G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Azaphen
CAS:24853-80-3
Azaphen (Pipofezin hydrochloride) is the reuptake of serotonin inhibitor.with antidepressant action and has sedative effects, …
Formula:
C16H21Cl2N5O
Purity:
97.62%
Color and Shape:
Solid
Molecular weight:
370.28
Ref: TM-T7521
| 1ml | 45.00 € | ||
| 25mg | 46.00 € | ||
| 50mg | 60.00 € | ||
| 100mg | 86.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
Nomifensine maleate
CAS:32795-47-4
Nomifensine maleate (Nomifensine (maleate)) is a selective inhibitor of dopamine uptake. Nomifensine maleate is used …
Formula:
C20H22N2O4
Purity:
98.46%
Color and Shape:
Solid
Molecular weight:
354.4
Ref: TM-T7070
| 10mg | 44.00 € | ||
| 25mg | 64.00 € | ||
| 50mg | 94.00 € | ||
| 100mg | 152.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
Pregnenolone acetate
CAS:1778-02-5
Pregnenolone acetate inhibits CB1 receptors, blocking THC effects and shielding the brain from cannabis intoxication.
Formula:
C23H34O3
Purity:
99.66%
Color and Shape:
White To Light Yellow Crystalline Powder
Molecular weight:
358.51
Ref: TM-TC0019
| 5mg | 35.00 € | ||
| 10mg | 52.00 € | ||
| 25mg | 82.00 € | ||
| 50mg | 109.00 € | ||
| 100mg | 163.00 € | ||
| 200mg | 232.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
SNAP 94847 hydrochloride
CAS:1781934-47-1
SNAP 94847 hydrochloride is a melanin-concentrating hormonereceptor1 (MCHR1) antagonist(Ki= 2.2 nM)
Formula:
C29H33ClF2N2O2
Purity:
100% - 99.85%
Color and Shape:
Solid
Molecular weight:
515.03
Ref: TM-T8004
| 2mg | 41.00 € | ||
| 5mg | 62.00 € | ||
| 10mg | 93.00 € | ||
| 25mg | 181.00 € | ||
| 50mg | 306.00 € | ||
| 100mg | 440.00 € | ||
| 200mg | 613.00 € | ||
| 1mL*10mM (DMSO) | 69.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
ONO-AE3-208
CAS:402473-54-5
ONO-AE3-208 (AE 3-208) is an EP4 antagonist. It suppresses cell migration, invasion, and metastasis of …
Formula:
C24H21FN2O3
Purity:
98% - 98.04%
Color and Shape:
Solid
Molecular weight:
404.43
Ref: TM-TQ0290
| 2mg | 41.00 € | ||
| 5mg | 62.00 € | ||
| 10mg | 89.00 € | ||
| 25mg | 151.00 € | ||
| 50mg | 216.00 € | ||
| 100mg | To inquire | ||
| 1mL*10mM (DMSO) | 68.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
Piboserod
CAS:152811-62-6
Piboserod (SB-207266) (SB 207266) is a selective 5-HT(4) receptor antagonist.
Formula:
C22H31N3O2
Purity:
98.09% - 99.49%
Color and Shape:
Solid
Molecular weight:
369.5
Ref: TM-T2278
| 1mg | 40.00 € | ||
| 2mg | 57.00 € | ||
| 5mg | 91.00 € | ||
| 10mg | 127.00 € | ||
| 25mg | 233.00 € | ||
| 50mg | 421.00 € | ||
| 100mg | 605.00 € | ||
| 500mg | 1,236.00 € | ||
| 1mL*10mM (DMSO) | 126.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
SX-682
CAS:1648843-04-2
SX-682 is an orally available allosteric inhibitor of CXCR1 and CXCR2.Cost-effective and quality-assured.
Formula:
C19H14BF4N3O4S
Purity:
98.88% - 99.57%
Color and Shape:
Solid
Molecular weight:
467.2
Ref: TM-T8497
| 1mg | 40.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 118.00 € | ||
| 25mg | 213.00 € | ||
| 50mg | 353.00 € | ||
| 100mg | 470.00 € | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
Piribedil
CAS:3605-01-4
Piribedil (Trivastan) is a dopamine D2 agonist, used in the treatment of Parkinson's disease.
Formula:
C16H18N4O2
Purity:
99.83% - 99.91%
Color and Shape:
Solid
Molecular weight:
298.34
Ref: TM-T3278
| 25mg | 62.00 € | ||
| 50mg | 80.00 € | ||
| 100mg | 93.00 € | ||
| 200mg | 156.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
JNJ-7777120
CAS:459168-41-3
JNJ-7777120 is the first potent and selective non-imidazole histamine H4 receptor antagonist, exhibits >1000-fold selectivity …
Formula:
C14H16ClN3O
Purity:
99.71% - 99.93%
Color and Shape:
Solid
Molecular weight:
277.75
Ref: TM-T2232
| 5mg | 69.00 € | ||
| 10mg | 94.00 € | ||
| 25mg | 167.00 € | ||
| 50mg | 268.00 € | ||
| 100mg | 430.00 € | ||
| 500mg | 920.00 € | ||
| 1mL*10mM (DMSO) | 73.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
CGP71683 hydrochloride
CAS:192322-50-2
CGP71683 hydrochloride: NPY5 receptor antagonist, Ki=1.3 nM; inactive at Y1 (Ki >4000 nM) and Y2 …
Formula:
C26H30ClN5O2S
Purity:
99.92%
Color and Shape:
Solid
Molecular weight:
512.07
Ref: TM-T5587
| 1mg | 50.00 € | ||
| 5mg | 103.00 € | ||
| 10mg | 156.00 € | ||
| 25mg | 252.00 € | ||
| 50mg | 360.00 € | ||
| 100mg | 527.00 € | ||
| 1mL*10mM (DMSO) | 117.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
Perospirone
CAS:150915-41-6
Perospirone (Lullan) is an antagonist of serotonin 5HT2A receptors and dopamine D2 receptors.
Formula:
C23H30N4O2S
Purity:
98.86%
Color and Shape:
White Powder
Molecular weight:
426.57
Ref: TM-T4576
| 5mg | 43.00 € | ||
| 10mg | 65.00 € | ||
| 25mg | 107.00 € | ||
| 50mg | 189.00 € | ||
| 100mg | 322.00 € | ||
| 200mg | 451.00 € | ||
| 1mL*10mM (DMSO) | 46.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
CYM2503
CAS:1308833-36-4
CYM2503 is a GAL2 receptor PAM enhancing galanin-induced IP1 without binding the galanin site.
Formula:
C45H55N5O7
Purity:
97.04%
Color and Shape:
Solid
Molecular weight:
777.95
Ref: TM-T8963
| 1mg | 36.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 113.00 € | ||
| 25mg | 220.00 € | ||
| 50mg | 353.00 € | ||
| 100mg | 497.00 € | ||
| 200mg | 677.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
CYM50358
CAS:1314212-39-9
N-(4-(aminomethyl)-2,6-dimethylphenyl)-5 is a potent, selective antagonist of the sphingosine-1-phosphate receptor 4 (S1P4).
Formula:
C20H18Cl2N2O2
Purity:
98.05% - 99.76%
Color and Shape:
Solid
Molecular weight:
389.28
Ref: TM-T9464
| 1mg | 55.00 € | ||
| 5mg | 118.00 € | ||
| 10mg | 185.00 € | ||
| 25mg | 424.00 € | ||
| 50mg | 626.00 € | ||
| 100mg | 893.00 € | ||
| 1mL*10mM (DMSO) | 130.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
SBI-115
CAS:882366-16-7
SBI-115 is an antagonist of TGR5. SBI-115 decreases hepatic cystogenesis with polycystic liver diseases via …
Formula:
C14H13ClN2O4S
Purity:
99.53%
Color and Shape:
Solid
Molecular weight:
340.78
Ref: TM-T7428
| 5mg | 52.00 € | ||
| 10mg | 80.00 € | ||
| 25mg | 143.00 € | ||
| 50mg | 217.00 € | ||
| 100mg | 348.00 € | ||
| 1mL*10mM (DMSO) | 59.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
SB399885
CAS:402713-80-8
SB399885 is a potent, brain-penetrant, oral SR-6 antagonist with 200-fold selectivity for SR-6 receptors.
Formula:
C18H21Cl2N3O4S
Purity:
98.94%
Color and Shape:
Solid
Molecular weight:
446.35
Ref: TM-T19669
| 1mg | 94.00 € | ||
| 5mg | 169.00 € | ||
| 10mg | 244.00 € | ||
| 25mg | 402.00 € | ||
| 50mg | 542.00 € | ||
| 100mg | 762.00 € | ||
| 200mg | 1,025.00 € | ||
| 1mL*10mM (DMSO) | 200.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
LY334370
CAS:182563-08-2
LY334370 is a selective 5-HT1F receptor agonist with a Ki of 1.6 nM
Formula:
C21H22FN3O
Purity:
98.48%
Color and Shape:
Solid
Molecular weight:
351.42
Ref: TM-T4266
| 5mg | 45.00 € | ||
| 10mg | 65.00 € | ||
| 25mg | 130.00 € | ||
| 50mg | 187.00 € | ||
| 100mg | 272.00 € | ||
| 200mg | 375.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
Glucagon (19-29), human acetate
Glucagon (19-29), human acetate a COOH-terminal fragment processed from glucagon, is a potent and efficient …
Formula:
C63H93N15O20S
Purity:
98.11%
Color and Shape:
Solid
Molecular weight:
1412.57
Ref: TM-TP1863L
| 5mg | 64.00 € | ||
| 10mg | 94.00 € | ||
| 25mg | 162.00 € | ||
| 50mg | 234.00 € | ||
| 100mg | 354.00 € | ||
| 200mg | 528.00 € | ||
| 500mg | 789.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
CCG215022
CAS:1813527-81-9
CCG215022 is a G protein-coupled receptor kinases (GRKs) inhibitor with IC50s of 0.15±0.07 μM, 0.38±0.06 …
Formula:
C26H22FN7O3
Purity:
97.46% - 99.69%
Color and Shape:
Solid
Molecular weight:
499.5
Ref: TM-T3498
| 1mg | 94.00 € | ||
| 2mg | 138.00 € | ||
| 5mg | 231.00 € | ||
| 10mg | 369.00 € | ||
| 25mg | 616.00 € | ||
| 50mg | 877.00 € | ||
| 100mg | 1,196.00 € | ||
| 500mg | 2,385.00 € | ||
| 1mL*10mM (DMSO) | 257.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
ABT-724
CAS:70006-24-5
ABT-724 is an agonist of dopamine D4 receptor(EC50: 12.4 nM)
Formula:
C17H19N5
Purity:
99.73%
Color and Shape:
Solid
Molecular weight:
293.37
Ref: TM-T7834
| 5mg | 89.00 € | ||
| 25mg | 167.00 € | ||
| 50mg | 251.00 € | ||
| 1mL*10mM (DMSO) | 90.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
Grp94 Inhibitor-1
CAS:2234897-35-7
Grp94 Inhibitor-1 is a potent, selective Grp94 inhibitor (IC50 : 2 nM).
Formula:
C22H28N2O2
Purity:
97.02%
Color and Shape:
Solid
Molecular weight:
352.47
Ref: TM-T7261
| 5mg | 48.00 € | ||
| 10mg | 74.00 € | ||
| 25mg | 122.00 € | ||
| 50mg | 189.00 € | ||
| 100mg | 328.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
