G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
Read more
Vatinoxan hydrochloride
CAS:130466-38-5
Vatinoxan hydrochloride is an antagonist of the peripheral α2 adrenergic receptors.
Formula:
C20H27ClN4O4S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
454.97
Ref: TM-T13285
| 25mg | 1,967.00 € | ||
| 50mg | 2,598.00 € | ||
| 100mg | 3,458.00 € |
Estimated delivery in United States, on Friday 7 Feb 2025
LGD-6972
CAS:1207989-09-0
LGD-6972 is an antagonist of glucagon receptor.
Formula:
C43H46N2O5S
Purity:
98.8% - 99.33%
Color and Shape:
Solid
Molecular weight:
702.9
Ref: TM-T11845
| 1mg | 87.00 € | ||
| 5mg | 183.00 € | ||
| 10mg | 269.00 € | ||
| 25mg | 461.00 € | ||
| 50mg | 676.00 € | ||
| 100mg | 916.00 € | ||
| 1mL*10mM (DMSO) | 276.00 € |
Estimated delivery in United States, on Friday 14 Feb 2025
Vasopressin
CAS:11000-17-2
Vasopressin receptor agonist; antidiuretic
Formula:
C46H65N15O12S2
Purity:
Min. 95%
Color and Shape:
White Powder
Molecular weight:
1,084.23 g/mol
Ref: 3D-FV40959
| 1g | 1,160.00 € | ||
| 50mg | 310.00 € | ||
| 100mg | 436.00 € | ||
| 250mg | 647.00 € | ||
| 500mg | 863.00 € |
Estimated delivery in United States, on Friday 14 Feb 2025
SB-616234-A
CAS:908601-49-0
SB-616234-A is a selective and orally bioavailable antagonist of 5-HT1B receptor, with anxiolytic and antidepressant …
Formula:
C32H36ClN5O3
Purity:
99.68%
Color and Shape:
Solid
Molecular weight:
574.11
Ref: TM-T12847
| 1mg | 103.00 € | ||
| 5mg | 248.00 € | ||
| 10mg | 358.00 € | ||
| 25mg | 542.00 € | ||
| 50mg | 732.00 € | ||
| 100mg | 1,007.00 € | ||
| 200mg | 1,358.00 € | ||
| 1mL*10mM (DMSO) | 313.00 € |
Estimated delivery in United States, on Friday 21 Feb 2025
AMG 837 calcium hydrate
CAS:1259389-38-2
AMG 837 calcium hydrate is a potent GPR40 agonist with an EC50 of 13 nM.
Formula:
C52H44CaF6O8
Purity:
98.07%
Color and Shape:
Solid
Molecular weight:
950.97
Ref: TM-TQ0020
| 2mg | 36.00 € | ||
| 5mg | 51.00 € | ||
| 10mg | 78.00 € | ||
| 25mg | 145.00 € | ||
| 50mg | 280.00 € | ||
| 100mg | 400.00 € | ||
| 200mg | 547.00 € | ||
| 1mL*10mM (DMSO) | 56.00 € |
Estimated delivery in United States, on Friday 21 Feb 2025
SR 142948
CAS:184162-64-9
SR 142948 is a neurotensin (NT) receptor antagonist.
Formula:
C39H51N5O6
Purity:
98%
Color and Shape:
Solid
Molecular weight:
685.85
Ref: TM-T23386
| 10mg | 878.00 € |
Estimated delivery in United States, on Friday 21 Feb 2025
PSB 1115
CAS:152529-79-8
PSB 1115 is an A2B receptor antagonist and can counteract the inhibitory effect of NECA.
Formula:
C14H14N4O5S
Purity:
100% - 99.24%
Color and Shape:
Solid
Molecular weight:
350.35
Ref: TM-T23201
| 1mg | 66.00 € | ||
| 5mg | To inquire |
Estimated delivery in United States, on Friday 21 Feb 2025
Lumateperone
CAS:313368-91-1
Lumateperone (ITI 722) is a 5HT2A receptor antagonist and a dopamine receptor phosphoprotein modulator (DPPM).
Formula:
C24H28FN3O
Purity:
99.77%
Color and Shape:
Solid
Molecular weight:
393.5
Ref: TM-T21069
| 10mg | 39.00 € | ||
| 25mg | 57.00 € | ||
| 50mg | 83.00 € | ||
| 100mg | 115.00 € |
Estimated delivery in United States, on Friday 21 Feb 2025
16,16-Dimethyl prostaglandin E2
CAS:39746-25-3
16,16-Dimethyl prostaglandin E2 regulates hematopoietic stem cells via EP2/EP4 and Wnt, taken orally.
Formula:
C22H36O5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
380.52
Ref: TM-T10046
| 1mg | 204.00 € | ||
| 5mg | 947.00 € | ||
| 10mg | 1,783.00 € |
Estimated delivery in United States, on Friday 7 Mar 2025
GLPG0974
CAS:1391076-61-1
GLPG0974 is an antagonist of FFA2/GPR43 with IC50 of 9 nM.
Formula:
C25H25ClN2O4S
Purity:
99.58%
Color and Shape:
Solid
Molecular weight:
484.99
Ref: TM-T15388
| 1mg | 55.00 € | ||
| 5mg | 118.00 € | ||
| 10mg | 183.00 € | ||
| 25mg | 368.00 € | ||
| 50mg | 547.00 € | ||
| 1mL*10mM (DMSO) | 125.00 € |
Estimated delivery in United States, on Friday 7 Mar 2025
SB-423562
CAS:351490-27-2
SB-423562 is a calcium-sensing receptor (CaSR) antagonist and can be used in studies about osteoporosis.
Formula:
C26H32N2O4
Purity:
98.64%
Color and Shape:
Solid
Molecular weight:
436.54
Ref: TM-T12846
| 1mg | 38.00 € | ||
| 5mg | 82.00 € | ||
| 10mg | 122.00 € | ||
| 25mg | 214.00 € | ||
| 50mg | 325.00 € | ||
| 100mg | 450.00 € | ||
| 200mg | 616.00 € | ||
| 1mL*10mM (DMSO) | 91.00 € |
Estimated delivery in United States, on Friday 7 Mar 2025
SCH 563705
CAS:473728-58-4
SCH 563705 is a CXCR2 and CXCR1 antagonist used in the study of acute respiratory …
Formula:
C23H27N3O5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
425.48
Ref: TM-T16864
| 1mg | 309.00 € | ||
| 5mg | 738.00 € | ||
| 10mg | 1,154.00 € | ||
| 25mg | 1,716.00 € | ||
| 50mg | 2,326.00 € | ||
| 1mL*10mM (DMSO) | 828.00 € |
Estimated delivery in United States, on Friday 7 Mar 2025
Treprostinil diethanolamine
CAS:830354-48-8
Treprostinil diethanolamine (UT-15C) is a potent agonist of EP2, DP1 and IP, with values of …
Formula:
C27H45NO7
Purity:
98.21%
Color and Shape:
Liquid
Molecular weight:
495.65
Ref: TM-T63349
| 1mg | 110.00 € | ||
| 5mg | 440.00 € | ||
| 10mg | 647.00 € | ||
| 25mg | 994.00 € | ||
| 50mg | 1,341.00 € | ||
| 100mg | 1,810.00 € | ||
| 200mg | 2,420.00 € |
Estimated delivery in United States, on Friday 7 Mar 2025
SB 243213 dihydrochloride
CAS:1780372-25-9
SB 243213 dihydrochloride is an orally active, selective and high-affinity antagonist of 5-hydroxytryptamine (5-HT)2C receptor(pKi …
Formula:
C22H21Cl2F3N4O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
501.33
Ref: TM-T12859L
| 1mg | 108.00 € | ||
| 5mg | 313.00 € |
Estimated delivery in United States, on Friday 7 Mar 2025
MK-3207 Hydrochloride
CAS:957116-20-0
MK-3207 Hydrochloride (MK-3207 HCl) is a potent CGRP receptor antagonist with IC50 and Kiof 0.12 …
Formula:
C31H29F2N5O3·HCl
Purity:
98%
Color and Shape:
Solid
Molecular weight:
594.05
Ref: TM-T6590
| 1mg | 152.00 € | ||
| 5mg | 323.00 € | ||
| 10mg | 484.00 € | ||
| 25mg | 823.00 € | ||
| 50mg | 1,234.00 € | ||
| 100mg | 1,856.00 € | ||
| 1ml*10 (DMSO) | To inquire |
Estimated delivery in United States, on Friday 7 Mar 2025
Atumelnant
CAS:2392970-97-5
Atumelnant (CRN04894) is an MC2R antagonist used in the study of congenital adrenocortical hyperplasia (CAH) …
Formula:
C33H42F3N5O3
Purity:
98.41%
Color and Shape:
Liquid
Molecular weight:
613.71
Ref: TM-T86091
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Friday 7 Mar 2025
Aclidinium
CAS:727649-81-2
Aclidinium, a dual-action compound, serves as a long-acting muscarinic antagonist and a β2-adrenoceptor (β2-AR) agonist, …
Formula:
C26H30NO4S2
Color and Shape:
Liquid
Molecular weight:
484.65
Ref: TM-T200043
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Friday 7 Mar 2025
LSN3318839
CAS:2764704-18-7
LSN3318839 is a potent and orally available glucagon-like peptide-1 receptor (GLP-1R) modulator.LSN3318839 enhances GLP-1R G-protein-coupled …
Formula:
C26H23Cl2N3O2
Purity:
99.43%
Color and Shape:
Liquid
Molecular weight:
480.39
Ref: TM-T63166
| 1mg | 199.00 € | ||
| 5mg | 502.00 € | ||
| 10mg | 725.00 € | ||
| 25mg | 1,095.00 € | ||
| 50mg | 1,476.00 € | ||
| 100mg | 2,014.00 € |
Estimated delivery in United States, on Friday 7 Mar 2025
YGZ-331
CAS:1350113-04-0
YGZ-331, a sedative hypnotic, acts by elevating GABA levels as a derivative of the adenosine …
Formula:
C19H23N5O4
Color and Shape:
Liquid
Molecular weight:
385.42
Ref: TM-T200016
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Friday 7 Mar 2025
LY2794193
CAS:2173037-97-1
LY2794193 is a highly effective and selective agonist of the mGlu3 receptor (hmGlu3 Ki=0.927 nM,EC50=0.47 …
Formula:
C16H18N2O6
Color and Shape:
Solid
Molecular weight:
334.32
Ref: TM-T15807
| 5mg | 490.00 € | ||
| 25mg | 1,679.00 € | ||
| 50mg | 2,209.00 € | ||
| 100mg | 3,061.00 € |
Estimated delivery in United States, on Friday 7 Mar 2025
