G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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CCK Octapeptide, non-sulfated acetate
CCK Octapeptide, non-sulfated acetate is a synthetic desulfated peptide of cholecystokinin.
Formula:
C51H66N10O15S2
Purity:
98.97%
Color and Shape:
Solid
Molecular weight:
1123.26
Ref: TM-TP2204L
| 1mg | 85.00 € | ||
| 5mg | 158.00 € | ||
| 10mg | 253.00 € | ||
| 25mg | 415.00 € | ||
| 50mg | 582.00 € | ||
| 100mg | 787.00 € | ||
| 200mg | 1,063.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
7-FluorotryptaMine HCl
CAS:159730-09-3
7-FluorotryptaMine HCl is a potent aromatic monoamine GPRC5A agonist that induces GPRC5A-mediated β-arrestin recruitment.7-FluorotryptaMine HCl …
Formula:
C10H12ClFN2
Purity:
98.06%
Color and Shape:
Liquid
Molecular weight:
214.67
Ref: TM-T77673
| 1mg | 36.00 € | ||
| 5mg | 69.00 € | ||
| 10mg | 101.00 € | ||
| 25mg | 207.00 € | ||
| 50mg | 312.00 € | ||
| 100mg | 463.00 € | ||
| 500mg | 1,050.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
4-P-PDOT
CAS:134865-74-0
4-P-PDOT (4-phenyl-2- propionamidotetralin) is a potent, selective and affinity Melatonin receptor (MT2) antagonist.
Formula:
C19H21NO
Purity:
99.68%
Color and Shape:
Solid
Molecular weight:
279.38
Ref: TM-T14042
| 5mg | 50.00 € | ||
| 10mg | 72.00 € | ||
| 25mg | 126.00 € | ||
| 50mg | 227.00 € | ||
| 100mg | 362.00 € | ||
| 1mL*10mM (DMSO) | 50.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Dermorphin
CAS:77614-16-5
Dermorphin is agonist of μ-opioid receptor (MOR) agonist.
Formula:
C40H50N8O10
Purity:
98.82%
Color and Shape:
Solid
Molecular weight:
802.87
Ref: TM-T7404
| 1mg | 44.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
(Val3,Pro8)-Oxytocin
CAS:2134138-89-7
(Val3,Pro8)-Oxytocin functions primarily as a Gq-dependent pathway agonist and exhibits secondary activity as a reduced …
Formula:
C41H60N12O12S2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
977.12
Ref: TM-T80140
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 25 Nov 2024
RS 15385-198
CAS:121961-55-5
RS 15385-198 is a less active isomer of Delequamine. Delequamine is a selective alpha2-adrenergic receptor …
Formula:
C18H26N2O3S
Purity:
98.81%
Color and Shape:
Soild
Molecular weight:
350.48
Ref: TM-T68051L
| 1mg | 183.00 € | ||
| 5mg | 453.00 € | ||
| 10mg | 648.00 € | ||
| 25mg | 1,011.00 € | ||
| 50mg | 1,395.00 € | ||
| 100mg | 1,844.00 € | ||
| 500mg | 3,679.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Thrombin Receptor Activator for Peptide 5 (TRAP-5)
CAS:141685-53-2
Thrombin Receptor Activator for Peptide 5 (TRAP-5) is also called Coagulation Factor II Receptor (1-5), …
Formula:
C30H50N8O7
Purity:
98%
Color and Shape:
Solid
Molecular weight:
634.77
Ref: TM-T7496
| 1mg | 78.00 € | ||
| 5mg | 160.00 € | ||
| 10mg | 243.00 € | ||
| 25mg | 437.00 € | ||
| 50mg | 655.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Urotensin II, mouse TFA (9047-55-6 free base)
Urotensin II, mouse TFA is an endogenous ligand for the orphan GPR14 or SENR. It …
Formula:
C78H101N18F3O21S2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1747.88
Ref: TM-TP2166
| 100mg | To inquire | ||
| 500mg | To inquire |
Estimated delivery in United States, on Monday 25 Nov 2024
Dopamine D2 receptor agonist-2
CAS:1610591-93-9
Dopamine D2 receptor agonist-2 (Dopamine D2 Receptor) is a ligand targeting the dopamine D2 receptor.
Formula:
C25H31Cl2N5OS
Purity:
98.93%
Color and Shape:
Soild
Molecular weight:
520.52
Ref: TM-T60075
| 1mg | 37.00 € | ||
| 5mg | 69.00 € | ||
| 10mg | 88.00 € | ||
| 25mg | 144.00 € | ||
| 50mg | 204.00 € | ||
| 100mg | 304.00 € | ||
| 200mg | 436.00 € | ||
| 1mL*10mM (DMSO) | 88.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
PD 144418 oxalate
CAS:1794760-28-3
PD 144418 oxalate: σ1 receptor ligand, Ki=0.08 nM; 1377 nM for σ2, minimal affinity elsewhere; …
Formula:
C20H24N2O5
Purity:
99.08%
Color and Shape:
Solid
Molecular weight:
372.42
Ref: TM-T39211
| 1mg | 58.00 € | ||
| 5mg | 130.00 € | ||
| 10mg | 182.00 € | ||
| 25mg | 314.00 € | ||
| 50mg | 457.00 € | ||
| 100mg | 668.00 € | ||
| 200mg | 916.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
IRL-1038 acetate
IRL-1038 acetate is a potent ETB endothelin receptor antagonist.
Formula:
C70H96N14O17S2
Purity:
97.51%
Color and Shape:
Soild
Molecular weight:
1469.73
Ref: TM-TP2262L
| 1mg | 407.00 € | ||
| 5mg | 940.00 € | ||
| 10mg | 1,406.00 € | ||
| 25mg | 2,407.00 € | ||
| 50mg | 3,237.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
2-Oleoylglycerol
CAS:3443-84-3
2-Oleoylglycerol is a lipid found in palm kernels that acts as a GPR119 agonist with …
Formula:
C21H40O4
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
356.54
Ref: TM-T37526
| 1mg (28mM*100μL in Ethanol) | 92.00 € | ||
| 25mg (28mM*2.5mL in Ethanol) | To inquire |
Estimated delivery in United States, on Monday 25 Nov 2024
Tebufelone
CAS:112018-00-5
Tebufelone is a potent NSAID, inhibits CO, has anti-inflammatory and analgesic properties, and blocks lipoxygenase …
Formula:
C20H28O2
Purity:
99.5%
Color and Shape:
Liquid
Molecular weight:
300.44
Ref: TM-T68155
| 1mg | 56.00 € | ||
| 5mg | 119.00 € | ||
| 10mg | 170.00 € | ||
| 25mg | 277.00 € | ||
| 50mg | 424.00 € | ||
| 100mg | 612.00 € | ||
| 500mg | 1,265.00 € | ||
| 1mL*10mM (DMSO) | 186.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Esprolol
CAS:396654-09-4
Esprolol (ACC-9369 free base) is a novel beta-adrenergic antagonist used to study exertional angina.
Formula:
C17H27NO4
Purity:
100% - 99.16%
Color and Shape:
Soild
Molecular weight:
309.4
Ref: TM-T27286L
| 1mg | 125.00 € | ||
| 5mg | 295.00 € | ||
| 10mg | 436.00 € | ||
| 25mg | 717.00 € | ||
| 50mg | 1,007.00 € | ||
| 100mg | 1,351.00 € | ||
| 500mg | 2,692.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
![d[Leu4,Lys8]-VP acetate](https://static.cymitquimica.com/products/TM/thumb/TP1927L1.jpg)
d[Leu4,Lys8]-VP acetate
d[Leu4,Lys8]-VP acetate: Vasopressin V1b agonist. Ki: rat 0.16 nM, human 0.52 nM, mouse 1.38 nM. …
Formula:
C49H71N11O13S2
Purity:
98.86%
Color and Shape:
Solid
Molecular weight:
1086.28
Ref: TM-TP1927L1
| 1mg | 46.00 € | ||
| 2mg | 58.00 € | ||
| 5mg | 83.00 € | ||
| 10mg | 118.00 € | ||
| 25mg | 204.00 € | ||
| 50mg | 306.00 € | ||
| 100mg | 460.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Zalospirone
CAS:114298-18-9
Zalospirone is a 5-HT1A receptor agonist that can be used to study anxiety disorders and …
Formula:
C24H29N5O2
Purity:
100% - 99%
Color and Shape:
Solid
Molecular weight:
419.52
Ref: TM-T68172
| 1mg | 326.00 € | ||
| 5mg | 769.00 € | ||
| 10mg | 1,049.00 € | ||
| 25mg | 1,486.00 € | ||
| 50mg | 1,838.00 € | ||
| 100mg | 2,336.00 € | ||
| 500mg | 4,564.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Dynorphin B (1-9)
CAS:126050-26-8
Dynorphin B (1-9), a neuropeptide and the N-terminal cleavage product of dynorphin B, has its …
Formula:
C54H78N16O12
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1143.3
Ref: TM-T80463
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 25 Nov 2024
Galanin-Like Peptide (human)
CAS:245114-99-2
Galanin-Like Peptide (human) is a neuropeptide consisting of 60 amino acids, instrumental in regulating feeding, …
Formula:
C292H451N83O84S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
6500.28
Ref: TM-T80144
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 25 Nov 2024
SDF-1α (human)
CAS:1268129-65-2
SDF-1α (human) serves as a chemotactic agent for mononuclear cells through its interaction with the …
Formula:
C356H578N106O93S4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
7959.34
Ref: TM-T80130
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 25 Nov 2024
Mifentidine
CAS:83184-43-4
Mifentidine (DA 4577) is an orally available H2 receptor antagonist for the study of gastric …
Formula:
C13H16N4
Purity:
100% - 99.20%
Color and Shape:
Liquid
Molecular weight:
228.29
Ref: TM-T68100
| 1mg | 182.00 € | ||
| 5mg | 451.00 € | ||
| 10mg | 646.00 € | ||
| 25mg | 1,007.00 € | ||
| 50mg | 1,390.00 € | ||
| 100mg | 1,837.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
