G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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SB-674042
CAS:483313-22-0
SB-674042 is a nonpeptide dual antagonist of the appetite peptides OX1 and OX2 receptors.SB-674042 is …
Formula:
C24H21FN4O2S
Purity:
99.9%
Color and Shape:
Solid
Molecular weight:
448.51
Ref: TM-T16854
| 1mg | 49.00 € | ||
| 1mL*10mM (DMSO) | 92.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
MRGPRX4 modulator-2
CAS:2492595-24-9
MRGPRX4 modulator-2 (compound 1-55) is a highly potent antagonist of MRGPRX4 with an IC50 value …
Formula:
C15H9ClF4O3
Purity:
99.24%
Color and Shape:
Liquid
Molecular weight:
348.68
Ref: TM-T61183
| 1mg | 61.00 € | ||
| 5mg | 129.00 € | ||
| 10mg | 199.00 € | ||
| 25mg | To inquire |
Estimated delivery in United States, on Friday 13 Dec 2024
Gastrin I, human
CAS:10047-33-3
Gastrin I, human (Gastrin I (human)) is an endogenous peptide produced in the stomach that …
Formula:
C97H124N20O31S
Purity:
98.62%
Color and Shape:
Coa
Molecular weight:
2098.2
Ref: TM-TP2030
| 1mg | 106.00 € | ||
| 5mg | 398.00 € | ||
| 10mg | 626.00 € | ||
| 25mg | 1,058.00 € | ||
| 50mg | 1,423.00 € | ||
| 100mg | 1,853.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
Rolofylline
CAS:136199-02-5
Rolofylline (KW-3902) is an adenosine A1 receptor antagonist used to study acute congestive heart failure …
Formula:
C20H28N4O2
Purity:
99.53%
Color and Shape:
Solid
Molecular weight:
356.46
Ref: TM-T16782
| 1mg | 46.00 € | ||
| 5mg | 90.00 € | ||
| 10mg | 115.00 € | ||
| 25mg | 185.00 € | ||
| 50mg | 274.00 € | ||
| 100mg | 405.00 € | ||
| 1mL*10mM (DMSO) | 106.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
Asenapine hydrochloride
CAS:1261398-77-9
Asenapine hydrochloride (Org 5222 hydrochloride) is an antagonist of 5-hydroxytryptamine, adrenergic, dopamine, and histamine receptors …
Formula:
C17H17Cl2NO
Color and Shape:
Solid
Molecular weight:
322.23
Ref: TM-T22589
| 1mg | 76.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
Omidenepag
CAS:1187451-41-7
Omidenepag (UR-7276) is an EP2 agonist and a novel topical ocular hypotensive agent.Omidenepag can be …
Formula:
C23H22N6O4S
Purity:
99.67%
Color and Shape:
Solid
Molecular weight:
478.52
Ref: TM-T16389
| 1mg | 76.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
Fenoterol hydrobromide
CAS:1944-12-3
Fenoterol hydrobromide is a beta2-adrenergic receptor agonist and bronchodilator used in the study of cardiovascular …
Formula:
C17H22BrNO4
Color and Shape:
Solid
Molecular weight:
384.27
Ref: TM-T22331
| 10mg | 35.00 € | ||
| 1mL*10mM (DMSO) | 80.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
NCRW0005-F05
CAS:342779-66-2
NCRW0005-F05 is a potent agonist of orphan G-protein coupled receptor GPR139 with an IC 50 …
Formula:
C16H13F2NO2
Purity:
99.48%
Color and Shape:
Liquid
Molecular weight:
289.28
Ref: TM-T60199
| 5mg | 46.00 € | ||
| 10mg | 77.00 € | ||
| 25mg | 144.00 € | ||
| 50mg | 222.00 € | ||
| 100mg | To inquire | ||
| 1mL*10mM (DMSO) | 50.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
Falcarinol
CAS:21852-80-2
Falcarinol, also known as Panaxynol, is a naturally occurring compound that acts as an orally …
Formula:
C17H24O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
244.37
Ref: TM-TN2360
| 20mg | 410.00 € | ||
| 1mL*10mM (DMSO) | 199.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
Trabodenoson
CAS:871108-05-3
Trabodenoson (INO-8875) is a selective and potent adenosine A1 receptor agonist, an adenosine analog, for …
Formula:
C15H20N6O6
Purity:
99.94%
Color and Shape:
Solid
Molecular weight:
380.36
Ref: TM-T34914
| 1mg | 128.00 € | ||
| 2mg | 182.00 € | ||
| 5mg | 307.00 € | ||
| 10mg | 460.00 € | ||
| 25mg | 736.00 € | ||
| 50mg | 1,000.00 € | ||
| 100mg | 1,336.00 € | ||
| 1mL*10mM (DMSO) | 343.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
Atogepant
CAS:1374248-81-3
Atogepant (MK-8031) is an orally available, selective and potent calcitonin gene-related peptide receptor (CGRP) antagonist …
Formula:
C29H23F6N5O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
603.52
Ref: TM-T26682
| 1mg | 159.00 € | ||
| 5mg | 383.00 € | ||
| 10mg | 568.00 € | ||
| 25mg | 888.00 € | ||
| 50mg | 1,205.00 € | ||
| 100mg | 1,621.00 € | ||
| 500mg | 3,295.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
Agomelatine (L(+)-Tartaric acid)
CAS:824393-18-2
Agomelatine (S-20098) L(+)-Tartaric acid is a specific agonist of MT1 and MT2 receptors (Kis: 0.1, …
Formula:
C19H23NO8
Color and Shape:
Solid
Molecular weight:
393.39
Ref: TM-T10267
| 2mg | 40.00 € | ||
| 5mg | 57.00 € | ||
| 1mL*10mM (DMSO) | 64.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
MRS-3777 hemioxalate
CAS:1186195-57-2
MRS-3777 hemioxalate, a selective adenosine A3 receptor antagonist, reverses the anti-injury perception effects of its …
Formula:
C17H19N5OC2H2O4
Purity:
97.10%
Color and Shape:
Solid
Molecular weight:
354.39
Ref: TM-T12107
| 1mg | 77.00 € | ||
| 5mg | To inquire |
Estimated delivery in United States, on Friday 13 Dec 2024
Degarelix
CAS:214766-78-6
Degarelix is a competitive and reversible gonadotropin-releasing hormone receptor (GnRHR) antagonist.
Formula:
C82H103ClN18O16
Color and Shape:
Solid
Molecular weight:
1632.26
Ref: TM-T10988
| 50mg | 793.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
BMS-986224
CAS:2055200-88-7
BMS-986224 is an orally active, potent and selective APJ receptor agonist.BMS-986224 is a candidate compound …
Formula:
C24H23ClN4O6
Purity:
98.61% - 98.82%
Color and Shape:
Solid
Molecular weight:
498.92
Ref: TM-T39448
| 1mg | 379.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
PD176252
CAS:204067-01-6
PD176252 is a BB1 and BB2 antagonist, GRPR inhibitor, and FPR1/FPR2 agonist that inhibits the …
Formula:
C32H36N6O5
Purity:
99.18%
Color and Shape:
Solid
Molecular weight:
584.67
Ref: TM-T16449
| 1mg | 35.00 € | ||
| 5mg | 67.00 € | ||
| 10mg | To inquire | ||
| 25mg | To inquire | ||
| 1mL*10mM (DMSO) | 88.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
Taranabant racemate
CAS:701977-00-6
Taranabant racemate is an antagonist and/or inverse agonist of the Cannabinoid-1 (CB1) receptor.
Formula:
C27H25ClF3N3O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
515.95
Ref: TM-T13081
| 2mg | 50.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
Argipressin
CAS:113-79-1
Argipressin is a vasoconstrictive and antidiuretic hormone, binding to V1 receptors with Kd ~1.4 nM …
Formula:
C46H65N15O12S2
Purity:
98%
Color and Shape:
White Powder
Molecular weight:
1084.23
Ref: TM-T7434
| 1mg | 50.00 € | ||
| 5mg | 89.00 € | ||
| 10mg | 118.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
GW-1100
CAS:306974-70-9
GW-1100 is a selective GPR40 and FFAR1 antagonist for the study of diabetes and metabolic …
Formula:
C27H25FN4O4S
Purity:
97.01%
Color and Shape:
Solid
Molecular weight:
520.58
Ref: TM-T15448
| 1mg | 36.00 € | ||
| 5mg | To inquire |
Estimated delivery in United States, on Friday 13 Dec 2024
UCSF924
CAS:1434515-70-4
UCSF924 is a potent and specific agonist of dopamine D4 receptor (DRD4) partial (EC50: 4.2 …
Formula:
C20H22N2O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
322.4
Ref: TM-T13245
| 2mg | 91.00 € | ||
| 1mL*10mM (DMSO) | 205.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
