G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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SB 216641
CAS:170230-39-4
SB 216641 is a 5-HT (1B/1D) antagonist with anxiolytic activity for the study of anxiety …
Formula:
C28H30N4O4
Purity:
98.01%
Color and Shape:
Solid
Molecular weight:
486.56
Ref: TM-T85323
| 1mg | 196.00 € | ||
| 5mg | 486.00 € | ||
| 10mg | 682.00 € | ||
| 25mg | 1,064.00 € | ||
| 50mg | 1,467.00 € | ||
| 100mg | 1,878.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
CI 169369
CAS:85273-96-7
CI 169369 is a selective 5-HT2 receptor antagonist used in the study of anxiety and …
Formula:
C19H21ClN2S
Purity:
100%
Color and Shape:
Soild
Molecular weight:
344.9
Ref: TM-T84289
| 1mg | 199.00 € | ||
| 5mg | 493.00 € | ||
| 10mg | 692.00 € | ||
| 25mg | 1,080.00 € | ||
| 50mg | 1,489.00 € | ||
| 100mg | 1,907.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
![Des-Arg9-[Leu8]-Bradykinin acetate](https://static.cymitquimica.com/products/TM/thumb/T80072.jpg)
Des-Arg9-[Leu8]-Bradykinin acetate
CAS:115035-45-5
Des-Arg9-[Leu8]-Bradykinin acetate is a potent antagonist of the bradykinin receptor 1 (B1R), utilized in renal …
Formula:
C43H67N11O12
Purity:
98%
Color and Shape:
Solid
Molecular weight:
930.06
Ref: TM-T80072
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Ac-(d-Arg)-CEH-(d-Phe)-RWC-NH2
CAS:819048-44-7
Ac-DArg-c[Cys-Glu-His-DPhe-Arg-Trp-Cys]-NH2 is a synthetic cyclic octapeptide that exhibits melanocortin-4 receptor (MC4R) agonism and has been …
Formula:
C51H70N18O11S2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1175.35
Ref: TM-T80121
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Semaglutide TFA (910463-68-2 free base)
Semaglutide TFA is a agonist of glucagon-like peptide-1 (GLP-1) receptor,with a potential for type 2 …
Formula:
NA
Purity:
98%
Color and Shape:
Solid
Molecular weight:
4210.63
Ref: TM-T12878
| 1mg | 219.00 € | ||
| 5mg | 758.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Esprolol
CAS:396654-09-4
Esprolol (ACC-9369 free base) is a novel beta-adrenergic antagonist used to study exertional angina.
Formula:
C17H27NO4
Purity:
100% - 99.16%
Color and Shape:
Soild
Molecular weight:
309.4
Ref: TM-T27286L
| 1mg | 125.00 € | ||
| 5mg | 295.00 € | ||
| 10mg | 436.00 € | ||
| 25mg | 717.00 € | ||
| 50mg | 1,007.00 € | ||
| 100mg | 1,351.00 € | ||
| 500mg | 2,692.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
PU-WS13 hydrobromide
PU-WS13 hydrobromide is a GRP94 inhibitor with anti-inflammatory activity and inhibits the proliferation of M2-like …
Formula:
C17H21BrCl2N6S
Purity:
98%
Color and Shape:
Soild
Molecular weight:
492.26
Ref: TM-T5351L
| 1mg | 42.00 € | ||
| 5mg | 85.00 € | ||
| 10mg | 94.00 € | ||
| 25mg | 217.00 € | ||
| 50mg | 420.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
ABT 724 trihydrochloride
CAS:587870-77-7
ABT-724 trihydrochloride: selective D4 agonist; EC50=12.4nM(human),14.3nM(rat),23.2nM(ferret); for erectile dysfunction research.
Formula:
C17H22Cl3N5
Purity:
99.72%
Color and Shape:
Solid
Molecular weight:
402.75
Ref: TM-T22019
| 1ml | 43.00 € | ||
| 5mg | 39.00 € | ||
| 10mg | 63.00 € | ||
| 25mg | 122.00 € | ||
| 50mg | 182.00 € | ||
| 100mg | 272.00 € | ||
| 200mg | 405.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
GRP (14-27) (human, porcine, canine)
CAS:81608-29-9
GRP (14-27) (human, porcine, canine) functions as a ligand for bombesin receptors, with its specific …
Formula:
C75H110N24O16S2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1667.96
Ref: TM-T80148
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Talquetamab
CAS:2226212-40-2
Talquetamab (JNJ-64407564) is a T-cell retargeting GPRC5D bispecific antibody with antitumor activity for the treatment …
Color and Shape:
Solid
Ref: TM-T76882
| 1mg | 273.00 € | ||
| 2mg | 413.00 € | ||
| 5mg | 682.00 € | ||
| 10mg | 1,094.00 € | ||
| 25mg | 1,622.00 € | ||
| 50mg | 2,188.00 € | ||
| 100mg | 2,951.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
β-Endorphin (6-31), human
CAS:77761-27-4
β-Endorphin is an endogenous opioid neuropeptide and opioid receptor agonist that preferentially binds to μ-opioid …
Formula:
C131H218N34O40
Purity:
98%
Color and Shape:
Solid
Molecular weight:
2909.38
Ref: TM-T76285
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
p-MPPF
CAS:155204-26-5
p-MPPF is a 5-HT antagonist that can be used to study neurological diseases.
Formula:
C25H27FN4O2
Purity:
99.79%
Color and Shape:
Solid
Molecular weight:
434.51
Ref: TM-T69750L
| 1mg | 192.00 € | ||
| 5mg | 476.00 € | ||
| 10mg | 668.00 € | ||
| 25mg | 1,041.00 € | ||
| 50mg | 1,437.00 € | ||
| 100mg | 1,839.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
(d(CH2)51,Tyr(Me)2,Dab5,Arg8)-Vasopressin
CAS:176714-12-8
(d(CH2)5[Tyr(Me)2, Dab5]AVP), a vasopressin V1a receptor-specific antagonist, demonstrates a pA2 value of 6.71 [1].
Formula:
C52H76N14O11S2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1137.38
Ref: TM-T80137
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Survodutide
CAS:2805997-46-8
Survodutide (BI 456906) is a dual agonist of glucagon and glucagon-like peptide 1 (GLP-1) receptor …
Formula:
C192H289N47O61
Purity:
99.83%
Color and Shape:
Solid
Molecular weight:
4231.62
Ref: TM-T76559
| 1mg | 102.00 € | ||
| 5mg | 212.00 € | ||
| 10mg | 322.00 € | ||
| 25mg | 535.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
N-Desmethyl Pimavanserin
CAS:639863-77-7
N-Desmethyl Pimavanserin (AC-279) is the active metabolite of Pimavanserin and is used in the treatment …
Formula:
C24H32FN3O2
Purity:
98.02%
Color and Shape:
Solid
Molecular weight:
413.53
Ref: TM-T37979
| 1mg | 69.00 € | ||
| 1ml | 238.00 € | ||
| 2mg | 117.00 € | ||
| 5mg | 263.00 € | ||
| 10mg | 375.00 € | ||
| 25mg | 631.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
CB2R agonist 3
CB2R agonist 3, a potent activator of cannabinoid receptor 2 (CB2R), exhibits an EC50 value …
Purity:
98%
Ref: TM-T82769
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
1-Oleoyl Lysophosphatidic Acid
CAS:65528-98-5
1-Oleoyl Lysophosphatidic Acid (1-Oleoyl LPA) is a biologically active phospholipid that can be used to …
Formula:
C21H41O7P
Color and Shape:
Solid
Molecular weight:
436.52
Ref: TM-T36907
| 22.91mM*1 | 379.00 € | ||
| 22.91mM*100 | 68.00 € | ||
| 22.91mM*2.5 | 795.00 € | ||
| 22.91mM*500 | 231.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
(Val3,Pro8)-Oxytocin
CAS:2134138-89-7
(Val3,Pro8)-Oxytocin functions primarily as a Gq-dependent pathway agonist and exhibits secondary activity as a reduced …
Formula:
C41H60N12O12S2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
977.12
Ref: TM-T80140
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Capeserod
CAS:769901-96-4
Capeserod is a potential 5-HT4 receptor (5-hydroxytryptamine receptor 4) agonist for the study of digestive …
Formula:
C23H25ClN4O4
Purity:
98.82% - 99.37%
Color and Shape:
Solid
Molecular weight:
456.92
Ref: TM-T68035
| 1mg | 182.00 € | ||
| 5mg | 449.00 € | ||
| 10mg | 643.00 € | ||
| 25mg | 1,004.00 € | ||
| 50mg | 1,385.00 € | ||
| 100mg | 1,831.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Enrasentan
CAS:167256-08-8
Enrasentan (sb-217242) is a mixed antagonist of ET(A) and ET(B) receptors that reduces blood pressure …
Formula:
C29H30O8
Purity:
97.90% - 97.96%
Color and Shape:
Solid
Molecular weight:
506.54
Ref: TM-T31640
| 1mg | 181.00 € | ||
| 5mg | 447.00 € | ||
| 10mg | 640.00 € | ||
| 25mg | 1,004.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
