G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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![d[Leu4,Lys8]-VP acetate](https://static.cymitquimica.com/products/TM/thumb/TP1927L1.jpg)
d[Leu4,Lys8]-VP acetate
d[Leu4,Lys8]-VP acetate: Vasopressin V1b agonist. Ki: rat 0.16 nM, human 0.52 nM, mouse 1.38 nM. …
Formula:
C49H71N11O13S2
Purity:
98.86%
Color and Shape:
Solid
Molecular weight:
1086.28
Ref: TM-TP1927L1
| 1mg | 46.00 € | ||
| 2mg | 58.00 € | ||
| 5mg | 83.00 € | ||
| 10mg | 118.00 € | ||
| 25mg | 204.00 € | ||
| 50mg | 306.00 € | ||
| 100mg | 460.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Invopressin
CAS:1488411-60-4
Invopressin (Compound 42), a vasopressin V1A receptor partial agonist (EC50: 1.0 nM), is utilized in …
Formula:
C110H161N31O27S2
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
2413.78
Ref: TM-T80270
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 11 Dec 2024
A 77636 hydrochloride
CAS:145307-34-2
A 77636 hydrochloride is a potent, orally active, selective and long acting dopamine D1 receptor …
Formula:
C20H28ClNO3
Purity:
99.62%
Color and Shape:
Solid
Molecular weight:
365.89
Ref: TM-T21782
| 1mg | 94.00 € | ||
| 5mg | 213.00 € | ||
| 10mg | 310.00 € | ||
| 25mg | 523.00 € | ||
| 50mg | 736.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
(D-Arg8)-Inotocin
CAS:745816-74-4
'(D-Arg8)-Inotocin is a potent, selective, and competitive antagonist of the vasopressin receptor (V 1a R), …
Formula:
C39H68N14O11S2
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
973.17
Ref: TM-T80138
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Adenosine receptor agonist 1
Compound 6m, an A3 adenosine receptor (AR) partial agonist, exhibits a K i value of …
Formula:
C12H14ClN5O2Se
Color and Shape:
Liquid
Molecular weight:
374.68
Ref: TM-T89890
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 11 Dec 2024
CXCL-CXCR1/2-IN-1
CAS:2415653-55-1
CXCL-CXCR1/2-IN-1 is an ELR+CXCL-CXCR1/2 pathway inhibitor with anticancer activity and can be used in the …
Formula:
C14H8Cl2N4O3S
Purity:
99.40%
Color and Shape:
Soild
Molecular weight:
383.21
Ref: TM-T84325
| 5mg | 47.00 € | ||
| 10mg | 69.00 € | ||
| 25mg | 124.00 € | ||
| 50mg | 198.00 € | ||
| 100mg | 295.00 € | ||
| 500mg | 705.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Neocarzinostatin
CAS:9014-02-2
Neocarzinostatin is an effective DNA-damaging, anti-tumor antibiotic.
Purity:
98%
Color and Shape:
Solid
Molecular weight:
N/A
Ref: TM-T16283
| 100mg | To inquire | ||
| 500mg | To inquire |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Y1 receptor antagonist 1 formic
H 409-22 isomer formic, a formate salt of Y1 receptor antagonist 1, is an antagonist …
Formula:
C29H35N5O5
Color and Shape:
Liquid
Molecular weight:
533.62
Ref: TM-T200259
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Capeserod
CAS:769901-96-4
Capeserod is a potential 5-HT4 receptor (5-hydroxytryptamine receptor 4) agonist for the study of digestive …
Formula:
C23H25ClN4O4
Purity:
98.82% - 99.37%
Color and Shape:
Liquid
Molecular weight:
456.92
Ref: TM-T68035
| 1mg | 182.00 € | ||
| 5mg | 449.00 € | ||
| 10mg | 643.00 € | ||
| 25mg | 1,004.00 € | ||
| 50mg | 1,385.00 € | ||
| 100mg | 1,831.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
(Val3,Pro8)-Oxytocin
CAS:2134138-89-7
(Val3,Pro8)-Oxytocin functions primarily as a Gq-dependent pathway agonist and exhibits secondary activity as a reduced …
Formula:
C41H60N12O12S2
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
977.12
Ref: TM-T80140
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Guanylin TFA (mouse,rat)
Guanylin (mouse, rat) TFA is a peptide composed of 15 amino acids and acts as …
Formula:
C60H90N16O22S4·xC2HF3O2
Color and Shape:
Liquid
Molecular weight:
1515.71 (free base)
Ref: TM-TP2847
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 11 Dec 2024
(d(CH2)51,Tyr(Me)2,Dab5,Arg8)-Vasopressin
CAS:176714-12-8
(d(CH2)5[Tyr(Me)2, Dab5]AVP), a vasopressin V1a receptor-specific antagonist, demonstrates a pA2 value of 6.71 [1].
Formula:
C52H76N14O11S2
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
1137.38
Ref: TM-T80137
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 11 Dec 2024
GRP (14-27) (human, porcine, canine)
CAS:81608-29-9
GRP (14-27) (human, porcine, canine) functions as a ligand for bombesin receptors, with its specific …
Formula:
C75H110N24O16S2
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
1667.96
Ref: TM-T80148
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 11 Dec 2024
LCKLSL hydrochloride
LCKLSL hydrochloride is an AnxA2 inhibitor with potential anti-angiogenic activity and inhibits the development of …
Formula:
C30H58ClN7O8S
Color and Shape:
Liquid
Molecular weight:
712.34
Ref: TM-T78015
| 1mg | 90.00 € | ||
| 5mg | 184.00 € | ||
| 10mg | 346.00 € | ||
| 25mg | 640.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Ac-(d-Arg)-CEH-(d-Phe)-RWC-NH2
CAS:819048-44-7
Ac-DArg-c[Cys-Glu-His-DPhe-Arg-Trp-Cys]-NH2 is a synthetic cyclic octapeptide that exhibits melanocortin-4 receptor (MC4R) agonism and has been …
Formula:
C51H70N18O11S2
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
1175.35
Ref: TM-T80121
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 11 Dec 2024
KwFwLL-NH2
CAS:942266-38-8
KwFwLL-NH2 is a hexapeptide that serves as a ligand for the ghrelin receptor (ghrelin receptor). …
Formula:
C49H66N10O6
Color and Shape:
Liquid
Molecular weight:
891.11
Ref: TM-TP2863
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 11 Dec 2024
NPS ALX Compound 4a hydrochloride(1:1)
NPS ALX Compound 4a hydrochloride(1:1) is a potent and selective 5-hydroxytryptamine6 (5-HT6) receptor antagonist, with …
Formula:
C25H26ClN3O2S
Purity:
99.8%
Color and Shape:
Soild
Molecular weight:
468.01
Ref: TM-T12262L1
| 1mg | 51.00 € | ||
| 5mg | 110.00 € | ||
| 10mg | 165.00 € | ||
| 25mg | 272.00 € | ||
| 50mg | 394.00 € | ||
| 100mg | 539.00 € | ||
| 200mg | 713.00 € | ||
| 1mL*10mM (DMSO) | 132.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
β-CGRP (mouse)
β-CGRP (mouse), a calcitonin gene-related peptide, induces vasodilation and is applicable in research areas including …
Formula:
C165H265N49O55S2
Color and Shape:
Liquid
Molecular weight:
3879.29
Ref: TM-TP2859
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 11 Dec 2024
AB21 oxalate
AB21 oxalate, a potent and selective S1R antagonist, exhibits binding affinities (Kis) of 13 nM …
Formula:
C25H30N2O5
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
438.52
Ref: TM-T78916
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 11 Dec 2024
BMS 193885
CAS:679839-66-8
BMS 193885 is a selective and competitive neuropeptide Y(1) receptor antagonist with affinity of 3.3 …
Formula:
C36H48N4O9
Purity:
98%
Color and Shape:
Solid
Molecular weight:
680.79
Ref: TM-T22608
| 10mg | 797.00 € | ||
| 50mg | 3,187.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
