G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Atipamezole hydrochloride
CAS:104075-48-1
Atipamezole is a synthetic α2 adrenergic receptor antagonist.
Formula:
C14H16N2·HCl
Purity:
96.71%
Color and Shape:
Solid
Molecular weight:
248.75
Ref: TM-T6765
| 5mg | 56.00 € | ||
| 10mg | 78.00 € | ||
| 25mg | 135.00 € | ||
| 50mg | 231.00 € | ||
| 100mg | 341.00 € | ||
| 200mg | 528.00 € | ||
| 500mg | 824.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Nociceptin
CAS:170713-75-4
Nociceptin (Orphanin FQ) is a 17-amino-acid polypeptide that is structurally related to the opioid peptide …
Formula:
C79H129N27O22
Purity:
99.35%
Color and Shape:
Solid
Molecular weight:
1809.04
Ref: TM-TP1071
| 1mg | 80.00 € | ||
| 5mg | 222.00 € | ||
| 10mg | 360.00 € | ||
| 25mg | 603.00 € | ||
| 50mg | 861.00 € | ||
| 100mg | 1,170.00 € | ||
| 500mg | 2,341.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
BRL 54443
CAS:57477-39-1
BRL 54443 is a potent 5-HT1E/1F receptor agonist (pKi values are 8.7 and 8.9 respectively).
Formula:
C14H18N2O
Purity:
99.95%
Color and Shape:
Solid
Molecular weight:
230.31
Ref: TM-T2459
| 5mg | 52.00 € | ||
| 10mg | 82.00 € | ||
| 25mg | 154.00 € | ||
| 50mg | 234.00 € | ||
| 100mg | 393.00 € | ||
| 1mL*10mM (DMSO) | 59.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
PF-06882961 Tris
CAS:2230198-03-3
PF-06882961 Tris (UNII-2HJV78O0SS) is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.
Formula:
C35H41FN6O7
Purity:
98.11% - 99.52%
Color and Shape:
Solid
Molecular weight:
676.7
Ref: TM-T8876
| 1mg | 129.00 € | ||
| 5mg | 282.00 € | ||
| 10mg | 424.00 € | ||
| 25mg | 694.00 € | ||
| 50mg | 975.00 € | ||
| 100mg | 1,318.00 € | ||
| 500mg | 2,626.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Ac-RYYRWK-NH2 acetate
Ac-RYYRWK-NH2 acetate is a potent partial agonist of the nociceptin receptor(NOP), which is the endogenous …
Formula:
C51H73N15O11
Purity:
98.60%
Color and Shape:
Solid
Molecular weight:
1072.22
Ref: TM-TP1941L1
| 1mg | 155.00 € | ||
| 5mg | 337.00 € | ||
| 10mg | 506.00 € | ||
| 25mg | 760.00 € | ||
| 50mg | 1,018.00 € | ||
| 100mg | 1,358.00 € | ||
| 200mg | 1,798.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
CPI-444
CAS:1202402-40-1
CPI-444 (V81444) is an antagonist of the adenosine A2A receptor.It reduces tumor area in mouse …
Formula:
C20H21N7O3
Purity:
98.78%
Color and Shape:
Solid
Molecular weight:
407.43
Ref: TM-T7183
| 1mg | 40.00 € | ||
| 2mg | 35.00 € | ||
| 5mg | 88.00 € | ||
| 10mg | 120.00 € | ||
| 25mg | 211.00 € | ||
| 50mg | 353.00 € | ||
| 100mg | 528.00 € | ||
| 200mg | 438.00 € | ||
| 1mL*10mM (DMSO) | 79.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
CID 16020046
CAS:834903-43-4
CID 16020046 (C390-0219) is a selective GPR55 antagonist, inhibiting GPR55 constitutive activity with IC50 of …
Formula:
C25H19N3O4
Purity:
99.59%
Color and Shape:
Solid
Molecular weight:
425.44
Ref: TM-T4478
| 2mg | 39.00 € | ||
| 5mg | 60.00 € | ||
| 10mg | 87.00 € | ||
| 25mg | 157.00 € | ||
| 50mg | 222.00 € | ||
| 100mg | 322.00 € | ||
| 1mL*10mM (DMSO) | 68.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
6-fluoro-DL-Tryptophan
CAS:7730-20-3
6-fluoro-DL-Tryptophan is an inhibitor of serotonin (5-HT) synthesis.
Formula:
C11H11FN2O2
Purity:
99.25%
Color and Shape:
Off-White Powder
Molecular weight:
222.22
Ref: TM-T7694
| 50mg | 48.00 € | ||
| 100mg | 71.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
GUANABENZ
CAS:5051-62-7
GUANABENZ is a Central alpha-2 Adrenergic Agonist. The mechanism of action of guanabenz is as …
Formula:
C8H8Cl2N4
Purity:
98.6%
Color and Shape:
White Solid From Acetonitrile Solid
Molecular weight:
231.08
Ref: TM-T5471
| 2mg | 35.00 € | ||
| 5mg | 48.00 € | ||
| 10mg | 63.00 € | ||
| 25mg | 102.00 € | ||
| 50mg | 144.00 € | ||
| 100mg | 209.00 € | ||
| 200mg | 310.00 € | ||
| 1mL*10mM (DMSO) | 50.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Neuromedin N acetate(92169-45-4 free base)
Neuromedin N acetate(92169-45-4 free base) is a neuropeptide derived from the same precursor polypeptide as …
Formula:
C40H67N7O10
Purity:
99.95%
Color and Shape:
Solid
Molecular weight:
805.9
Ref: TM-TP1085L
| 1mg | 35.00 € | ||
| 5mg | 59.00 € | ||
| 10mg | 85.00 € | ||
| 25mg | 161.00 € | ||
| 50mg | 226.00 € | ||
| 100mg | 337.00 € | ||
| 200mg | 479.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
BPTU
CAS:870544-59-5
BPTU (BMS-646786) is an allosteric antagonist of P2Y1 (EC50 = 0.06-0.3 μM).
Formula:
C23H22F3N3O3
Purity:
99.37% - 99.89%
Color and Shape:
Solid
Molecular weight:
445.43
Ref: TM-T4132
| 1mg | 38.00 € | ||
| 2mg | 49.00 € | ||
| 5mg | 71.00 € | ||
| 10mg | 115.00 € | ||
| 25mg | 233.00 € | ||
| 50mg | 403.00 € | ||
| 100mg | 600.00 € | ||
| 1mL*10mM (DMSO) | 72.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Prazosin
CAS:19216-56-9
Prazosin (Prazosine), an α1-blocker, acts as an inverse agonist at alpha-1 adrenergic receptors and is …
Formula:
C19H21N5O4
Purity:
99.29%
Color and Shape:
White To Tan Powder Solid
Molecular weight:
383.4
Ref: TM-T22406
| 10mg | 49.00 € | ||
| 25mg | 71.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
PSN 375963
CAS:388575-52-8
PSN 375963 (PSN 375963 hydrochloride) hydrochloride is a synthetic agonist of the endogenous ligand for …
Formula:
C17H23N3O
Purity:
99.24%
Color and Shape:
Solid
Molecular weight:
285.38
Ref: TM-T23204
| 5mg | 44.00 € | ||
| 10mg | 63.00 € | ||
| 25mg | 112.00 € | ||
| 50mg | 181.00 € | ||
| 100mg | 296.00 € | ||
| 200mg | 422.00 € | ||
| 1mL*10mM (DMSO) | 62.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Alprenolol hydrochloride
CAS:13707-88-5
Alprenolol hydrochloride is a non-selective blocker of beta, and also is a antagonist of5-HT1A receptor.
Formula:
C15H24ClNO2
Purity:
99.79%
Color and Shape:
Solid
Molecular weight:
285.81
Ref: TM-T22236
| 50mg | 41.00 € | ||
| 100mg | 63.00 € | ||
| 500mg | 195.00 € | ||
| 1mL*10mM (DMSO) | 35.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
3-Hydroxyoctanoic Acid
CAS:14292-27-4
3-Hydroxyoctanoic Acid, an energy metabolism intermediate, activates orphan receptor GPR109B.
Formula:
C8H16O3
Purity:
97.82% - ≥98%
Color and Shape:
Solid
Molecular weight:
160.21
Ref: TM-T9719
| 5mg | 37.00 € | ||
| 10mg | 57.00 € | ||
| 25mg | 87.00 € | ||
| 50mg | 136.00 € | ||
| 100mg | 187.00 € | ||
| 500mg | 486.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Betazole dihydrochloride
CAS:138-92-1
Betazole dihydrochloride (Betazole hydrochloride) is an agonist of H2 receptor.
Formula:
C5H11Cl2N3
Purity:
99.12%
Color and Shape:
Solid
Molecular weight:
184.067
Ref: TM-T8599
| 1mg | 35.00 € | ||
| 5mg | 59.00 € | ||
| 10mg | 93.00 € | ||
| 25mg | 171.00 € | ||
| 50mg | 299.00 € | ||
| 100mg | 387.00 € | ||
| 200mg | 553.00 € | ||
| 1mL*10mM (DMSO) | 59.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
SKF 38393 hydrochloride
CAS:62717-42-4
SKF 38393 hydrochloride (SKF38393 HCl) is a selective dopamine D1/D5 receptor agonist.
Formula:
C16H17NO2·HCl
Purity:
98.70% - 99.1%
Color and Shape:
Solid
Molecular weight:
291.77
Ref: TM-T6988
| 25mg | 54.00 € | ||
| 50mg | 77.00 € | ||
| 1mL*10mM (DMSO) | 85.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
E7046
CAS:1369489-71-3
E7046 is a specific, orally bioavailable EP4 antagonist (IC50: 13.5 nM, Ki: 23.14 nM), exhibiting …
Formula:
C22H18F5N3O4
Purity:
99.86%
Color and Shape:
Solid
Molecular weight:
483.4
Ref: TM-TQ0025
| 5mg | 52.00 € | ||
| 10mg | 74.00 € | ||
| 25mg | 126.00 € | ||
| 50mg | 209.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
![[D-Phe12]-Bombesin acetate](https://static.cymitquimica.com/products/TM/thumb/TP2239L.jpg)
[D-Phe12]-Bombesin acetate
[D-Phe12]-Bombesin acetate inhibits bombesin-stimulated secretion.
Formula:
C76H116N22O20S
Purity:
99.81%
Color and Shape:
Liquid
Molecular weight:
1689.94
Ref: TM-TP2239L
| 1mg | 157.00 € | ||
| 5mg | 343.00 € | ||
| 10mg | 513.00 € | ||
| 25mg | 923.00 € | ||
| 50mg | 1,380.00 € | ||
| 100mg | 2,074.00 € | ||
| 200mg | 3,111.00 € | ||
| 500mg | 4,714.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Amylin, amide, rat acetate(124447-81-0,free base)
Amylin, amide, rat acetate is a potent and high affinity ligand of AMY1 and AMY3 …
Formula:
C169H276N52O55S2
Purity:
98.5%
Color and Shape:
Solid
Molecular weight:
3980.45
Ref: TM-TP1232L
| 1mg | 171.00 € | ||
| 5mg | 403.00 € | ||
| 10mg | 547.00 € | ||
| 25mg | 843.00 € | ||
| 50mg | 1,090.00 € | ||
| 100mg | 1,533.00 € | ||
| 200mg | 2,060.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
