G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Sertraline hydrochloride
CAS:79559-97-0
Sertraline hydrochloride (Sertraline HCl) is a selective serotonin uptake inhibitor that is used in the …
Formula:
C17H18Cl3N
Purity:
99.12% - 99.89%
Color and Shape:
Solid Powder
Molecular weight:
342.691
Ref: TM-T0482
| 5mg | 51.00 € | ||
| 10mg | 63.00 € | ||
| 25mg | 103.00 € | ||
| 50mg | 180.00 € | ||
| 100mg | 235.00 € | ||
| 200mg | 304.00 € | ||
| 500mg | 515.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
CE3F4
CAS:143703-25-7
CE3F4 is a selective antagonist of exchange protein directly activated by cAMP (Epac1; IC50s of …
Formula:
C11H10Br2FNO
Purity:
97.15% - 98.06%
Color and Shape:
Solid
Molecular weight:
351.01
Ref: TM-T12616L
| 5mg | 51.00 € | ||
| 10mg | 88.00 € | ||
| 25mg | 154.00 € | ||
| 50mg | 274.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
Eletriptan hydrobromide
CAS:177834-92-3
Eletriptan hydrobromide (Eletriptan HBr) is an orally active agonist with specific affinity for the 5-hydroxytriptamine1B/1D …
Formula:
C22H27BrN2O2S
Purity:
100% - 99.69%
Color and Shape:
Tan Solid
Molecular weight:
463.43
Ref: TM-T0216
| 2mg | 39.00 € | ||
| 5mg | 57.00 € | ||
| 10mg | 70.00 € | ||
| 25mg | 134.00 € | ||
| 50mg | 235.00 € | ||
| 100mg | 427.00 € | ||
| 200mg | 555.00 € | ||
| 500mg | 890.00 € | ||
| 1mL*10mM (DMSO) | 63.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
Betaxolol hydrochloride
CAS:63659-19-8
Betaxolol HCl (SL 75212) is a cardioselective beta-blocker for hypertension without reported liver injury.
Formula:
C18H30ClNO3
Purity:
99.48% - 99.56%
Color and Shape:
Solid
Molecular weight:
343.89
Ref: TM-T0226
| 25mg | 38.00 € | ||
| 50mg | 50.00 € | ||
| 100mg | 85.00 € | ||
| 200mg | 96.00 € | ||
| 500mg | 159.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
Sumatriptan succinate
CAS:103628-48-4
Sumatriptan succinate (GR 43175), a serotonin1 (5-HT1) receptor agonist, is used in the acute treatment …
Formula:
C18H27N3O6S
Purity:
97.53% - 99.51%
Color and Shape:
White Powder
Molecular weight:
413.49
Ref: TM-T0203
| 25mg | 37.00 € | ||
| 50mg | 52.00 € | ||
| 100mg | 74.00 € | ||
| 500mg | 169.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
Spiperone
CAS:749-02-0
Spiperone (Spiropitan) is a spiro butyrophenone analog similar to HALOPERIDOL and other related compounds.
Formula:
C23H26FN3O2
Purity:
99.34% - 99.89%
Color and Shape:
Solid
Molecular weight:
395.47
Ref: TM-T0280
| 5mg | 47.00 € | ||
| 10mg | 64.00 € | ||
| 25mg | 90.00 € | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
Rimonabant
CAS:168273-06-1
Rimonabant (SR141716) is an inverse agonist for the cannabinoid receptor CB1.
Formula:
C22H21Cl3N4O
Purity:
98% - 99.91%
Color and Shape:
White Or Almost White Crystalline Powder
Molecular weight:
463.79
Ref: TM-T1519L
| 10mg | 49.00 € | ||
| 25mg | 90.00 € | ||
| 50mg | 130.00 € | ||
| 100mg | 187.00 € | ||
| 1mL*10mM (DMSO) | 59.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
Buflomedil hydrochloride
CAS:35543-24-9
Buflomedil hydrochloride (Fonzylane), a vasodilator, is used in therapy of claudication or the symptoms of …
Formula:
C17H26ClNO4
Purity:
99.67% - 99.7%
Color and Shape:
White Or Off-White Crystalline Powder
Molecular weight:
343.85
Ref: TM-T0317
| 1g | 86.00 € | ||
| 5g | 180.00 € | ||
| 100mg | 42.00 € | ||
| 500mg | 59.00 € | ||
| 1mL*10mM (DMSO) | 35.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
Pizotifen Malate
CAS:5189-11-7
Pizotifen Malate (BC-105 malate), a highly selective 5-HT receptor blocking agent, is a drug based …
Formula:
C19H21NS·C4H6O5
Purity:
100%
Color and Shape:
Solid
Molecular weight:
429.53
Ref: TM-T0225
| 50mg | 34.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
Fluvoxamine maleate
CAS:61718-82-9
Fluvoxamine maleate (DU-23000 (maleate)) is a selective serotonin reuptake inhibitor that is used in the …
Formula:
C19H25F3N2O6
Purity:
99.92% - 99.94%
Color and Shape:
White Crystalline Powder
Molecular weight:
434.41
Ref: TM-T1077
| 10mg | 51.00 € | ||
| 25mg | 69.00 € | ||
| 50mg | 85.00 € | ||
| 100mg | 115.00 € | ||
| 200mg | 170.00 € | ||
| 500mg | 278.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
Nadolol
CAS:42200-33-9
Nadolol is a non-selective beta-adrenergic antagonist with antihypertensive and antiarrhythmic activities.
Formula:
C17H27NO4
Purity:
99.87% - 99.92%
Color and Shape:
White To Off-White Crystalline Powder Solid
Molecular weight:
309.4
Ref: TM-T1203
| 25mg | 48.00 € | ||
| 50mg | 72.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
Metaraminol tartrate
CAS:33402-03-8
Metaraminol tartrate (Metaradrine tartrate) is a sympathomimetic agent that acts predominantly at alpha-1 adrenergic receptors.
Formula:
C13H19NO8
Purity:
99.68%
Color and Shape:
White Powder
Molecular weight:
317.29
Ref: TM-T0279
| 50mg | 46.00 € | ||
| 100mg | 55.00 € | ||
| 200mg | 87.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
Cyproheptadine hydrochloride sesquihydrate
CAS:41354-29-4
Cyproheptadine hydrochloride sesquihydrate (Peritol), an antihistamine, is an antagonist of serotonin and histamine2.
Formula:
C21H24ClNO
Purity:
100% - 99.77%
Color and Shape:
White To Slightly Yellowish Crystalline Solid
Molecular weight:
341.88
Ref: TM-T0174
| 500mg | 34.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
Fluoxetine
CAS:54910-89-3
Fluoxetine (LY-110140), a specific serotonin inhibitor, serves as an antidepressant with fewer side-effects.
Formula:
C17H18F3NO
Purity:
99.07% - 99.28%
Color and Shape:
Solid
Molecular weight:
309.33
Ref: TM-T0450
| 10mg | 35.00 € | ||
| 25mg | 48.00 € | ||
| 50mg | 63.00 € | ||
| 100mg | 81.00 € | ||
| 200mg | 120.00 € | ||
| 500mg | 213.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
Quetiapine
CAS:111974-69-7
Quetiapine treats schizophrenia and bipolar I, targeting serotonin, dopamine, and adrenoreceptor subtypes, plus H1 histamine …
Formula:
C21H25N3O2S
Purity:
100% - 99.14%
Color and Shape:
White To Off-White Crystalline Powder
Molecular weight:
383.51
Ref: TM-T0162
| 10mg | 55.00 € | ||
| 50mg | 88.00 € | ||
| 100mg | 115.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
LY2940094
CAS:1307245-86-8
LY2940094 (LY-2940094) decreases ethanol self-administration in animal models.
Formula:
C22H23ClF2N4O2S
Purity:
99.40%
Color and Shape:
Solid
Molecular weight:
480.96
Ref: TM-T15799
| 1mg | 81.00 € | ||
| 2mg | 106.00 € | ||
| 5mg | 163.00 € | ||
| 10mg | 274.00 € | ||
| 25mg | 542.00 € | ||
| 50mg | 778.00 € | ||
| 100mg | 1,074.00 € | ||
| 1mL*10mM (DMSO) | 180.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
Blonanserin
CAS:132810-10-7
Blonanserin (AD-5423), approved in Japan (2008), is an atypical antipsychotic with fewer side effects like …
Formula:
C23H30FN3
Purity:
99.85%
Color and Shape:
Solid
Molecular weight:
367.5
Ref: TM-T1180
| 5mg | 37.00 € | ||
| 10mg | 52.00 € | ||
| 25mg | 93.00 € | ||
| 50mg | 124.00 € | ||
| 100mg | 172.00 € | ||
| 200mg | 299.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
Naftopidil
CAS:57149-07-2
Naftopidil (KT-611) (INN, marketed under the brand name Flivas), an antihypertensive medicine, is used as …
Formula:
C24H28N2O3
Purity:
99.60% - 99.97%
Color and Shape:
White Crystalline Powder
Molecular weight:
392.49
Ref: TM-T0696
| 1g | 70.00 € | ||
| 500mg | 48.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
Urapidil hydrochloride
CAS:64887-14-5
Urapidil hydrochloride (Urapidil HCl) is 5-HT1A receptor agonist and an α1-adrenoceptor antagonist.
Formula:
C20H29N5O3·HCl
Purity:
99.58%
Color and Shape:
White Or Off-White Crystalline Powder
Molecular weight:
423.94
Ref: TM-T0088
| 1g | 137.00 € | ||
| 100mg | 47.00 € | ||
| 200mg | 62.00 € | ||
| 500mg | 94.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
Mebhydrolin napadisylate
CAS:6153-33-9
Mebhydrolin napadisylate (Incidal) is an antihistamine used to relieve allergic symptoms caused by histamine release, …
Formula:
C19H20N2C10H8O6S2
Purity:
99.35% - 99.77%
Color and Shape:
White Or Almost White Crystalline
Molecular weight:
420.52
Ref: TM-T0113
| 1g | 64.00 € | ||
| 5g | 136.00 € | ||
| 10g | 188.00 € | ||
| 500mg | 47.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
