G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Cortistatin 14, human, rat acetate
Cortistatin 14, human, rat acetate is a neuropeptide having structural similarity to somatostatin-14 and shows …
Formula:
C80H112N18O19S2
Purity:
97.86%
Color and Shape:
Solid
Molecular weight:
1693.98
Ref: TM-TP1188L
| 1mg | 106.00 € | ||
| 5mg | 229.00 € | ||
| 10mg | 340.00 € | ||
| 25mg | 543.00 € | ||
| 50mg | 730.00 € | ||
| 100mg | 979.00 € | ||
| 200mg | 1,309.00 € |
Estimated delivery in United States, on Monday 7 Oct 2024
PF-06655075 TFA
PF-06655075 (TFA) is the trifluoroacetic acid (TFA) salt of PF-06655075, a novel, non-brain-penetrant oxytocin receptor …
Purity:
98%
Ref: TM-T81501
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 7 Oct 2024
D3R/MOR antagonist 1
Compound 114 (D3R/MOR antagonist 1) exhibits dual antagonistic activity at dopamine D3 receptors (D3R) and …
Formula:
C22H27Cl2N3O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
420.38
Ref: TM-T78778
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 7 Oct 2024
BQ-3020 ammonium
BQ-3020 ammonium, a selective endothelin receptor (ET B receptor) agonist, demonstrates inhibition of [125 I] …
Formula:
C96H140N20O25S·xNH3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
2006.32 (free base)
Ref: TM-T78096
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 7 Oct 2024
PF-06478939 TFA
PF-06478939 TFA is a peptide that acts as a non-brain-penetrating agonist at the oxytocin (OT) …
Formula:
C78H134N14O22S2·xC2HF3O2
Purity:
98%
Color and Shape:
Solid
Ref: TM-T79174
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 7 Oct 2024
FGH31
FGH31 (Compound 24), a dopamine D4 agonist, exhibits potent and selective GRK2-dependency with a K …
Formula:
C33H36N4O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
520.66
Ref: TM-T79312
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 7 Oct 2024
Xanthine amine congener trihydrochloride
CAS:2459963-12-1
Xanthine amine congener trihydrochloride: potent adenosine antagonist, reverses effects of N6-cyclohexyladenosine on urine, sodium excretion, …
Formula:
C21H29ClN6O4
Purity:
97.85%
Color and Shape:
Solid
Molecular weight:
464.95
Ref: TM-T23535L
| 1mg | 73.00 € | ||
| 5mg | 138.00 € | ||
| 10mg | 185.00 € | ||
| 25mg | 327.00 € | ||
| 50mg | 458.00 € | ||
| 100mg | 648.00 € |
Estimated delivery in United States, on Monday 7 Oct 2024
![[Des-Arg9]-Bradykinin acetate](https://static.cymitquimica.com/products/TM/thumb/TP1445.jpg)
[Des-Arg9]-Bradykinin acetate
CAS:23827-91-0
[Des-Arg9]-Bradykinin acetate is a selective agonist of Bradykinin B1 receptor.
Formula:
C46H65N11O12
Purity:
99.05%
Color and Shape:
Solid
Molecular weight:
964.07
Ref: TM-TP1445
| 5mg | 35.00 € | ||
| 10mg | 49.00 € | ||
| 25mg | 101.00 € | ||
| 50mg | 150.00 € | ||
| 100mg | 216.00 € | ||
| 200mg | 315.00 € |
Estimated delivery in United States, on Monday 7 Oct 2024
GLP-1R Antagonist 1
CAS:488097-06-9
GLP-1R Antagonist 1 is an orally active, CNS penetrant and non-competitive glucagon-like peptide 1 receptor …
Formula:
C16H11ClF6N4O2
Purity:
90%
Color and Shape:
Solid
Molecular weight:
440.73
Ref: TM-T15387
| 1mg | 45.00 € | ||
| 1ml | 95.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 142.00 € | ||
| 25mg | 267.00 € | ||
| 50mg | 423.00 € |
Estimated delivery in United States, on Monday 7 Oct 2024
Ceruletide Ammonium acetate
Ceruletide Ammonium acetate (FI-6934 Ammonium acetate) is a cholecystokinin (CCK) receptor agonist.
Formula:
C60H77N13O23S2
Purity:
99.73%
Color and Shape:
Solid
Molecular weight:
1412.46
Ref: TM-T14932L
| 1mg | 234.00 € | ||
| 5mg | 476.00 € | ||
| 10mg | 691.00 € | ||
| 25mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 7 Oct 2024
EP4-IN-1
CAS:2455480-28-9
EP4-IN-1: Potent EP4 receptor inhibitor with anti-tumor, anti-inflammatory, and analgesic properties.
Formula:
C27H24N2O4
Purity:
100%
Color and Shape:
Soild
Molecular weight:
440.49
Ref: TM-T77699
| 2mg | 41.00 € | ||
| 5mg | 61.00 € | ||
| 10mg | 90.00 € |
Estimated delivery in United States, on Monday 7 Oct 2024
Spns2-IN-1
Spns2-IN-1 is a potent Spns2 inhibitor, effectively impeding Spns2-dependent S1P transport with an IC50 value …
Purity:
98%
Ref: TM-T81114
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 7 Oct 2024
(S)-(-)-Atenolol
CAS:93379-54-5
(S)-(-)-Atenolol has beta-adrenergic blocking effects.
Formula:
C14H22N2O3
Purity:
100% - 100%
Color and Shape:
Solid
Molecular weight:
266.34
Ref: TM-T35833
| 1mg | 73.00 € | ||
| 5mg | 151.00 € | ||
| 10mg | 213.00 € | ||
| 25mg | 359.00 € | ||
| 50mg | 534.00 € | ||
| 100mg | 763.00 € |
Estimated delivery in United States, on Monday 7 Oct 2024
hNTS1R agonist-1
Compound 10, an hNTS1R agonist-1, acts as a full agonist with a strong affinity for …
Formula:
C37H62N10O9
Purity:
98%
Color and Shape:
Solid
Molecular weight:
790.95
Ref: TM-T78954
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 7 Oct 2024
Thrombin Receptor Activator for Peptide 5 (TRAP-5)
CAS:141685-53-2
Thrombin Receptor Activator for Peptide 5 (TRAP-5) is also called Coagulation Factor II Receptor (1-5), …
Formula:
C30H50N8O7
Purity:
98%
Color and Shape:
Solid
Molecular weight:
634.77
Ref: TM-T7496
| 1mg | 78.00 € | ||
| 5mg | 160.00 € | ||
| 10mg | 243.00 € | ||
| 25mg | 437.00 € | ||
| 50mg | 655.00 € |
Estimated delivery in United States, on Monday 7 Oct 2024
NUCC-390 dihydrochloride (1060524-97-1 free base)
NUCC-390 dihydrochloride is selective agonist of small-molecule CXCR4 receptor.
Formula:
C23H35Cl2N5O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
468.46
Ref: TM-T12269L
| 100mg | To inquire | ||
| 500mg | To inquire |
Estimated delivery in United States, on Monday 7 Oct 2024
TCMCB07 TFA
TCMCB07 TFA is a cyclic nonapeptide and an orally active, brain-penetrating antagonist of the melanocortin …
Formula:
C63H87N15O11·xC2HF3O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1230.46 (free base)
Ref: TM-T80541
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 7 Oct 2024
Apelin-12 acetate
Apelin-12 acetate possesses a high affinity to orphan receptor APJ receptor.
Formula:
C66H107N21O16S
Purity:
98.82%
Color and Shape:
Solid
Molecular weight:
1482.75
Ref: TM-T39823L
| 1mg | 212.00 € | ||
| 1ml | 751.00 € | ||
| 5mg | 298.00 € | ||
| 10mg | 465.00 € | ||
| 25mg | 740.00 € | ||
| 50mg | 1,049.00 € | ||
| 100mg | 1,412.00 € |
Estimated delivery in United States, on Monday 7 Oct 2024
AB21 oxalate
AB21 oxalate, a potent and selective S1R antagonist, exhibits binding affinities (Kis) of 13 nM …
Formula:
C25H30N2O5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
438.52
Ref: TM-T78916
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 7 Oct 2024
Hemopressin(human, mouse) TFA
CAS:1431329-48-4
Hemopressin TFA: nonapeptide from hemoglobin, oral CB1 inverse agonist, eases inflammatory pain.
Formula:
C52H80F3N13O14
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1168.27
Ref: TM-T75799
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 7 Oct 2024
