
Color and Shape:
Solid
Molecular weight:
318.37
Ref: TM-T15655
| 1mg | 366.00 € | ||
| 5mg | 855.00 € | ||
| 10mg | 1,164.00 € | ||
| 25mg | 1,694.00 € | ||
| 50mg | 2,211.00 € | ||
| 100mg | 2,879.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Nolomirole HCl
CAS:138531-51-8
Nolomirole HCl (CHF 1035) is a novel selective dopamine agonist with oral activity and inhibitory …
Formula:
C19H28ClNO4
Purity:
100% - 99.12%
Color and Shape:
Solid
Molecular weight:
369.88
Ref: TM-T33711L
| 1mg | 493.00 € | ||
| 5mg | 1,093.00 € | ||
| 25mg | 1,683.00 € | ||
| 50mg | 2,224.00 € | ||
| 100mg | 2,877.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
AR-08
CAS:226081-74-9
AR-08 is a potent α2-adrenergic receptor agonist for the study of ADHD and attention deficit.
Formula:
C12H12N6
Purity:
99.7%
Color and Shape:
Solid
Molecular weight:
240.26
Ref: TM-T10052
| 1mg | 650.00 € | ||
| 5mg | 1,671.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
XL413 hydrochloride
CAS:2062200-97-7
XL413 hydrochloride (BMS-863233 Hydrochloride) is a potent, selective and ATP competitive inhibitor of Cdc7. XL413 …
Formula:
C14H13Cl2N3O2
Purity:
98.81% - 99.82%
Color and Shape:
Solid
Molecular weight:
326.18
Ref: TM-T6735
| 1mg | 52.00 € | ||
| 1ml | 159.00 € | ||
| 5mg | 113.00 € | ||
| 10mg | 158.00 € | ||
| 25mg | 276.00 € | ||
| 50mg | 462.00 € | ||
| 100mg | 694.00 € | ||
| 200mg | 917.00 € | ||
| 500mg | 1,417.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Gastrin/CCK antagonist 1
CAS:162271-52-5
Gastrin/CCK antagonist 1 is a potent gastrin/CCK antagonist for the study of metabolic system-related diseases.
Formula:
C28H32FN5O4
Purity:
98.33%
Color and Shape:
Solid
Molecular weight:
521.58
Ref: TM-T13260
| 1mg | 650.00 € | ||
| 5mg | 1,671.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Vidupiprant
CAS:1169483-24-2
Vidupiprant (AMG 853) is an effective dual antagonist of CRTH2 and prostanoid D receptor with …
Formula:
C28H27Cl2FN2O6S
Purity:
97.16%
Color and Shape:
Solid
Molecular weight:
609.49
Ref: TM-T17232
| 1mg | 66.00 € | ||
| 1ml | 187.00 € | ||
| 5mg | 142.00 € | ||
| 10mg | 214.00 € | ||
| 25mg | 388.00 € | ||
| 50mg | 578.00 € | ||
| 100mg | 822.00 € | ||
| 500mg | 1,660.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Ubrogepant
CAS:1374248-77-7
Ubrogepant (MK-1602) is an antagonist of calcitonin gene-related peptide receptor that can be used in …
Formula:
C29H26F3N5O3
Purity:
99.79%
Color and Shape:
Solid
Molecular weight:
549.54
Ref: TM-T17194
| 1mg | 150.00 € | ||
| 1ml | 484.00 € | ||
| 5mg | 369.00 € | ||
| 10mg | 583.00 € | ||
| 25mg | 914.00 € | ||
| 50mg | 1,198.00 € | ||
| 100mg | 1,643.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Phentolamine Analogue 1
CAS:47142-51-8
Phentolamine Analogue 1 is an analogue of phentolamine. Phentolamine is a nonselective antagonist of α-adrenergic.
Formula:
C17H19N3O
Purity:
98.54%
Color and Shape:
Solid
Molecular weight:
281.35
Ref: TM-T12444
| 1mg | 83.00 € | ||
| 1ml | 166.00 € | ||
| 5mg | 172.00 € | ||
| 10mg | 249.00 € | ||
| 25mg | 410.00 € | ||
| 50mg | 577.00 € | ||
| 100mg | 780.00 € | ||
| 200mg | 1,034.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
RTI-13951-33
CAS:2244884-08-8
RTI-13951-33 is an effective and brain-penetrant GPR88 agonist (EC50: 25 nM, in GPR88 cAMP functional …
Formula:
C28H33N3O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
459.58
Ref: TM-T12778L
| 25mg | 1,688.00 € | ||
| 50mg | 2,225.00 € | ||
| 100mg | 2,897.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Firuglipel
CAS:1371591-51-3
Firuglipel is an orally available and selective agonist of GPR119.
Formula:
C25H26FN3O5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
467.49
Ref: TM-T15283
| 25mg | 1,688.00 € | ||
| 50mg | 2,217.00 € | ||
| 100mg | 2,888.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
LY2922470
CAS:1423018-12-5
LY2922470: Selective GPR40 agonist; EC50=7nM (human), 1nM (mouse), 3nM (rat); lowers glucose, boosts insulin/GLP-1.
Formula:
C28H29NO4S
Purity:
93.34% - 96%
Color and Shape:
Solid
Molecular weight:
475.6
Ref: TM-T15810
| 1mg | 113.00 € | ||
| 1ml | 247.00 € | ||
| 5mg | 232.00 € | ||
| 10mg | 348.00 € | ||
| 25mg | 603.00 € | ||
| 50mg | 860.00 € | ||
| 100mg | 1,177.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
PAC1R antagonist 1
CAS:2305204-24-2
PAC1R antagonist 1 is a PAC1 receptor antagonist that inhibits the activation of peptides by …
Formula:
C17H17ClN6O2
Purity:
98.43%
Color and Shape:
Solid
Molecular weight:
372.81
Ref: TM-T78105
| 1mg | 143.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
CB1 antagonist 1
CAS:890037-68-0
CB1 antagonist 1 is a CB1 receptor antagonist, used in the research of obesity and …
Formula:
C26H22Cl2N4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
461.39
Ref: TM-T10510
| 25mg | 1,967.00 € | ||
| 50mg | 2,598.00 € | ||
| 100mg | 3,458.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Osemozotan HCl
CAS:137275-80-0
Osemozotan is a 5-HT1A receptor agonist potentially for the treatment of generalized anxiety disorder.
Formula:
C19H22ClNO5
Purity:
98.87% - 99.63%
Color and Shape:
Solid
Molecular weight:
379.84
Ref: TM-T28270
| 1mg | 350.00 € | ||
| 5mg | 837.00 € | ||
| 10mg | 1,144.00 € | ||
| 25mg | 1,688.00 € | ||
| 50mg | 2,287.00 € | ||
| 100mg | 3,061.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
(+)-Fluprostenol
CAS:54276-17-4
(+)-Fluprostenol (AL-5848), an analogue of prostaglandin F2 alpha, is a prostaglandin F2α receptor PTGFR agonist …
Formula:
C23H29F3O6
Purity:
99.56%
Color and Shape:
Solid
Molecular weight:
458.47
Ref: TM-T21224
| 1mg | 83.00 € | ||
| 1ml | 211.00 € | ||
| 5mg | 177.00 € | ||
| 10mg | 291.00 € | ||
| 25mg | 537.00 € | ||
| 50mg | 774.00 € | ||
| 100mg | 1,068.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
mPGES1-IN-3
CAS:1469976-70-2
mPGES1-IN-3 is a potent and selective inhibitor of microsomal prostaglandin E2 synthase-1 (mPGES-1) .
Formula:
C24H16ClF5N4O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
538.85
Ref: TM-T12100
| 25mg | 1,827.00 € | ||
| 50mg | 2,413.00 € | ||
| 100mg | 3,180.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
