G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Isobutyryl-L-carnitine
CAS:25518-49-4
Isobutyryl-L-carnitine is a member of the class of compounds known as acylcarnitines. Isobutyryl-L-carnitine is a …
Formula:
C11H21NO4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
231.29
Ref: TM-T19381
| 100mg | To inquire | ||
| 500mg | To inquire |
Estimated delivery in United States, on Monday 31 Mar 2025
GLP-1 (9-36) amide
CAS:161748-29-4
GLP-1 (9-36) amide is an antagonist at the human GLP-1 receptor.
Formula:
C140H214N36O43
Purity:
97%
Color and Shape:
Solid
Molecular weight:
3089.41
Ref: TM-TP2252
| 1mg | 88.00 € | ||
| 5mg | 243.00 € | ||
| 10mg | 359.00 € | ||
| 25mg | 595.00 € | ||
| 50mg | 838.00 € | ||
| 100mg | 1,130.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
Upidosin
CAS:152735-23-4
Upidosin (SB-216469), a uroselective α1 blocker: Ki α1a=0.34 nM, α1b=3.9 nM, α1d=1.5 nM, α2=33.3 nM.
Formula:
C31H33N3O4
Purity:
99.26%
Color and Shape:
Solid
Molecular weight:
511.61
Ref: TM-T9762
| 5mg | 44.00 € | ||
| 10mg | 62.00 € | ||
| 25mg | 90.00 € | ||
| 50mg | 129.00 € | ||
| 100mg | 187.00 € | ||
| 200mg | 281.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
NF-56-EJ40 hydrochloride
CAS:2728500-80-7
NF-56-EJ40 HCl is a selective human SUCNR1 antagonist, IC50 = 25 nM, Ki = 33 …
Formula:
C27H31Cl2N3O3
Purity:
97.02%
Color and Shape:
Soild
Molecular weight:
516.46
Ref: TM-T12216L
| 5mg | 55.00 € | ||
| 10mg | 82.00 € | ||
| 25mg | 126.00 € | ||
| 50mg | 182.00 € | ||
| 100mg | 273.00 € | ||
| 200mg | 409.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
Cortistatin 14, human, rat acetate
Cortistatin 14, human, rat acetate is a neuropeptide having structural similarity to somatostatin-14 and shows …
Formula:
C80H112N18O19S2
Purity:
97.86%
Color and Shape:
Solid
Molecular weight:
1693.98
Ref: TM-TP1188L
| 1mg | 109.00 € | ||
| 5mg | 238.00 € | ||
| 10mg | 353.00 € | ||
| 25mg | 563.00 € | ||
| 50mg | 758.00 € | ||
| 100mg | 1,017.00 € | ||
| 200mg | 1,359.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
Ceruletide Ammonium acetate
Ceruletide Ammonium acetate (FI-6934 Ammonium acetate) is a cholecystokinin (CCK) receptor agonist.
Formula:
C60H77N13O23S2
Purity:
99.73%
Color and Shape:
Solid
Molecular weight:
1412.46
Ref: TM-T14932L
| 1mg | 239.00 € | ||
| 5mg | 487.00 € | ||
| 10mg | 705.00 € | ||
| 25mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 31 Mar 2025
Spantide acetate
Spantide acetate is a selective antagonist of NK1 receptor with Kis of 230 nM and …
Formula:
C77H112N20O15
Purity:
98.92%
Color and Shape:
Liquid
Molecular weight:
1557.84
Ref: TM-T20413L
| 1mg | 129.00 € | ||
| 5mg | 329.00 € | ||
| 10mg | 525.00 € | ||
| 25mg | 848.00 € | ||
| 50mg | 1,159.00 € | ||
| 100mg | 1,568.00 € | ||
| 500mg | 3,117.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
RF9 acetate
RF9 acetate is an effective and selective antagonist of Neuropeptide FF receptor with Ki values …
Formula:
C28H42N6O5
Purity:
99.35%
Color and Shape:
Liquid
Molecular weight:
542.67
Ref: TM-T16738L
| 1mg | 65.00 € | ||
| 5mg | 125.00 € | ||
| 10mg | 182.00 € | ||
| 25mg | 325.00 € | ||
| 50mg | 467.00 € | ||
| 100mg | 645.00 € | ||
| 200mg | 868.00 € | ||
| 1mL*10mM (DMSO) | 167.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
Homoeriodictyol
CAS:446-71-9
Homoeriodictyol, a naturally occurring, bitter-masking flavanone, as a promising agent to increase appetite and food …
Formula:
C16H14O6
Purity:
98.16% - 99.96%
Color and Shape:
Solid
Molecular weight:
302.28
Ref: TM-TN1740
| 1mg | 127.00 € | ||
| 5mg | 264.00 € | ||
| 10mg | 432.00 € | ||
| 25mg | 697.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
YNT-185
CAS:1804978-81-1
YNT-185 is a nonpeptide, selective agonist of the orexin type-2 receptor (OX2R), demonstrating EC50 values …
Formula:
C33H37N5O5S
Purity:
98.6%
Color and Shape:
Liquid
Molecular weight:
615.74
Ref: TM-T39229
| 1mg | 66.00 € | ||
| 5mg | 144.00 € | ||
| 10mg | 227.00 € | ||
| 25mg | 454.00 € | ||
| 50mg | 733.00 € | ||
| 100mg | 998.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
Thioperamide maleate
CAS:148440-81-7
Thioperamide maleate (MR-12842 maleate) is an effective and selective antagonist of H3 receptor (Ki = …
Formula:
C19H28N4O4S
Purity:
99.88%
Color and Shape:
Solid
Molecular weight:
408.52
Ref: TM-T41247
| 1mg | 42.00 € | ||
| 5mg | 88.00 € | ||
| 10mg | 127.00 € | ||
| 25mg | To inquire | ||
| 1mL*10mM (DMSO) | 99.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
Dermorphin
CAS:77614-16-5
Dermorphin is agonist of μ-opioid receptor (MOR) agonist.
Formula:
C40H50N8O10
Purity:
98.82%
Color and Shape:
Solid
Molecular weight:
802.87
Ref: TM-T7404
| 1mg | 44.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
LY83583
CAS:91300-60-6
LY83583 is a soluble guanylate cyclase competitive inhibitor with IC50 of 2 µM.
Formula:
C15H10N2O2
Purity:
98.2% - 98.71%
Color and Shape:
Solid
Molecular weight:
250.25
Ref: TM-T21576
| 5mg | 60.00 € | ||
| 10mg | 87.00 € | ||
| 25mg | 170.00 € | ||
| 50mg | 274.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
UFP-101 acetate
UFP-101 acetate is a selective and competitive antagonist of the NOP receptor (pKi = 10.24) …
Formula:
C84H142N32O23
Purity:
95.92%
Color and Shape:
Solid
Molecular weight:
1968.23
Ref: TM-TP2105L
| 1mg | 301.00 € | ||
| 2mg | 545.00 € | ||
| 5mg | 852.00 € | ||
| 10mg | 1,169.00 € | ||
| 25mg | 1,730.00 € | ||
| 50mg | 2,337.00 € | ||
| 100mg | 3,125.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
SphK1&2-IN-1
CAS:1415662-57-5
SphK1&2-IN-1 is a sphingosine kinase inhibitor with anti-inflammatory, antitumor and hemostatic effects.
Formula:
C14H14N2O3S
Purity:
99.27%
Color and Shape:
Liquid
Molecular weight:
290.34
Ref: TM-T9992
| 1mg | 46.00 € | ||
| 5mg | 89.00 € | ||
| 10mg | 138.00 € | ||
| 25mg | 259.00 € | ||
| 50mg | 373.00 € | ||
| 100mg | 495.00 € | ||
| 200mg | 660.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
Urocortin (rat) acetate
Urocortin (rat) acetate: CRF receptor agonist; Ki=13nM (hCRF1), 1.5nM (rCRF2α), 0.97nM (mCRF2β); neuropeptide.
Purity:
97.76%
Color and Shape:
Soild
Ref: TM-TP1020L
| 1mg | 157.00 € | ||
| 5mg | 375.00 € | ||
| 10mg | 535.00 € | ||
| 25mg | 787.00 € | ||
| 50mg | 1,074.00 € | ||
| 100mg | 1,454.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
Myriceric acid C
CAS:162059-94-1
Myriceric acid C has cytotoxic activity against human lung carcinoma and breast carcinoma.
Formula:
C48H60O10
Purity:
98%
Color and Shape:
Solid
Molecular weight:
796.98
Ref: TM-TN4606
| 5mg | 675.00 € | ||
| 1mL*10mM (DMSO) | 1,026.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
CYM 50769
CAS:1421365-63-0
CYM 50769 is a neuropeptide W/B receptor 1 (NPBWR1, GPR7) antagonist(IC50 = 0.12 μM).
Formula:
C24H17ClN2O3
Purity:
98% - 98.76%
Color and Shape:
Solid
Molecular weight:
416.86
Ref: TM-T22702
| 1mg | 52.00 € | ||
| 5mg | 97.00 € | ||
| 10mg | 170.00 € | ||
| 25mg | 378.00 € | ||
| 50mg | 560.00 € | ||
| 100mg | 800.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
Detomidine carboxylic acid
CAS:115664-39-6
Detomidine carboxylic acid, a urine metabolite of detomidine, is a synthetic α2-agonist, animal analgesic, with …
Formula:
C12H12N2O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
216.24
Ref: TM-T11010
| 25mg | 2,585.00 € | ||
| 50mg | 3,402.00 € | ||
| 100mg | 4,655.00 € | ||
| 500mg | To inquire |
Estimated delivery in United States, on Monday 31 Mar 2025
PAR-4 Agonist Peptide, amide
CAS:352017-71-1
PAR-4 Agonist Peptide, amide (AY-NH2) is an agonist of proteinase-activated receptor-4 (PAR-4).
Formula:
C34H48N8O7
Purity:
98%
Color and Shape:
Solid
Molecular weight:
680.79
Ref: TM-T7623
| 1mg | 90.00 € | ||
| 5mg | 144.00 € | ||
| 10mg | 235.00 € | ||
| 25mg | 398.00 € | ||
| 50mg | 567.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
