G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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LUF6096
CAS:1116652-18-6
LUF6096 (CF-602) is a potent allosteric enhancer of the adenosine A3 receptor, exhibiting the capability …
Formula:
C22H21Cl2N3O
Purity:
100%
Color and Shape:
Solid
Molecular weight:
414.33
Ref: TM-T9180
| 1mg | 53.00 € | ||
| 2mg | 79.00 € | ||
| 5mg | 114.00 € | ||
| 10mg | 182.00 € | ||
| 25mg | 311.00 € | ||
| 50mg | 439.00 € | ||
| 100mg | 624.00 € | ||
| 500mg | To inquire | ||
| 1mL*10mM (DMSO) | 132.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
(Rac)-AMXT-1501 4HCl
CAS:2771343-93-0
AMXT-1501 tetrahydrochloride is an inhibitor of polyamine transport.
Formula:
C32H72Cl4N6O2
Purity:
98.31%
Color and Shape:
Solid
Molecular weight:
714.77
Ref: TM-T10313
| 1mg | 170.00 € | ||
| 2mg | 250.00 € | ||
| 5mg | 430.00 € | ||
| 10mg | 657.00 € | ||
| 25mg | 1,442.00 € | ||
| 50mg | 2,225.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
CXCR4-IN-2
CXCR4-IN-2 (compound A1), a potent bifunctional fluorinated small molecule, inhibits CXCR4 and exhibits anticancer properties …
Formula:
C21H20F6N4S
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
474.47
Ref: TM-T78879
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 11 Dec 2024
BAM (8-22) acetate
BAM (8-22) acetate, a proenkephalin A derivative, stimulates MrgprC11, hMrgprX1, and causes scratching in mice.
Formula:
C93H131N25O25S
Purity:
98.85%
Color and Shape:
Solid
Molecular weight:
2031.25
Ref: TM-TP1914L1
| 1mg | 292.00 € | ||
| 5mg | 547.00 € | ||
| 10mg | 730.00 € | ||
| 25mg | 1,089.00 € | ||
| 50mg | 1,464.00 € | ||
| 100mg | 1,985.00 € | ||
| 200mg | 2,681.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
CCK Octapeptide, non-sulfated acetate
CCK Octapeptide, non-sulfated acetate is a synthetic desulfated peptide of cholecystokinin.
Formula:
C51H66N10O15S2
Purity:
98.97%
Color and Shape:
Liquid
Molecular weight:
1123.26
Ref: TM-TP2204L
| 1mg | 128.00 € | ||
| 5mg | 258.00 € | ||
| 10mg | 427.00 € | ||
| 25mg | 702.00 € | ||
| 50mg | 985.00 € | ||
| 100mg | 1,332.00 € | ||
| 500mg | 2,645.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Vasopressin Dimer (anti-parallel) (TFA)
Vasopressin Dimer (anti-parallel) TFA, an anti-parallel dimer form of vasopressin, has the capability to activate …
Formula:
C94H131F3N30O26S4
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
2282.49
Ref: TM-T80198
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Apitegromab
CAS:2278276-46-1
Apitegromab (SRK-015) is a new myostatin inhibitor, an antibody targeting myostatin precursor, which can be …
Purity:
95%
Color and Shape:
Liquid
Ref: TM-T77445
| 1mg | 207.00 € | ||
| 5mg | 608.00 € | ||
| 10mg | 917.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Ceruletide Ammonium Salt
Ceruletide Ammonium Salt is a decapeptide, originating from the skin of tropical frogs, which is …
Formula:
C58H77N14O21S2
Purity:
98.47%
Color and Shape:
Soild
Molecular weight:
1370.44
Ref: TM-T14932L1
| 1mg | 96.00 € | ||
| 5mg | 323.00 € | ||
| 10mg | 480.00 € | ||
| 25mg | 769.00 € | ||
| 50mg | 1,013.00 € | ||
| 100mg | 1,374.00 € | ||
| 500mg | 2,719.00 € | ||
| 1mL*10mM (DMSO) | 36.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
B-Raf IN 14
CAS:326918-98-3
B-Raf IN 14 is a BRAF inhibitor.
Formula:
C15H14BrN5O3S
Purity:
98.32%
Color and Shape:
Liquid
Molecular weight:
424.27
Ref: TM-T72070
| 1mg | 182.00 € | ||
| 5mg | 411.00 € | ||
| 10mg | 602.00 € | ||
| 25mg | 917.00 € | ||
| 50mg | 1,299.00 € | ||
| 100mg | 1,737.00 € | ||
| 500mg | 3,463.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Picumeterol FA
picumeterol FA is a potent and selective β2-adrenergic receptor agonist.
Formula:
C22H31Cl2N3O4
Purity:
99.80%
Color and Shape:
Soild
Molecular weight:
472.4
Ref: TM-T68129L1
| 1mg | 182.00 € | ||
| 5mg | 452.00 € | ||
| 10mg | 647.00 € | ||
| 25mg | 1,009.00 € | ||
| 50mg | 1,384.00 € | ||
| 100mg | 1,828.00 € | ||
| 500mg | 3,648.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
α-CGRP (mouse, rat) TFA
α-CGRP (mouse, rat) TFA, a neuropeptide belonging to the calcitonin gene-related peptide (CGRP) family, is …
Formula:
C162H262N50O52S2·C2HF3O2
Purity:
98%
Color and Shape:
Liquid
Ref: TM-T78540
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 11 Dec 2024
RS 56812
CAS:143137-37-5
RS 56812 is a 5-HT3 receptor antagonist and agonist used in the study of cognitive …
Formula:
C18H21N3O2
Purity:
98.78%
Color and Shape:
Soild
Molecular weight:
311.38
Ref: TM-T23264L
| 1mg | 200.00 € | ||
| 2mg | 295.00 € | ||
| 5mg | 494.00 € | ||
| 10mg | 693.00 € | ||
| 25mg | 1,082.00 € | ||
| 50mg | 1,493.00 € | ||
| 100mg | 1,911.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Dopamine D2 receptor agonist-2
CAS:1610591-93-9
Dopamine D2 receptor agonist-2 (Dopamine D2 Receptor) is a ligand targeting the dopamine D2 receptor.
Formula:
C25H31Cl2N5OS
Purity:
98.93%
Color and Shape:
Soild
Molecular weight:
520.52
Ref: TM-T60075
| 1mg | 37.00 € | ||
| 5mg | 69.00 € | ||
| 10mg | 88.00 € | ||
| 25mg | 144.00 € | ||
| 50mg | 204.00 € | ||
| 100mg | 304.00 € | ||
| 200mg | 436.00 € | ||
| 1mL*10mM (DMSO) | 88.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Dermorphin
CAS:77614-16-5
Dermorphin is agonist of μ-opioid receptor (MOR) agonist.
Formula:
C40H50N8O10
Purity:
98.82%
Color and Shape:
Solid
Molecular weight:
802.87
Ref: TM-T7404
| 1mg | 44.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Galanin-Like Peptide (rat)
CAS:245114-97-0
Galanin-Like Peptide (rat), a neuropeptide comprising 60 amino acids, plays a crucial role in regulating …
Formula:
C288H461N87O83S
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
6502.34
Ref: TM-T80146
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 11 Dec 2024
LY83583
CAS:91300-60-6
LY83583 is a soluble guanylate cyclase competitive inhibitor with IC50 of 2 µM.
Formula:
C15H10N2O2
Purity:
98.2% - 98.71%
Color and Shape:
Solid
Molecular weight:
250.25
Ref: TM-T21576
| 5mg | 59.00 € | ||
| 10mg | 96.00 € | ||
| 25mg | 172.00 € | ||
| 50mg | 270.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
L-796,778
CAS:217480-25-6
L-796,778 is an SST3 agonist and a selective ligand of SST3, which can increase the …
Formula:
C29H40N6O7
Purity:
98%
Color and Shape:
Solid
Molecular weight:
584.66
Ref: TM-T32511
| 1mg | 182.00 € | ||
| 5mg | 416.00 € | ||
| 10mg | 614.00 € | ||
| 25mg | 920.00 € | ||
| 50mg | 1,287.00 € | ||
| 100mg | 1,754.00 € | ||
| 500mg | 3,531.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Tropanserin
CAS:85181-40-4
Tropanserin (MDL 72422) is a 5-hydroxytryptamine receptor antagonist with anxiolytic activity that is used to …
Formula:
C17H23NO2
Purity:
99.74%
Color and Shape:
Solid
Molecular weight:
273.37
Ref: TM-T8451
| 1mg | 45.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 138.00 € | ||
| 25mg | 222.00 € | ||
| 50mg | 333.00 € | ||
| 100mg | 491.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Org 13011
CAS:142494-12-0
Org 13011 has CNS activity and induces conditioned taste aversion by mediating 5-HT 1A receptors.
Formula:
C18H25F3N4O
Purity:
98.98%
Color and Shape:
Soild
Molecular weight:
370.41
Ref: TM-T28258L
| 1mg | 185.00 € | ||
| 5mg | 459.00 € | ||
| 10mg | 657.00 € | ||
| 25mg | 1,025.00 € | ||
| 50mg | 1,413.00 € | ||
| 100mg | 1,869.00 € | ||
| 1mL*10mM (DMSO) | 466.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Vasopressin Dimer (parallel) (TFA)
Vasopressin Dimer (parallel) TFA, a parallel dimer of Vasopressin, has the capability to activate four …
Formula:
C94H131F3N30O26S4
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
2282.49
Ref: TM-T80197
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 11 Dec 2024
