G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Solabegron
CAS:252920-94-8
Solabegron (GW 427353) is a selective agonist of β3-adrenergic receptor, stimulating cAMP accumulation in Chinese …
Formula:
C23H23ClN2O3
Purity:
98.99%
Color and Shape:
Solid
Molecular weight:
410.89
Ref: TM-T12970
| 1mg | 96.00 € | ||
| 1ml | 281.00 € | ||
| 5mg | 259.00 € | ||
| 10mg | 423.00 € | ||
| 25mg | 769.00 € | ||
| 50mg | 1,041.00 € | ||
| 100mg | 1,392.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
hGPR91 antagonist 1
CAS:1314796-00-3
hGPR91 antagonist 1 is a potent and selective hGPR91 antagonist (IC50: 7 μM).
Formula:
C31H23F4N3O
Purity:
98.89%
Color and Shape:
Solid
Molecular weight:
529.53
Ref: TM-T11560
| 1mg | 94.00 € | ||
| 1ml | 221.00 € | ||
| 5mg | 199.00 € | ||
| 10mg | 293.00 € | ||
| 25mg | 495.00 € | ||
| 50mg | 676.00 € | ||
| 100mg | 916.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Labetalol
CAS:36894-69-6
Labetalol: mixed alpha/beta blocker for hypertension, oral or IV; affected by CYP2C19 genetics.
Formula:
C19H24N2O3
Purity:
99.87% - 99.89%
Color and Shape:
Solid
Molecular weight:
328.41
Ref: TM-T20570
| 1ml | 47.00 € | ||
| 10mg | 46.00 € | ||
| 25mg | 78.00 € | ||
| 50mg | 109.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
JNJ-18038683
CAS:851376-05-1
JNJ-18038683 is a 5-Hydroxytryptamine Type 7 (5-HT7) receptor antagonist, with pKis of 8.19, 8.20 for …
Formula:
C26H28ClN3O7
Purity:
98.31%
Color and Shape:
Solid
Molecular weight:
529.97
Ref: TM-T11720
| 1mg | 39.00 € | ||
| 1ml | 92.00 € | ||
| 2mg | 50.00 € | ||
| 5mg | 82.00 € | ||
| 10mg | 134.00 € | ||
| 25mg | 270.00 € | ||
| 50mg | 425.00 € | ||
| 100mg | 624.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
JMV 2959 hydrochloride (925238-89-7 free base)
CAS:2448414-54-6
JMV 2959 hydrochloride (925238-89-7 free base) is a growth hormone secretagogue receptor type 1a (GHS-R1a) …
Formula:
C30H33ClN6O2
Purity:
98.09%
Color and Shape:
Solid
Molecular weight:
545.08
Ref: TM-T11719
| 1mg | 41.00 € | ||
| 1ml | 96.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 125.00 € | ||
| 25mg | 258.00 € | ||
| 50mg | 384.00 € | ||
| 100mg | 547.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Tegaserod maleate
CAS:189188-57-6
Tegaserod (SDZ-HTF-919), a 5-HT4 agonist for irritable bowel syndrome, was withdrawn by FDA on March …
Formula:
C20H27N5O5
Purity:
98% - 99.06%
Color and Shape:
White Powder
Molecular weight:
417.46
Ref: TM-T1551
| 1ml | 51.00 € | ||
| 10mg | 46.00 € | ||
| 25mg | 78.00 € | ||
| 50mg | 118.00 € | ||
| 100mg | 194.00 € | ||
| 200mg | 295.00 € | ||
| 500mg | 497.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Paroxetine hydrochloride
CAS:78246-49-8
Paroxetine hydrochloride (Paroxetine HCl) is a serotonin uptake inhibitor that is effective in the treatment …
Formula:
C19H21ClFNO3
Purity:
98% - 99.91%
Color and Shape:
White Crystalline Powder
Molecular weight:
365.826
Ref: TM-T1636
| 1ml | 55.00 € | ||
| 25mg | 54.00 € | ||
| 50mg | 63.00 € | ||
| 100mg | 89.00 € | ||
| 200mg | 113.00 € | ||
| 500mg | 153.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Dipivefrin hydrochloride
CAS:64019-93-8
Dipivefrin hydrochloride (Dipivefrin HCl) that is available as an ophthalmic solution is a prodrug of …
Formula:
C19H27NO5·HCl
Purity:
99.22% - 99.92%
Color and Shape:
Less Gas With A Sweet Odor Colorless Gas With A Sweet Odor
Molecular weight:
387.9
Ref: TM-T0103
| 1ml | 34.00 € | ||
| 10mg | 46.00 € | ||
| 25mg | 51.00 € | ||
| 50mg | 82.00 € | ||
| 100mg | 112.00 € | ||
| 200mg | 169.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Aripiprazole
CAS:129722-12-9
Aripiprazole (OPC-14597) is a piperazine/quinolone antipsychotic, partial agonist at 5-HT1A/D2, and antagonist at 5-HT2A.
Formula:
C23H27Cl2N3O2
Purity:
99.43% - 99.62%
Color and Shape:
Colourless Flake Crystalline Solid
Molecular weight:
448.39
Ref: TM-T1566
| 1g | 130.00 € | ||
| 1ml | 55.00 € | ||
| 100mg | 63.00 € | ||
| 200mg | 82.00 € | ||
| 500mg | 99.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Alfuzosin hydrochloride
CAS:81403-68-1
Alfuzosin hydrochloride (Alfuzosin HCl) is an α1 adrenergic receptor antagonist. It applies to treat benign …
Formula:
C19H27N5O4·HCl
Purity:
99.61%
Color and Shape:
White To Off-White Solid
Molecular weight:
425.91
Ref: TM-T0091
| 1ml | 49.00 € | ||
| 5mg | 45.00 € | ||
| 10mg | 68.00 € | ||
| 25mg | 106.00 € | ||
| 50mg | 171.00 € | ||
| 100mg | 246.00 € | ||
| 500mg | 601.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Betahistine mesylate
CAS:54856-23-4
Betahistine mesylate (Extovyl), an H1 agonist and vasodilator, treats Meniere's disease and vascular headaches; risks …
Formula:
C8H12N2·2(CH4O3S)
Purity:
98%
Color and Shape:
Coa
Molecular weight:
328.4
Ref: TM-T0246L
| 1ml | 51.00 € | ||
| 10mg | 35.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Fluphenazine dihydrochloride
CAS:146-56-5
Fluphenazine dihydrochloride (Prolixin) is an inhibitor of phenothiazine-class D1DR and D2DR. Fluphenazine can be used …
Formula:
C22H28Cl2F3N3OS
Purity:
100%
Color and Shape:
Off-White Solid
Molecular weight:
510.44
Ref: TM-T0068
| 1ml | 55.00 € | ||
| 50mg | 55.00 € | ||
| 100mg | 61.00 € | ||
| 200mg | 86.00 € | ||
| 500mg | 115.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
6-Iodopravadoline
CAS:164178-33-0
6-Iodopravadoline (AM630) is an antagonist of CB2 (Ki: 31.2 nM). And it shows 165-fold selectivity …
Formula:
C23H25IN2O3
Purity:
99.86%
Color and Shape:
Off-White Solid
Molecular weight:
504.36
Ref: TM-T14204
| 1mg | 40.00 € | ||
| 1ml | 104.00 € | ||
| 2mg | 50.00 € | ||
| 5mg | 72.00 € | ||
| 10mg | 94.00 € | ||
| 25mg | 207.00 € | ||
| 50mg | 337.00 € | ||
| 100mg | 539.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Desipramine hydrochloride
CAS:58-28-6
Desipramine hydrochloride (Norimipramine) ,a secondary amine tricyclic antidepressant (TCA), is the hydrochloride salt form of …
Formula:
C18H23ClN2
Purity:
99.58% - 99.94%
Color and Shape:
White To Off-White Powder
Molecular weight:
302.842
Ref: TM-T0991
| 1ml | 36.00 € | ||
| 50mg | 41.00 € | ||
| 100mg | 52.00 € | ||
| 200mg | 66.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Terlipressin Acetate
CAS:1884420-36-3
Terlipressin Acetate, a highly selective vasopressin V1 receptor agonist, on OGD/R-induced damage in intestinal epithelial …
Formula:
C56H82N16O19S2
Purity:
99.69%
Color and Shape:
Solid
Molecular weight:
1347.5
Ref: TM-T13920L
| 5mg | 48.00 € | ||
| 10mg | 60.00 € | ||
| 25mg | 101.00 € | ||
| 50mg | 133.00 € | ||
| 100mg | 203.00 € | ||
| 200mg | 305.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Ethamsylate
CAS:2624-44-4
Ethamsylate (Dicynene) enhances capillary stability, platelet adhesion, and blocks prostaglandins to act as a hemostatic …
Formula:
C10H17NO5S
Purity:
99.98%
Color and Shape:
White Crystals Or Crystalline Powder
Molecular weight:
263.31
Ref: TM-T0002
| 1ml | 41.00 € | ||
| 10mg | 43.00 € | ||
| 25mg | 55.00 € | ||
| 50mg | 72.00 € | ||
| 100mg | 99.00 € | ||
| 200mg | 146.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Dapoxetine hydrochloride
CAS:129938-20-1
Dapoxetine hydrochloride (LY-210448 hydrochloride) is a selectivity short-acting serotonin reuptake inhibitor, used for the therapy …
Formula:
C21H23NO·HCl
Purity:
100% - 99%
Color and Shape:
White To Off-White Crystalline Solid
Molecular weight:
341.87
Ref: TM-T6461
| 1ml | 65.00 € | ||
| 10mg | 35.00 € | ||
| 25mg | 57.00 € | ||
| 50mg | 74.00 € | ||
| 100mg | 99.00 € | ||
| 200mg | 154.00 € | ||
| 500mg | 241.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Fluoxetine hydrochloride
CAS:56296-78-7
Fluoxetine HCl (Lilly110140), a selective serotonin reuptake inhibitor (SSRI), is an antidepressant with fewer side …
Formula:
C17H19ClF3NO
Purity:
99.6% - 99.98%
Color and Shape:
White To Off-White Crystalline Solid White To Off-White Powder
Molecular weight:
345.787
Ref: TM-T0450L
| 1ml | 69.00 € | ||
| 25mg | 57.00 € | ||
| 50mg | 74.00 € | ||
| 100mg | 93.00 € | ||
| 200mg | 148.00 € | ||
| 500mg | 239.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
JP1302 dihydrochloride
CAS:1259314-65-2
JP1302 dihydrochloride: selective α2C-adrenoceptor antagonist; Ki=28 nM, Kb=16 nM.
Formula:
C24H26Cl2N4
Purity:
99.61%
Color and Shape:
Solid
Molecular weight:
441.4
Ref: TM-T11726
| 1mg | 45.00 € | ||
| 1ml | 95.00 € | ||
| 2mg | 59.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 124.00 € | ||
| 25mg | 230.00 € | ||
| 50mg | 370.00 € | ||
| 100mg | 553.00 € | ||
| 500mg | 1,196.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Filorexant
CAS:1088991-73-4
Filorexant (MK-6096) is an orally bioavailable effective and selective reversible antagonist of OX1 and OX2 …
Formula:
C24H25FN4O2
Purity:
99.33%
Color and Shape:
Solid
Molecular weight:
420.48
Ref: TM-T16096
| 1mg | 52.00 € | ||
| 1ml | 123.00 € | ||
| 5mg | 109.00 € | ||
| 10mg | 183.00 € | ||
| 25mg | 308.00 € | ||
| 50mg | 460.00 € | ||
| 100mg | 675.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
