G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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NCRW0005-F05
CAS:342779-66-2
NCRW0005-F05 is a potent agonist of orphan G-protein coupled receptor GPR139 with an IC 50 …
Formula:
C16H13F2NO2
Purity:
99.48%
Color and Shape:
Solid
Molecular weight:
289.28
Ref: TM-T60199
| 5mg | 46.00 € | ||
| 10mg | 77.00 € | ||
| 25mg | 144.00 € | ||
| 50mg | 222.00 € | ||
| 100mg | To inquire | ||
| 1mL*10mM (DMSO) | 50.00 € |
Estimated delivery in United States, on Wednesday 27 Nov 2024
CGP 20712 A
CAS:105737-62-0
CGP 20712 A (CGP 20712 mesylate) is a β1-adrenergic receptor antagonist with antihypertensive activity that …
Formula:
C24H29F3N4O8S
Purity:
99.37%
Color and Shape:
Solid
Molecular weight:
590.57
Ref: TM-T10778
| 1mg | 95.00 € | ||
| 5mg | 271.00 € | ||
| 10mg | 401.00 € | ||
| 25mg | 654.00 € | ||
| 50mg | 907.00 € | ||
| 100mg | 1,199.00 € | ||
| 200mg | 1,649.00 € |
Estimated delivery in United States, on Wednesday 27 Nov 2024
Poly-D-lysine hydrobromide (MW 30000-70000)
CAS:27964-99-4
Poly-D-lysine hydrobromide (MW 30000-70000) (Poly-D-lysine HBr) is a peptide CaSR agonist that removes proteinase K-resistant …
Formula:
(C6H14N2O2)x·xHBr
Color and Shape:
Solid
Molecular weight:
227.102
Ref: TM-T40363
| 5mg | 35.00 € | ||
| 10mg | 52.00 € | ||
| 25mg | 95.00 € | ||
| 50mg | 150.00 € | ||
| 100mg | 212.00 € |
Estimated delivery in United States, on Wednesday 27 Nov 2024
Dihydromunduletone
CAS:674786-20-0
Dihydromunduletone (DHM) is an adhesion G protein-coupled receptor (aGPCR) antagonist inhibits GPR56 and GPR114/ADGRG5, which …
Formula:
C25H28O6
Purity:
99.96%
Color and Shape:
Solid
Molecular weight:
424.49
Ref: TM-T11044
| 1mg | 172.00 € |
Estimated delivery in United States, on Wednesday 27 Nov 2024
Maropitant citrate
CAS:359875-09-5
Maropitant citrate is a useful organic compound for research related to life sciences. The catalog …
Formula:
C38H50N2O9
Color and Shape:
Solid
Molecular weight:
678.81
Ref: TM-T35344
| 500mg | 1,282.00 € |
Estimated delivery in United States, on Wednesday 27 Nov 2024
AF-710B
CAS:1235733-73-9
AF710B is an enantiomer of AF710. AF-710B is also a sigma and M1 muscarinic receptors …
Formula:
C20H27N3OS
Purity:
98.62% - 99.89%
Color and Shape:
Solid
Molecular weight:
357.51
Ref: TM-T23649
| 1mg | 311.00 € | ||
| 2mg | 462.00 € | ||
| 5mg | 737.00 € | ||
| 10mg | 1,044.00 € | ||
| 25mg | 1,549.00 € | ||
| 50mg | 2,039.00 € |
Estimated delivery in United States, on Wednesday 27 Nov 2024
(R)-Mirtazapine
CAS:61364-37-2
(R)-Mirtazapine ((R)-Org3770) is a 5-HT3 receptor antagonist, a potential analgesic with anti-injury perception properties.
Formula:
C17H19N3
Purity:
99.75%
Color and Shape:
Solid
Molecular weight:
265.35
Ref: TM-T12632
| 1mg | 56.00 € | ||
| 5mg | 119.00 € | ||
| 10mg | 185.00 € | ||
| 25mg | 324.00 € | ||
| 50mg | 481.00 € | ||
| 100mg | 685.00 € |
Estimated delivery in United States, on Wednesday 27 Nov 2024
Rizatriptan
CAS:144034-80-0
Rizatriptan (Risatriptan) is a selective 5-hydroxytryptamine 1B/1D receptor agonist used in the study of migraine.
Formula:
C15H19N5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
269.35
Ref: TM-T1734L
| 5mg | 35.00 € | ||
| 10mg | 47.00 € | ||
| 25mg | 68.00 € | ||
| 50mg | 88.00 € | ||
| 100mg | 131.00 € |
Estimated delivery in United States, on Wednesday 27 Nov 2024
Falcarinol
CAS:21852-80-2
Falcarinol, also known as Panaxynol, is a naturally occurring compound that acts as an orally …
Formula:
C17H24O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
244.37
Ref: TM-TN2360
| 20mg | 410.00 € | ||
| 1mL*10mM (DMSO) | 199.00 € |
Estimated delivery in United States, on Wednesday 27 Nov 2024
GRK6-IN-2
CAS:2677786-27-3
GRK6-IN-2 is a potent G protein-coupled receptor kinase 6 (GRK6) inhibitor with potential antitumor activity.GRK6-IN-2 …
Formula:
C21H21FN6
Purity:
98.94%
Color and Shape:
Solid
Molecular weight:
376.43
Ref: TM-T61556
| 2mg | 61.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 157.00 € | ||
| 25mg | 301.00 € | ||
| 50mg | 462.00 € | ||
| 100mg | 694.00 € |
Estimated delivery in United States, on Wednesday 27 Nov 2024
Calcitonin (salmon)
CAS:47931-85-1
Calcitonin (salmon), a calcium regulating hormone, is used to treat osteoporosis in women who are …
Formula:
C145H240N44O48S2
Purity:
99.41%
Color and Shape:
Powder
Molecular weight:
3431.85
Ref: TM-TP1040
| 1mg | 95.00 € | ||
| 5mg | 184.00 € | ||
| 10mg | 268.00 € | ||
| 25mg | 413.00 € |
Estimated delivery in United States, on Wednesday 27 Nov 2024
Fenoprofen
CAS:29679-58-1
Fenoprofen (LILLY-5385) is a non-steroidal anti-inflammatory compound and a modifier enhancer of the melanocortin receptor, …
Formula:
C15H14O3
Color and Shape:
Solid
Molecular weight:
242.27
Ref: TM-T0184L
| 10mg | 35.00 € | ||
| 25mg | 52.00 € | ||
| 50mg | 66.00 € | ||
| 100mg | 94.00 € | ||
| 500mg | 196.00 € |
Estimated delivery in United States, on Wednesday 27 Nov 2024
Atosiban
CAS:90779-69-4
Atosiban (RW22164), an oxytocin/vasopressin inhibitor, halts premature labor as an intravenous tocolytic, reducing uterine contractions …
Formula:
C43H67N11O12S2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
994.19
Ref: TM-T4996
| 5mg | 67.00 € | ||
| 10mg | 90.00 € | ||
| 50mg | 203.00 € | ||
| 100mg | 295.00 € |
Estimated delivery in United States, on Wednesday 27 Nov 2024
Spiroxatrine
CAS:1054-88-2
Spiroxatrine (R 5188) is a 5-HT1α and α2-adrenergic dual antagonist with sedative activity for the …
Formula:
C22H25N3O3
Purity:
99.83%
Color and Shape:
Solid
Molecular weight:
379.45
Ref: TM-T23382
| 5mg | 86.00 € | ||
| 10mg | 123.00 € | ||
| 25mg | 245.00 € | ||
| 50mg | 392.00 € | ||
| 100mg | 569.00 € |
Estimated delivery in United States, on Wednesday 27 Nov 2024
Sumanirole maleate
CAS:179386-44-8
Sumanirole maleate (U-95666E) is a highly selective full agonist of the D2 receptor (ED50: 46 …
Formula:
C15H17N3O5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
319.31
Ref: TM-TQ0140
| 2mg | 89.00 € |
Estimated delivery in United States, on Wednesday 27 Nov 2024
Citalopram
CAS:59729-33-8
Citalopram (Lu 10-171), a serotonin and 5-HT reuptake inhibitor.Citalopram has antidepressant activity and may be …
Formula:
C20H21FN2O
Purity:
99.89%
Color and Shape:
Solid
Molecular weight:
324.39
Ref: TM-T20828
| 25mg | 35.00 € | ||
| 50mg | 48.00 € | ||
| 100mg | 69.00 € | ||
| 500mg | 147.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Wednesday 27 Nov 2024
Atipamezole
CAS:104054-27-5
Atipamezole (Antisedan) is a synthetic α2 adrenergic receptor antagonist. It has also been researched in …
Formula:
C14H16N2
Purity:
99.76%
Color and Shape:
Off-White To Light Yellow Crystal Powder
Molecular weight:
212.29
Ref: TM-T6766
| 5mg | 35.00 € | ||
| 10mg | 48.00 € | ||
| 25mg | 92.00 € | ||
| 50mg | 145.00 € | ||
| 100mg | 210.00 € | ||
| 200mg | 312.00 € | ||
| 1mL*10mM (DMSO) | 35.00 € |
Estimated delivery in United States, on Wednesday 27 Nov 2024
MRS-3777 hemioxalate
CAS:1186195-57-2
MRS-3777 hemioxalate, a selective adenosine A3 receptor antagonist, reverses the anti-injury perception effects of its …
Formula:
C17H19N5OC2H2O4
Purity:
97.10%
Color and Shape:
Solid
Molecular weight:
354.39
Ref: TM-T12107
| 1mg | 75.00 € | ||
| 5mg | To inquire |
Estimated delivery in United States, on Wednesday 27 Nov 2024
BMS-986278
CAS:2170126-74-4
BMS-986278 is an orally active and potent hemophosphatidic acid receptor 1 (LPA1) antagonist with Kb …
Formula:
C22H31N5O5
Purity:
99.86%
Color and Shape:
Solid
Molecular weight:
445.51
Ref: TM-T39647
| 1mg | 68.00 € | ||
| 5mg | 148.00 € | ||
| 10mg | 200.00 € | ||
| 25mg | 362.00 € | ||
| 50mg | 492.00 € | ||
| 1mL*10mM (DMSO) | 160.00 € |
Estimated delivery in United States, on Wednesday 27 Nov 2024
Fedovapagon
CAS:347887-36-9
Fedovapagon (VA106483) is a pressin V2 receptor (V2R) agonist for the study of overactive bladder …
Formula:
C27H34N4O3
Purity:
99.33%
Color and Shape:
Solid
Molecular weight:
462.58
Ref: TM-T15273
| 5mg | 109.00 € | ||
| 10mg | 172.00 € | ||
| 25mg | 364.00 € | ||
| 50mg | 640.00 € | ||
| 100mg | 904.00 € | ||
| 1mL*10mM (DMSO) | 123.00 € |
Estimated delivery in United States, on Wednesday 27 Nov 2024
