G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Deltorphin I
CAS:122752-15-2
Deltorphin I is an agonist of δ-opioid receptor.
Formula:
C37H52N8O10
Purity:
100%
Color and Shape:
Solid
Molecular weight:
768.86
Ref: TM-T7637
| 1mg | 62.00 € | ||
| 5mg | 140.00 € | ||
| 10mg | 203.00 € | ||
| 25mg | 343.00 € | ||
| 50mg | 505.00 € | ||
| 100mg | 720.00 € | ||
| 1mL*10mM (DMSO) | 199.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Protease-Activated Receptor-2, amide
CAS:190383-13-2
Protease-Activated Receptor-2, amide (SLIGKV-NH2) is an agonist of PAR2 (IC50 : 10.4 M)
Formula:
C28H54N8O7
Purity:
100%
Color and Shape:
Solid
Molecular weight:
614.78
Ref: TM-T7513
| 2mg | 52.00 € | ||
| 5mg | 75.00 € | ||
| 10mg | 114.00 € | ||
| 25mg | 187.00 € | ||
| 50mg | 282.00 € | ||
| 100mg | 421.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Prucalopride Succinate
CAS:179474-85-2
Prucalopride Succinate is a 5-HT4 receptor agonist with Ki 2.5 nM (5-HT4a) and 8 nM …
Formula:
C18H26ClN3O3·C4H6O4
Purity:
99.24%
Color and Shape:
Solid
Molecular weight:
485.96
Ref: TM-T6958
| 10mg | 47.00 € | ||
| 25mg | 54.00 € | ||
| 50mg | 73.00 € | ||
| 100mg | 111.00 € | ||
| 200mg | 169.00 € | ||
| 1mL*10mM (DMSO) | 36.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Talnetant
CAS:174636-32-9
Talnetant (SB 223412) is a selective NK3 receptor antagonist that can penetrate the brain and …
Formula:
C25H22N2O2
Purity:
≥95%
Color and Shape:
Solid
Molecular weight:
382.45
Ref: TM-T7549
| 1mg | 42.00 € | ||
| 2mg | 55.00 € | ||
| 5mg | 91.00 € | ||
| 10mg | 127.00 € | ||
| 25mg | 261.00 € | ||
| 50mg | 479.00 € | ||
| 100mg | 728.00 € | ||
| 1mL*10mM (DMSO) | 142.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
TC-G 1005
CAS:1415407-60-1
TC-G 1005 is a potent and selective GPBA agonist (EC50 :0.72 nM; hTGR5).
Formula:
C25H25N3O2
Purity:
98.2% - 99.23%
Color and Shape:
Solid
Molecular weight:
399.48
Ref: TM-T8818
| 1mg | 35.00 € | ||
| 2mg | 45.00 € | ||
| 5mg | 68.00 € | ||
| 10mg | 94.00 € | ||
| 25mg | 184.00 € | ||
| 50mg | 277.00 € | ||
| 100mg | 414.00 € | ||
| 1mL*10mM (DMSO) | 76.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Dexmedetomidine hydrochloride
CAS:145108-58-3
Dexmedetomidine hydrochloride (Precedex) is a potent, selective, orally active α2-adrenoceptor agonist.Cost-effective and quality-assured.
Formula:
C13H16N2·HCl
Purity:
100.00% - 99.86%
Color and Shape:
White Or Almost White Crystalline Powder
Molecular weight:
236.74
Ref: TM-T6466
| 5mg | 41.00 € | ||
| 10mg | 54.00 € | ||
| 25mg | 87.00 € | ||
| 50mg | 157.00 € | ||
| 100mg | 222.00 € | ||
| 200mg | 333.00 € | ||
| 500mg | 551.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Ganirelix Acetate
CAS:123246-29-7
Ganirelix Acetate is a gonadotropin-releasing hormone (GnRH) receptor antagonist
Formula:
C82H117ClN18O15
Purity:
96.05%
Color and Shape:
Solid
Molecular weight:
1630.4
Ref: TM-TP2337
| 1mg | 84.00 € | ||
| 5mg | 171.00 € | ||
| 10mg | 248.00 € | ||
| 25mg | 408.00 € | ||
| 50mg | 574.00 € | ||
| 100mg | 776.00 € | ||
| 200mg | 1,029.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
AM211
CAS:1175526-27-8
AM211 (AM211 free acid) is a potent and orally bioavailable antagonist of prostaglandin D2 (PGD2) …
Formula:
C27H27F3N2O4
Purity:
≥95%
Color and Shape:
Solid
Molecular weight:
500.51
Ref: TM-T7652
| 1mg | 37.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 118.00 € | ||
| 25mg | 230.00 € | ||
| 50mg | 352.00 € | ||
| 100mg | 520.00 € | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Cinaciguat
CAS:329773-35-5
Cinaciguat (BAY 58-2667) is a pioneering sGC activator for acute heart failure treatment.
Formula:
C36H39NO5
Purity:
98% - 99.82%
Color and Shape:
Solid
Molecular weight:
565.7
Ref: TM-T1984
| 1mg | 47.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 142.00 € | ||
| 25mg | 206.00 € | ||
| 50mg | 285.00 € | ||
| 100mg | 404.00 € | ||
| 200mg | 552.00 € | ||
| 1mL*10mM (DMSO) | 106.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
JD-5037
CAS:1392116-14-1
JD-5037 is a novel, peripherally restricted CB1R antagonist with an IC50 of 1.5 nM.
Formula:
C27H27Cl2N5O3S
Purity:
98.14% - 98.87%
Color and Shape:
Solid
Molecular weight:
572.51
Ref: TM-T4453
| 1mg | 43.00 € | ||
| 2mg | 57.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 139.00 € | ||
| 25mg | 241.00 € | ||
| 50mg | 362.00 € | ||
| 100mg | 538.00 € | ||
| 1mL*10mM (DMSO) | 106.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
3-CPMT
CAS:14008-79-8
3-CPMT (FC-1) is a dopamine uptake inhibitor and a potent long-acting antihistaminic agent.
Formula:
C21H25Cl2NO
Purity:
99.03%
Color and Shape:
Solid
Molecular weight:
378.33
Ref: TM-T22508
| 1mg | 44.00 € | ||
| 2mg | 54.00 € | ||
| 5mg | 74.00 € | ||
| 10mg | 95.00 € | ||
| 25mg | 220.00 € | ||
| 50mg | 417.00 € | ||
| 100mg | 616.00 € | ||
| 1mL*10mM (DMSO) | 91.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
5-O-Demethylnobiletin
CAS:2174-59-6
5-O-Demethylnobiletin is a natural anti-inflammatory that inhibits 5-LOX without altering COX-2 expression.
Formula:
C20H20O8
Purity:
99.83% - ≥95%
Color and Shape:
Solid
Molecular weight:
388.37
Ref: TM-T5714
| 1mg | 64.00 € | ||
| 5mg | 125.00 € | ||
| 10mg | 204.00 € | ||
| 25mg | 357.00 € | ||
| 50mg | 499.00 € | ||
| 100mg | 739.00 € | ||
| 500mg | 1,613.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
JMS-17-2
CAS:1380392-05-1
JMS-17-2 is a potent and selective antagonist of CX3CR1( IC50 : 0.32 nM).
Formula:
C25H26ClN3O
Purity:
98.70% - ≥98%
Color and Shape:
Solid
Molecular weight:
419.95
Ref: TM-T5849
| 1mg | 40.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 85.00 € | ||
| 10mg | 128.00 € | ||
| 25mg | 218.00 € | ||
| 50mg | 337.00 € | ||
| 100mg | 500.00 € | ||
| 1mL*10mM (DMSO) | 96.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
5-HT1A modulator 2 hydrochloride
CAS:3880-76-0
5-HT1A modulator 2 hydrochloride is a modulator of 5-HT1A showing an affinity of 53 nM …
Formula:
C11H16ClNO
Purity:
97%
Color and Shape:
Solid
Molecular weight:
213.7
Ref: TM-T37197
| 50mg | 34.00 € | ||
| 1mL*10mM (DMSO) | 50.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Tetrahydroberberine
CAS:522-97-4
Tetrahydroberberine (Canadine) is an isoquinoline alkaloid isolated from corydalis tuber, has a micromolar affinity for …
Formula:
C20H21NO4
Purity:
96.65% - 99.89%
Color and Shape:
Solid
Molecular weight:
339.39
Ref: TM-T2874
| 5mg | 47.00 € | ||
| 10mg | 62.00 € | ||
| 25mg | 91.00 € | ||
| 50mg | 134.00 € | ||
| 100mg | 184.00 € | ||
| 500mg | 477.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Danirixin
CAS:954126-98-8
Danirixin (GSK1325756) is a potent antagonist of CXCR2 that inhibits IL-8 binding to CXCR2 (IC50: …
Formula:
C19H21ClFN3O4S
Purity:
100.00% - 99.78%
Color and Shape:
Solid
Molecular weight:
441.9
Ref: TM-T5193
| 1mg | 60.00 € | ||
| 5mg | 109.00 € | ||
| 10mg | 176.00 € | ||
| 25mg | 328.00 € | ||
| 50mg | 522.00 € | ||
| 100mg | 736.00 € | ||
| 1mL*10mM (DMSO) | 133.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Fosaprepitant dimeglumine
CAS:265121-04-8
Fosaprepitant dimeglumine (MK-0517) is a soluble prodrug of aprepitant, which prevents nausea by blocking NK1 …
Formula:
C37H56F7N6O16P
Purity:
97.39% - 98.75%
Color and Shape:
Solid
Molecular weight:
1004.83
Ref: TM-T1790
| 5mg | 49.00 € | ||
| 10mg | 66.00 € | ||
| 25mg | 119.00 € | ||
| 50mg | 208.00 € | ||
| 100mg | 343.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
L-765314
CAS:189349-50-6
L-765314: potent α1B adrenergic receptor antagonist, used for blood pressure research.
Formula:
C27H34N6O5
Purity:
99.73%
Color and Shape:
Solid
Molecular weight:
522.6
Ref: TM-T5511
| 2mg | 35.00 € | ||
| 5mg | 51.00 € | ||
| 10mg | 72.00 € | ||
| 25mg | 132.00 € | ||
| 50mg | 203.00 € | ||
| 100mg | 300.00 € | ||
| 1mL*10mM (DMSO) | 64.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Decloxizine dihydrochloride
CAS:13073-96-6
Decloxizine dihydrochloride (UCB 1402 dihydrochloride) is a histamine 1 receptor antagonist.
Formula:
C21H28N2O2·2ClH
Purity:
99.73%
Color and Shape:
Solid
Molecular weight:
413.39
Ref: TM-T5495
| 10mg | 45.00 € | ||
| 25mg | 67.00 € | ||
| 50mg | 95.00 € | ||
| 100mg | 131.00 € | ||
| 500mg | 462.00 € | ||
| 1mL*10mM (DMSO) | 95.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
ML221
CAS:877636-42-5
ML221 is a potent apelin /APJ functional antagonist, inhibiting apelin-13-mediated activation of APJ, with IC50s …
Formula:
C17H11N3O6S
Purity:
97.74%
Color and Shape:
Solid
Molecular weight:
385.35
Ref: TM-T4390
| 5mg | 54.00 € | ||
| 10mg | 84.00 € | ||
| 25mg | 163.00 € | ||
| 50mg | 240.00 € | ||
| 100mg | 435.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
