G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Guanylin (mouse, rat)
CAS:145257-03-0
Guanylin (mouse, rat), a peptide consisting of 15 amino acids, acts as an activator of …
Formula:
C60H90N16O22S4
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
1515.71
Ref: TM-T80150
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 10 Dec 2024
N-0500 HCl
CAS:100935-99-7
N-0500 HCl, a potent DA receptor agonist, displaces [3H]DP_x005f_x0002_5,6-ADTN with an IC50 of 3nM.
Formula:
C15H22ClNO2
Purity:
98.3% - 98.42%
Color and Shape:
Liquid
Molecular weight:
283.79
Ref: TM-T60107
| 5mg | 35.00 € | ||
| 10mg | 54.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Seglitide acetate
CAS:99248-33-6
Seglitide acetate (MK-678) is a selective agonist of sst2 somatostatin receptor.
Formula:
C46H60N8O9
Purity:
98.87%
Color and Shape:
Solid
Molecular weight:
869.02
Ref: TM-T28743
| 1mg | 111.00 € | ||
| 2mg | 159.00 € | ||
| 5mg | 247.00 € | ||
| 10mg | 362.00 € | ||
| 25mg | 543.00 € | ||
| 50mg | 763.00 € | ||
| 100mg | 1,026.00 € | ||
| 200mg | 1,392.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
GV-150013X
CAS:151386-96-8
GV-150013X ((S)-1-(1-(adamantan-1-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydro-1H-benzo[b][1,4]diazepin-3-yl)-3-phenylurea) is a potent CCKB antiagonist, pKi
Formula:
C33H34N4O3
Purity:
100%
Color and Shape:
Soild
Molecular weight:
534.65
Ref: TM-T27503L
| 1mg | 183.00 € | ||
| 5mg | 444.00 € | ||
| 10mg | 608.00 € | ||
| 25mg | 919.00 € | ||
| 50mg | 1,235.00 € | ||
| 100mg | 1,625.00 € | ||
| 1mL*10mM (DMSO) | 638.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
TAK-615
CAS:1664335-55-0
TAK-615 is commonly used to study pulmonary fibrosis and is a negative allosteric modulator of …
Formula:
C25H22FNO4
Purity:
99.36%
Color and Shape:
Solid
Molecular weight:
419.44
Ref: TM-T9699
| 1mg | 75.00 € | ||
| 5mg | 166.00 € | ||
| 10mg | 254.00 € | ||
| 25mg | 420.00 € | ||
| 50mg | 592.00 € | ||
| 100mg | 799.00 € | ||
| 500mg | 1,591.00 € | ||
| 1mL*10mM (DMSO) | 180.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
PAR-4 Agonist Peptide, amide
CAS:352017-71-1
PAR-4 Agonist Peptide, amide (AY-NH2) is an agonist of proteinase-activated receptor-4 (PAR-4).
Formula:
C34H48N8O7
Purity:
98%
Color and Shape:
Solid
Molecular weight:
680.79
Ref: TM-T7623
| 1mg | 51.00 € | ||
| 5mg | 142.00 € | ||
| 10mg | 230.00 € | ||
| 25mg | 391.00 € | ||
| 50mg | 563.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
GSK270822A
CAS:864082-23-5
GSK270822A is a selective ROCK1 inhibitor. GSK270822A exhibits IC50 of 9nM, 1100nM, 1550nM for ROCK1, …
Formula:
C24H20N4O2
Purity:
98.13% - 98.77%
Color and Shape:
Liquid
Molecular weight:
396.44
Ref: TM-T27467
| 1mg | 222.00 € | ||
| 5mg | 542.00 € | ||
| 10mg | 721.00 € | ||
| 25mg | 1,089.00 € | ||
| 50mg | 1,461.00 € | ||
| 100mg | 1,964.00 € | ||
| 1mL*10mM (DMSO) | 564.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
BMS-193885
CAS:186185-03-5
BMS-193885 is a selective, brain-penetrant, and competitive antagonist of the neuropeptide Y1 receptor with a …
Formula:
C33H42N4O6
Purity:
98%
Color and Shape:
Solid
Molecular weight:
590.71
Ref: TM-T14671
| 1mg | 34.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 112.00 € | ||
| 25mg | 218.00 € | ||
| 50mg | 324.00 € | ||
| 100mg | 472.00 € | ||
| 1mL*10mM (DMSO) | 90.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
L 152804
CAS:6508-43-6
L 152804: Y5 receptor antagonist, reduces food intake/boosts energy, leads to weight loss in obese …
Formula:
C23H26O4
Purity:
99.65%
Color and Shape:
Solid
Molecular weight:
366.45
Ref: TM-T15679
| 5mg | 50.00 € | ||
| 10mg | 78.00 € | ||
| 25mg | 114.00 € | ||
| 50mg | 174.00 € | ||
| 100mg | 253.00 € | ||
| 200mg | 359.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
NOX-6-18
CAS:898211-21-7
NOX-6-18 (GPR132-B-160) is a GPR132 antagonist with insulin-promoting activity and reduced weight gain.
Formula:
C18H17NO5S
Purity:
99.29%
Color and Shape:
Soild
Molecular weight:
359.4
Ref: TM-T83972
| 1mg | 75.00 € | ||
| 5mg | 160.00 € | ||
| 10mg | 250.00 € | ||
| 25mg | 502.00 € | ||
| 50mg | 809.00 € | ||
| 100mg | 1,290.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Upidosin
CAS:152735-23-4
Upidosin (SB-216469), a uroselective α1 blocker: Ki α1a=0.34 nM, α1b=3.9 nM, α1d=1.5 nM, α2=33.3 nM.
Formula:
C31H33N3O4
Purity:
99.26%
Color and Shape:
Solid
Molecular weight:
511.61
Ref: TM-T9762
| 5mg | 43.00 € | ||
| 10mg | 60.00 € | ||
| 25mg | 88.00 € | ||
| 50mg | 125.00 € | ||
| 100mg | 181.00 € | ||
| 200mg | 272.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
NESS 0327
CAS:494844-07-4
NESS 0327 is a high selectivity antagonist of the cannabinoid CB1 receptor. NESS 0327 is …
Formula:
C24H23Cl3N4O
Purity:
99.74%
Color and Shape:
Solid
Molecular weight:
489.82
Ref: TM-T22114
| 1mg | 123.00 € | ||
| 5mg | 300.00 € | ||
| 10mg | 429.00 € | ||
| 25mg | 643.00 € | ||
| 50mg | 867.00 € | ||
| 100mg | 1,156.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Pro8-Oxytocin TFA
Pro8-Oxytocin TFA, a modified oxytocin (OXT) ligand, exhibits greater potency and efficacy than the standard …
Formula:
C42H62N12O12S2·xC2HF3O2
Purity:
98%
Color and Shape:
Liquid
Ref: TM-T80134
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Nα-Methylhistamine FA
Nα-Methylhistamine FA is a histamine H3 receptor agonist
Formula:
C7H13N3O2
Purity:
100%
Color and Shape:
Liquid
Molecular weight:
171.2
Ref: TM-T23038L
| 1mg | 190.00 € | ||
| 5mg | 469.00 € | ||
| 10mg | 672.00 € | ||
| 25mg | 1,048.00 € | ||
| 50mg | 1,446.00 € | ||
| 100mg | 1,912.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
NF546 hydrate
NF546 (hydrate), a selective non-nucleotide P2Y11 agonist, exhibits a pEC50 value of 6.27 and induces …
Formula:
C47H44N6Na4O17P4·5H2O
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
1424.01
Ref: TM-T78079
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 10 Dec 2024
CB2R/FAAH modulator-3
CAS:2876918-67-9
CB2R/FAAH modulator-3 (compound 27) is a modulator targeting at CB2R and FAAH.
Formula:
C22H31NO2
Purity:
99.02%
Color and Shape:
Soild
Molecular weight:
341.49
Ref: TM-T67747
| 2mg | 38.00 € | ||
| 5mg | 57.00 € | ||
| 10mg | 89.00 € | ||
| 25mg | 160.00 € | ||
| 50mg | 253.00 € | ||
| 100mg | 373.00 € | ||
| 200mg | 531.00 € | ||
| 1mL*10mM (DMSO) | 62.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
cAC 253 acetate
cAC 253 acetate (TP2135 Free base) is an amylin antagonist. cAC 253 acetate inhibits 125I-adrenomedullin …
Formula:
C128H206N42O42S2
Purity:
98.16% - 99.99%
Color and Shape:
Soild
Molecular weight:
3069.39
Ref: TM-TP2135L
| 1mg | 182.00 € | ||
| 5mg | 415.00 € | ||
| 10mg | 616.00 € | ||
| 25mg | 920.00 € | ||
| 50mg | 1,290.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
L-796,778 acetate
L-796,778 acetate is a slective somatostatin receptor agonist with IC50 of 24nM for sst3, for …
Formula:
C31H44N6O9
Purity:
98%
Color and Shape:
Soild
Molecular weight:
644.72
Ref: TM-T32511L
| 1mg | 185.00 € | ||
| 5mg | 422.00 € | ||
| 10mg | 637.00 € | ||
| 25mg | 1,089.00 € | ||
| 50mg | 1,630.00 € | ||
| 100mg | 2,449.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
TCMCB07
CAS:1456699-27-6
TCMCB07, a cyclic nonapeptide, serves as an orally active, brain-penetrant antagonist of the melanocortin receptor …
Formula:
C63H87N15O11
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
1230.46
Ref: TM-T80540
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Picumeterol
CAS:130641-36-0
Picumeterol(GR 114297A) is a potent and selective β2 adrenergic receptor agonist. In vitro and in …
Formula:
C21H29Cl2N3O2
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
426.38
Ref: TM-T68129
| Undefined size | To inquire |
Estimated delivery in United States, on Tuesday 10 Dec 2024
