G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Maropitant citrate
CAS:359875-09-5
Maropitant citrate is a synthetic neurokinin-1 receptor antagonist and substance P inhibitor, used for controlling …
Formula:
C38H50N2O9
Purity:
98.91%
Color and Shape:
Liquid
Molecular weight:
678.81
Ref: TM-T35344
| 1mg | 58.00 € | ||
| 5mg | 116.00 € | ||
| 10mg | 170.00 € | ||
| 25mg | 274.00 € | ||
| 50mg | 408.00 € | ||
| 100mg | 607.00 € | ||
| 200mg | 845.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
GPR41 agonist-1
CAS:506417-09-0
GPR41 agonist-1 is a GPR41 agonist, used for studying metabolic diseases such as diabetes and …
Formula:
C24H23N3O4
Purity:
98.40%
Color and Shape:
Liquid
Molecular weight:
417.46
Ref: TM-T62173
| 2mg | 69.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
Octreotide
CAS:83150-76-9
Octreotide (SMS 201-995) is a potent inhibitor of growth hormone, glucagon, and insulin.
Formula:
C49H66N10O10S2
Purity:
99.64%
Color and Shape:
White Powder
Molecular weight:
1019.24
Ref: TM-T2584
| 1mg | 50.00 € | ||
| 5mg | 105.00 € | ||
| 10mg | 170.00 € | ||
| 25mg | 284.00 € | ||
| 50mg | 425.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
Docosahexaenoic acid ethyl ester
CAS:81926-94-5
Docosahexaenoic acid ethyl ester (Ethyl docosahexaenoate) enhances 6-hydroxydopamine-induced neuronal damage by inducing lipid peroxidation in …
Formula:
C24H36O2
Color and Shape:
Solid
Molecular weight:
356.54
Ref: TM-T41321
| 50mg | 40.00 € | ||
| 100mg | 52.00 € | ||
| 500mg | 137.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
TUG-770
CAS:1402601-82-4
TUG-770 is a highly potent agonist of free fatty acid receptor 1 (FFA1/GPR40, EC50: 6 …
Formula:
C19H14FNO2
Purity:
97.6%
Color and Shape:
Solid
Molecular weight:
307.32
Ref: TM-TQ0241
| 1mg | 64.00 € | ||
| 5mg | 137.00 € | ||
| 10mg | 210.00 € | ||
| 25mg | 408.00 € | ||
| 50mg | 652.00 € | ||
| 100mg | 938.00 € | ||
| 500mg | 1,882.00 € | ||
| 1mL*10mM (DMSO) | 202.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
(Rac)-Rotigotine hydrochloride
CAS:102120-99-0
(Rac)-Rotigotine hydrochloride is a racemate of Rotigotine. Rotigotine is a full agonist of dopamine receptor, …
Formula:
C19H26ClNOS
Color and Shape:
Solid
Molecular weight:
351.93
Ref: TM-T12676
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
(R,S)-Ivosidenib
CAS:2070009-31-1
(R,S)-Ivosidenib is the less active enantiomer of Ivosidenib .
Formula:
C28H22ClF3N6O3
Color and Shape:
Solid
Molecular weight:
582.96
Ref: TM-T13438
| 2mg | 379.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
GW-1100
CAS:306974-70-9
GW-1100 is a selective GPR40 and FFAR1 antagonist for the study of diabetes and metabolic …
Formula:
C27H25FN4O4S
Purity:
97.01%
Color and Shape:
Solid
Molecular weight:
520.58
Ref: TM-T15448
| 1mg | 37.00 € | ||
| 5mg | To inquire |
Estimated delivery in United States, on Monday 31 Mar 2025
PD128907 HCl
CAS:112960-16-4
PD128907 HCl is a potent and selective dopamine D3 receptor agonist, with EC50 of 0.64 …
Formula:
C14H20ClNO3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
285.77
Ref: TM-T6142
| 1mg | 49.00 € | ||
| 5mg | 105.00 € | ||
| 10mg | 162.00 € | ||
| 25mg | 264.00 € | ||
| 50mg | 393.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
Motixafortide
CAS:664334-36-5
Motixafortide (BKT140 4-fluorobenzoyl) is an antagonist of CXCR4 (IC50: 1 nM).
Formula:
C97H144FN33O19S2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
2159.52
Ref: TM-T14665
| 25mg | 710.00 € | ||
| 50mg | 1,130.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
Endomorphin 2 TFA
CAS:1276124-00-5
Endomorphin 2 TFA, displays reasonable affinities for kappa3 binding sites, with Ki value between 20 …
Formula:
C34H38F3N5O7
Color and Shape:
Solid
Molecular weight:
685.69
Ref: TM-T11198
| 2mg | 90.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
Asimadoline
CAS:153205-46-0
Asimadoline (EMD-61753) is a proprietary small molecule therapeutic, originally discovered by Merck KGaA of Darmstadt, …
Formula:
C27H30N2O2
Color and Shape:
Solid
Molecular weight:
414.54
Ref: TM-T4633
| 5mg | 73.00 € | ||
| 25mg | 283.00 € | ||
| 1mL*10mM (DMSO) | 79.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
Zagociguat
CAS:2201048-82-8
Zagociguat (CY6463) is a stimulator of guanylate cyclase that increases nitric oxide (NO) signaling and …
Formula:
C16H10F4N6
Purity:
99.37%
Color and Shape:
Liquid
Molecular weight:
362.28
Ref: TM-T39673
| 1mg | 107.00 € | ||
| 5mg | 254.00 € | ||
| 10mg | 408.00 € | ||
| 25mg | 796.00 € | ||
| 50mg | 1,195.00 € | ||
| 100mg | 1,617.00 € | ||
| 200mg | 2,176.00 € | ||
| 1mL*10mM (DMSO) | 280.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
Sumanirole maleate
CAS:179386-44-8
Sumanirole maleate (U-95666E) is a highly selective full agonist of the D2 receptor (ED50: 46 …
Formula:
C15H17N3O5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
319.31
Ref: TM-TQ0140
| 2mg | 90.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
SB-200646A
CAS:143797-62-0
SB-200646A: oral 5-HT2B/2C antagonist; higher affinity than 5-HT2A (pKi: 7.5, 6.9 vs 5.2); anxiolytic with …
Formula:
C15H15ClN4O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
302.76
Ref: TM-T22423
| 2mg | 42.00 € | ||
| 1mL*10mM (DMSO) | 84.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
WZ4141
CAS:1222776-76-2
WZ4141 is an intermediate in compound synthesis.
Formula:
C16H13N3O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
279.29
Ref: TM-T19604
| 5mg | 445.00 € | ||
| 1mL*10mM (DMSO) | 435.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
CB1/2 agonist 3
CAS:2772655-86-2
CB1/2 agonist 3 is a competitive and potent CB1/CB2 agonist with high affinity for hCB1 …
Formula:
C25H41NO2
Purity:
98.78%
Color and Shape:
Liquid
Molecular weight:
387.6
Ref: TM-T61736
| 1mg | 42.00 € | ||
| 5mg | 88.00 € | ||
| 10mg | 131.00 € | ||
| 25mg | 207.00 € | ||
| 50mg | 309.00 € | ||
| 100mg | 459.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
Eticlopride hydrochloride
CAS:97612-24-3
Eticlopride, an antipsychotic, is a Selective dopamine D2/D3 receptor antagonist (Ki: 0.5/0.16 nM).
Formula:
C17H25ClN2O3·HCl
Purity:
98%
Color and Shape:
Solid
Molecular weight:
377.31
Ref: TM-T4007
| 1mg | 49.00 € | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
AF-710B
CAS:1235733-73-9
AF710B is an enantiomer of AF710. AF-710B is also a sigma and M1 muscarinic receptors …
Formula:
C20H27N3OS
Purity:
98.62% - 99.89%
Color and Shape:
Solid
Molecular weight:
357.51
Ref: TM-T23649
| 1mg | 316.00 € | ||
| 2mg | 470.00 € | ||
| 5mg | 750.00 € | ||
| 10mg | 1,064.00 € | ||
| 25mg | 1,586.00 € | ||
| 50mg | 2,072.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
S1RA
CAS:878141-96-9
S1RA (E-52862)(E-52862) is a potent, selective antagonist of the sigma-1 receptor (σ1R, Ki=17 nM), demonstrating …
Formula:
C20H23N3O2
Purity:
99.45%
Color and Shape:
Solid
Molecular weight:
337.42
Ref: TM-T1865
| 1mg | 38.00 € | ||
| 5mg | 80.00 € | ||
| 10mg | 133.00 € | ||
| 25mg | 215.00 € | ||
| 50mg | 319.00 € | ||
| 1mL*10mM (DMSO) | 88.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
