G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Trimebutine
CAS:39133-31-8
Trimebutine (Mebutin) is a spasmolytic agent that regulates intestinal and colonic motility and relieves abdominal …
Formula:
C22H29NO5
Purity:
98.13% - 99.49%
Color and Shape:
Solid
Molecular weight:
387.47
Ref: TM-T0918
| 1g | 36.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Tegaserod maleate
CAS:189188-57-6
Tegaserod (SDZ-HTF-919), a 5-HT4 agonist for irritable bowel syndrome, was withdrawn by FDA on March …
Formula:
C20H27N5O5
Purity:
98% - 99.06%
Color and Shape:
White Powder
Molecular weight:
417.46
Ref: TM-T1551
| 10mg | 46.00 € | ||
| 25mg | 78.00 € | ||
| 50mg | 118.00 € | ||
| 100mg | 194.00 € | ||
| 200mg | 295.00 € | ||
| 500mg | 497.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Tiapride hydrochloride
CAS:51012-33-0
Tiapride is a selective blocker of D2/3 dopamine receptors in the brain.
Formula:
C15H24N2O4S·HCl
Purity:
98.86% - 99.4%
Color and Shape:
Solid
Molecular weight:
364.89
Ref: TM-T1292
| 50mg | 43.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Deoxycholic acid
CAS:83-44-3
Deoxycholic acid (Cholanoic Acid) is a bile acid formed by bacterial action from cholate.
Formula:
C24H40O4
Purity:
99.35%
Color and Shape:
Crystals From Alc Solid
Molecular weight:
392.57
Ref: TM-T2965
| 100mg | 57.00 € | ||
| 500mg | 78.00 € | ||
| 1mL*10mM (DMSO) | 63.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Protriptyline hydrochloride
CAS:1225-55-4
Protriptyline HCl: a tricyclic antidepressant that increases norepinephrine and serotonin levels and has anticholinergic effects.
Formula:
C19H21N·HCl
Purity:
98.54% - 99.98%
Color and Shape:
Solid
Molecular weight:
299.84
Ref: TM-T0204
| 10mg | 49.00 € | ||
| 25mg | 93.00 € | ||
| 50mg | 153.00 € | ||
| 1mL*10mM (DMSO) | 36.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Paroxetine hydrochloride
CAS:78246-49-8
Paroxetine hydrochloride (Paroxetine HCl) is a serotonin uptake inhibitor that is effective in the treatment …
Formula:
C19H21ClFNO3
Purity:
98% - 99.91%
Color and Shape:
White Crystalline Powder
Molecular weight:
365.826
Ref: TM-T1636
| 25mg | 54.00 € | ||
| 50mg | 63.00 € | ||
| 100mg | 89.00 € | ||
| 200mg | 113.00 € | ||
| 500mg | 153.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Tropisetron hydrochloride
CAS:105826-92-4
Tropisetron hydrochloride (Tropisetron HCl) is a selective, competitive serotonin 5-HT3 receptor antagonist, with antinauseant and …
Formula:
C17H21ClN2O2
Purity:
99.65% - 99.83%
Color and Shape:
Solid
Molecular weight:
320.82
Ref: TM-T1173
| 10mg | 52.00 € | ||
| 25mg | 70.00 € | ||
| 50mg | 88.00 € | ||
| 100mg | 105.00 € | ||
| 200mg | 162.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
N6-Ethyladenosine
CAS:14357-08-5
N6-Ethyladenosine is an adenosine derivative, acts as an agonist of Adenosine receptor(hA1AR and hA3AR with …
Formula:
C12H17N5O4
Purity:
99.96%
Color and Shape:
Solid
Molecular weight:
295.29
Ref: TM-T12161
| 2mg | 34.00 € | ||
| 5mg | 49.00 € | ||
| 10mg | 78.00 € | ||
| 25mg | 126.00 € | ||
| 50mg | 205.00 € | ||
| 100mg | 302.00 € | ||
| 200mg | 435.00 € | ||
| 1mL*10mM (DMSO) | 83.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Amitraz
CAS:33089-61-1
Amitraz (NSC 324552): white monoclinic crystals, mp 86-87°C, water-insoluble, used as acaricide and in canine …
Formula:
C19H23N3
Purity:
99.62%
Color and Shape:
White/Pale Yellow Crystalline Solid
Molecular weight:
293.41
Ref: TM-T1632
| 1g | 87.00 € | ||
| 200mg | 40.00 € | ||
| 500mg | 60.00 € | ||
| 1mL*10mM (DMSO) | 46.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Abarelix
CAS:183552-38-7
Abarelix (PPI 149) is a potent gonadotrophin-releasing hormone (GnRH) antagonist, which is used for prostate …
Formula:
C72H95ClN14O14
Purity:
100%
Color and Shape:
Solid
Molecular weight:
1416.06
Ref: TM-T10217L
| 2mg | 41.00 € | ||
| 5mg | 61.00 € | ||
| 10mg | 96.00 € | ||
| 25mg | 176.00 € | ||
| 50mg | 277.00 € | ||
| 100mg | 424.00 € | ||
| 1mL*10mM (DMSO) | 90.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
AH 6809
CAS:33458-93-4
AH 6809 blocks EP1, EP2, EP3, DP receptors (Ki: 1217-1597 nM human, 350 nM mouse …
Formula:
C17H14O5
Purity:
97.59%
Color and Shape:
Solid
Molecular weight:
298.29
Ref: TM-T14148
| 2mg | 45.00 € | ||
| 5mg | 67.00 € | ||
| 10mg | 87.00 € | ||
| 25mg | 170.00 € | ||
| 50mg | 315.00 € | ||
| 100mg | 506.00 € | ||
| 1mL*10mM (DMSO) | 72.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Betahistine mesylate
CAS:54856-23-4
Betahistine mesylate (Extovyl), an H1 agonist and vasodilator, treats Meniere's disease and vascular headaches; risks …
Formula:
C8H12N2·2(CH4O3S)
Purity:
98%
Color and Shape:
Coa
Molecular weight:
328.4
Ref: TM-T0246L
| 10mg | 35.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Dopexamine hydrochloride
CAS:86484-91-5
Dopexamine hydrochloride (FPL60278AR) is a β2-adrenoceptor agonist that modulates inflammation and protects organs without affecting …
Formula:
C22H34Cl2N2O2
Purity:
98.55%
Color and Shape:
Solid
Molecular weight:
429.42
Ref: TM-T11318
| 1mg | 52.00 € | ||
| 2mg | 74.00 € | ||
| 5mg | 109.00 € | ||
| 10mg | 171.00 € | ||
| 25mg | 346.00 € | ||
| 50mg | 516.00 € | ||
| 100mg | 727.00 € | ||
| 1mL*10mM (DMSO) | 123.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Ethamsylate
CAS:2624-44-4
Ethamsylate (Dicynene) enhances capillary stability, platelet adhesion, and blocks prostaglandins to act as a hemostatic …
Formula:
C10H17NO5S
Purity:
99.98%
Color and Shape:
White Crystals Or Crystalline Powder
Molecular weight:
263.31
Ref: TM-T0002
| 5g | 88.00 € | ||
| 1mL*10mM (DMSO) | 36.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Amiselimod hydrochloride
CAS:942398-84-7
Amiselimod hydrochloride (MT-1303 hydrochloride) is a sphingosine 1-phosphate receptor-1 (S1P1) modulator.
Formula:
C19H31ClF3NO3
Purity:
99.55%
Color and Shape:
Solid
Molecular weight:
413.9
Ref: TM-T10305
| 1mg | 38.00 € | ||
| 5mg | 79.00 € | ||
| 10mg | 118.00 € | ||
| 25mg | 210.00 € | ||
| 50mg | 345.00 € | ||
| 100mg | 499.00 € | ||
| 1mL*10mM (DMSO) | 88.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
EHP-101
CAS:1818428-24-8
EHP-101 is a PPARγ/CB2 dual agonist with anti-inflammatory properties, inhibits fat formation, and combats diet-related …
Formula:
C28H35NO3
Purity:
99.22%
Color and Shape:
Solid
Molecular weight:
433.58
Ref: TM-T13289
| 1mg | 105.00 € | ||
| 5mg | 222.00 € | ||
| 10mg | 369.00 € | ||
| 25mg | 610.00 € | ||
| 50mg | 848.00 € | ||
| 100mg | 1,142.00 € | ||
| 1mL*10mM (DMSO) | 249.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Dapoxetine hydrochloride
CAS:129938-20-1
Dapoxetine hydrochloride (LY-210448 hydrochloride) is a selectivity short-acting serotonin reuptake inhibitor, used for the therapy …
Formula:
C21H23NO·HCl
Purity:
100% - 99%
Color and Shape:
White To Off-White Crystalline Solid
Molecular weight:
341.87
Ref: TM-T6461
| 10mg | 35.00 € | ||
| 25mg | 57.00 € | ||
| 50mg | 74.00 € | ||
| 100mg | 99.00 € | ||
| 200mg | 154.00 € | ||
| 500mg | 241.00 € | ||
| 1mL*10mM (DMSO) | 65.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Filorexant
CAS:1088991-73-4
Filorexant (MK-6096) is an orally bioavailable effective and selective reversible antagonist of OX1 and OX2 …
Formula:
C24H25FN4O2
Purity:
99.33%
Color and Shape:
Solid
Molecular weight:
420.48
Ref: TM-T16096
| 1mg | 35.00 € | ||
| 5mg | 73.00 € | ||
| 10mg | 113.00 € | ||
| 25mg | 183.00 € | ||
| 50mg | 276.00 € | ||
| 100mg | 404.00 € | ||
| 1mL*10mM (DMSO) | 81.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
VUF11207 fumarate
CAS:1785665-61-3
VUF11207 fumarate is an agonist of CXCR7 and a high-potency ligand of CXCR7 (pKi: 8.1).
Formula:
C31H39FN2O8
Purity:
99.5%
Color and Shape:
Solid
Molecular weight:
586.65
Ref: TM-T13324
| 1mg | 42.00 € | ||
| 2mg | 55.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 135.00 € | ||
| 25mg | 270.00 € | ||
| 50mg | 467.00 € | ||
| 100mg | 672.00 € | ||
| 200mg | 934.00 € | ||
| 1mL*10mM (DMSO) | 96.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Olodaterol
CAS:868049-49-4
Olodaterol is a novel, long-acting beta2-adrenergic agonist (LABA) that exerts its pharmacological effect by binding …
Formula:
C21H26N2O5
Purity:
98.9%
Color and Shape:
Solid
Molecular weight:
386.45
Ref: TM-T3457
| 1mg | 50.00 € | ||
| 5mg | 87.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
