G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Fenoprofen
CAS:29679-58-1
Fenoprofen (LILLY-5385) is a non-steroidal anti-inflammatory compound and a modifier enhancer of the melanocortin receptor, …
Formula:
C15H14O3
Purity:
98.4%
Color and Shape:
Solid
Molecular weight:
242.27
Ref: TM-T0184L
| 10mg | 35.00 € | ||
| 25mg | 52.00 € | ||
| 50mg | 66.00 € | ||
| 100mg | 95.00 € | ||
| 500mg | 198.00 € |
Estimated delivery in United States, on Thursday 6 Mar 2025
SB-674042
CAS:483313-22-0
SB-674042 is a nonpeptide dual antagonist of the appetite peptides OX1 and OX2 receptors.SB-674042 is …
Formula:
C24H21FN4O2S
Purity:
99.9%
Color and Shape:
Solid
Molecular weight:
448.51
Ref: TM-T16854
| 1mg | 49.00 € | ||
| 1mL*10mM (DMSO) | 93.00 € |
Estimated delivery in United States, on Thursday 6 Mar 2025
Calcitonin (salmon)
CAS:47931-85-1
Calcitonin (salmon), a calcium regulating hormone, is used to treat osteoporosis in women who are …
Formula:
C145H240N44O48S2
Purity:
99.41%
Color and Shape:
Powder
Molecular weight:
3431.85
Ref: TM-TP1040
| 1mg | 97.00 € | ||
| 5mg | 188.00 € | ||
| 10mg | 274.00 € | ||
| 25mg | 423.00 € |
Estimated delivery in United States, on Thursday 6 Mar 2025
AF-710B
CAS:1235733-73-9
AF710B is an enantiomer of AF710. AF-710B is also a sigma and M1 muscarinic receptors …
Formula:
C20H27N3OS
Purity:
98.62% - 99.89%
Color and Shape:
Solid
Molecular weight:
357.51
Ref: TM-T23649
| 1mg | 316.00 € | ||
| 2mg | 470.00 € | ||
| 5mg | 750.00 € | ||
| 10mg | 1,064.00 € | ||
| 25mg | 1,586.00 € | ||
| 50mg | 2,072.00 € |
Estimated delivery in United States, on Thursday 6 Mar 2025
GW-1100
CAS:306974-70-9
GW-1100 is a selective GPR40 and FFAR1 antagonist for the study of diabetes and metabolic …
Formula:
C27H25FN4O4S
Purity:
97.01%
Color and Shape:
Solid
Molecular weight:
520.58
Ref: TM-T15448
| 1mg | 34.00 € | ||
| 5mg | To inquire |
Estimated delivery in United States, on Thursday 6 Mar 2025
Fexofenadine-d6
CAS:548783-71-7
Fexofenadine D6 is an antihistamine pharmaceutical drug.Fexofenadine D6 is deuterium labeled is Fexofenadine.
Formula:
C32H39NO4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
507.69
Ref: TM-T11276
| 1mg | 160.00 € | ||
| 5mg | 512.00 € |
Estimated delivery in United States, on Thursday 6 Mar 2025
MRGPRX4 modulator-2
CAS:2492595-24-9
MRGPRX4 modulator-2 (compound 1-55) is a highly potent antagonist of MRGPRX4 with an IC50 value …
Formula:
C15H9ClF4O3
Purity:
99.24%
Color and Shape:
Liquid
Molecular weight:
348.68
Ref: TM-T61183
| 1mg | 62.00 € | ||
| 5mg | 130.00 € | ||
| 10mg | 204.00 € | ||
| 25mg | To inquire |
Estimated delivery in United States, on Thursday 6 Mar 2025
Agomelatine (L(+)-Tartaric acid)
CAS:824393-18-2
Agomelatine (S-20098) L(+)-Tartaric acid is a specific agonist of MT1 and MT2 receptors (Kis: 0.1, …
Formula:
C19H23NO8
Color and Shape:
Solid
Molecular weight:
393.39
Ref: TM-T10267
| 2mg | 40.00 € | ||
| 5mg | 57.00 € | ||
| 1mL*10mM (DMSO) | 64.00 € |
Estimated delivery in United States, on Thursday 6 Mar 2025
PF-543 Citrate
CAS:1415562-83-2
PF-543 Citrate is an inhibitor of sphingosine-competitive SPHK1(IC50 of 2 nM ).
Formula:
C33H39NO11S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
657.73
Ref: TM-T12436
| 2mg | 52.00 € | ||
| 5mg | 84.00 € |
Estimated delivery in United States, on Thursday 6 Mar 2025
Atogepant
CAS:1374248-81-3
Atogepant (MK-8031) is an orally available, selective and potent calcitonin gene-related peptide receptor (CGRP) antagonist …
Formula:
C29H23F6N5O3
Purity:
99.66%
Color and Shape:
Solid
Molecular weight:
603.52
Ref: TM-T26682
| 1mg | 166.00 € | ||
| 5mg | 401.00 € | ||
| 10mg | 595.00 € | ||
| 25mg | 932.00 € | ||
| 50mg | 1,264.00 € | ||
| 100mg | 1,700.00 € | ||
| 500mg | 3,457.00 € |
Estimated delivery in United States, on Thursday 6 Mar 2025
Tamsulosin
CAS:106133-20-4
Tamsulosin: an alpha1A blocker for easing urination in BPH by relaxing prostate and bladder muscles.
Formula:
C20H28N2O5S
Purity:
99.94%
Color and Shape:
White Crystals
Molecular weight:
408.51
Ref: TM-T0210L
| 10mg | 35.00 € | ||
| 25mg | 52.00 € | ||
| 50mg | 74.00 € | ||
| 100mg | 97.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Thursday 6 Mar 2025
Degarelix
CAS:214766-78-6
Degarelix is a competitive and reversible gonadotropin-releasing hormone receptor (GnRHR) antagonist.
Formula:
C82H103ClN18O16
Color and Shape:
Solid
Molecular weight:
1632.26
Ref: TM-T10988
| 50mg | 805.00 € |
Estimated delivery in United States, on Thursday 6 Mar 2025
(S)-Mirtazapine
CAS:61337-87-9
(S)-Mirtazapine ((S)-Org3770) is a 5-HT2 receptor antagonist with pro-nociceptive effects that can be used to …
Formula:
C17H19N3
Purity:
99.37%
Color and Shape:
Solid
Molecular weight:
265.35
Ref: TM-T12632L
| 1mg | 57.00 € | ||
| 5mg | 120.00 € | ||
| 10mg | 188.00 € | ||
| 25mg | 432.00 € | ||
| 50mg | 622.00 € | ||
| 100mg | 873.00 € |
Estimated delivery in United States, on Thursday 6 Mar 2025
Apraclonidine hydrochloride
CAS:73218-79-8
Apraclonidine hydrochloride (ALO 2145) is an α2-adrenergic agonist and a weak α-1 adrenergic receptor agonist.
Formula:
C9H11Cl3N4
Purity:
98.01%
Color and Shape:
Solid
Molecular weight:
281.57
Ref: TM-T21371
| 10mg | 52.00 € | ||
| 25mg | 88.00 € | ||
| 50mg | 116.00 € | ||
| 100mg | 168.00 € | ||
| 200mg | 235.00 € | ||
| 1mL*10mM (DMSO) | 35.00 € |
Estimated delivery in United States, on Thursday 6 Mar 2025
BMS-986224
CAS:2055200-88-7
BMS-986224 is an orally active, potent and selective APJ receptor agonist.BMS-986224 is a candidate compound …
Formula:
C24H23ClN4O6
Purity:
98.61% - 98.82%
Color and Shape:
Solid
Molecular weight:
498.92
Ref: TM-T39448
| 1mg | 379.00 € |
Estimated delivery in United States, on Thursday 6 Mar 2025
Taranabant racemate
CAS:701977-00-6
Taranabant racemate is an antagonist and/or inverse agonist of the Cannabinoid-1 (CB1) receptor.
Formula:
C27H25ClF3N3O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
515.95
Ref: TM-T13081
| 2mg | 50.00 € |
Estimated delivery in United States, on Thursday 6 Mar 2025
Nebentan potassium
CAS:342005-82-7
Nebentan potassium (YM598) is an ETA receptor antagonist that inhibits pulmonary arterial hypertension and is …
Formula:
C24H20KN5O5S
Purity:
98.92%
Color and Shape:
Solid
Molecular weight:
529.61
Ref: TM-T36008
| 1mg | 92.00 € | ||
| 2mg | 120.00 € | ||
| 5mg | 188.00 € | ||
| 10mg | 311.00 € | ||
| 25mg | 550.00 € | ||
| 50mg | 882.00 € | ||
| 100mg | 1,198.00 € | ||
| 500mg | 2,403.00 € | ||
| 1mL*10mM (DMSO) | 226.00 € |
Estimated delivery in United States, on Thursday 6 Mar 2025
cis-(Z)-Flupentixol dihydrochloride
CAS:51529-01-2
cis-(Z)-Flupentixol dihydrochloride (Emergil) is a dopamine receptor antagonist.
Formula:
C23H27Cl2F3N2OS
Purity:
98.07%
Color and Shape:
Solid
Molecular weight:
507.44
Ref: TM-T2564
| 5mg | 59.00 € | ||
| 10mg | 87.00 € | ||
| 25mg | 167.00 € | ||
| 50mg | 265.00 € |
Estimated delivery in United States, on Thursday 6 Mar 2025
Kynurenic acid
CAS:492-27-3
Kynurenic acid (Quinurenic acid) is an NMDA, glutamate, α7 nicotinic acetylcholine receptor triple antagonist and …
Formula:
C10H7NO3
Purity:
99.69%
Color and Shape:
Liquid
Molecular weight:
189.17
Ref: TM-T65135
| 50mg | 37.00 € |
Estimated delivery in United States, on Thursday 6 Mar 2025
Docosahexaenoic acid ethyl ester
CAS:81926-94-5
Docosahexaenoic acid ethyl ester (Ethyl docosahexaenoate) enhances 6-hydroxydopamine-induced neuronal damage by inducing lipid peroxidation in …
Formula:
C24H36O2
Color and Shape:
Solid
Molecular weight:
356.54
Ref: TM-T41321
| 50mg | 37.00 € | ||
| 100mg | 52.00 € | ||
| 500mg | 127.00 € |
Estimated delivery in United States, on Thursday 6 Mar 2025
