G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Cholecystokinin (26-33) free acid
CAS:103974-46-5
Cholecystokinin (26-33) free acid is part of CCK and induces mild taste aversion conditioning in …
Formula:
C49H61N9O14S2
Purity:
99.14%
Color and Shape:
Soild
Molecular weight:
1064.19
Ref: TM-TP2500
| 1mg | 48.00 € | ||
| 5mg | 93.00 € | ||
| 10mg | 141.00 € | ||
| 25mg | 226.00 € | ||
| 50mg | 339.00 € | ||
| 100mg | 502.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
7-Desmethyl-3-hydroxyagomelatine
CAS:166527-00-0
7-Desmethyl-3-hydroxyagomelatine, less active than parent drug Agomelatine, is a melatonergic agonist and 5-HT2C antagonist.
Formula:
C14H15NO3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
245.27
Ref: TM-T10192
| 100mg | To inquire | ||
| 500mg | To inquire |
Estimated delivery in United States, on Wednesday 11 Dec 2024
SphK1&2-IN-1
CAS:1415662-57-5
SphK1&2-IN-1 is a sphingosine kinase inhibitor with anti-inflammatory, antitumor and hemostatic effects.
Formula:
C14H14N2O3S
Purity:
99.27%
Color and Shape:
Liquid
Molecular weight:
290.34
Ref: TM-T9992
| 1mg | 44.00 € | ||
| 5mg | 97.00 € | ||
| 10mg | 134.00 € | ||
| 25mg | 250.00 € | ||
| 50mg | 359.00 € | ||
| 100mg | 477.00 € | ||
| 200mg | 636.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
2'-Hydroxydaidzein
CAS:7678-85-5
2'-Hydroxydaidzein is an isoflavonoid phytonutrient found in plant species, when a natural compound. 2'-Hydroxydaidzein has …
Formula:
C15H10O5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
270.24
Ref: TM-TN2766
| 1mg | To inquire |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Prostaglandin F2α 1,11-lactone
CAS:62410-84-8
Prostaglandin F2α 1,11-lactone (PGF2α 1,11-lactone) is a lipid-soluble prodrug of Prostaglandin F2α and can be …
Formula:
C20H32O4
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
336.47
Ref: TM-T37326
| 10mg | 1,613.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Urocortin (rat) acetate
Urocortin (rat) acetate: CRF receptor agonist; Ki=13nM (hCRF1), 1.5nM (rCRF2α), 0.97nM (mCRF2β); neuropeptide.
Purity:
97.76%
Color and Shape:
Soild
Ref: TM-TP1020L
| 1mg | 154.00 € | ||
| 5mg | 369.00 € | ||
| 10mg | 526.00 € | ||
| 25mg | 774.00 € | ||
| 50mg | 1,056.00 € | ||
| 100mg | 1,429.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
A3AR agonist 1
A3AR Agonist 1 (Compound 12), with a Ki of 25.8 nM, is a potent A3 …
Formula:
C28H34N6O6
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
550.61
Ref: TM-T79372
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Lys-(Des-Arg9,Leu8)-Bradykinin
CAS:71800-37-8
Lys-(Des-Arg9,Leu8)-Bradykinin is a selective antagonist of the bradykinin B1 receptor [1].
Formula:
C47H75N13O11
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
998.18
Ref: TM-T80117
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 11 Dec 2024
CB2R/FAAH modulator-2
CAS:2876918-68-0
CB2R/FAAH modulator-2 (compound 26) is a dual modulator targeting at CB2R and FAAH.
Formula:
C24H33NO2
Purity:
99.52%
Color and Shape:
Soild
Molecular weight:
367.52
Ref: TM-T67745
| 1mg | 36.00 € | ||
| 5mg | 79.00 € | ||
| 10mg | 120.00 € | ||
| 25mg | 188.00 € | ||
| 50mg | 282.00 € | ||
| 100mg | 430.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
SB 216641
CAS:170230-39-4
SB 216641 is a 5-HT (1B/1D) antagonist with anxiolytic activity for the study of anxiety …
Formula:
C28H30N4O4
Purity:
98.01%
Color and Shape:
Liquid
Molecular weight:
486.56
Ref: TM-T85323
| 1mg | 196.00 € | ||
| 5mg | 486.00 € | ||
| 10mg | 682.00 € | ||
| 25mg | 1,064.00 € | ||
| 50mg | 1,467.00 € | ||
| 100mg | 1,878.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
DPDPE
CAS:88373-73-3
DPDPE is selective δ-opioid receptor agonist peptide.
Formula:
C30H39N5O7S2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
645.79
Ref: TM-TP2036
| 1mg | 376.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Mibenratide TFA
Mibenratide TFA, a small cyclic peptide, functions as an adrenergic β1 receptor antagonist and has …
Purity:
98%
Ref: TM-T81798
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 11 Dec 2024
TDI-10229
CAS:2810887-45-5
TDI-10229: potent oral sAC inhibitor, IC50=195 nM. Good mouse pharmacokinetics for in vivo use.
Formula:
C16H16ClN5
Purity:
97.77%
Color and Shape:
Soild
Molecular weight:
313.78
Ref: TM-T64355
| 1mg | 41.00 € | ||
| 5mg | 159.00 € | ||
| 10mg | 233.00 € | ||
| 25mg | 416.00 € | ||
| 50mg | 625.00 € | ||
| 100mg | 903.00 € | ||
| 200mg | 1,246.00 € | ||
| 1mL*10mM (DMSO) | 171.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
(Leu31,Pro34)-Peptide YY (human) (TFA)
"(Leu31,Pro34)-Peptide YY (human) (TFA) is the trifluoroacetic acid (TFA) form of (Leu31,Pro34)-Peptide YY (human), a …
Formula:
C195H296N54O56·xC2HF3O2
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
4292.75 (free base)
Ref: TM-T80087
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Binospirone
CAS:102908-59-8
Binospirone (MDL 73005EF) is a 5-HT1A receptor agonist with anxiolytic activity used in the study …
Formula:
C20H26N2O4
Purity:
98.05% - 99.11%
Color and Shape:
Soild
Molecular weight:
358.43
Ref: TM-T71138L
| 1mg | 185.00 € | ||
| 5mg | 459.00 € | ||
| 10mg | 657.00 € | ||
| 25mg | 1,025.00 € | ||
| 50mg | 1,413.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Fosopamine(HCl)
CAS:135962-35-5
Fosopamine(HCl) is a DRDs agonist that can be used to study hypertension.
Formula:
C9H15ClNO5P
Purity:
100%
Color and Shape:
Liquid
Molecular weight:
283.65
Ref: TM-T68076L
| 1mg | 95.00 € | ||
| 5mg | 234.00 € | ||
| 10mg | 307.00 € | ||
| 25mg | 547.00 € | ||
| 50mg | 710.00 € | ||
| 100mg | 994.00 € | ||
| 500mg | 1,978.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Ala5-Galanin (2-11)
CAS:859843-84-8
Ala5-Galanin (2-11) is a specific agonist for the galanin receptor 2 (GAL2R) with an affinity …
Formula:
C54H81N13O13
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
1120.3
Ref: TM-T80517
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Propiram fumarate HCl
CAS:945013-73-0
Propiram fumarate HClis an orally available Opioid receptors agonist with analgesic activity for the study …
Formula:
C16H25N3O·xClH
Purity:
99.25%
Color and Shape:
Soild
Ref: TM-T28453L
| 1mg | 183.00 € | ||
| 5mg | 401.00 € | ||
| 10mg | 591.00 € | ||
| 25mg | 916.00 € | ||
| 50mg | 1,271.00 € | ||
| 100mg | 1,710.00 € | ||
| 500mg | 3,416.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
NXT-10796
NXT-10796 is an orally active, intestinally restricted agonist of the EP4 receptor [1].
Formula:
C23H31N3O6
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
445.51
Ref: TM-T79432
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Des His1, Glu8 Exendin-4
Des His1, Glu8 Exendin-4 is a glucagon-like peptide-1 receptor (GLP1R) antagonist that regulates blood glucose …
Formula:
C179H277N47O59S
Color and Shape:
Liquid
Molecular weight:
4063.46
Ref: TM-T76291
| 1mg | 227.00 € | ||
| 5mg | 499.00 € | ||
| 10mg | 747.00 € | ||
| 25mg | 1,268.00 € | ||
| 50mg | 1,902.00 € | ||
| 100mg | 2,564.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
