G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Ac-RYYRIK-NH2 acetate
Ac-RYYRIK-NH2 acetate is an agonist at nociceptin/orphanin FQ(noc/OFQ) receptors, affecting spontaneous locomotor activity.
Formula:
C46H74N14O11
Purity:
99.84%
Color and Shape:
Solid
Molecular weight:
999.17
Ref: TM-TP1940L1
| 1mg | 274.00 € | ||
| 2mg | 412.00 € | ||
| 5mg | 620.00 € | ||
| 10mg | 926.00 € | ||
| 25mg | 1,375.00 € | ||
| 50mg | 1,855.00 € | ||
| 100mg | 2,499.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Bradykinin (2-9)
CAS:16875-11-9
Bradykinin (2-9) (Des-Arg1-bradykinin) is an amino-truncated peptide compound that is a metabolite of Bradykinin.
Formula:
C44H61N11O10
Purity:
100%
Color and Shape:
Solid
Molecular weight:
904.02
Ref: TM-TP1181
| 1mg | 52.00 € | ||
| 1ml | 175.00 € | ||
| 2mg | 68.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 162.00 € | ||
| 25mg | 263.00 € | ||
| 50mg | 394.00 € | ||
| 100mg | 572.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
JTC-801
CAS:244218-51-7
JTC-801 is a selective opioid receptor-like1 (ORL1) receptor antagonist with IC50 of 94 nM, weakly …
Formula:
C26H25N3O2·HCl
Purity:
98% - 99.27%
Color and Shape:
Solid
Molecular weight:
447.96
Ref: TM-T6553
| 1ml | 71.00 € | ||
| 5mg | 48.00 € | ||
| 10mg | 71.00 € | ||
| 25mg | 139.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Dynorphin A acetate(80448-90-4 free base)
Dynorphin A acetate is an Endogenous kappa receptor agonist.
Formula:
C101H159N31O25
Purity:
99.69%
Color and Shape:
Solid
Molecular weight:
2207.58
Ref: TM-TP2040L
| 1mg | 70.00 € | ||
| 5mg | 234.00 € | ||
| 10mg | 321.00 € | ||
| 25mg | 541.00 € | ||
| 50mg | 774.00 € | ||
| 100mg | 1,067.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Nelotanserin
CAS:839713-36-9
Nelotanserin (APD125): strong 5-HT2A inverse agonist (IC50: 1.7 nM), moderate 5-HT2C (79 nM), weak 5-HT2B …
Formula:
C18H15BrF2N4O2
Purity:
98.01% - 98.42%
Color and Shape:
Solid
Molecular weight:
437.24
Ref: TM-T7350
| 1mg | 40.00 € | ||
| 1ml | 84.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 86.00 € | ||
| 10mg | 118.00 € | ||
| 25mg | 185.00 € | ||
| 50mg | 343.00 € | ||
| 100mg | 510.00 € | ||
| 500mg | 1,109.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Naftopidil dihydrochloride
CAS:57149-08-3
Naftopidil dihydrochloride (KT-611 2HCl) is a selective 5-HT1A and α1-adrenergic receptor antagonist with IC50 of …
Formula:
C24H28N2O3·2HCl
Purity:
99.95%
Color and Shape:
White Solid
Molecular weight:
465.41
Ref: TM-T6600
| 1ml | 52.00 € | ||
| 50mg | 58.00 € | ||
| 100mg | 95.00 € | ||
| 200mg | 170.00 € | ||
| 500mg | 290.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
5-Iodotubercidin
CAS:24386-93-4
5-Iodotubercidin (NSC-113939) is a potent adenosine kinase inhibitor with IC50 of 26 nM.
Formula:
C11H13IN4O4
Purity:
99.98%
Color and Shape:
Tan Solid
Molecular weight:
392.15
Ref: TM-T6745
| 1mg | 45.00 € | ||
| 1ml | 96.00 € | ||
| 2mg | 56.00 € | ||
| 5mg | 90.00 € | ||
| 10mg | 151.00 € | ||
| 25mg | 337.00 € | ||
| 50mg | 499.00 € | ||
| 100mg | 718.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Perospirone
CAS:150915-41-6
Perospirone (Lullan) is an antagonist of serotonin 5HT2A receptors and dopamine D2 receptors.
Formula:
C23H30N4O2S
Purity:
98.86%
Color and Shape:
White Powder
Molecular weight:
426.57
Ref: TM-T4576
| 1ml | 46.00 € | ||
| 5mg | 43.00 € | ||
| 10mg | 65.00 € | ||
| 25mg | 107.00 € | ||
| 50mg | 189.00 € | ||
| 100mg | 322.00 € | ||
| 200mg | 451.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Vericiguat
CAS:1350653-20-1
Vericiguat (BAY1021189) is a potent and orally available guanylate cyclase stimulator.
Formula:
C19H16F2N8O2
Purity:
98.86% - 99.6%
Color and Shape:
Solid
Molecular weight:
426.38
Ref: TM-T17226
| 1mg | 47.00 € | ||
| 1ml | 113.00 € | ||
| 5mg | 102.00 € | ||
| 10mg | 142.00 € | ||
| 25mg | 256.00 € | ||
| 50mg | 414.00 € | ||
| 100mg | 591.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
BETP
CAS:1371569-69-5
BETP is an agonist of GLP-1 receptor (EC50s: 0.66 and 0.755 μM for human and …
Formula:
C20H17F3N2O2S
Purity:
97.92%
Color and Shape:
Solid
Molecular weight:
406.42
Ref: TM-TQ0124
| 1mg | 47.00 € | ||
| 1ml | 96.00 € | ||
| 5mg | 91.00 € | ||
| 10mg | 137.00 € | ||
| 25mg | 258.00 € | ||
| 50mg | 414.00 € | ||
| 100mg | 661.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Phenylbiguanide
CAS:102-02-3
Phenylbiguanide (N-Phenylbiguanide) is a 5-HT3 receptor selective agonist(EC50 : 3.0±0.1 μM)
Formula:
C8H11N5
Purity:
99.87%
Color and Shape:
Solid
Molecular weight:
177.21
Ref: TM-T7135
| 1g | 82.00 € | ||
| 1ml | 34.00 € | ||
| 200mg | 38.00 € | ||
| 500mg | 56.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Puerarin
CAS:3681-99-0
Puerarin (Kakonein), also known as Kakonein, is a member of the class of compounds known …
Formula:
C21H20O9
Purity:
98.9% - 99.84%
Color and Shape:
Yellow Brown Fine Powder
Molecular weight:
416.38
Ref: TM-T2815
| 1ml | 87.00 € | ||
| 5mg | 51.00 € | ||
| 10mg | 91.00 € | ||
| 25mg | 162.00 € | ||
| 50mg | 235.00 € | ||
| 100mg | 351.00 € | ||
| 500mg | 812.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Sotagliflozin
CAS:1018899-04-1
Sotagliflozin (LP-802034) is an orally bioavailable inhibitor of the sodium-glucose co-transporter subtype 1 (SGLT1) and …
Formula:
C21H25ClO5S
Purity:
98% - 99.37%
Color and Shape:
Solid
Molecular weight:
424.94
Ref: TM-T3547
| 1mg | 45.00 € | ||
| 1ml | 88.00 € | ||
| 2mg | 56.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 129.00 € | ||
| 25mg | 244.00 € | ||
| 50mg | 369.00 € | ||
| 100mg | 548.00 € | ||
| 500mg | 1,175.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
PEN (human) aceate
PEN (human) aceate, one of the most abundant hypothalamic neuropeptide and derived from the proprotein …
Formula:
C99H163N27O34
Purity:
99.25%
Color and Shape:
Solid
Molecular weight:
2275.51
Ref: TM-TP1949L
| 1mg | 143.00 € | ||
| 5mg | 312.00 € | ||
| 10mg | 464.00 € | ||
| 25mg | 834.00 € | ||
| 50mg | 1,264.00 € | ||
| 100mg | 1,866.00 € | ||
| 200mg | 2,778.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
ACTH 11-24 acetate(4237-93-8 free base)
CAS:79190-56-0
ACTH 11-24 acetate is a cortisol-stimulating adrenocorticotrophin fragment and a competitive antagonist of ACTH 1-39 …
Formula:
C79H138N24O18
Purity:
100%
Color and Shape:
Solid
Molecular weight:
1712.12
Ref: TM-TP1248L
| 1mg | 51.00 € | ||
| 5mg | 93.00 € | ||
| 10mg | 113.00 € | ||
| 25mg | 195.00 € | ||
| 50mg | 293.00 € | ||
| 100mg | 422.00 € | ||
| 200mg | 589.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Paltusotine
CAS:2172870-89-0
Paltusotine: nonpeptide SST2 agonist, orally bioavailable, regulates GH/IGF-1 in acromegaly.
Formula:
C27H22F2N4O
Purity:
99.77%
Color and Shape:
Solid
Molecular weight:
456.49
Ref: TM-T9692
| 1mg | 171.00 € | ||
| 5mg | 413.00 € | ||
| 10mg | 597.00 € | ||
| 25mg | 903.00 € | ||
| 50mg | 1,220.00 € | ||
| 100mg | 1,645.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
TUG-1375
CAS:2247372-59-2
TUG-1375 is an Agonist of Thiazolidine Free Fatty Acid Receptor 2
Formula:
C22H19ClN2O4S
Purity:
97.72% - 99.41%
Color and Shape:
Solid
Molecular weight:
442.92
Ref: TM-T7796
| 1mg | 86.00 € | ||
| 1ml | 205.00 € | ||
| 5mg | 186.00 € | ||
| 10mg | 305.00 € | ||
| 25mg | 476.00 € | ||
| 50mg | 638.00 € | ||
| 100mg | 858.00 € | ||
| 200mg | 1,154.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
AM1241
CAS:444912-48-5
AM-1241 is a selective cannabinoid CB2 receptor agonist with Ki of 3.4 nM, exhibits 82-fold …
Formula:
C22H22IN3O3
Purity:
98.82% - 99.10%
Color and Shape:
Solid
Molecular weight:
503.33
Ref: TM-T6755
| 1ml | 92.00 € | ||
| 2mg | 38.00 € | ||
| 5mg | 51.00 € | ||
| 10mg | 88.00 € | ||
| 25mg | 168.00 € | ||
| 50mg | 284.00 € | ||
| 100mg | 512.00 € | ||
| 500mg | 1,112.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Ponesimod
CAS:854107-55-4
Ponesimod (ACT-128800) is an orally available sphingosine-1-phosphate receptor 1 (S1PR1, S1P1) agonist with potential immunomodulating …
Formula:
C23H25ClN2O4S
Purity:
98.22% - 99.42%
Color and Shape:
Solid
Molecular weight:
460.97
Ref: TM-T3258
| 1mg | 45.00 € | ||
| 1ml | 96.00 € | ||
| 2mg | 58.00 € | ||
| 5mg | 92.00 € | ||
| 10mg | 128.00 € | ||
| 25mg | 229.00 € | ||
| 50mg | 397.00 € | ||
| 100mg | 583.00 € | ||
| 500mg | 1,254.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
![Lys-[Des-Arg9]Bradykinin acetate](https://static.cymitquimica.com/products/TM/thumb/TP1918L1.jpg)
Lys-[Des-Arg9]Bradykinin acetate
Lys-[Des-Arg9]Bradykinin acetate is an endogenous potent and highly selective bradykinin B1 receptor agonist (Ki values …
Formula:
C52H77N13O13
Purity:
99.93%
Color and Shape:
Solid
Molecular weight:
1092.27
Ref: TM-TP1918L1
| 1mg | 87.00 € | ||
| 5mg | 171.00 € | ||
| 10mg | 257.00 € | ||
| 25mg | 468.00 € | ||
| 50mg | 680.00 € | ||
| 100mg | 956.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
