G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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WIN 51,708
CAS:144177-30-0
WIN 51,708 is an antagonist of neurokinin-1 receptor.
Formula:
C29H33N3O
Purity:
99%
Color and Shape:
Solid
Molecular weight:
439.59
Ref: TM-T29157
| 1mg | 279.00 € | ||
| 2mg | 414.00 € | ||
| 5mg | 685.00 € | ||
| 10mg | 938.00 € | ||
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
NCRW0005-F05
CAS:342779-66-2
NCRW0005-F05 is a potent agonist of orphan G-protein coupled receptor GPR139 with an IC 50 …
Formula:
C16H13F2NO2
Purity:
99.48%
Color and Shape:
Liquid
Molecular weight:
289.28
Ref: TM-T60199
| 10mg | 50.00 € | ||
| 25mg | 87.00 € | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 35.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
BAN ORL 24 dihydrochloride
CAS:1401463-54-4
BAN ORL 24 dihydrochloride is a highly potent nociceptin/orphan FQ (N/OFQ) receptor (NOP) antagonist that …
Formula:
C27H37Cl2N3O2
Purity:
95.03%
Color and Shape:
Solid
Molecular weight:
506.51
Ref: TM-T10457
| 2mg | 81.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
Ozanimod hydrochloride
CAS:1618636-37-5
Ozanimod (RPC-1063) HCl is a selective S1P1/S1P5 modulator with high affinity, used in relapsing MS …
Formula:
C23H25ClN4O3
Purity:
99.81%
Color and Shape:
Liquid
Molecular weight:
440.92
Ref: TM-T62552
| 1mg | 66.00 € | ||
| 5mg | 139.00 € | ||
| 10mg | 202.00 € | ||
| 25mg | 416.00 € | ||
| 50mg | 652.00 € | ||
| 100mg | 938.00 € | ||
| 500mg | 1,872.00 € | ||
| 1mL*10mM (DMSO) | 154.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
Neurotensin(8-13)
CAS:60482-95-3
Neurotensin(8-13) is Neurotensin (NT) fragment, Neurotensin(8-13) results in a decrease in cell-surface NT1 receptors (NTR1) …
Formula:
C38H64N12O8
Purity:
99.95%
Color and Shape:
Solid
Molecular weight:
816.99
Ref: TM-T7617
| 1mg | 170.00 € | ||
| 2mg | 274.00 € | ||
| 5mg | 406.00 € | ||
| 10mg | 787.00 € | ||
| 25mg | To inquire | ||
| 50mg | To inquire | ||
| 100mg | To inquire |
Estimated delivery in United States, on Monday 31 Mar 2025
Dehydroaripiprazole
CAS:129722-25-4
Dehydroaripiprazole (DM-14857), aripiprazole's active metabolite, is formed by CYP3A4 and CYP2D6, with similar antipsychotic effects.
Formula:
C23H25Cl2N3O2
Purity:
97.05%
Color and Shape:
Solid
Molecular weight:
446.37
Ref: TM-T10989
| 1mg | 37.00 € | ||
| 5mg | 79.00 € | ||
| 10mg | 119.00 € | ||
| 25mg | 235.00 € | ||
| 50mg | 349.00 € | ||
| 100mg | 515.00 € | ||
| 500mg | 1,103.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
Argipressin
CAS:113-79-1
Argipressin is a vasoconstrictive and antidiuretic hormone, binding to V1 receptors with Kd ~1.4 nM …
Formula:
C46H65N15O12S2
Purity:
98%
Color and Shape:
White Powder
Molecular weight:
1084.23
Ref: TM-T7434
| 1mg | 50.00 € | ||
| 5mg | 89.00 € | ||
| 10mg | 118.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
Clothiapine
CAS:2058-52-8
Clothiapine is an atypical antipsychotic of the dibenzothiazepine chemical class.
Formula:
C18H18ClN3S
Purity:
99.93%
Color and Shape:
Solid
Molecular weight:
343.87
Ref: TM-T23900
| 1mg | 98.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
L-α-lysophosphatidylinositol sodium
CAS:796963-91-2
L-α-lysophosphatidylinositol sodium is an endogenous ligand of GPR55 and an endocannabinoid neurotransmitter.
Formula:
C25H48NaO12P
Color and Shape:
Liquid
Molecular weight:
594.6
Ref: TM-T77212
| 1mg | To inquire |
Estimated delivery in United States, on Monday 31 Mar 2025
PD176252
CAS:204067-01-6
PD176252 is a BB1 and BB2 antagonist, GRPR inhibitor, and FPR1/FPR2 agonist that inhibits the …
Formula:
C32H36N6O5
Purity:
99.18%
Color and Shape:
Solid
Molecular weight:
584.67
Ref: TM-T16449
| 1mg | 35.00 € | ||
| 5mg | 67.00 € | ||
| 10mg | To inquire | ||
| 25mg | To inquire | ||
| 1mL*10mM (DMSO) | 88.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
Levocetirizine Dihydrochloride
CAS:130018-87-0
Levocetirizine Dihydrochloride is a third-gen antihistamine targeting H1-receptors, treating allergies and urticaria.
Formula:
C21H27Cl3N2O3
Purity:
99.75%
Color and Shape:
White Or Off-White Crystalline Powder
Molecular weight:
461.81
Ref: TM-T22354
| 1g | 692.00 € | ||
| 10mg | 50.00 € | ||
| 25mg | 86.00 € | ||
| 50mg | 131.00 € | ||
| 100mg | 188.00 € | ||
| 200mg | 283.00 € | ||
| 500mg | 487.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
(S)-Mirtazapine
CAS:61337-87-9
(S)-Mirtazapine ((S)-Org3770) is a 5-HT2 receptor antagonist with pro-nociceptive effects that can be used to …
Formula:
C17H19N3
Purity:
99.37%
Color and Shape:
Solid
Molecular weight:
265.35
Ref: TM-T12632L
| 1mg | 57.00 € | ||
| 5mg | 120.00 € | ||
| 10mg | 188.00 € | ||
| 25mg | 432.00 € | ||
| 50mg | 622.00 € | ||
| 100mg | 873.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
Poly-D-lysine hydrobromide (MW 30000-70000)
CAS:27964-99-4
Poly-D-lysine hydrobromide (MW 30000-70000) (Poly-D-lysine HBr) is a peptide CaSR agonist that removes proteinase K-resistant …
Formula:
(C6H14N2O2)x·xHBr
Color and Shape:
Liquid
Molecular weight:
227.102
Ref: TM-T40363
| 5mg | 35.00 € | ||
| 10mg | 52.00 € | ||
| 25mg | 97.00 € | ||
| 50mg | 154.00 € | ||
| 100mg | 216.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
Canagliflozin hemihydrate
CAS:928672-86-0
Canagliflozin hemihydrate (TA 7284) treats type 2 diabetes by blocking SGLT2, leading to glucose excretion …
Formula:
C48H52F2O11S2
Purity:
99.42% - 99.96%
Color and Shape:
Solid
Molecular weight:
907.05
Ref: TM-T1782L
| 1g | 120.00 € | ||
| 100mg | 37.00 € | ||
| 500mg | 88.00 € | ||
| 1mL*10mM (DMSO) | 42.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
Alfuzosin
CAS:81403-80-7
Alfuzosin (SL 77499) is an alpha-1 adrenergic antagonist used to treat benign prostatic hypertrophy and …
Formula:
C19H27N5O4
Purity:
99.64%
Color and Shape:
White Crystaline Powder
Molecular weight:
389.45
Ref: TM-T22232
| 10mg | 48.00 € | ||
| 25mg | 81.00 € | ||
| 50mg | 120.00 € | ||
| 100mg | 187.00 € | ||
| 500mg | 472.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
BW 723C86
CAS:160521-72-2
BW 723C86 is a 5-HT2B receptor agonist with anxiolytic effects, inducing overeating and reduced grooming …
Formula:
C16H19ClN2OS
Purity:
99.35%
Color and Shape:
Solid
Molecular weight:
322.85
Ref: TM-T21625
| 2mg | 62.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
BMS-986278
CAS:2170126-74-4
BMS-986278 is an orally active and potent hemophosphatidic acid receptor 1 (LPA1) antagonist with Kb …
Formula:
C22H31N5O5
Purity:
99.86%
Color and Shape:
Liquid
Molecular weight:
445.51
Ref: TM-T39647
| 1mg | 70.00 € | ||
| 5mg | 154.00 € | ||
| 10mg | 207.00 € | ||
| 25mg | 376.00 € | ||
| 50mg | 512.00 € | ||
| 1mL*10mM (DMSO) | 166.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
Fexofenadine-d6
CAS:548783-71-7
Fexofenadine D6 is an antihistamine pharmaceutical drug.Fexofenadine D6 is deuterium labeled is Fexofenadine.
Formula:
C32H39NO4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
507.69
Ref: TM-T11276
| 1mg | 160.00 € | ||
| 5mg | 512.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
Ketanserin tartrate
CAS:83846-83-7
Ketanserin tartrate (KJK-945 tartrate) is a 5-HT2A receptor and α1-adrenergic receptor antagonist for the study …
Formula:
C26H28FN3O9
Purity:
99.68%
Color and Shape:
Solid
Molecular weight:
545.51
Ref: TM-T1066L
| 25mg | 37.00 € | ||
| 50mg | 52.00 € | ||
| 100mg | 67.00 € | ||
| 1mL*10mM (DMSO) | 35.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
UCM 608
CAS:151889-03-1
UCM 608 (2-Phenylmelatonin) is an antagonist of melatonin-induced contractile responses at low concentrations and induces …
Formula:
C19H20N2O2
Purity:
98.88%
Color and Shape:
Solid
Molecular weight:
308.37
Ref: TM-T22499
| 2mg | 50.00 € | ||
| 5mg | 79.00 € | ||
| 10mg | 97.00 € | ||
| 25mg | 165.00 € | ||
| 50mg | 235.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
