G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Deslorelin acetate(57773-65-6 free base)
Deslorelin acetate(57773-65-6 free base) is a gonadotropin releasing hormone super-agonist (GnRH agonist)
Formula:
C66H87N17O14
Purity:
99.84%
Color and Shape:
Solid
Molecular weight:
1342.5
Ref: TM-TP2323L
| 1mg | 91.00 € | ||
| 2mg | 118.00 € | ||
| 5mg | 165.00 € | ||
| 10mg | 222.00 € | ||
| 25mg | 399.00 € | ||
| 50mg | 591.00 € | ||
| 100mg | 824.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
TUG-891
CAS:1374516-07-0
TUG-891 is a G protein-coupled receptor expressed in intestine, adipocytes, and pro-inflammatory macrophages that is …
Formula:
C23H21FO3
Purity:
98.28% - 99.21%
Color and Shape:
Solid
Molecular weight:
364.41
Ref: TM-T3433
| 1mg | 40.00 € | ||
| 2mg | 51.00 € | ||
| 5mg | 83.00 € | ||
| 10mg | 114.00 € | ||
| 25mg | 221.00 € | ||
| 50mg | 369.00 € | ||
| 100mg | 540.00 € | ||
| 500mg | 1,143.00 € | ||
| 1mL*10mM (DMSO) | 93.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
JNJ-10229570
CAS:524923-88-4
JNJ-10229570 (UNII-N9IX402L35) is an antagonist of melanocortin receptor 1 (MC1R) and melanocortin receptor 5 (MC5R), …
Formula:
C22H19N3O2S
Purity:
99.06%
Color and Shape:
Solid
Molecular weight:
389.47
Ref: TM-T5464
| 1mg | 108.00 € | ||
| 5mg | 184.00 € | ||
| 10mg | 291.00 € | ||
| 25mg | 461.00 € | ||
| 50mg | 640.00 € | ||
| 100mg | 828.00 € | ||
| 1mL*10mM (DMSO) | 210.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
AR-M 1000390 hydrochloride
CAS:209808-47-9
ARM-390 HCl is a δ-opioid receptor agonist, brain-penetrant, nonpeptidic, prevents hyperalgesia without desensitization. Derived from …
Formula:
C23H29ClN2O
Purity:
99.68%
Color and Shape:
Solid
Molecular weight:
384.94
Ref: TM-T4236
| 5mg | 69.00 € | ||
| 10mg | 102.00 € | ||
| 25mg | 204.00 € | ||
| 50mg | 368.00 € | ||
| 100mg | 553.00 € | ||
| 1mL*10mM (DMSO) | 77.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Neuropeptide SF(mouse,rat) acetate
Neuropeptide SF (mouse,rat) acetate is a NPFF receptor agonist with Ki of 48.4 nM (NPFF1) …
Formula:
C42H69N13O12
Purity:
98.37%
Color and Shape:
Solid
Molecular weight:
948.08
Ref: TM-TP1884L1
| 1mg | 85.00 € | ||
| 5mg | 172.00 € | ||
| 10mg | 249.00 € | ||
| 25mg | 410.00 € | ||
| 50mg | 577.00 € | ||
| 100mg | 780.00 € | ||
| 200mg | 1,034.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
CYM-5541
CAS:945128-26-7
CYM-5541 (ML249) is a selective and allosteric S1P3 receptor agonist.
Formula:
C19H28N2O2
Purity:
97.34% - 98.39%
Color and Shape:
Solid
Molecular weight:
316.44
Ref: TM-T3961
| 2mg | 38.00 € | ||
| 5mg | 56.00 € | ||
| 10mg | 91.00 € | ||
| 25mg | 157.00 € | ||
| 50mg | 249.00 € | ||
| 100mg | 365.00 € | ||
| 500mg | 855.00 € | ||
| 1mL*10mM (DMSO) | 64.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Lys-Bradykinin acetate(342-10-9 free base)
CAS:84640-50-6
Lys-Bradykinin acetate is an endogenous bradykinin receptor agonist.
Formula:
C58H89N17O14
Purity:
99.86%
Color and Shape:
Solid
Molecular weight:
1248.43
Ref: TM-TP2268L
| 1mg | 96.00 € | ||
| 5mg | 210.00 € | ||
| 10mg | 313.00 € | ||
| 25mg | 528.00 € | ||
| 50mg | 743.00 € | ||
| 100mg | 1,051.00 € | ||
| 500mg | 2,098.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
ATI-2341 acetate(1337878-62-2 free base)
ATI-2341 acetate is an effective allosteric agonist of CXCR4, it activates Gα1 instead of Gα13.
Formula:
C106H182N26O27S2
Purity:
97.14%
Color and Shape:
Solid
Molecular weight:
2316.87
Ref: TM-T6764L
| 1mg | 84.00 € | ||
| 5mg | 248.00 € | ||
| 10mg | 365.00 € | ||
| 25mg | 543.00 € | ||
| 50mg | 763.00 € | ||
| 100mg | 1,026.00 € | ||
| 200mg | 1,392.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
I-191
CAS:1690172-25-8
I-191 is a potent antagonist of protease-activated receptor 2 (PAR2), inhibits multiple signaling functions in …
Formula:
C23H26FN5O2
Purity:
99.80%
Color and Shape:
Solid
Molecular weight:
423.48
Ref: TM-T7137
| 1mg | 88.00 € | ||
| 2mg | 114.00 € | ||
| 5mg | 185.00 € | ||
| 10mg | 277.00 € | ||
| 25mg | 463.00 € | ||
| 50mg | 673.00 € | ||
| 100mg | 920.00 € | ||
| 1mL*10mM (DMSO) | 209.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Mesdopetam hemitartrate
CAS:2562346-14-7
Mesdopetam hemitartrate antagonizes dopamine D3 receptor (Ki=90 nM; IC50=9.8 μM) and stabilizes psychomotor function.
Formula:
C28H42F2N2O12S2
Purity:
99.98%
Color and Shape:
Solid
Molecular weight:
700.77
Ref: TM-T9409
| 1mg | 40.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 110.00 € | ||
| 25mg | 213.00 € | ||
| 50mg | 402.00 € | ||
| 100mg | 600.00 € | ||
| 500mg | 1,276.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Teduglutide acetate
Teduglutide acetate, a GLP-2 analogue, maximizes small intestinal mucosal hypertrophy.
Formula:
C166H256N44O56S
Purity:
97.39%
Color and Shape:
Soild
Molecular weight:
3812.13
Ref: TM-T35337L
| 1mg | 108.00 € | ||
| 5mg | 213.00 € | ||
| 10mg | 341.00 € | ||
| 25mg | 575.00 € | ||
| 50mg | 816.00 € | ||
| 100mg | 1,109.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Pamoic acid
CAS:130-85-8
Pamoic acid is the orphan G protein-coupled receptor GPR35 agonist. Pamoic acid activates ERK and …
Formula:
C23H16O6
Purity:
99.99%
Color and Shape:
Fine Yellow Powder
Molecular weight:
388.37
Ref: TM-T8353
| 1g | 48.00 € | ||
| 1ml*10 (DMSO) | 49.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Carcinine ditrifluoroacetate Acetate
Carcinine ditrifluoroacetate Acetate (β-Alanylhistamine dihydrochloride) is an H3 receptor antagonist.
Formula:
C14H20F6N4O7
Purity:
98.18%
Color and Shape:
Liquid
Molecular weight:
470.32
Ref: TM-T22624L
| 1mg | 62.00 € | ||
| 5mg | 113.00 € | ||
| 10mg | 171.00 € | ||
| 25mg | 308.00 € | ||
| 50mg | 435.00 € | ||
| 100mg | 604.00 € | ||
| 200mg | 821.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Ticagrelor metabolite M5
CAS:1251765-07-7
Ticagrelor metabolite M5 (T437700) is a metabolite of Ticagrelor, the first reversible oral antagonist of …
Formula:
C14H22N6O4S
Purity:
99.35%
Color and Shape:
Solid
Molecular weight:
370.43
Ref: TM-T21059
| 1mg | 41.00 € | ||
| 2mg | 51.00 € | ||
| 5mg | 88.00 € | ||
| 10mg | 113.00 € | ||
| 25mg | 218.00 € | ||
| 50mg | 323.00 € | ||
| 100mg | 436.00 € | ||
| 200mg | 610.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
![[Met5]-Enkephalin, amide TFA](https://static.cymitquimica.com/products/TM/thumb/TP1254.jpg)
[Met5]-Enkephalin, amide TFA
[Met5]-Enkephalin, amide TFA (5-Methionine-enkephalin amide (TFA)) is a δ opioid receptors agonist as well as …
Formula:
C29H37F3N6O8S
Purity:
99.81%
Color and Shape:
Solid
Molecular weight:
686.7
Ref: TM-TP1254
| 10mg | 35.00 € | ||
| 25mg | 62.00 € | ||
| 50mg | 91.00 € | ||
| 100mg | 119.00 € | ||
| 200mg | 173.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Hemokinin 1 (mouse) acetate(208041-90-1 free base)
Mouse Hemokinin-1 acetate: NK1 receptor agonist, Ki=0.175 nM; NK2 Ki=560 nM.
Formula:
C63H104N22O17S
Purity:
98.33%
Color and Shape:
Solid
Molecular weight:
1473.72
Ref: TM-TP1772L
| 1mg | 139.00 € | ||
| 5mg | 387.00 € | ||
| 10mg | 575.00 € | ||
| 25mg | 917.00 € | ||
| 50mg | 1,238.00 € | ||
| 100mg | 1,670.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Gastrin I (human) acetate
Gastrin I (human) acetate (Gastrin-17 acetate) is the endogenous peptide produced in the stomach, and …
Formula:
C99H128N20O33S
Purity:
98.84%
Color and Shape:
Solid
Molecular weight:
2158.25
Ref: TM-TP2030L1
| 1mg | 78.00 € | ||
| 5mg | 260.00 € | ||
| 10mg | 381.00 € | ||
| 25mg | 594.00 € | ||
| 50mg | 803.00 € | ||
| 100mg | 1,081.00 € | ||
| 200mg | 1,456.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
β-MSH (1-22) (human) acetate
Beta-MSH (1-22) (human) acetate (Beta-MSH (1-22) (human) acetate (17908-57-5 Free base)) , is an endogenous …
Formula:
C120H178N34O37S
Purity:
99.64%
Color and Shape:
Liquid
Molecular weight:
2720.97
Ref: TM-TP1004L
| 1mg | 162.00 € | ||
| 5mg | 456.00 € | ||
| 10mg | 668.00 € | ||
| 25mg | 1,044.00 € | ||
| 50mg | 1,375.00 € | ||
| 100mg | 1,850.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Fenoldopam mesylate
CAS:67227-57-0
Fenoldopam mesylate (Corlopam mesylate) is a selective dopamine-1 receptor (DA1) agonist with natriuretic/diuretic properties.
Formula:
C16H16ClNO3·CH4O3S
Purity:
99.19%
Color and Shape:
Solid
Molecular weight:
401.86
Ref: TM-T6835
| 10mg | 50.00 € | ||
| 25mg | 88.00 € | ||
| 50mg | 147.00 € | ||
| 100mg | 206.00 € | ||
| 200mg | 315.00 € | ||
| 1mL*10mM (DMSO) | 53.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
ML401
CAS:1597489-14-9
ML401 is a selectively EBI2(GPR183) receptor antagonist(IC50 of 1.03 nM) .
Formula:
C20H20BrClN2O
Purity:
99.13%
Color and Shape:
Solid
Molecular weight:
419.74
Ref: TM-T8234
| 1mg | 130.00 € | ||
| 2mg | 155.00 € | ||
| 5mg | 186.00 € | ||
| 10mg | 304.00 € | ||
| 25mg | 484.00 € | ||
| 50mg | 650.00 € | ||
| 100mg | 841.00 € | ||
| 500mg | 1,715.00 € | ||
| 1mL*10mM (DMSO) | 205.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
