G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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V-0219
CAS:878453-71-5
V-0219 is a positive allosteric modulator of GLP-1 and can be used in studies about …
Formula:
C20H25F3N4O2
Purity:
100%
Color and Shape:
Soild
Molecular weight:
410.43
Ref: TM-T60047
| 2mg | 108.00 € |
Estimated delivery in United States, on Wednesday 9 Oct 2024
SYL-4
CAS:6222-65-7
SYL-4 is a potential P2Y12 receptor antagonist with a Ki value of 7.35 ± 1.72 …
Formula:
C20H15N3O5S
Purity:
95.76%
Color and Shape:
Soild
Molecular weight:
409.42
Ref: TM-T83637
| 1mg | 815.00 € | ||
| 25mg | 2,514.00 € |
Estimated delivery in United States, on Wednesday 9 Oct 2024
Pramipexole dihydrochloride
CAS:104632-25-9
Pramipexole dihydrochloride could be used to treat Parkinson disease.
Formula:
C10H18ClN3S
Purity:
98%
Color and Shape:
White Crystalline Powder
Molecular weight:
247.79
Ref: TM-T1476L
| 5mg | 36.00 € | ||
| 10mg | 59.00 € |
Estimated delivery in United States, on Wednesday 9 Oct 2024
(S)-Mirtazapine
CAS:61337-87-9
(S)-Mirtazapine ((S)-Org3770) is a 5-HT2 receptor antagonist with pro-nociceptive effects that can be used to …
Formula:
C17H19N3
Purity:
99.37%
Color and Shape:
Solid
Molecular weight:
265.35
Ref: TM-T12632L
| 1mg | 56.00 € | ||
| 5mg | 119.00 € | ||
| 10mg | 185.00 € | ||
| 25mg | 425.00 € | ||
| 50mg | 612.00 € | ||
| 100mg | 857.00 € |
Estimated delivery in United States, on Wednesday 9 Oct 2024
Neurotensin(8-13)
CAS:60482-95-3
Neurotensin(8-13) is Neurotensin (NT) fragment, Neurotensin(8-13) results in a decrease in cell-surface NT1 receptors (NTR1) …
Formula:
C38H64N12O8
Purity:
99.95%
Color and Shape:
Solid
Molecular weight:
816.99
Ref: TM-T7617
| 1mg | 50.00 € | ||
| 2mg | 63.00 € | ||
| 5mg | 81.00 € | ||
| 10mg | 126.00 € | ||
| 25mg | 271.00 € | ||
| 50mg | 346.00 € | ||
| 100mg | 457.00 € |
Estimated delivery in United States, on Wednesday 9 Oct 2024
Asenapine hydrochloride
CAS:1261398-77-9
Asenapine hydrochloride (Org 5222 hydrochloride) is an antagonist of 5-hydroxytryptamine, adrenergic, dopamine, and histamine receptors …
Formula:
C17H17Cl2NO
Color and Shape:
Solid
Molecular weight:
322.23
Ref: TM-T22589
| 1mg | 76.00 € |
Estimated delivery in United States, on Wednesday 9 Oct 2024
Dynorphin A acetate(80448-90-4 free base)
Dynorphin A acetate is an Endogenous kappa receptor agonist.
Formula:
C101H159N31O25
Purity:
99.69%
Color and Shape:
Solid
Molecular weight:
2207.58
Ref: TM-TP2040L
| 1mg | 70.00 € | ||
| 5mg | 234.00 € | ||
| 10mg | 321.00 € | ||
| 25mg | 541.00 € | ||
| 50mg | 774.00 € | ||
| 100mg | 1,067.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Guanabenz hydrochloride
CAS:23113-43-1
Guanabenz hydrochloride (NE56490) is an orally active α2-adrenoceptor agonist with hypotensive effects.
Formula:
C8H9Cl3N4
Purity:
99.45%
Color and Shape:
Solid
Molecular weight:
267.54
Ref: TM-T21957
| 1ml | 34.00 € | ||
| 50mg | 44.00 € | ||
| 100mg | 78.00 € | ||
| 200mg | 102.00 € | ||
| 500mg | 169.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Siponimod
CAS:1230487-00-9
Siponimod (BAF312) modulates S1P1/S1P5 with EC50s of 0.39/0.98 nM; >1000x selectivity over S1P2-4.
Formula:
C29H35F3N2O3
Purity:
97.08% - 99.29%
Color and Shape:
Solid
Molecular weight:
516.59
Ref: TM-T6403
| 1ml | 65.00 € | ||
| 2mg | 44.00 € | ||
| 5mg | 61.00 € | ||
| 10mg | 90.00 € | ||
| 25mg | 142.00 € | ||
| 50mg | 224.00 € | ||
| 100mg | 304.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Albiglutide TFA (782500-75-8 free base)
Albiglutide TFA (782500-75-8 free base) (Albiglutide TFA) is a long acting GLP-1 receptor agonist for …
Formula:
C150H225F3N40O47
Purity:
100%
Color and Shape:
Solid
Molecular weight:
3397.63
Ref: TM-TP1796
| 1mg | 95.00 € | ||
| 5mg | 269.00 € | ||
| 10mg | 391.00 € | ||
| 25mg | 598.00 € | ||
| 50mg | 814.00 € | ||
| 100mg | 1,081.00 € | ||
| 200mg | 1,447.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Deltorphin I
CAS:122752-15-2
Deltorphin I is an agonist of δ-opioid receptor.
Formula:
C37H52N8O10
Purity:
100%
Color and Shape:
Solid
Molecular weight:
768.86
Ref: TM-T7637
| 1mg | 62.00 € | ||
| 1ml | 199.00 € | ||
| 5mg | 140.00 € | ||
| 10mg | 203.00 € | ||
| 25mg | 343.00 € | ||
| 50mg | 505.00 € | ||
| 100mg | 720.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Protease-Activated Receptor-2, amide
CAS:190383-13-2
Protease-Activated Receptor-2, amide (SLIGKV-NH2) is an agonist of PAR2 (IC50 : 10.4 M)
Formula:
C28H54N8O7
Purity:
100%
Color and Shape:
Solid
Molecular weight:
614.78
Ref: TM-T7513
| 2mg | 52.00 € | ||
| 5mg | 75.00 € | ||
| 10mg | 114.00 € | ||
| 25mg | 187.00 € | ||
| 50mg | 282.00 € | ||
| 100mg | 421.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Prucalopride Succinate
CAS:179474-85-2
Prucalopride Succinate is a 5-HT4 receptor agonist with Ki 2.5 nM (5-HT4a) and 8 nM …
Formula:
C18H26ClN3O3·C4H6O4
Purity:
99.24%
Color and Shape:
Solid
Molecular weight:
485.96
Ref: TM-T6958
| 1ml | 36.00 € | ||
| 10mg | 47.00 € | ||
| 25mg | 54.00 € | ||
| 50mg | 73.00 € | ||
| 100mg | 111.00 € | ||
| 200mg | 169.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Talnetant
CAS:174636-32-9
Talnetant (SB 223412) is a selective NK3 receptor antagonist that can penetrate the brain and …
Formula:
C25H22N2O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
382.45
Ref: TM-T7549
| 1mg | 42.00 € | ||
| 1ml | 142.00 € | ||
| 2mg | 55.00 € | ||
| 5mg | 91.00 € | ||
| 10mg | 127.00 € | ||
| 25mg | 261.00 € | ||
| 50mg | 479.00 € | ||
| 100mg | 728.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
TC-G 1005
CAS:1415407-60-1
TC-G 1005 is a potent and selective GPBA agonist (EC50 :0.72 nM; hTGR5).
Formula:
C25H25N3O2
Purity:
98.2% - 99.23%
Color and Shape:
Solid
Molecular weight:
399.48
Ref: TM-T8818
| 1mg | 35.00 € | ||
| 1ml | 76.00 € | ||
| 2mg | 45.00 € | ||
| 5mg | 68.00 € | ||
| 10mg | 94.00 € | ||
| 25mg | 184.00 € | ||
| 50mg | 277.00 € | ||
| 100mg | 414.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Dexmedetomidine hydrochloride
CAS:145108-58-3
Dexmedetomidine hydrochloride (Precedex) is an imidazole derivative that is an agonist of the adrenergic α2 …
Formula:
C13H16N2·HCl
Purity:
100.00% - 99.86%
Color and Shape:
White Or Almost White Crystalline Powder
Molecular weight:
236.74
Ref: TM-T6466
| 1ml | 51.00 € | ||
| 5mg | 41.00 € | ||
| 10mg | 54.00 € | ||
| 25mg | 87.00 € | ||
| 50mg | 157.00 € | ||
| 100mg | 222.00 € | ||
| 200mg | 333.00 € | ||
| 500mg | 551.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Ganirelix Acetate
CAS:123246-29-7
Ganirelix Acetate is a gonadotropin-releasing hormone (GnRH) receptor antagonist
Formula:
C82H117ClN18O15
Purity:
96.05%
Color and Shape:
Solid
Molecular weight:
1630.4
Ref: TM-TP2337
| 1mg | 84.00 € | ||
| 5mg | 171.00 € | ||
| 10mg | 248.00 € | ||
| 25mg | 408.00 € | ||
| 50mg | 574.00 € | ||
| 100mg | 776.00 € | ||
| 200mg | 1,029.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
AM211
CAS:1175526-27-8
AM211 (AM211 free acid) is a potent and orally bioavailable antagonist of prostaglandin D2 (PGD2) …
Formula:
C27H27F3N2O4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
500.51
Ref: TM-T7652
| 1mg | 37.00 € | ||
| 1ml | 87.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 118.00 € | ||
| 25mg | 230.00 € | ||
| 50mg | 352.00 € | ||
| 100mg | 520.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Cinaciguat
CAS:329773-35-5
Cinaciguat (BAY 58-2667) is a pioneering sGC activator for acute heart failure treatment.
Formula:
C36H39NO5
Purity:
98% - 99.82%
Color and Shape:
Solid
Molecular weight:
565.7
Ref: TM-T1984
| 1mg | 71.00 € | ||
| 1ml | 173.00 € | ||
| 2mg | 94.00 € | ||
| 5mg | 142.00 € | ||
| 10mg | 230.00 € | ||
| 25mg | 352.00 € | ||
| 50mg | 484.00 € | ||
| 100mg | 687.00 € | ||
| 500mg | 1,395.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
JD-5037
CAS:1392116-14-1
JD-5037 is a novel, peripherally restricted CB1R antagonist with an IC50 of 1.5 nM.
Formula:
C27H27Cl2N5O3S
Purity:
98.14% - 98.87%
Color and Shape:
Solid
Molecular weight:
572.51
Ref: TM-T4453
| 1mg | 43.00 € | ||
| 1ml | 106.00 € | ||
| 2mg | 57.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 139.00 € | ||
| 25mg | 241.00 € | ||
| 50mg | 362.00 € | ||
| 100mg | 538.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
