G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Oxmetidine FA
Oxmetidine FA is an orally available specific histamine H2 receptor antagonist with antiulcerogenic properties.
Formula:
C20H23N5O5S
Purity:
97.34%
Color and Shape:
Soild
Molecular weight:
445.49
Ref: TM-T68122L
| 1mg | 182.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Somatostatin acetate
Somatostatin acetate is an endogenously secreted inhibitor of cell proliferation with potential antitumor activity for …
Ref: TM-TP1302L
| 1mg | 59.00 € | ||
| 5mg | 121.00 € | ||
| 10mg | 169.00 € | ||
| 25mg | 282.00 € | ||
| 50mg | 419.00 € | ||
| 100mg | 619.00 € | ||
| 500mg | 1,312.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Spiroglumide
CAS:137795-35-8
Spiroglumide, a CCKB-gastrin antagonist that inhibits dose-dependent pentagastrin-induced acid hypersecretion with an ID50 of 20.1 …
Formula:
C21H26Cl2N2O4
Purity:
98.34%
Color and Shape:
Soild
Molecular weight:
441.35
Ref: TM-T68016
| 1mg | 152.00 € | ||
| 5mg | 363.00 € | ||
| 10mg | 552.00 € | ||
| 25mg | 876.00 € | ||
| 50mg | 1,196.00 € | ||
| 100mg | 1,616.00 € | ||
| 500mg | 3,214.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Saterinone
CAS:102669-89-6
Saterinone: PDE III inhibitor, α-1-adrenoceptor antagonist, vasodilator, used for acute chronic heart failure, IC50 2.3x10^-5 …
Formula:
C27H30N4O4
Purity:
98.23%
Color and Shape:
Solid
Molecular weight:
474.55
Ref: TM-T68138
| 1mg | 152.00 € | ||
| 1ml | 433.00 € | ||
| 5mg | 365.00 € | ||
| 10mg | 548.00 € | ||
| 25mg | 875.00 € | ||
| 50mg | 1,188.00 € | ||
| 100mg | 1,606.00 € | ||
| 500mg | 3,212.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Binospirone
CAS:102908-59-8
Binospirone (MDL 73005EF) is a 5-HT1A receptor agonist with anxiolytic activity used in the study …
Formula:
C20H26N2O4
Purity:
98.05% - 99.11%
Color and Shape:
Soild
Molecular weight:
358.43
Ref: TM-T71138L
| 1mg | 185.00 € | ||
| 1ml | 47.00 € | ||
| 5mg | 459.00 € | ||
| 10mg | 657.00 € | ||
| 25mg | 1,025.00 € | ||
| 50mg | 1,413.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
difelikefalin acetate(1024828-77-0 Free base)
is a ketone and a building block.
Formula:
C38H57N7O8
Purity:
96.94%
Color and Shape:
Solid
Molecular weight:
739.9
Ref: TM-TP2485
| 1mg | 162.00 € | ||
| 5mg | 325.00 € | ||
| 10mg | 506.00 € | ||
| 25mg | 821.00 € | ||
| 50mg | 1,105.00 € | ||
| 100mg | 1,514.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Isocupressic acid
CAS:1909-91-7
Isocupressic acid triggers cow abortions in the last trimester by halting angiogenesis and inducing corpus …
Formula:
C20H32O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
320.47
Ref: TM-TN4277
| 1ml | To inquire | ||
| 5mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
(D-Arg8)-Inotocin
CAS:745816-74-4
'(D-Arg8)-Inotocin is a potent, selective, and competitive antagonist of the vasopressin receptor (V 1a R), …
Formula:
C39H68N14O11S2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
973.17
Ref: TM-T80138
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
ITIC
CAS:1664293-06-4
"ITIC, a non-fullerene acceptor with high Tg of 180°C, shows excellent thermal stability and a …
Formula:
C94H82N4O2S4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1427.96
Ref: TM-T19386
| 25mg | 1,435.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
S1R agonist 2
CAS:150085-21-5
S1R agonist 2 is a selective S1R agonist with a Ki of 88 nM for …
Formula:
C21H27NO
Purity:
99.04%
Color and Shape:
Solid
Molecular weight:
309.45
Ref: TM-T72059
| 1mg | 46.00 € | ||
| 5mg | 90.00 € | ||
| 10mg | 143.00 € | ||
| 25mg | 267.00 € | ||
| 50mg | 406.00 € | ||
| 100mg | 600.00 € | ||
| 500mg | 1,268.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
![[Ala17]-MCH acetate](https://static.cymitquimica.com/products/TM/thumb/TP1997L.jpg)
[Ala17]-MCH acetate
[Ala17]-MCH acetate is a selective ligand for MCHR1 with a Ki of 0.16 nM and …
Formula:
C99H159N29O28S4
Purity:
98.92%
Color and Shape:
Solid
Molecular weight:
2331.76
Ref: TM-TP1997L
| 1mg | 112.00 € | ||
| 5mg | 269.00 € | ||
| 10mg | 392.00 € | ||
| 25mg | 598.00 € | ||
| 50mg | 813.00 € | ||
| 100mg | 1,080.00 € | ||
| 200mg | 1,446.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Tolnapersine TFA
Tolnapersine TFA is a mixed dopamine agonist and alpha adrenergic receptor antagonist.
Formula:
C23H27F3N2O3
Purity:
98.10%
Color and Shape:
Soild
Molecular weight:
436.47
Ref: TM-T68023L
| 1mg | 182.00 € | ||
| 5mg | 399.00 € | ||
| 10mg | 591.00 € | ||
| 25mg | 920.00 € | ||
| 50mg | 1,267.00 € | ||
| 100mg | 1,710.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Pafenolol
CAS:75949-61-0
Pafenolol is a P-glycoprotein modulator with a Ki value of 5.5 µM. pafenolol is an …
Formula:
C18H31N3O3
Purity:
98.43%
Color and Shape:
Solid
Molecular weight:
337.46
Ref: TM-T68124
| 1mg | 93.00 € | ||
| 5mg | 186.00 € | ||
| 10mg | 279.00 € | ||
| 25mg | 544.00 € | ||
| 50mg | 743.00 € | ||
| 100mg | 1,019.00 € | ||
| 500mg | 2,070.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Eldelumab
CAS:946414-98-8
Eldelumab (BMS-936557) is an anti-IP-10 IgG 1 monoclonal antibody.Eldelumab has anti-inflammatory activity and is used …
Purity:
95%
Color and Shape:
Solid
Ref: TM-T76741
| 1mg | 226.00 € | ||
| 2mg | 333.00 € | ||
| 5mg | 554.00 € | ||
| 10mg | 841.00 € | ||
| 25mg | 1,273.00 € | ||
| 50mg | 1,716.00 € | ||
| 100mg | 2,310.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Relamorelin
CAS:661472-41-9
Relamorelin (RM-131) is a growth hormone-releasing peptide/growth hormone secretagogue receptor agonist, a 5 amino acid …
Formula:
C43H50N8O5S
Purity:
99.26% - 99.85%
Color and Shape:
Solid
Molecular weight:
790.97
Ref: TM-T34281
| 1mg | 468.00 € | ||
| 5mg | 1,082.00 € | ||
| 10mg | 1,458.00 € | ||
| 25mg | 2,163.00 € | ||
| 50mg | 2,793.00 € | ||
| 100mg | 3,940.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Neurokinin A(4-10)
CAS:97559-35-8
Neurokinin A(4-10)(TFA) is an agonist of tachykinin NK2 receptor .
Formula:
C34H54N8O10S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
766.91
Ref: TM-T7559
| 1mg | 123.00 € | ||
| 5mg | 243.00 € | ||
| 10mg | 427.00 € | ||
| 25mg | 850.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
KB-5492 FA
KB-5492 FA is a selective sigma receptor inhibitor with antiulcerogenic effects.CAS 번호128-52-56-8
Formula:
C24H32N2O8
Purity:
98.54%
Color and Shape:
Solid
Molecular weight:
476.52
Ref: TM-T62396L
| 1ml | 68.00 € | ||
| 5mg | 62.00 € | ||
| 10mg | 97.00 € | ||
| 25mg | 189.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
PACAP-38 (31-38), human, mouse, rat acetate
PACAP-38 (31-38) acetate stimulates PAC1 receptor and boosts NPY and catecholamine in sympathetic neurons.
Formula:
C49H87N17O13
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1122.32
Ref: TM-TP1618L
| 1mg | 132.00 € | ||
| 5mg | 383.00 € | ||
| 10mg | 555.00 € | ||
| 25mg | 891.00 € | ||
| 50mg | 1,203.00 € | ||
| 100mg | 1,606.00 € | ||
| 500mg | 3,240.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Somatostatin 1-28 acetate
Somatostatin 1-28 acetate circulates in human plasma.
Purity:
99.51%
Color and Shape:
Soild
Ref: TM-TP2124L
| 1mg | 465.00 € | ||
| 5mg | 943.00 € | ||
| 10mg | 1,272.00 € | ||
| 25mg | 1,903.00 € | ||
| 50mg | 2,571.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Retatrutide
CAS:2381089-83-2
Retatrutide (LY3437943) is a triple agonist of GCGR, GIPR and GLP-1R that can be used …
Formula:
C221H342N46O68
Purity:
98.31%
Color and Shape:
Solid
Molecular weight:
4731.33
Ref: TM-T76279
| 1mg | 231.00 € | ||
| 5mg | 581.00 € | ||
| 10mg | 932.00 € | ||
| 25mg | 1,374.00 € | ||
| 50mg | 1,847.00 € | ||
| 100mg | 2,513.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
