G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Mogamulizumab
CAS:1159266-37-1
Mogamulizumab is a monoclonal antibody targeting CC chemokine receptor 4 with anticancer effects, used in …
Purity:
SDS-PAGE:97.3%;SEC-HPLC:99.4%
Color and Shape:
Liquid
Molecular weight:
146.43 kDa
Ref: TM-T76782
| 1mg | 445.00 € | ||
| 5mg | 916.00 € | ||
| 10mg | 1,281.00 € | ||
| 25mg | 1,839.00 € | ||
| 50mg | 2,591.00 € | ||
| 100mg | 3,533.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Samidorphan HCl
CAS:2328045-02-7
Samidorphan HCl is an orally active and highly potent modulator of the opioid system that …
Formula:
C21H27ClN2O4
Purity:
98.25% - 99.60%
Color and Shape:
Soild
Molecular weight:
406.9
Ref: TM-T67888L
| 1mg | 162.00 € | ||
| 5mg | 386.00 € | ||
| 10mg | 573.00 € | ||
| 25mg | 909.00 € | ||
| 50mg | 1,225.00 € | ||
| 100mg | 1,652.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Galcanezumab
CAS:1578199-75-3
Galcanezumab: humanized IgG4 antibody that targets CGRP for migraine and cluster headache prevention/treatment.
Purity:
> 95%
Color and Shape:
Liquid
Molecular weight:
144.08 kDa
Ref: TM-T76682
| 1mg | 125.00 € | ||
| 5mg | 370.00 € | ||
| 10mg | 594.00 € | ||
| 25mg | 919.00 € | ||
| 50mg | 1,233.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
PF-9184
CAS:1221971-47-6
PF-9184 inhibits human mPGES-1 selectively, with an IC50 of 16.5 nM, and reduces IL-1β-stimulated PGE2 …
Formula:
C21H14Cl2N2O4S
Purity:
97.64%
Color and Shape:
Solid
Molecular weight:
461.32
Ref: TM-T21738
| 1mg | 35.00 € | ||
| 5mg | 75.00 € | ||
| 10mg | 102.00 € | ||
| 25mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 16 Dec 2024
Anatibant 2HCl
CAS:209788-45-4
Anatibant 2HCl is a small molecule bradykinin B2 receptor antagonist for the treatment of neurological …
Formula:
C34H36Cl2N6O5S·2ClH
Purity:
99.18% - 99.71%
Color and Shape:
Soild
Molecular weight:
784.58
Ref: TM-T26627L
| 1mg | 327.00 € | ||
| 5mg | 901.00 € | ||
| 10mg | 1,119.00 € | ||
| 25mg | 1,477.00 € | ||
| 50mg | 1,839.00 € | ||
| 100mg | 2,322.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
6'-GNTI dihydrochloride
CAS:2410327-94-3
6'-GNTI dihydrochloride is a κ-opioid receptor (KOR) agonist that favors activation of G-protein-mediated signaling over …
Formula:
C27H29N5O3·2ClH
Purity:
99.08%
Color and Shape:
Liquid
Molecular weight:
544.47
Ref: TM-T39988
| 1mg | 325.00 € | ||
| 5mg | 788.00 € | ||
| 10mg | 1,082.00 € | ||
| 25mg | 1,606.00 € | ||
| 50mg | 2,164.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Sergliflozin A
CAS:360775-96-8
Sergliflozin A is a selective SGLT2 inhibitor that induces diabetes in a dose-dependent manner. It …
Formula:
C20H24O7
Purity:
100.00%
Color and Shape:
Liquid
Molecular weight:
376.4
Ref: TM-T68174
| 1mg | 108.00 € | ||
| 5mg | 242.00 € | ||
| 10mg | 363.00 € | ||
| 25mg | 609.00 € | ||
| 50mg | 865.00 € | ||
| 100mg | 1,170.00 € | ||
| 500mg | 2,348.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Gevotroline
CAS:107266-06-8
Gevotroline, a chemical in palm wine that can be used to treat psychosis, is a …
Formula:
C19H20FN3
Purity:
98.79%
Color and Shape:
Liquid
Molecular weight:
309.38
Ref: TM-T68080
| 1mg | 87.00 € | ||
| 5mg | 196.00 € | ||
| 10mg | 288.00 € | ||
| 25mg | 547.00 € | ||
| 50mg | 734.00 € | ||
| 100mg | 1,007.00 € | ||
| 500mg | 2,042.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
![[Des-Arg9]-Bradykinin](https://static.cymitquimica.com/products/TM/thumb/T7645.jpg)
[Des-Arg9]-Bradykinin
CAS:15958-92-6
[Des-Arg9]-Bradykinin ([Des-Arg9]-Bradykinin(2TFA))(2TFA) is an agonist of Bradykinin (B1) receptor.
Formula:
C44H61N11O10
Purity:
98%
Color and Shape:
Solid
Molecular weight:
904.02
Ref: TM-T7645
| 5mg | 252.00 € | ||
| 10mg | 444.00 € | ||
| 25mg | 936.00 € | ||
| 50mg | 1,470.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
IRAK inhibitor 4 trans
IRAK inhibitor 4 targets and blocks IRAK4 activity; refers to its trans molecular configuration.
Formula:
C33H35F3N6O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
620.66
Ref: TM-T11671
| 2mg | 374.00 € | ||
| 5mg | 560.00 € | ||
| 10mg | To inquire | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 763.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
HAEGTFTSD acetate(926018-45-3 free base)
HAEGTFTSD acetate is the first N-terminal 1-9 residues of GLP-1 peptide.The GLP-1 (7-36) amide is …
Formula:
C42H61N11O19
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1024.01
Ref: TM-TP1452L1
| 1mg | 251.00 € | ||
| 5mg | 513.00 € | ||
| 10mg | 777.00 € | ||
| 25mg | 1,398.00 € | ||
| 50mg | 2,095.00 € | ||
| 100mg | 3,143.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Ezlopitant
CAS:147116-64-1
Ezlopitant (CJ-11974) is a small molecule neurokinin-1-receptor (NK1) antagonist used to treat nausea, vomiting and …
Formula:
C31H38N2O
Purity:
97.03%
Color and Shape:
Liquid
Molecular weight:
454.65
Ref: TM-T68068
| 1mg | 91.00 € | ||
| 5mg | 196.00 € | ||
| 10mg | 288.00 € | ||
| 25mg | 544.00 € | ||
| 50mg | 729.00 € | ||
| 100mg | 1,013.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Losulazine
CAS:72141-57-2
Losulazine: a new antihypertensive, requires functional sympathetic nervous system; mechanism undefined.
Formula:
C27H22F4N4O3S
Purity:
99.80%
Color and Shape:
Liquid
Molecular weight:
558.55
Ref: TM-T68095
| 1mg | 92.00 € | ||
| 5mg | 195.00 € | ||
| 10mg | 288.00 € | ||
| 25mg | 544.00 € | ||
| 50mg | 725.00 € | ||
| 100mg | 1,013.00 € | ||
| 500mg | 2,023.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
(S, R)-LSN 3318839
CAS:2765539-92-0
(S,R)-LSN 3318839 enhances GLP-1R, shows strong blood sugar lowering in animals, works with sitagliptin.
Formula:
C26H23Cl2N3O2
Purity:
99.57%
Color and Shape:
Soild
Molecular weight:
480.39
Ref: TM-T63166L
| 1mg | 182.00 € | ||
| 5mg | 400.00 € | ||
| 10mg | 591.00 € | ||
| 25mg | 917.00 € | ||
| 50mg | 1,268.00 € | ||
| 100mg | 1,699.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
PF-03382792
CAS:1400811-63-3
PF-03382792 is a small molecule 5-HT4 receptor activator for the study of Alzheimer's disease.
Formula:
C23H32FN3O4
Purity:
98.09%
Color and Shape:
Solid
Molecular weight:
433.52
Ref: TM-T33940
| 1mg | 224.00 € | ||
| 5mg | 558.00 € | ||
| 10mg | 794.00 € | ||
| 25mg | 1,189.00 € | ||
| 50mg | 1,635.00 € | ||
| 100mg | 2,192.00 € | ||
| 500mg | 4,419.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
(R)-CJ 11974
CAS:187281-35-2
(R)-CJ 11974: non-peptide NK1 receptor antagonist, may relieve pain and prevent chemo-induced vomiting.
Formula:
C31H38N2O
Purity:
97.03%
Color and Shape:
Soild
Molecular weight:
454.65
Ref: TM-T68068L
| 1mg | 182.00 € | ||
| 5mg | 400.00 € | ||
| 10mg | 591.00 € | ||
| 25mg | 917.00 € | ||
| 50mg | 1,263.00 € | ||
| 100mg | 1,706.00 € | ||
| 500mg | 3,418.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
DPTN dihydrochloride
CAS:325767-87-1
DPTN dihydrochloride is a potent and selective A3AR antagonist with Ki values of 1.65, 9.61 …
Formula:
C22H20Cl2N4OS
Purity:
100%
Color and Shape:
Soild
Molecular weight:
459.39
Ref: TM-T72067
| 1mg | 50.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 162.00 € | ||
| 25mg | 339.00 € | ||
| 50mg | 524.00 € | ||
| 100mg | 738.00 € | ||
| 500mg | 1,557.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Semaglutide TFA (910463-68-2 free base)
Semaglutide TFA is a agonist of glucagon-like peptide-1 (GLP-1) receptor,with a potential for type 2 …
Formula:
C189H290F3N45O61
Purity:
99.69%
Color and Shape:
Solid
Molecular weight:
4225.6482
Ref: TM-T12878
| 1mg | 219.00 € | ||
| 5mg | 758.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
N-0500 HCl
CAS:100935-99-7
N-0500 HCl, a potent DA receptor agonist, displaces [3H]DP_x005f_x0002_5,6-ADTN with an IC50 of 3nM.
Formula:
C15H22ClNO2
Purity:
98.3% - 98.42%
Color and Shape:
Liquid
Molecular weight:
283.79
Ref: TM-T60107
| 5mg | 35.00 € | ||
| 10mg | 54.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Met-RANTES,human,acetate
Met-RANTES (human) acetate is the acetate salt form of Met-RANTES (human). It acts as an …
Ref: TM-T200698
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 16 Dec 2024
