G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Lintitript
CAS:136381-85-6
Lintitript (SR 27897) is a selective antagonist of CCK1 with EC50s of 6 nM and …
Formula:
C20H14ClN3O3S
Purity:
98.48%
Color and Shape:
Solid
Molecular weight:
411.86
Ref: TM-T15759
| 1mg | 113.00 € | ||
| 2mg | 154.00 € | ||
| 5mg | 230.00 € | ||
| 10mg | 344.00 € | ||
| 25mg | 549.00 € | ||
| 50mg | 741.00 € | ||
| 100mg | 994.00 € | ||
| 1mL*10mM (DMSO) | 258.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Mesoridazine Besylate
CAS:32672-69-8
Mesoridazine Besylate (Serentil), a piperidine antipsychotic and phenothiazine, treats schizophrenia; it's a thioridazine metabolite.
Formula:
C27H32N2O4S3
Purity:
99.58%
Color and Shape:
Solid
Molecular weight:
544.75
Ref: TM-T3086
| 5mg | 75.00 € | ||
| 10mg | 127.00 € | ||
| 1mL*10mM (DMSO) | 36.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
CXCR7 antagonist-1
CAS:1613021-99-0
CXCR7 antagonist-1 is a specific antagonist of the binding of the SDF-1 chemokine or I-TAC …
Formula:
C21H19FN6O
Purity:
99.51%
Color and Shape:
Liquid
Molecular weight:
390.41
Ref: TM-T39078
| 1mg | 175.00 € | ||
| 5mg | 444.00 € | ||
| 10mg | 643.00 € | ||
| 25mg | 1,003.00 € | ||
| 50mg | 1,380.00 € | ||
| 100mg | 1,831.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Muscarinic toxin 3
CAS:873336-87-9
Muscarinic toxin 3 (MT3), a potent non-competitive antagonist of mAChR and adrenoceptors, exhibits pIC50 values …
Formula:
C319H489N89O97S8
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
7379.35
Ref: TM-T80477
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 11 Dec 2024
rac Desmethyl Citalopram Hydrochloride
CAS:97743-99-2
rac Desmethyl Citalopram Hydrochloride is a 5-hydroxy tryptamine uptake inhibitor with IC50 value of 0.013 …
Formula:
C19H20ClFN2O
Purity:
96.14%
Color and Shape:
Liquid
Molecular weight:
346.83
Ref: TM-T67851
| 1mg | 95.00 € | ||
| 5mg | 413.00 € | ||
| 10mg | 509.00 € | ||
| 25mg | 810.00 € | ||
| 50mg | 1,112.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
KSK67
CAS:2566715-93-1
KSK67 is a selective dual antagonist of sigma-2 and histamine H3 receptors with inhibitory effects …
Formula:
C22H27N3O2
Purity:
99.11%
Color and Shape:
Soild
Molecular weight:
365.47
Ref: TM-T77593
| 1mg | 73.00 € | ||
| 5mg | 158.00 € | ||
| 10mg | 226.00 € | ||
| 25mg | 456.00 € | ||
| 50mg | 785.00 € | ||
| 100mg | 1,355.00 € | ||
| 500mg | 2,732.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
SB 258585
CAS:209480-63-7
SB 258585: Selective 5-HT6 antagonist, binds human receptors, used in cognitive and antipsychotic assays.
Formula:
C18H22IN3O3S
Purity:
99.8%
Color and Shape:
Soild
Molecular weight:
487.36
Ref: TM-T23318L
| 1mg | 48.00 € | ||
| 5mg | 92.00 € | ||
| 10mg | 158.00 € | ||
| 25mg | 272.00 € | ||
| 50mg | 479.00 € | ||
| 100mg | 688.00 € | ||
| 500mg | 1,421.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
H4R antagonist 3
CAS:1003091-20-0
H4R antagonist 3 is a novel histamine-4 receptor (H4R) antagonist with an EC50 <10 mM.H4R …
Formula:
C19H21ClN4S
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
372.92
Ref: TM-T77715
| 1mg | 183.00 € | ||
| 5mg | 452.00 € | ||
| 10mg | 648.00 € | ||
| 25mg | 1,011.00 € | ||
| 50mg | 1,394.00 € | ||
| 100mg | 1,843.00 € | ||
| 500mg | 3,676.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
D3R/MOR antagonist 2
Compound 121, a D3R/MOR antagonist with K i values of 361 nM and 85.2 nM …
Formula:
C25H31ClN2O
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
410.98
Ref: TM-T78779
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Desmethyl cariprazine
CAS:839712-15-1
Desmethyl cariprazine is a Cariprazine active metabolite. Cariprazine, an antipsychotic drug candidate, shows a high …
Formula:
C20H30Cl2N4O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
413.38
Ref: TM-T15100
| 100mg | To inquire | ||
| 500mg | To inquire |
Estimated delivery in United States, on Wednesday 11 Dec 2024
UFP-101 acetate
UFP-101 acetate is a selective and competitive antagonist of the NOP receptor (pKi = 10.24) …
Formula:
C84H142N32O23
Purity:
95.92%
Color and Shape:
Solid
Molecular weight:
1968.23
Ref: TM-TP2105L
| 1mg | 295.00 € | ||
| 2mg | 532.00 € | ||
| 5mg | 833.00 € | ||
| 10mg | 1,142.00 € | ||
| 25mg | 1,691.00 € | ||
| 50mg | 2,284.00 € | ||
| 100mg | 3,056.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Galanin-Like Peptide (porcine)
CAS:245114-96-9
Galanin-Like Peptide (porcine) is a 60 amino acid neuropeptide originally isolated from the porcine hypothalamus.
Formula:
C281H443N81O78
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
6204.02
Ref: TM-T80145
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 11 Dec 2024
PG 931 acetate
PG 931 acetate is a potent agonist of melanocortin 4 (MC4) receptors.
Formula:
C61H89N15O13
Purity:
98.74%
Color and Shape:
Liquid
Molecular weight:
1240.45
Ref: TM-TP1953L
| 1mg | 399.00 € | ||
| 5mg | 898.00 € | ||
| 10mg | 1,218.00 € | ||
| 25mg | 1,813.00 € | ||
| 50mg | 2,446.00 € | ||
| 100mg | 3,290.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
CP 866087
CAS:519052-02-9
CP 866087 is an opioid receptor antagonist for the study of female sexual dysfunction.
Formula:
C24H30N2O3S
Purity:
99.28% - 99.52%
Color and Shape:
Solid
Molecular weight:
426.57
Ref: TM-T31081L
| 1mg | 183.00 € | ||
| 5mg | 452.00 € | ||
| 10mg | 647.00 € | ||
| 25mg | 1,010.00 € | ||
| 50mg | 1,393.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
ITIC
CAS:1664293-06-4
"ITIC, a non-fullerene acceptor with high Tg of 180°C, shows excellent thermal stability and a …
Formula:
C94H82N4O2S4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1427.96
Ref: TM-T19386
| 25mg | 1,435.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Evofolin B
CAS:1961305-60-1
Evofolin B is a natural compound isolated from the stem bark of Zanthoxylum ailanthoides.
Formula:
C17H18O6
Purity:
98%
Color and Shape:
Solid
Molecular weight:
318.32
Ref: TM-TN2408
| 5mg | 3,360.00 € | ||
| 1mL*10mM (DMSO) | 4,037.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
AC-263093
CAS:849459-86-5
AC-263093 is an NPFFR2 agonist with anxiolytic activity that increases c-Fos protein expression in the …
Formula:
C8H8Br2N4
Purity:
99.78%
Color and Shape:
Soild
Molecular weight:
319.98
Ref: TM-T83651
| 5mg | 47.00 € | ||
| 10mg | 69.00 € | ||
| 25mg | 124.00 € | ||
| 50mg | 193.00 € | ||
| 100mg | 305.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
AD186
AD186, a potent and selective S1R agonist, exhibits dissociation constants (Kis) of 2.7 nM for …
Formula:
C22H28N2
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
320.47
Ref: TM-T78915
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Nelivaptan
CAS:439687-69-1
Nelivaptan (SR 149415) is a vasopressin V1b receptor antagonist that can eliminate CHS-induced GE damage.Cost-effective …
Formula:
C30H32ClN3O8S
Purity:
98% - 98.39%
Color and Shape:
Solid
Molecular weight:
630.11
Ref: TM-T28153
| 1mg | 77.00 € | ||
| 5mg | 147.00 € | ||
| 10mg | 205.00 € | ||
| 25mg | 343.00 € | ||
| 50mg | 508.00 € | ||
| 100mg | 730.00 € | ||
| 500mg | 1,514.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Neurokinin B acetate(86933-75-7 free base)
Neurokinin B acetate, a tachykinin, interacts with NK1R, NK2R, & NK3R receptors to exert biological …
Formula:
C57H83N13O16S2
Purity:
98.53%
Color and Shape:
Solid
Molecular weight:
1270.48
Ref: TM-TP1363L
| 1mg | 86.00 € | ||
| 5mg | 309.00 € | ||
| 10mg | 552.00 € | ||
| 25mg | 880.00 € | ||
| 50mg | 1,196.00 € | ||
| 100mg | 1,616.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
