G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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AC-263093
CAS:849459-86-5
AC-263093 is an NPFFR2 agonist with anxiolytic activity that increases c-Fos protein expression in the …
Formula:
C8H8Br2N4
Purity:
99.78%
Color and Shape:
Soild
Molecular weight:
319.98
Ref: TM-T83651
| 5mg | 47.00 € | ||
| 10mg | 69.00 € | ||
| 25mg | 124.00 € | ||
| 50mg | 193.00 € | ||
| 100mg | 305.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Gancaonin I
CAS:126716-36-7
Gancaonin I exhibits anti-BsFtsZ GTPase activities; it also shows significant inhibitory activity against B. subtilis, …
Formula:
C21H22O5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
354.4
Ref: TM-TN4098
| 5mg | 1,879.00 € | ||
| 1mL*10mM (DMSO) | 2,349.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
![[Ala17]-MCH acetate](https://static.cymitquimica.com/products/TM/thumb/TP1997L.jpg)
[Ala17]-MCH acetate
[Ala17]-MCH acetate is a selective ligand for MCHR1 with a Ki of 0.16 nM and …
Formula:
C99H159N29O28S4
Purity:
98.92%
Color and Shape:
Liquid
Molecular weight:
2331.76
Ref: TM-TP1997L
| 1mg | 112.00 € | ||
| 5mg | 269.00 € | ||
| 10mg | 392.00 € | ||
| 25mg | 598.00 € | ||
| 50mg | 813.00 € | ||
| 100mg | 1,080.00 € | ||
| 200mg | 1,446.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
(d(CH2)51,Tyr(Me)2,Dab5,Arg8)-Vasopressin
CAS:176714-12-8
(d(CH2)5[Tyr(Me)2, Dab5]AVP), a vasopressin V1a receptor-specific antagonist, demonstrates a pA2 value of 6.71 [1].
Formula:
C52H76N14O11S2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1137.38
Ref: TM-T80137
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 25 Nov 2024
MCUF-651
CAS:2747162-85-0
MCUF-651 is a guanylyl cyclase A receptor positive allosteric modulators, EC50=0.45 μM.
Formula:
C17H22F2N4OS
Purity:
99.57%
Color and Shape:
Soild
Molecular weight:
368.44
Ref: TM-T67734
| 1mg | 96.00 € | ||
| 5mg | 200.00 € | ||
| 10mg | 308.00 € | ||
| 25mg | 533.00 € | ||
| 50mg | 836.00 € | ||
| 100mg | 1,274.00 € | ||
| 1mL*10mM (DMSO) | 413.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
FGH31
FGH31 (Compound 24), a dopamine D4 agonist, exhibits potent and selective GRK2-dependency with a K …
Formula:
C33H36N4O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
520.66
Ref: TM-T79312
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 25 Nov 2024
YT 146
CAS:90596-75-1
YT 146 is a biochemical.
Formula:
C18H25N5O4
Purity:
98.81% - 99.72%
Color and Shape:
Solid
Molecular weight:
375.42
Ref: TM-T35282
| 1mg | 274.00 € | ||
| 5mg | 673.00 € | ||
| 10mg | 920.00 € | ||
| 25mg | 1,417.00 € | ||
| 50mg | 1,846.00 € | ||
| 100mg | 2,572.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Adrenocorticotropic Hormone (ACTH) (4-10), human
CAS:4037-01-8
Adrenocorticotropic Hormone (ACTH) (4-10) is an agonist of potent melanocortin(MC4R) receptor .
Formula:
C44H59N13O10S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
962.09
Ref: TM-T7627
| 2mg | 52.00 € | ||
| 5mg | 82.00 € | ||
| 10mg | 115.00 € | ||
| 25mg | 226.00 € | ||
| 50mg | 293.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
SphK1&2-IN-1
CAS:1415662-57-5
SphK1&2-IN-1 is a sphingosine kinase inhibitor with anti-inflammatory, antitumor and hemostatic effects.
Formula:
C14H14N2O3S
Purity:
99.27%
Color and Shape:
Liquid
Molecular weight:
290.34
Ref: TM-T9992
| 1mg | 44.00 € | ||
| 5mg | 97.00 € | ||
| 10mg | 134.00 € | ||
| 25mg | 250.00 € | ||
| 50mg | 359.00 € | ||
| 100mg | 477.00 € | ||
| 200mg | 636.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
KSK94 FA
KSK94 FA is a potent histamine H3 receptor antagonist that inhibits H3 receptors and is …
Formula:
C26H28N4O3
Purity:
98.13%
Color and Shape:
Soild
Molecular weight:
444.53
Ref: TM-T79500L
| 1mg | 183.00 € | ||
| 5mg | 452.00 € | ||
| 10mg | 647.00 € | ||
| 25mg | 1,010.00 € | ||
| 50mg | 1,393.00 € | ||
| 100mg | 1,841.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Tirzepatide
CAS:2023788-19-2
Tirzepatide (LY-3298176) is a dual agonist of GIP and GLP-1 receptors with neuroprotective activity and …
Formula:
C225H348N48O68
Purity:
99.52% - 99.99%
Color and Shape:
Solid
Molecular weight:
4813.45
Ref: TM-TP1111
| 1mg | 247.00 € | ||
| 5mg | 648.00 € | ||
| 10mg | 927.00 € | ||
| 25mg | 1,372.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
4-Methylhistamine
CAS:36507-31-0
4-Methylhistamine serves as a potent agonist for the histamine 4 receptor (H4R), holding promise for …
Formula:
C6H11N3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
125.17
Ref: TM-T80645
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 25 Nov 2024
Brexpiprazole S-oxide
CAS:1191900-51-2
Brexpiprazole S-oxide is the main metabolite of Brexpiprazole, a human 5-HT1A and dopamine receptor partial …
Formula:
C25H27N3O3S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
449.57
Ref: TM-T10612
| 100mg | To inquire | ||
| 500mg | To inquire |
Estimated delivery in United States, on Monday 25 Nov 2024
Mapenterol hydrochloride
CAS:54238-51-6
Mapenterol hydrochloride is an agonist of β2-adrenergic receptor.
Formula:
C14H21Cl2F3N2O
Purity:
99.31% - 99.85%
Color and Shape:
Solid
Molecular weight:
361.23
Ref: TM-T40622
| 1mg | 52.00 € | ||
| 5mg | 105.00 € | ||
| 10mg | 155.00 € | ||
| 25mg | 257.00 € | ||
| 50mg | 369.00 € | ||
| 100mg | 536.00 € | ||
| 500mg | 1,068.00 € | ||
| 1mL*10mM (DMSO) | 112.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Tizanidine
CAS:51322-75-9
Tizanidine, an α2-adrenergic receptor agonist, suppresses the release of neurotransmitters from central nervous system (CNS) …
Formula:
C9H8ClN5S
Purity:
99.75%
Color and Shape:
White Solid
Molecular weight:
253.71
Ref: TM-T7065
| 5mg | 35.00 € | ||
| 10mg | 52.00 € | ||
| 25mg | 72.00 € | ||
| 50mg | 95.00 € | ||
| 100mg | 104.00 € | ||
| 500mg | 247.00 € | ||
| 1mL*10mM (DMSO) | 46.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Tirzepatide monosodium salt
Tirzepatide sodium salt (LY3298176 sodium salt) is a GIP and GLP-1 receptor agonist with neuroprotective …
Formula:
C225H347N48O68Na
Purity:
99.69%
Color and Shape:
Soild
Molecular weight:
4835.51
Ref: TM-TP1111L1
| 1mg | 249.00 € | ||
| 5mg | 652.00 € | ||
| 10mg | 1,069.00 € | ||
| 25mg | 1,598.00 € | ||
| 50mg | 2,193.00 € | ||
| 100mg | 2,959.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Cericlamine
CAS:112922-55-1
Cericlamine is a selective 5-hydroxytryptamine (5-HT) reuptake blocker with antidepressant activity.
Formula:
C12H17Cl2NO
Purity:
98.57%
Color and Shape:
Solid
Molecular weight:
262.18
Ref: TM-T68040
| 1mg | 125.00 € | ||
| 5mg | 299.00 € | ||
| 10mg | 446.00 € | ||
| 25mg | 730.00 € | ||
| 50mg | 1,003.00 € | ||
| 100mg | 1,380.00 € | ||
| 500mg | 2,759.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
EP3 antagonist 4
CAS:2408297-80-1
EP3 antagonist 4: hEP inhibitor, Ki = 2 nM, low clearance, high oral AUC, good …
Formula:
C22H20Cl3FN4O3S2
Purity:
98%
Color and Shape:
Soild
Molecular weight:
577.91
Ref: TM-T77630
| 1mg | 184.00 € | ||
| 5mg | 405.00 € | ||
| 10mg | 612.00 € | ||
| 25mg | 1,044.00 € | ||
| 50mg | 1,580.00 € | ||
| 100mg | 2,388.00 € | ||
| 500mg | 5,254.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Somatostatin acetate
Somatostatin acetate is an endogenously secreted inhibitor of cell proliferation with potential antitumor activity for …
Ref: TM-TP1302L
| 1mg | 59.00 € | ||
| 5mg | 121.00 € | ||
| 10mg | 169.00 € | ||
| 25mg | 282.00 € | ||
| 50mg | 419.00 € | ||
| 100mg | 619.00 € | ||
| 500mg | 1,312.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
FFN246
CAS:2210244-83-8
FFN246, a fluorescent probe, concurrently targets the serotonin transporter (SERT) and vesicular monoamine transporter 2 …
Formula:
C15H13FN2O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
256.27
Ref: TM-T78684
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 25 Nov 2024
