G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Ticagrelor
CAS:274693-27-5
Ticagrelor (AR-C 126532XX), produced by AstraZeneca, is an inhibitor of platelet aggregation.
Formula:
C23H28F2N6O4S
Purity:
100%
Color and Shape:
Solid
Molecular weight:
522.57
Ref: TM-T0179
| 1g | 364.00 € | ||
| 10mg | 48.00 € | ||
| 25mg | 66.00 € | ||
| 50mg | 81.00 € | ||
| 100mg | 109.00 € | ||
| 200mg | 154.00 € | ||
| 500mg | 245.00 € | ||
| 1mL*10mM (DMSO) | 59.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Phentolamine mesylate
CAS:65-28-1
Phentolamine mesylate: nonselective alpha-blocker for hypertension, pheochromocytoma, Raynaud's, frostbite, impotence, and vascular issues.
Formula:
C17H19N3O·CH4O3S
Purity:
99.77% - 99.9%
Color and Shape:
By The Metabolic Processes Of Bacillus Subtilis And Licheniformis
Molecular weight:
377.46
Ref: TM-T1275
| 100mg | 56.00 € | ||
| 200mg | 73.00 € | ||
| 500mg | 150.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Rimonabant
CAS:168273-06-1
Rimonabant (SR141716) is an inverse agonist for the cannabinoid receptor CB1.
Formula:
C22H21Cl3N4O
Purity:
98% - 99.91%
Color and Shape:
White Or Almost White Crystalline Powder
Molecular weight:
463.79
Ref: TM-T1519L
| 10mg | 49.00 € | ||
| 25mg | 90.00 € | ||
| 50mg | 130.00 € | ||
| 100mg | 187.00 € | ||
| 1mL*10mM (DMSO) | 59.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Nicergoline
CAS:27848-84-6
Nicergoline (Nicergolinum) is an ergot derivative used to treat senile dementia and other disorders with …
Formula:
C24H26BrN3O3
Purity:
100% - 99.53%
Color and Shape:
Solid
Molecular weight:
484.39
Ref: TM-T1132
| 5mg | 35.00 € | ||
| 10mg | 51.00 € | ||
| 25mg | 67.00 € | ||
| 50mg | 85.00 € | ||
| 100mg | 104.00 € | ||
| 200mg | 145.00 € | ||
| 500mg | 234.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
LY2510924 acetate(1088715-84-7 free base)
Ly2510924 acetate is an potent and selective CXCR4 antagonist. It prevents the binding of SDF-1 …
Formula:
C64H91N13O13
Purity:
97.32%
Color and Shape:
Solid
Molecular weight:
1250.49
Ref: TM-T15805L
| 1mg | 159.00 € | ||
| 5mg | 306.00 € | ||
| 10mg | 459.00 € | ||
| 25mg | 750.00 € | ||
| 50mg | 1,026.00 € | ||
| 100mg | 1,415.00 € | ||
| 1mL*10mM (DMSO) | 730.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
CYM50308
CAS:1345858-76-5
CYM50308 is a high affinity agonist of sphingosine-1-phosphate receptor 4 (S1P4-R) (EC50: 56 nM).
Formula:
C20H21F2N3O2S
Purity:
99.43% - 99.63%
Color and Shape:
Solid
Molecular weight:
405.46
Ref: TM-T15032
| 1mg | 62.00 € | ||
| 5mg | 140.00 € | ||
| 10mg | 202.00 € | ||
| 25mg | 324.00 € | ||
| 50mg | 455.00 € | ||
| 100mg | 597.00 € | ||
| 200mg | 842.00 € | ||
| 500mg | 1,225.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Fexofenadine hydrochloride
CAS:138452-21-8
Fexofenadine Hydrochloride is a carboxylated metabolic derivative of terfenadine and long-lasting selective histamine H1 receptor …
Formula:
C32H40ClNO4
Purity:
100%
Color and Shape:
White Crystalline Powder
Molecular weight:
538.12
Ref: TM-T1470L
| 10mg | 50.00 € | ||
| 25mg | 74.00 € | ||
| 50mg | 105.00 € | ||
| 100mg | 140.00 € | ||
| 200mg | 190.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Acetophenazine dimaleate
CAS:5714-00-1
Acetophenazine dimaleate is an antipsychotic agent, effective in anxious depression. Acetophenazine dimaleate primarily targets the …
Formula:
C31H37N3O10S
Purity:
99.39% - 99.48%
Color and Shape:
Solid
Molecular weight:
643.71
Ref: TM-T10232
| 2mg | 42.00 € | ||
| 5mg | 59.00 € | ||
| 10mg | 85.00 € | ||
| 25mg | 127.00 € | ||
| 50mg | 183.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Motixafortide TFA(664334-36-5,Free)
Motixafortide TFA is a CXCR4 antagonist with ~1 nM IC50, promoting AML apoptosis by modulating …
Formula:
C99H145F4N33O21S2
Purity:
100%
Color and Shape:
Solid
Molecular weight:
2273.54
Ref: TM-T14665L
| 1mg | 74.00 € | ||
| 5mg | 188.00 € | ||
| 10mg | 283.00 € | ||
| 25mg | 452.00 € | ||
| 50mg | 638.00 € | ||
| 100mg | 848.00 € | ||
| 200mg | 1,121.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Granisetron hydrochloride
CAS:107007-99-8
Granisetron hydrochloride (Granisetron HCl) is a serotonin receptor (5HT-3 selective) antagonist that has been used …
Formula:
C18H25ClN4O
Purity:
99.88% - 99.94%
Color and Shape:
White To Off-White Crystalline Solid
Molecular weight:
348.87
Ref: TM-T1042
| 10mg | 38.00 € | ||
| 25mg | 56.00 € | ||
| 50mg | 81.00 € | ||
| 100mg | 127.00 € | ||
| 200mg | 178.00 € | ||
| 500mg | 304.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Amitraz
CAS:33089-61-1
Amitraz (NSC 324552): white monoclinic crystals, mp 86-87°C, water-insoluble, used as acaricide and in canine …
Formula:
C19H23N3
Purity:
99.62%
Color and Shape:
White/Pale Yellow Crystalline Solid
Molecular weight:
293.41
Ref: TM-T1632
| 1g | 52.00 € | ||
| 500mg | 39.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Fluvoxamine maleate
CAS:61718-82-9
Fluvoxamine maleate (DU-23000 (maleate)) is a selective serotonin reuptake inhibitor that is used in the …
Formula:
C19H25F3N2O6
Purity:
99.92% - 99.94%
Color and Shape:
White Crystalline Powder
Molecular weight:
434.41
Ref: TM-T1077
| 10mg | 51.00 € | ||
| 25mg | 69.00 € | ||
| 50mg | 85.00 € | ||
| 100mg | 115.00 € | ||
| 200mg | 170.00 € | ||
| 500mg | 278.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Isoxsuprine hydrochloride
CAS:579-56-6
Isoxsuprine hydrochloride (Isolait) is a beta-adrenergic agonist that causes direct relaxation of uterine and vascular …
Formula:
C18H24ClNO3
Purity:
99.31%
Color and Shape:
Crystals From Water Solid
Molecular weight:
337.84
Ref: TM-T0324
| 200mg | 35.00 € | ||
| 500mg | 51.00 € | ||
| 1mL*10mM (DMSO) | 39.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Amiselimod hydrochloride
CAS:942398-84-7
Amiselimod hydrochloride (MT-1303 hydrochloride) is a sphingosine 1-phosphate receptor-1 (S1P1) modulator.
Formula:
C19H31ClF3NO3
Purity:
99.55%
Color and Shape:
Solid
Molecular weight:
413.9
Ref: TM-T10305
| 1mg | 38.00 € | ||
| 5mg | 80.00 € | ||
| 10mg | 120.00 € | ||
| 25mg | 215.00 € | ||
| 50mg | 354.00 € | ||
| 100mg | 512.00 € | ||
| 1mL*10mM (DMSO) | 88.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Protriptyline hydrochloride
CAS:1225-55-4
Protriptyline HCl: a tricyclic antidepressant that increases norepinephrine and serotonin levels and has anticholinergic effects.
Formula:
C19H21N·HCl
Purity:
98.54% - 99.98%
Color and Shape:
Solid
Molecular weight:
299.84
Ref: TM-T0204
| 5mg | 34.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Filorexant
CAS:1088991-73-4
Filorexant (MK-6096) is an orally bioavailable effective and selective reversible antagonist of OX1 and OX2 …
Formula:
C24H25FN4O2
Purity:
99.33%
Color and Shape:
Solid
Molecular weight:
420.48
Ref: TM-T16096
| 1mg | 35.00 € | ||
| 5mg | 74.00 € | ||
| 10mg | 116.00 € | ||
| 25mg | 188.00 € | ||
| 50mg | 284.00 € | ||
| 100mg | 415.00 € | ||
| 1mL*10mM (DMSO) | 84.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Midodrine hydrochloride
CAS:3092-17-9
Midodrine, metabolized to desglymidodrine, activates alpha-1 receptors, raising blood pressure without CNS effects. It's a …
Formula:
C12H19ClN2O4
Purity:
99.06% - 99.36%
Color and Shape:
Crystalline Solid
Molecular weight:
290.74
Ref: TM-T1577
| 5mg | 47.00 € | ||
| 10mg | 70.00 € | ||
| 25mg | 126.00 € | ||
| 50mg | 183.00 € | ||
| 100mg | 273.00 € | ||
| 1mL*10mM (DMSO) | 50.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Diphenylpyraline hydrochloride
CAS:132-18-3
Diphenylpyraline hydrochloride treats Parkinsonism. It's an antihistamine with anticholinergic properties and inhibits dopamine reuptake.
Formula:
C19H23NO·HCl
Purity:
99.22%
Color and Shape:
Solid
Molecular weight:
317.85
Ref: TM-T0059
| 500mg | 35.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Ritodrine hydrochloride
CAS:23239-51-2
Ritodrine hydrochloride (NSC 291565), a phenethylamine derivative, reduces uterine contractions by increasing cAMP and decreasing …
Formula:
C17H21NO3·HCl
Purity:
99% - 99.89%
Color and Shape:
Solid
Molecular weight:
323.82
Ref: TM-T1433
| 1g | 52.00 € | ||
| 200mg | 35.00 € | ||
| 500mg | 42.00 € | ||
| 1mL*10mM (DMSO) | 35.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
CB1 antagonist 2
CAS:614726-85-1
CB1 antagonist 2 (AM4113) is caimabinoid 1 (CB1) antagonist which inhibits CB1 in vivo with …
Formula:
C17H12Cl3N3O
Purity:
99.75%
Color and Shape:
Solid
Molecular weight:
380.66
Ref: TM-T14881
| 2mg | 35.00 € | ||
| 5mg | 52.00 € | ||
| 10mg | 80.00 € | ||
| 25mg | 145.00 € | ||
| 50mg | 250.00 € | ||
| 100mg | 406.00 € | ||
| 500mg | 919.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
