G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Arotinolol hydrochloride
CAS:68377-91-3
Arotinolol HCl is a non-selective α/β-blocker, anti-hypertensive, anti-obesity, and improves aortic stiffness.
Formula:
C15H22ClN3O2S3
Purity:
99.84%
Color and Shape:
Solid
Molecular weight:
408
Ref: TM-T30140
| 1mg | 52.00 € | ||
| 5mg | 104.00 € | ||
| 10mg | 157.00 € | ||
| 25mg | 250.00 € | ||
| 50mg | 366.00 € | ||
| 100mg | 546.00 € | ||
| 500mg | 1,161.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Tolamolol
CAS:38103-61-6
Tolamolol is a selective β-adrenergic blocker that significantly reduces the degree of exercise-induced inhibition of …
Formula:
C19H24N2O4
Purity:
97.58%
Color and Shape:
Solid
Molecular weight:
344.4
Ref: TM-T68164
| 1mg | 101.00 € | ||
| 5mg | 186.00 € | ||
| 10mg | 260.00 € | ||
| 25mg | 470.00 € | ||
| 50mg | 613.00 € | ||
| 100mg | 910.00 € | ||
| 500mg | 1,831.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Tienoxolol FA
Tienoxolol FA, a beta-blocker for treating heart disease, hypertension, and ischemia.
Formula:
C22H30N2O7S
Purity:
97.05% - 99.47%
Color and Shape:
Soild
Molecular weight:
466.55
Ref: TM-T68161L
| 1mg | 182.00 € | ||
| 5mg | 401.00 € | ||
| 10mg | 591.00 € | ||
| 25mg | 917.00 € | ||
| 50mg | 1,263.00 € | ||
| 100mg | 1,700.00 € | ||
| 500mg | 3,415.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
CB2R/FAAH modulator-3
CAS:2876918-67-9
CB2R/FAAH modulator-3 (compound 27) is a modulator targeting at CB2R and FAAH.
Formula:
C22H31NO2
Purity:
99.02%
Color and Shape:
Soild
Molecular weight:
341.49
Ref: TM-T67747
| 1mg | 45.00 € | ||
| 1ml | 95.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 135.00 € | ||
| 25mg | 258.00 € | ||
| 50mg | 423.00 € | ||
| 100mg | 625.00 € | ||
| 500mg | 1,328.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Neurokinin B acetate(86933-75-7 free base)
Neurokinin B acetate, a tachykinin, interacts with NK1R, NK2R, & NK3R receptors to exert biological …
Formula:
C57H83N13O16S2
Purity:
98.53%
Color and Shape:
Solid
Molecular weight:
1270.48
Ref: TM-TP1363L
| 1mg | 86.00 € | ||
| 5mg | 309.00 € | ||
| 10mg | 552.00 € | ||
| 25mg | 880.00 € | ||
| 50mg | 1,196.00 € | ||
| 100mg | 1,616.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
S1PR1 modulator 1
CAS:2328109-05-1
S1PR1 modulator 1 is a selective inhibitor of S1PR1 with a pIC50 of 7.6.
Formula:
C23H24N2O3S
Purity:
99.44%
Color and Shape:
Solid
Molecular weight:
408.51
Ref: TM-T12821
| 1mg | 64.00 € | ||
| 1ml | 138.00 € | ||
| 5mg | 118.00 € | ||
| 10mg | 167.00 € | ||
| 25mg | 267.00 € | ||
| 50mg | 394.00 € | ||
| 100mg | 584.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
L-796,778 acetate
L-796,778 acetate is a slective somatostatin receptor agonist with IC50 of 24nM for sst3, for …
Formula:
C31H44N6O9
Purity:
98%
Color and Shape:
Soild
Molecular weight:
644.72
Ref: TM-T32511L
| 1mg | 185.00 € | ||
| 5mg | 422.00 € | ||
| 10mg | 637.00 € | ||
| 25mg | 1,089.00 € | ||
| 50mg | 1,630.00 € | ||
| 100mg | 2,449.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Invopressin
CAS:1488411-60-4
Invopressin (Compound 42), a vasopressin V1A receptor partial agonist (EC50: 1.0 nM), is utilized in …
Formula:
C110H161N31O27S2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
2413.78
Ref: TM-T80270
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
PACAP (6-27) (human, chicken, mouse, ovine, porcine, rat) (trifluoroacetate salt)
PACAP (6-27) is an antagonist for PACAP receptors with varying IC50s; blocks cAMP in neuroblastoma …
Ref: TM-T36427
| 500µg | 422.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Vasopressin Dimer (parallel) (TFA)
Vasopressin Dimer (parallel) TFA, a parallel dimer of Vasopressin, has the capability to activate four …
Formula:
C94H131F3N30O26S4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
2282.49
Ref: TM-T80197
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
![[D-Ala2]leucine-enkephalin acetate](https://static.cymitquimica.com/products/TM/thumb/TP1367L.jpg)
[D-Ala2]leucine-enkephalin acetate
[D-Ala2]leucine-enkephalin acetate ([D-Ala2]leucine-enkephalin acetate (64963-01-5 free base)) is a delta opioid agonist used to study …
Formula:
C31H43N5O9
Purity:
98%
Color and Shape:
Solid
Molecular weight:
629.65
Ref: TM-TP1367L
| 5mg | 55.00 € | ||
| 10mg | 66.00 € | ||
| 25mg | 99.00 € | ||
| 50mg | 160.00 € | ||
| 100mg | 232.00 € | ||
| 200mg | 349.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Cericlamine
CAS:112922-55-1
Cericlamine is a selective 5-hydroxytryptamine (5-HT) reuptake blocker with antidepressant activity.
Formula:
C12H17Cl2NO
Purity:
98.57%
Color and Shape:
Solid
Molecular weight:
262.18
Ref: TM-T68040
| 1mg | 125.00 € | ||
| 5mg | 299.00 € | ||
| 10mg | 446.00 € | ||
| 25mg | 730.00 € | ||
| 50mg | 1,003.00 € | ||
| 100mg | 1,380.00 € | ||
| 500mg | 2,759.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
EP3 antagonist 4
CAS:2408297-80-1
EP3 antagonist 4: hEP inhibitor, Ki = 2 nM, low clearance, high oral AUC, good …
Formula:
C22H20Cl3FN4O3S2
Purity:
98%
Color and Shape:
Soild
Molecular weight:
577.91
Ref: TM-T77630
| 1mg | 184.00 € | ||
| 5mg | 405.00 € | ||
| 10mg | 612.00 € | ||
| 25mg | 1,044.00 € | ||
| 50mg | 1,580.00 € | ||
| 100mg | 2,388.00 € | ||
| 500mg | 5,254.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Cortistatin-8 acetate
Cortistatin-8 acetate: synthetic corticosteroid analog, GHS-R antagonist; doesn't affect acyl GH release or hesperidin response.
Formula:
C49H72N12O11S2
Purity:
99.01%
Color and Shape:
Soild
Molecular weight:
1069.3
Ref: TM-TP2236L
| 1mg | 223.00 € | ||
| 5mg | 548.00 € | ||
| 10mg | 783.00 € | ||
| 25mg | 1,189.00 € | ||
| 50mg | 1,613.00 € | ||
| 100mg | 2,172.00 € | ||
| 500mg | 4,353.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Galanin-Like Peptide (rat)
CAS:245114-97-0
Galanin-Like Peptide (rat), a neuropeptide comprising 60 amino acids, plays a crucial role in regulating …
Formula:
C288H461N87O83S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
6502.34
Ref: TM-T80146
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
PACAP-related Peptide (human) (trifluoroacetate salt)
Endogenous 29-amino acid PRP belongs to secretin/glucagon family, found in pancreas, adrenal glands, and some …
Ref: TM-T36428
| 1mg | 839.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Gancaonin I
CAS:126716-36-7
Gancaonin I exhibits anti-BsFtsZ GTPase activities; it also shows significant inhibitory activity against B. subtilis, …
Formula:
C21H22O5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
354.4
Ref: TM-TN4098
| 1ml | 2,349.00 € | ||
| 5mg | 1,879.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
LHRH
CAS:35263-73-1
Luteinizing hormone-releasing hormone (LHRH) is a neuropeptide produced in the hypothalamus that plays a pivotal …
Formula:
C55H74N16O14
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1183.27
Ref: TM-T80116
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
(Iso)-Landipirdine
CAS:1000308-09-7
(Iso)-Landipirdine((Iso)-RO5025181) is a selective and potent 5-HT6R antagonist.
Formula:
C18H19FN2O3S
Purity:
97.27%
Color and Shape:
Soild
Molecular weight:
362.42
Ref: TM-T27795L
| 1mg | 182.00 € | ||
| 5mg | 449.00 € | ||
| 10mg | 643.00 € | ||
| 25mg | 1,003.00 € | ||
| 50mg | 1,384.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
CYM 50769
CAS:1421365-63-0
CYM 50769 is a neuropeptide W/B receptor 1 (NPBWR1, GPR7) antagonist(IC50 = 0.12 μM).
Formula:
C24H17ClN2O3
Purity:
98% - 98.76%
Color and Shape:
Solid
Molecular weight:
416.86
Ref: TM-T22702
| 1mg | 52.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 171.00 € | ||
| 25mg | 369.00 € | ||
| 50mg | 551.00 € | ||
| 100mg | 783.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
