G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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ACT-462206
CAS:1361321-96-1
ACT-462206 is a Orexin 1/Orexin 2 receptor antagonist.ACT-462206 is highly potent and can be used …
Formula:
C20H24N2O4S
Purity:
99.45%
Color and Shape:
Solid
Molecular weight:
388.48
Ref: TM-T26559
| 1mg | 44.00 € | ||
| 1ml | 92.00 € | ||
| 5mg | 92.00 € | ||
| 10mg | 135.00 € | ||
| 25mg | 274.00 € | ||
| 50mg | 439.00 € | ||
| 100mg | 697.00 € | ||
| 500mg | 1,393.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
L-798106
CAS:244101-02-8
L-798106 (CM9) is an EP3 receptor antagonist that inhibits EP4, EP1, and EP2 receptors and …
Formula:
C27H22BrNO4S
Purity:
98.97%
Color and Shape:
Solid
Molecular weight:
536.44
Ref: TM-T15689
| 1mg | 51.00 € | ||
| 1ml | 127.00 € | ||
| 5mg | 108.00 € | ||
| 10mg | 171.00 € | ||
| 25mg | 341.00 € | ||
| 50mg | 536.00 € | ||
| 100mg | 858.00 € | ||
| 500mg | 1,655.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
PD176252
CAS:204067-01-6
PD176252 is a BB1 and BB2 antagonist, GRPR inhibitor, and FPR1/FPR2 agonist that inhibits the …
Formula:
C32H36N6O5
Purity:
99.18%
Color and Shape:
Solid
Molecular weight:
584.67
Ref: TM-T16449
| 1mg | 35.00 € | ||
| 1ml | 88.00 € | ||
| 5mg | 67.00 € | ||
| 10mg | To inquire | ||
| 25mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Argipressin
CAS:113-79-1
Argipressin is a vasoconstrictive and antidiuretic hormone, binding to V1 receptors with Kd ~1.4 nM …
Formula:
C46H65N15O12S2
Purity:
98%
Color and Shape:
White Powder
Molecular weight:
1084.23
Ref: TM-T7434
| 1mg | 50.00 € | ||
| 2mg | 63.00 € | ||
| 5mg | 89.00 € | ||
| 10mg | 118.00 € | ||
| 25mg | 154.00 € | ||
| 50mg | 177.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Tandospirone
CAS:87760-53-0
Tandospirone (SM-3997) is a selective 5-HT1A partial agonist, Ki: 27 nM, with low affinity for …
Formula:
C21H29N5O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
383.49
Ref: TM-TQ0315
| 1ml | 96.00 € | ||
| 2mg | 47.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
cis-(Z)-Flupentixol dihydrochloride
CAS:51529-01-2
cis-(Z)-Flupentixol dihydrochloride (Emergil) is a dopamine receptor antagonist.
Formula:
C23H27Cl2F3N2OS
Purity:
98.07%
Color and Shape:
Solid
Molecular weight:
507.44
Ref: TM-T2564
| 5mg | 64.00 € | ||
| 10mg | 87.00 € | ||
| 25mg | 176.00 € | ||
| 50mg | 268.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Falcarinol
CAS:21852-80-2
Falcarinol, also known as Panaxynol, is a naturally occurring compound that acts as an orally …
Formula:
C17H24O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
244.37
Ref: TM-TN2360
| 1ml | 199.00 € | ||
| 20mg | 410.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
(Rac)-Rotigotine hydrochloride
CAS:102120-99-0
(Rac)-Rotigotine hydrochloride is a racemate of Rotigotine. Rotigotine is a full agonist of dopamine receptor, …
Formula:
C19H26ClNOS
Color and Shape:
Solid
Molecular weight:
351.93
Ref: TM-T12676
| 1ml | 57.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Eplivanserin (mixture)
CAS:130581-13-4
Eplivanserin mixture is a selective serotonin reuptake inhibitor and a 5-HT2A receptor antagonist,
Formula:
C19H21FN2O2
Color and Shape:
Solid
Molecular weight:
328.387
Ref: TM-T11216
| 2mg | 35.00 € | ||
| 5mg | 49.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Virodhamine
CAS:287937-12-6
Virodhamine (O-arachidonoyl ethanolamine), an endocannabinoid, is an antagonist of CB1 receptor and an agonist of …
Formula:
C22H37NO2
Purity:
98%
Color and Shape:
Soild
Molecular weight:
347.53
Ref: TM-T64371
| 2mg | 52.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
AF-710B
CAS:1235733-73-9
AF710B is an enantiomer of AF710. AF-710B is also a sigma and M1 muscarinic receptors …
Formula:
C20H27N3OS
Purity:
98.62% - 99.89%
Color and Shape:
Solid
Molecular weight:
357.51
Ref: TM-T23649
| 1mg | 311.00 € | ||
| 2mg | 462.00 € | ||
| 5mg | 737.00 € | ||
| 10mg | 1,044.00 € | ||
| 25mg | 1,549.00 € | ||
| 50mg | 2,039.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
SB 243213
CAS:200940-22-3
SB 243213 is a 5-HT2C receptor antagonist with anxiolytic and antidepressant activity used in schizophrenia …
Formula:
C22H19F3N4O2
Purity:
100% - 100%
Color and Shape:
Solid
Molecular weight:
428.41
Ref: TM-T37816
| 1mg | 38.00 € | ||
| 1ml | 87.00 € | ||
| 5mg | 79.00 € | ||
| 10mg | 119.00 € | ||
| 25mg | 270.00 € | ||
| 50mg | 502.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
MRS-3777 hemioxalate
CAS:1186195-57-2
MRS-3777 hemioxalate, a selective adenosine A3 receptor antagonist, reverses the anti-injury perception effects of its …
Formula:
C17H19N5OC2H2O4
Purity:
97.10%
Color and Shape:
Solid
Molecular weight:
354.39
Ref: TM-T12107
| 1mg | 79.00 € | ||
| 5mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
S1RA
CAS:878141-96-9
S1RA (E-52862)(E-52862) is a potent, selective antagonist of the sigma-1 receptor (σ1R, Ki=17 nM), demonstrating …
Formula:
C20H23N3O2
Purity:
99.45%
Color and Shape:
Solid
Molecular weight:
337.42
Ref: TM-T1865
| 1mg | 38.00 € | ||
| 1ml | 86.00 € | ||
| 5mg | 79.00 € | ||
| 10mg | 131.00 € | ||
| 25mg | 212.00 € | ||
| 50mg | 315.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
WZ4141
CAS:1222776-76-2
WZ4141 is an intermediate in compound synthesis.
Formula:
C16H13N3O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
279.29
Ref: TM-T19604
| 1ml | 433.00 € | ||
| 5mg | 439.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Rolofylline
CAS:136199-02-5
Rolofylline (KW-3902) is an adenosine A1 receptor antagonist used to study acute congestive heart failure …
Formula:
C20H28N4O2
Purity:
99.53%
Color and Shape:
Solid
Molecular weight:
356.46
Ref: TM-T16782
| 1mg | 46.00 € | ||
| 1ml | 106.00 € | ||
| 5mg | 90.00 € | ||
| 10mg | 115.00 € | ||
| 25mg | 185.00 € | ||
| 50mg | 274.00 € | ||
| 100mg | 405.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
SB-200646A
CAS:143797-62-0
SB-200646A: oral 5-HT2B/2C antagonist; higher affinity than 5-HT2A (pKi: 7.5, 6.9 vs 5.2); anxiolytic with …
Formula:
C15H15ClN4O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
302.76
Ref: TM-T22423
| 1ml | 83.00 € | ||
| 2mg | 41.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
TP-16
CAS:2332972-26-4
TP-16 is a novel potent and selective EP4 antagonist that blocks the function of IMCs …
Formula:
C24H22FNO4S
Purity:
98.83% - 99.33%
Color and Shape:
Solid
Molecular weight:
439.5
Ref: TM-T62525
| 1mg | 432.00 € | ||
| 5mg | 1,013.00 € | ||
| 25mg | 2,016.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Calcitonin (salmon)
CAS:47931-85-1
Calcitonin (salmon), a calcium regulating hormone, is used to treat osteoporosis in women who are …
Formula:
C145H240N44O48S2
Purity:
99.41%
Color and Shape:
Powder
Molecular weight:
3431.85
Ref: TM-TP1040
| 1mg | 95.00 € | ||
| 5mg | 184.00 € | ||
| 10mg | 268.00 € | ||
| 25mg | 413.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Eticlopride hydrochloride
CAS:97612-24-3
Eticlopride, an antipsychotic, is a Selective dopamine D2/D3 receptor antagonist (Ki: 0.5/0.16 nM).
Formula:
C17H25ClN2O3·HCl
Purity:
98%
Color and Shape:
Solid
Molecular weight:
377.31
Ref: TM-T4007
| 1mg | 49.00 € | ||
| 1ml | 87.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
