G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Mebhydrolin napadisylate
CAS:6153-33-9
Mebhydrolin napadisylate (Incidal) is an antihistamine used to relieve allergic symptoms caused by histamine release, …
Formula:
C19H20N2C10H8O6S2
Purity:
99.35% - 99.77%
Color and Shape:
White Or Almost White Crystalline
Molecular weight:
420.52
Ref: TM-T0113
| 1g | 62.00 € | ||
| 5g | 131.00 € | ||
| 10g | 182.00 € | ||
| 500mg | 45.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Levodropropizine
CAS:99291-25-5
Levodropropizine ((S)-(-)-Dropropizine) is a histamine receptor inhibitor. It is used as an effective and very …
Formula:
C13H20N2O2
Purity:
100% - 99.93%
Color and Shape:
White Or Off White Crystalline Powder
Molecular weight:
236.31
Ref: TM-T0217
| 1g | 49.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Ifenprodil
CAS:23210-56-2
Ifenprodil (RC61-91) inhibits NMDA receptor subunits GluN1 & GluN2B, GIRK channels, and affects alpha1, serotonin, …
Formula:
C21H27NO2
Purity:
99.78%
Color and Shape:
White Crystalline Powder
Molecular weight:
325.44
Ref: TM-T1186L
| 1mg | 106.00 € | ||
| 5mg | 208.00 € | ||
| 10mg | 312.00 € | ||
| 25mg | 502.00 € | ||
| 50mg | 676.00 € | ||
| 100mg | 897.00 € | ||
| 200mg | 1,235.00 € | ||
| 1mL*10mM (DMSO) | 217.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Midodrine hydrochloride
CAS:3092-17-9
Midodrine, metabolized to desglymidodrine, activates alpha-1 receptors, raising blood pressure without CNS effects. It's a …
Formula:
C12H19ClN2O4
Purity:
99.06% - 99.36%
Color and Shape:
Crystalline Solid
Molecular weight:
290.74
Ref: TM-T1577
| 5mg | 51.00 € | ||
| 10mg | 74.00 € | ||
| 25mg | 128.00 € | ||
| 50mg | 185.00 € | ||
| 100mg | 274.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Azasetron hydrochloride
CAS:123040-16-4
Azasetron hydrochloride (Y-25130 HCl) is a 5-HT3 receptor antagonist which is used as an anti-emetic.
Formula:
C17H20ClN3O3·HCl
Purity:
99.85%
Color and Shape:
Solid
Molecular weight:
386.27
Ref: TM-T1528
| 5mg | 40.00 € | ||
| 10mg | 57.00 € | ||
| 25mg | 93.00 € | ||
| 50mg | 168.00 € | ||
| 100mg | 275.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
(R)-Elagolix
CAS:834153-87-6
(R)-Elagolix (NBI-56418) is an orally active, highly selective, short-term potent antagonist of the non-peptide gonadotropin-releasing …
Formula:
C32H30F5N3O5
Purity:
97.63%
Color and Shape:
Solid
Molecular weight:
631.59
Ref: TM-T11174
| 1mg | 38.00 € | ||
| 2mg | 49.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 109.00 € | ||
| 25mg | 184.00 € | ||
| 50mg | 323.00 € | ||
| 100mg | 477.00 € | ||
| 200mg | 680.00 € | ||
| 1mL*10mM (DMSO) | 95.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Diphenylpyraline hydrochloride
CAS:132-18-3
Diphenylpyraline hydrochloride treats Parkinsonism. It's an antihistamine with anticholinergic properties and inhibits dopamine reuptake.
Formula:
C19H23NO·HCl
Purity:
99.22%
Color and Shape:
Solid
Molecular weight:
317.85
Ref: TM-T0059
| 500mg | 35.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Tolazoline hydrochloride
CAS:59-97-2
Tolazoline hydrochloride (NSC35110 (hydrochloride)) is a non-selective competitive α-adrenergic receptor antagonist used in treatment of …
Formula:
C10H13ClN2
Purity:
100%
Color and Shape:
Pale Yellow Crystalline Solid
Molecular weight:
196.68
Ref: TM-T1680
| 1g | 47.00 € | ||
| 5g | 89.00 € | ||
| 10g | 128.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
GSK256073
CAS:862892-90-8
GSK256073 is an orally active GPR109A agonist.
Formula:
C10H13ClN4O2
Purity:
98.03%
Color and Shape:
Solid
Molecular weight:
256.69
Ref: TM-T15432
| 1mg | 72.00 € | ||
| 2mg | 95.00 € | ||
| 5mg | 157.00 € | ||
| 10mg | 245.00 € | ||
| 25mg | 430.00 € | ||
| 50mg | 633.00 € | ||
| 100mg | 900.00 € | ||
| 1mL*10mM (DMSO) | 168.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Olanzapine
CAS:132539-06-1
Olanzapine (LY170053) is an atypical antipsychotic that is used currently in the treatment of schizophrenia …
Formula:
C17H20N4S
Purity:
100% - ≥95%
Color and Shape:
Yellowish Crystalline Powder
Molecular weight:
312.43
Ref: TM-T1567
| 25mg | 40.00 € | ||
| 50mg | 51.00 € | ||
| 100mg | 64.00 € | ||
| 200mg | 87.00 € | ||
| 500mg | 133.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Ritodrine hydrochloride
CAS:23239-51-2
Ritodrine hydrochloride (NSC 291565), a phenethylamine derivative, reduces uterine contractions by increasing cAMP and decreasing …
Formula:
C17H21NO3·HCl
Purity:
99% - 99.89%
Color and Shape:
Solid
Molecular weight:
323.82
Ref: TM-T1433
| 1g | 52.00 € | ||
| 200mg | 36.00 € | ||
| 500mg | 42.00 € | ||
| 1mL*10mM (DMSO) | 36.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
A3AR agonist 2
Compound 19, a selective A3 Adenosine Receptor (A3AR) agonist (K i : 22.1 nM), effectively …
Formula:
C34H34N6O6
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
622.67
Ref: TM-T79373
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 10 Dec 2024
GRK2-IN-1 hydrochloride (2055990-90-2 free base)
GRKs-IN-1 hydrochloride has remarkable potency against and selectivity for G protein-coupled receptor kinase 2 GRK2 …
Formula:
C24H26ClFN4O4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
488.94
Ref: TM-T13714L
| 1mg | 106.00 € | ||
| 2mg | 169.00 € | ||
| 5mg | 294.00 € | ||
| 10mg | 459.00 € | ||
| 25mg | 824.00 € | ||
| 50mg | 1,372.00 € | ||
| 100mg | 1,870.00 € | ||
| 200mg | To inquire | ||
| 500mg | To inquire | ||
| 1mL*10mM (DMSO) | 316.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Serazapine
CAS:115313-22-9
Serazapine is a highly specific serotonin (5-HT2) binding inhibitor with anxiolytic activity for the treatment …
Formula:
C22H23N3O2
Purity:
98.06% - 99%
Color and Shape:
Liquid
Molecular weight:
361.44
Ref: TM-T68142
| 1mg | 197.00 € | ||
| 5mg | 505.00 € | ||
| 10mg | 723.00 € | ||
| 25mg | 1,103.00 € | ||
| 50mg | 1,504.00 € | ||
| 100mg | 2,023.00 € | ||
| 500mg | 4,057.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
β-Endorphin (1-27) (human)
CAS:76622-84-9
β-Endorphin (1-27) (human) is an opioid antagonist that selectively binds to μ-, δ-, and κ-opioid …
Formula:
C139H217N33O40S
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
3022.47
Ref: TM-T80515
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Semaglutide TFA (910463-68-2 free base)
Semaglutide TFA is a agonist of glucagon-like peptide-1 (GLP-1) receptor,with a potential for type 2 …
Formula:
NA
Purity:
99.69%
Color and Shape:
Solid
Molecular weight:
4210.63
Ref: TM-T12878
| 1mg | 219.00 € | ||
| 5mg | 758.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Catalpalactone
CAS:1585-68-8
Catalpalactone: antitermitic, cytotoxic, inhibits NO in cells (IC50 9.80µM), reduces dopamine synthesis, hinders TPA-induced EBV-EA …
Formula:
C15H14O4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
258.27
Ref: TM-TN3607
| 5mg | 1,378.00 € | ||
| 1mL*10mM (DMSO) | To inquire |
Estimated delivery in United States, on Tuesday 10 Dec 2024
GLP-1 (9-36) amide
CAS:161748-29-4
GLP-1 (9-36) amide is an antagonist at the human GLP-1 receptor.
Formula:
C140H214N36O43
Purity:
97%
Color and Shape:
Solid
Molecular weight:
3089.41
Ref: TM-TP2252
| 1mg | 88.00 € | ||
| 5mg | 238.00 € | ||
| 10mg | 353.00 € | ||
| 25mg | 584.00 € | ||
| 50mg | 823.00 € | ||
| 100mg | 1,109.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Deltorphin
CAS:119975-64-3
Deltorphin (Dermenkephalin) is Isolated from the skin of Phyllomedusa Sauvage. It also has an affinity …
Formula:
C44H62N10O10S2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
955.15
Ref: TM-T20166
| 1mg | 167.00 € | ||
| 5mg | 291.00 € | ||
| 10mg | 556.00 € | ||
| 25mg | 888.00 € | ||
| 50mg | 1,198.00 € | ||
| 100mg | 1,606.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Quipazine dimaleate
CAS:150323-78-7
Quipazine dimaleate is a selective 5-HT3 agonist.
Formula:
C21H23N3O8
Purity:
100%
Color and Shape:
Solid
Molecular weight:
445.42
Ref: TM-T23212
| 10mg | 35.00 € | ||
| 25mg | 52.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
