G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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TP-16
CAS:2332972-26-4
TP-16 is a novel potent and selective EP4 antagonist that blocks the function of IMCs …
Formula:
C24H22FNO4S
Purity:
98.83% - 99.33%
Color and Shape:
Liquid
Molecular weight:
439.5
Ref: TM-T62525
| 1mg | 439.00 € | ||
| 5mg | 1,017.00 € | ||
| 25mg | 2,023.00 € |
Estimated delivery in United States, on Thursday 6 Mar 2025
L-368,899 hydrochloride
CAS:160312-62-9
L-368,899 hydrochloride is an OXTR antagonist that prevents oxytocin-induced antiabnormal pain and anti-nausea, and may …
Formula:
C26H43ClN4O5S2
Purity:
99.59%
Color and Shape:
Solid
Molecular weight:
591.23
Ref: TM-T11794
| 2mg | 111.00 € | ||
| 5mg | 156.00 € | ||
| 10mg | 243.00 € | ||
| 25mg | 462.00 € | ||
| 50mg | 723.00 € | ||
| 100mg | 1,017.00 € | ||
| 1mL*10mM (DMSO) | 212.00 € |
Estimated delivery in United States, on Thursday 6 Mar 2025
Setiptiline
CAS:57262-94-9
Setiptiline (Org-8282) is a norepinephrine reuptake inhibitor, 2-adrenergic receptor antagonist, H1 receptor inverse agonist with …
Formula:
C19H19N
Purity:
98.07%
Color and Shape:
Solid
Molecular weight:
261.36
Ref: TM-T12900
| 5mg | 34.00 € | ||
| 1mL*10mM (DMSO) | 64.00 € |
Estimated delivery in United States, on Thursday 6 Mar 2025
Rizatriptan
CAS:144034-80-0
Rizatriptan (Risatriptan) is a selective 5-hydroxytryptamine 1B/1D receptor agonist used in the study of migraine.
Formula:
C15H19N5
Purity:
99.74%
Color and Shape:
Solid
Molecular weight:
269.35
Ref: TM-T1734L
| 5mg | 35.00 € | ||
| 10mg | 48.00 € | ||
| 25mg | 69.00 € | ||
| 50mg | 89.00 € | ||
| 100mg | 133.00 € |
Estimated delivery in United States, on Thursday 6 Mar 2025
SLIGRL-NH2
CAS:171436-38-7
SLIGRL-NH2 (Protease-Activated Receptor-2 Activating Peptide) is a PAR-2 agonist that induces non-histaminergic pruritus.
Formula:
C29H56N10O7
Purity:
98.29%
Color and Shape:
Solid
Molecular weight:
656.82
Ref: TM-TP1046
| 1mg | 98.00 € |
Estimated delivery in United States, on Thursday 6 Mar 2025
Motixafortide
CAS:664334-36-5
Motixafortide (BKT140 4-fluorobenzoyl) is an antagonist of CXCR4 (IC50: 1 nM).
Formula:
C97H144FN33O19S2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
2159.52
Ref: TM-T14665
| 25mg | 710.00 € | ||
| 50mg | 1,130.00 € |
Estimated delivery in United States, on Thursday 6 Mar 2025
Tegaserod
CAS:145158-71-0
Tegaserod is a 5-HT4R agonist and 5-HT2B receptor antagonist with antitumor activity used in the …
Formula:
C16H23N5O
Purity:
99.89%
Color and Shape:
Liquid
Molecular weight:
301.39
Ref: TM-T60680
| 2mg | 37.00 € |
Estimated delivery in United States, on Thursday 6 Mar 2025
LAS101057
CAS:925676-48-8
LAS101057 is a novel orally available and potent and selective A2B receptor antagonist for the …
Formula:
C18H14FN5O
Purity:
100%
Color and Shape:
Solid
Molecular weight:
335.34
Ref: TM-T15715
| 1mg | 42.00 € | ||
| 5mg | 88.00 € | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Thursday 6 Mar 2025
Endomorphin 2 TFA
CAS:1276124-00-5
Endomorphin 2 TFA, displays reasonable affinities for kappa3 binding sites, with Ki value between 20 …
Formula:
C34H38F3N5O7
Color and Shape:
Solid
Molecular weight:
685.69
Ref: TM-T11198
| 2mg | 90.00 € |
Estimated delivery in United States, on Thursday 6 Mar 2025
Meclizine
CAS:569-65-3
Meclizine, also known as Meclozine, is a piperazine class H1 antagonist with antihistamine properties that …
Formula:
C25H27ClN2
Purity:
95.16%
Color and Shape:
Solid
Molecular weight:
390.95
Ref: TM-T40652
| 1mg | 185.00 € | ||
| 5mg | 426.00 € | ||
| 10mg | 627.00 € | ||
| 25mg | 938.00 € | ||
| 50mg | 1,320.00 € | ||
| 100mg | 1,786.00 € |
Estimated delivery in United States, on Thursday 6 Mar 2025
Bucindolol
CAS:71119-11-4
Bucindolol (BMY 13105) is a novel and potent β1-adrenergic receptor blocker that mediates vasodilation and …
Formula:
C22H25N3O2
Purity:
99.9%
Color and Shape:
Solid
Molecular weight:
363.45
Ref: TM-T10631
| 1mg | 47.00 € |
Estimated delivery in United States, on Thursday 6 Mar 2025
ML 145
CAS:1164500-72-4
ML 145 is a selective antagonist of GPR35/CXCR8 (IC50/EC50 of 20.1 nM)
Formula:
C24H22N2O5S2
Purity:
97.74%
Color and Shape:
Solid
Molecular weight:
482.57
Ref: TM-T12074
| 2mg | 90.00 € | ||
| 5mg | 145.00 € | ||
| 10mg | 207.00 € | ||
| 25mg | 350.00 € | ||
| 50mg | 522.00 € | ||
| 100mg | 750.00 € | ||
| 200mg | 1,075.00 € |
Estimated delivery in United States, on Thursday 6 Mar 2025
Trabodenoson
CAS:871108-05-3
Trabodenoson (INO-8875) is a selective and potent adenosine A1 receptor agonist, an adenosine analog, for …
Formula:
C15H20N6O6
Purity:
99.94%
Color and Shape:
Solid
Molecular weight:
380.36
Ref: TM-T34914
| 1mg | 131.00 € | ||
| 2mg | 187.00 € | ||
| 5mg | 311.00 € | ||
| 10mg | 467.00 € | ||
| 25mg | 747.00 € | ||
| 50mg | 1,017.00 € | ||
| 100mg | 1,359.00 € | ||
| 1mL*10mM (DMSO) | 344.00 € |
Estimated delivery in United States, on Thursday 6 Mar 2025
Ketanserin tartrate
CAS:83846-83-7
Ketanserin tartrate (KJK-945 tartrate) is a 5-HT2A receptor and α1-adrenergic receptor antagonist for the study …
Formula:
C26H28FN3O9
Purity:
99.68%
Color and Shape:
Solid
Molecular weight:
545.51
Ref: TM-T1066L
| 25mg | 37.00 € | ||
| 50mg | 52.00 € | ||
| 100mg | 67.00 € | ||
| 1mL*10mM (DMSO) | 35.00 € |
Estimated delivery in United States, on Thursday 6 Mar 2025
UCM 608
CAS:151889-03-1
UCM 608 (2-Phenylmelatonin) is an antagonist of melatonin-induced contractile responses at low concentrations and induces …
Formula:
C19H20N2O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
308.37
Ref: TM-T22499
| 2mg | 54.00 € | ||
| 5mg | 85.00 € | ||
| 10mg | 105.00 € | ||
| 25mg | 173.00 € | ||
| 50mg | 254.00 € |
Estimated delivery in United States, on Thursday 6 Mar 2025
WIN 51,708
CAS:144177-30-0
WIN 51,708 is an antagonist of neurokinin-1 receptor.
Formula:
C29H33N3O
Purity:
99%
Color and Shape:
Solid
Molecular weight:
439.59
Ref: TM-T29157
| 1mg | 279.00 € | ||
| 2mg | 414.00 € | ||
| 5mg | 685.00 € | ||
| 10mg | 938.00 € | ||
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € |
Estimated delivery in United States, on Thursday 6 Mar 2025
Spiroxatrine
CAS:1054-88-2
Spiroxatrine (R 5188) is a 5-HT1α and α2-adrenergic dual antagonist with sedative activity for the …
Formula:
C22H25N3O3
Purity:
99.83%
Color and Shape:
Solid
Molecular weight:
379.45
Ref: TM-T23382
| 5mg | 88.00 € | ||
| 10mg | 126.00 € | ||
| 25mg | 250.00 € | ||
| 50mg | 400.00 € | ||
| 100mg | 582.00 € |
Estimated delivery in United States, on Thursday 6 Mar 2025
ACT-462206
CAS:1361321-96-1
ACT-462206 is a Orexin 1/Orexin 2 receptor antagonist.ACT-462206 is highly potent and can be used …
Formula:
C20H24N2O4S
Purity:
99.45%
Color and Shape:
Solid
Molecular weight:
388.48
Ref: TM-T26559
| 1mg | 44.00 € | ||
| 5mg | 93.00 € | ||
| 10mg | 137.00 € | ||
| 25mg | 279.00 € | ||
| 50mg | 445.00 € | ||
| 100mg | 707.00 € | ||
| 500mg | 1,415.00 € | ||
| 1mL*10mM (DMSO) | 93.00 € |
Estimated delivery in United States, on Thursday 6 Mar 2025
Clothiapine
CAS:2058-52-8
Clothiapine is an atypical antipsychotic of the dibenzothiazepine chemical class.
Formula:
C18H18ClN3S
Purity:
99.93%
Color and Shape:
Solid
Molecular weight:
343.87
Ref: TM-T23900
| 1mg | 98.00 € |
Estimated delivery in United States, on Thursday 6 Mar 2025
MS 15203
CAS:73912-52-4
MS 15203 is a GPR171 agonist that reduces chronic neuropathic and inflammatory pain in male …
Formula:
C12H11NO5
Purity:
99.53%
Color and Shape:
Liquid
Molecular weight:
249.22
Ref: TM-T37131
| 2mg | 46.00 € | ||
| 5mg | 66.00 € | ||
| 10mg | 104.00 € | ||
| 25mg | 210.00 € | ||
| 50mg | 311.00 € | ||
| 100mg | 467.00 € | ||
| 500mg | 1,017.00 € | ||
| 1mL*10mM (DMSO) | 74.00 € |
Estimated delivery in United States, on Thursday 6 Mar 2025
