G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Fluphenazine dihydrochloride
CAS:146-56-5
Fluphenazine dihydrochloride (Prolixin) is an inhibitor of phenothiazine-class D1DR and D2DR. Fluphenazine can be used …
Formula:
C22H28Cl2F3N3OS
Purity:
100%
Color and Shape:
Off-White Solid
Molecular weight:
510.44
Ref: TM-T0068
| 50mg | 55.00 € | ||
| 100mg | 61.00 € | ||
| 200mg | 86.00 € | ||
| 500mg | 115.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
6-Iodopravadoline
CAS:164178-33-0
6-Iodopravadoline (AM630) is an antagonist of CB2 (Ki: 31.2 nM). And it shows 165-fold selectivity …
Formula:
C23H25IN2O3
Purity:
99.86%
Color and Shape:
Off-White Solid
Molecular weight:
504.36
Ref: TM-T14204
| 1mg | 40.00 € | ||
| 2mg | 50.00 € | ||
| 5mg | 72.00 € | ||
| 10mg | 94.00 € | ||
| 25mg | 207.00 € | ||
| 50mg | 337.00 € | ||
| 100mg | 539.00 € | ||
| 1mL*10mM (DMSO) | 104.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
Olodaterol
CAS:868049-49-4
Olodaterol is a novel, long-acting beta2-adrenergic agonist (LABA) that exerts its pharmacological effect by binding …
Formula:
C21H26N2O5
Purity:
98.9%
Color and Shape:
Solid
Molecular weight:
386.45
Ref: TM-T3457
| 1mg | 50.00 € | ||
| 5mg | 87.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
Alprenolol
CAS:13655-52-2
Alprenolol (Alpheprol) is a non-selective β-adrenergic receptor (β-AR) antagonist that is also an antagonist of …
Formula:
C15H23NO2
Purity:
99.73% - 99.78%
Color and Shape:
Solid
Molecular weight:
249.35
Ref: TM-T4560
| 50mg | 52.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
Fenoterol
CAS:13392-18-2
Fenoterol is an agonist of β2-adrenergic receptor It is classed as sympathomimetic beta agonist and …
Formula:
C17H21NO4
Purity:
99.56%
Color and Shape:
Solid
Molecular weight:
303.35
Ref: TM-T8358
| 2mg | 38.00 € | ||
| 5mg | 54.00 € | ||
| 10mg | 88.00 € | ||
| 25mg | 158.00 € | ||
| 50mg | 227.00 € | ||
| 1mL*10mM (DMSO) | 71.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
Bisoprolol hemifumarate
CAS:104344-23-2
Bisoprolol, a selective beta-1 adrenergic receptor antagonist, selectively and competitively binds to and blocks beta-1 …
Formula:
C20H33NO6
Purity:
99% - 99.95%
Color and Shape:
White To Offf-White Powder
Molecular weight:
383.49
Ref: TM-T0143
| 50mg | 51.00 € | ||
| 1mL*10mM (DMSO) | 56.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
Metoprolol tartrate
CAS:56392-17-7
Metoprolol Tartrate is a blocker of the cardioselective β-adrenergic receptor.
Formula:
C15H25NO3C4H6O6
Purity:
99.72% - 99.93%
Color and Shape:
White To Off-White / Powder
Molecular weight:
684.81
Ref: TM-T0487
| 25mg | 116.00 € | ||
| 50mg | 168.00 € | ||
| 1mL*10mM (DMSO) | 67.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
Nadolol
CAS:42200-33-9
Nadolol is a non-selective beta-adrenergic antagonist with antihypertensive and antiarrhythmic activities.
Formula:
C17H27NO4
Purity:
99.87% - 99.92%
Color and Shape:
White To Off-White Crystalline Powder Solid
Molecular weight:
309.4
Ref: TM-T1203
| 25mg | 49.00 € | ||
| 50mg | 72.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
Terbutaline
CAS:23031-25-6
Terbutaline is a short-acting agonist of β2-adrenergic receptor (β2-AR) . It is an active metabolite …
Formula:
C12H19NO3
Purity:
99.46%
Color and Shape:
Solid
Molecular weight:
225.3
Ref: TM-T8810
| 5mg | 42.00 € | ||
| 10mg | 55.00 € | ||
| 25mg | 90.00 € | ||
| 50mg | 115.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
MRGPRX1 agonist 1
CAS:2377379-39-8
MRGPRX1 agonist 1 is a highly potent MRGPRX1 (Mas-related G-protein-coupled receptor X1)agonist(EC50 of 50 nM).
Formula:
C23H21N3O4S
Purity:
99.59%
Color and Shape:
Solid
Molecular weight:
435.5
Ref: TM-T12104
| 1mg | 87.00 € | ||
| 5mg | 206.00 € | ||
| 10mg | 330.00 € | ||
| 25mg | 599.00 € | ||
| 50mg | 820.00 € | ||
| 100mg | 1,169.00 € | ||
| 1mL*10mM (DMSO) | 228.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
Amisulpride
CAS:71675-85-9
Amisulpride (Solian/Deniban), a dopamine antagonist antipsychotic, treats psychosis and schizophrenia in Europe/Australia, not in the …
Formula:
C17H27N3O4S
Purity:
100%
Color and Shape:
White Or Almost White Crystalline Powder
Molecular weight:
369.48
Ref: TM-T0811
| 1g | 346.00 € | ||
| 25mg | 49.00 € | ||
| 50mg | 68.00 € | ||
| 100mg | 90.00 € | ||
| 200mg | 138.00 € | ||
| 500mg | 238.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
(3aR,9aR)-Fluparoxan
CAS:105182-47-6
(3aR,9aR)-Fluparoxan is a highly selective and potent adrenergic receptor α2B antagonist for the prevention, amelioration …
Formula:
C10H10FNO2
Purity:
98.68%
Color and Shape:
Soild
Molecular weight:
195.19
Ref: TM-T77566
| 1mg | 182.00 € | ||
| 5mg | 401.00 € | ||
| 10mg | 591.00 € | ||
| 25mg | 920.00 € | ||
| 50mg | 1,267.00 € | ||
| 100mg | 1,699.00 € | ||
| 500mg | 3,416.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
WAY-298630
CAS:303134-93-2
Fluorophenoxy benzimidazole, a CRTH2 blocker, IC50 < 10 μM for rhinitis, COPD, arthritis, eczema, conjunctivitis.
Formula:
C17H15FN2O3S
Purity:
97.13%
Color and Shape:
Liquid
Molecular weight:
346.38
Ref: TM-T77601
| 1mg | 181.00 € | ||
| 5mg | 400.00 € | ||
| 10mg | 595.00 € | ||
| 25mg | 917.00 € | ||
| 50mg | 1,263.00 € | ||
| 100mg | 1,710.00 € | ||
| 500mg | 3,428.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
GLP-1 (9-36) amide
CAS:161748-29-4
GLP-1 (9-36) amide is an antagonist at the human GLP-1 receptor.
Formula:
C140H214N36O43
Purity:
97%
Color and Shape:
Solid
Molecular weight:
3089.41
Ref: TM-TP2252
| 1mg | 88.00 € | ||
| 5mg | 238.00 € | ||
| 10mg | 353.00 € | ||
| 25mg | 584.00 € | ||
| 50mg | 823.00 € | ||
| 100mg | 1,109.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
GB-6
CAS:2413262-74-3
GB-6, a short linear peptide that selectively binds to the gastrin releasing peptide receptor (GRPR), …
Formula:
C32H45N11O8
Purity:
98%
Color and Shape:
Solid
Molecular weight:
711.77
Ref: TM-T80266
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 25 Nov 2024
AB21 HCl
AB21 HCl: σ1 receptor antagonist, Ki 13 nM; less potent at σ2 (102 nM). Reduces …
Formula:
C23H29ClN2O
Purity:
99.89%
Color and Shape:
Liquid
Molecular weight:
384.2
Ref: TM-T77340L
| 1mg | 182.00 € | ||
| 5mg | 401.00 € | ||
| 10mg | 593.00 € | ||
| 25mg | 917.00 € | ||
| 50mg | 1,268.00 € | ||
| 100mg | 1,706.00 € | ||
| 500mg | 3,418.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Nociceptin (1-13), amide
CAS:178064-02-3
Nociceptin (1-13), amide is a potent ORL1 (OP4) receptor agonist with a pEC50 of 7.9 …
Formula:
C61H100N22O15
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1381.59
Ref: TM-TP1793
| 5mg | 98.00 € | ||
| 10mg | 149.00 € | ||
| 25mg | 217.00 € | ||
| 50mg | 323.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Ac-(d-Arg)-CEH-(d-Phe)-RWC-NH2
CAS:819048-44-7
Ac-DArg-c[Cys-Glu-His-DPhe-Arg-Trp-Cys]-NH2 is a synthetic cyclic octapeptide that exhibits melanocortin-4 receptor (MC4R) agonism and has been …
Formula:
C51H70N18O11S2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1175.35
Ref: TM-T80121
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 25 Nov 2024
ITIC-4F
CAS:2097998-59-7
ITIC-4F: a postfullerene IDTT electron acceptor for high-efficiency PSCs, relevant in binary, ternary, and tandem …
Formula:
C94H78F4N4O2S4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1499.92
Ref: TM-T19385
| 50mg | To inquire | ||
| 100mg | To inquire |
Estimated delivery in United States, on Monday 25 Nov 2024
Adrenomedullin (AM) (22-52), human acetate
Adrenomedullin (AM) (22-52), human acetate is an antagonist of calcitonin generelated peptide receptor in the …
Formula:
C161H256N46O50
Purity:
99.42%
Color and Shape:
Liquid
Molecular weight:
3636.09
Ref: TM-TP1257L
| 1mg | 206.00 € | ||
| 5mg | 807.00 € | ||
| 10mg | 1,204.00 € | ||
| 25mg | 2,180.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
