G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Propiram fumarate HCl
CAS:945013-73-0
Propiram fumarate HClis an orally available Opioid receptors agonist with analgesic activity for the study …
Formula:
C16H25N3O·xClH
Purity:
99.25%
Color and Shape:
Soild
Ref: TM-T28453L
| 1mg | 185.00 € | ||
| 5mg | 409.00 € | ||
| 10mg | 605.00 € | ||
| 25mg | 938.00 € | ||
| 50mg | 1,293.00 € | ||
| 100mg | 1,738.00 € | ||
| 500mg | 3,496.00 € |
Estimated delivery in United States, on Monday 3 Mar 2025
D3R/MOR antagonist 2
Compound 121, a D3R/MOR antagonist with K i values of 361 nM and 85.2 nM …
Formula:
C25H31ClN2O
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
410.98
Ref: TM-T78779
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 3 Mar 2025
LUF6096
CAS:1116652-18-6
LUF6096 (CF-602) is a potent allosteric enhancer of the adenosine A3 receptor, exhibiting the capability …
Formula:
C22H21Cl2N3O
Purity:
100%
Color and Shape:
Solid
Molecular weight:
414.33
Ref: TM-T9180
| 1mg | 35.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 116.00 € | ||
| 25mg | 190.00 € | ||
| 50mg | 269.00 € | ||
| 100mg | 383.00 € | ||
| 1mL*10mM (DMSO) | 88.00 € |
Estimated delivery in United States, on Monday 3 Mar 2025
Evofolin B
CAS:1961305-60-1
Evofolin B is a natural compound isolated from the stem bark of Zanthoxylum ailanthoides.
Formula:
C17H18O6
Purity:
98%
Color and Shape:
Solid
Molecular weight:
318.32
Ref: TM-TN2408
| 5mg | 3,382.00 € | ||
| 1mL*10mM (DMSO) | 4,065.00 € |
Estimated delivery in United States, on Monday 3 Mar 2025
Prostaglandin F2α 1,11-lactone
CAS:62410-84-8
Prostaglandin F2α 1,11-lactone (PGF2α 1,11-lactone) is a lipid-soluble prodrug of Prostaglandin F2α and can be …
Formula:
C20H32O4
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
336.47
Ref: TM-T37326
| 10mg | 1,615.00 € |
Estimated delivery in United States, on Monday 3 Mar 2025
CCK Octapeptide, non-sulfated acetate
CCK Octapeptide, non-sulfated acetate is a synthetic desulfated peptide of cholecystokinin.
Formula:
C51H66N10O15S2
Purity:
98.97%
Color and Shape:
Liquid
Molecular weight:
1123.26
Ref: TM-TP2204L
| 1mg | 129.00 € | ||
| 5mg | 261.00 € | ||
| 10mg | 432.00 € | ||
| 25mg | 710.00 € | ||
| 50mg | 998.00 € | ||
| 100mg | 1,349.00 € | ||
| 500mg | 2,707.00 € |
Estimated delivery in United States, on Monday 3 Mar 2025
Nelivaptan
CAS:439687-69-1
Nelivaptan (SR 149415) is a vasopressin V1b receptor antagonist that can eliminate CHS-induced GE damage.Cost-effective …
Formula:
C30H32ClN3O8S
Purity:
98% - 98.39%
Color and Shape:
Solid
Molecular weight:
630.11
Ref: TM-T28153
| 1mg | 78.00 € | ||
| 5mg | 150.00 € | ||
| 10mg | 210.00 € | ||
| 25mg | 349.00 € | ||
| 50mg | 517.00 € | ||
| 100mg | 745.00 € | ||
| 500mg | 1,549.00 € |
Estimated delivery in United States, on Monday 3 Mar 2025
Galanin-Like Peptide (porcine)
CAS:245114-96-9
Galanin-Like Peptide (porcine) is a 60 amino acid neuropeptide originally isolated from the porcine hypothalamus.
Formula:
C281H443N81O78
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
6204.02
Ref: TM-T80145
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 3 Mar 2025
AD186
AD186, a potent and selective S1R agonist, exhibits dissociation constants (Kis) of 2.7 nM for …
Formula:
C22H28N2
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
320.47
Ref: TM-T78915
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 3 Mar 2025
CAY10678
CAS:1268709-57-4
CAY10678 is an mPGES-1 inhibitor that inhibits PD-1.CAY10678 reduces collagen deposition and T-cell depletion, and …
Formula:
C23H34N4O
Purity:
99.66%
Color and Shape:
Liquid
Molecular weight:
382.54
Ref: TM-T38369
| 1mg | 52.00 € | ||
| 5mg | 120.00 € | ||
| 10mg | 180.00 € | ||
| 25mg | 354.00 € | ||
| 50mg | 533.00 € | ||
| 100mg | 753.00 € | ||
| 500mg | 1,549.00 € |
Estimated delivery in United States, on Monday 3 Mar 2025
REV 5901A
CAS:92532-23-5
REV 5901A (REV 5901 HCl) is a leukotriene receptor antagonist and 5-LOX inhibitor with antimicrobial …
Formula:
C22H26ClNO2
Purity:
99.74%
Color and Shape:
Soild
Molecular weight:
371.90
Ref: TM-T21821L
| 1mg | 185.00 € | ||
| 5mg | 459.00 € | ||
| 10mg | 657.00 € | ||
| 25mg | 1,026.00 € | ||
| 50mg | 1,415.00 € | ||
| 100mg | 1,872.00 € |
Estimated delivery in United States, on Monday 3 Mar 2025
7-Desmethyl-3-hydroxyagomelatine
CAS:166527-00-0
7-Desmethyl-3-hydroxyagomelatine, less active than parent drug Agomelatine, is a melatonergic agonist and 5-HT2C antagonist.
Formula:
C14H15NO3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
245.27
Ref: TM-T10192
| 100mg | To inquire | ||
| 500mg | To inquire |
Estimated delivery in United States, on Monday 3 Mar 2025
SB 216641
CAS:170230-39-4
SB 216641 is a 5-HT (1B/1D) antagonist with anxiolytic activity for the study of anxiety …
Formula:
C28H30N4O4
Purity:
98.01%
Color and Shape:
Liquid
Molecular weight:
486.56
Ref: TM-T85323
| 1mg | 201.00 € | ||
| 5mg | 497.00 € | ||
| 10mg | 701.00 € | ||
| 25mg | 1,094.00 € | ||
| 50mg | 1,508.00 € | ||
| 100mg | 1,931.00 € |
Estimated delivery in United States, on Monday 3 Mar 2025
CI 169369
CAS:85273-96-7
CI 169369 is a selective 5-HT2 receptor antagonist used in the study of anxiety and …
Formula:
C19H21ClN2S
Purity:
100%
Color and Shape:
Soild
Molecular weight:
344.9
Ref: TM-T84289
| 1mg | 201.00 € | ||
| 5mg | 497.00 € | ||
| 10mg | 701.00 € | ||
| 25mg | 1,094.00 € | ||
| 50mg | 1,508.00 € | ||
| 100mg | 1,931.00 € |
Estimated delivery in United States, on Monday 3 Mar 2025
(-)-GSK598809 hydrochloride
CAS:863766-31-8
(-)-GSK598809 hydrochloride, a DRD3 selective antagonist, may correct reward deficits in substance dependence.
Formula:
C22H24ClF4N5OS
Purity:
97.66%
Color and Shape:
Soild
Molecular weight:
517.97
Ref: TM-T67913
| 1mg | 46.00 € | ||
| 5mg | 93.00 € | ||
| 10mg | 140.00 € | ||
| 25mg | 226.00 € | ||
| 50mg | 338.00 € | ||
| 100mg | 490.00 € | ||
| 1mL*10mM (DMSO) | 105.00 € |
Estimated delivery in United States, on Monday 3 Mar 2025
CB2 PET Radioligand 1
CB2 PET Radioligand 1 (compound [18F]9) is a positron emission tomography (PET) radioligand with high …
Formula:
C20H19F3N4O
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
388.39
Ref: TM-T79577
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 3 Mar 2025
Myriceric acid C
CAS:162059-94-1
Myriceric acid C has cytotoxic activity against human lung carcinoma and breast carcinoma.
Formula:
C48H60O10
Purity:
98%
Color and Shape:
Solid
Molecular weight:
796.98
Ref: TM-TN4606
| 5mg | 675.00 € | ||
| 1mL*10mM (DMSO) | 1,026.00 € |
Estimated delivery in United States, on Monday 3 Mar 2025
2'-Hydroxydaidzein
CAS:7678-85-5
2'-Hydroxydaidzein is an isoflavonoid phytonutrient found in plant species, when a natural compound. 2'-Hydroxydaidzein has …
Formula:
C15H10O5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
270.24
Ref: TM-TN2766
| 1mg | To inquire |
Estimated delivery in United States, on Monday 3 Mar 2025
CB2R/FAAH modulator-2
CAS:2876918-68-0
CB2R/FAAH modulator-2 (compound 26) is a dual modulator targeting at CB2R and FAAH.
Formula:
C24H33NO2
Purity:
99.52%
Color and Shape:
Soild
Molecular weight:
367.52
Ref: TM-T67745
| 1mg | 37.00 € | ||
| 5mg | 79.00 € | ||
| 10mg | 119.00 € | ||
| 25mg | 188.00 € | ||
| 50mg | 283.00 € | ||
| 100mg | 430.00 € |
Estimated delivery in United States, on Monday 3 Mar 2025
SKF-83566 hydrochloride
CAS:164265-49-0
SKF-83566 hydrochloride is a D1-like dopamine receptor antagonist, inhibiting dopamine transporters and mitigating GBP-induced CPP.
Formula:
C17H19BrClNO
Color and Shape:
Soild
Molecular weight:
368.69
Ref: TM-T8702L
| 1mg | 53.00 € | ||
| 5mg | 105.00 € | ||
| 10mg | 166.00 € | ||
| 25mg | 360.00 € | ||
| 50mg | 669.00 € |
Estimated delivery in United States, on Monday 3 Mar 2025
