G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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GW627368
CAS:439288-66-1
GW627368 (GW 627368X)X is a novel, potent and selective antagonist of prostanoid EP4 receptor.
Formula:
C30H28N2O6S
Purity:
99.54% - 99.92%
Color and Shape:
Solid
Molecular weight:
544.62
Ref: TM-T1978
| 1ml | 69.00 € | ||
| 2mg | 39.00 € | ||
| 5mg | 56.00 € | ||
| 10mg | 85.00 € | ||
| 25mg | 128.00 € | ||
| 50mg | 210.00 € | ||
| 100mg | 371.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
AP1189 acetate
CAS:959850-74-9
AP1189 acetate is a biased agonist at melanocortin 1 and melanocortin 3 receptors.
Formula:
C16H18N6O4
Purity:
98.73%
Color and Shape:
Solid
Molecular weight:
358.35
Ref: TM-T9596
| 1mg | 47.00 € | ||
| 1ml | 104.00 € | ||
| 5mg | 88.00 € | ||
| 10mg | 129.00 € | ||
| 25mg | 226.00 € | ||
| 50mg | 337.00 € | ||
| 100mg | 479.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Flibanserin
CAS:167933-07-5
Flibanserin (Girosa) is a serotonergic antidepressant used to treat hypoactive sexual desire disorder.
Formula:
C20H21F3N4O
Purity:
99.44% - 99.76%
Color and Shape:
White Powder
Molecular weight:
390.4
Ref: TM-T4297
| 1ml | 47.00 € | ||
| 5mg | 45.00 € | ||
| 10mg | 69.00 € | ||
| 25mg | 105.00 € | ||
| 50mg | 189.00 € | ||
| 100mg | 296.00 € | ||
| 500mg | 704.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
AF64394
CAS:1637300-25-4
AF64394 is a selective inverse agonist of GPR3(pIC50 : 7.3)
Formula:
C21H20ClN5O
Purity:
98.55%
Color and Shape:
Solid
Molecular weight:
393.87
Ref: TM-T8407
| 1mg | 39.00 € | ||
| 1ml | 88.00 € | ||
| 5mg | 80.00 € | ||
| 10mg | 109.00 € | ||
| 25mg | 184.00 € | ||
| 50mg | 276.00 € | ||
| 100mg | 430.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
1-Oleoyl lysophosphatidic acid sodium
CAS:325465-93-8
1-Oleoyl lysophosphatidic acid sodium (1-Oleoyl lysophosphatidic acid sodium salt) salt is an Endogenous agonist of …
Formula:
C21H40NaO7P
Purity:
98.75% - 99.24%
Color and Shape:
Solid
Molecular weight:
458.5
Ref: TM-T21654
| 1mg | 69.00 € | ||
| 5mg | 126.00 € | ||
| 10mg | 169.00 € | ||
| 25mg | 339.00 € | ||
| 50mg | 503.00 € | ||
| 100mg | 715.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
BAY 41-2272
CAS:256376-24-6
BAY 41-2272 is a direct and NO-independent soluble guanylate cyclase (sGC) stimulator.
Formula:
C20H17FN6
Purity:
99.54%
Color and Shape:
Solid
Molecular weight:
360.39
Ref: TM-T6775
| 1ml | 49.00 € | ||
| 2mg | 35.00 € | ||
| 5mg | 49.00 € | ||
| 10mg | 85.00 € | ||
| 25mg | 166.00 € | ||
| 50mg | 255.00 € | ||
| 100mg | 367.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Metergoline
CAS:17692-51-2
Metergoline (Methergoline) is a dopamine agonist and serotonin antagonist.
Formula:
C25H29N3O2
Purity:
99.7% - 99.83%
Color and Shape:
Solid
Molecular weight:
403.52
Ref: TM-T4008
| 1ml | 36.00 € | ||
| 10mg | 41.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Ciproxifan maleate
CAS:184025-19-2
Ciproxifan maleate (FUB 359)(FUB-359 maleate) is a highly potent and selective histamin H3-receptor antagonist with …
Formula:
C20H22N2O6
Purity:
99.45%
Color and Shape:
Solid
Molecular weight:
386.4
Ref: TM-T2004
| 1ml | 50.00 € | ||
| 2mg | 34.00 € | ||
| 5mg | 51.00 € | ||
| 10mg | 69.00 € | ||
| 25mg | 129.00 € | ||
| 50mg | 232.00 € | ||
| 100mg | 344.00 € | ||
| 200mg | 490.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Epinastine hydrochloride
CAS:108929-04-0
Epinastine hydrochloride (WAL-801CL HCl) is an antihistamine and mast cell stabilizer that is used in …
Formula:
C16H15N3·HCl
Purity:
99.62% - 99.92%
Color and Shape:
White Solid
Molecular weight:
285.77
Ref: TM-T6488
| 1ml | 47.00 € | ||
| 10mg | 39.00 € | ||
| 25mg | 59.00 € | ||
| 50mg | 75.00 € | ||
| 100mg | 99.00 € | ||
| 200mg | 175.00 € | ||
| 500mg | 315.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Darusentan
CAS:171714-84-4
Darusentan (Lu-135252) is a potent inhibitor of endothelin signaling and function in both large and …
Formula:
C22H22N2O6
Purity:
98.72%
Color and Shape:
Solid
Molecular weight:
410.43
Ref: TM-T5458
| 1ml | 69.00 € | ||
| 2mg | 44.00 € | ||
| 5mg | 67.00 € | ||
| 10mg | 102.00 € | ||
| 25mg | 177.00 € | ||
| 50mg | 293.00 € | ||
| 100mg | 423.00 € | ||
| 200mg | 594.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Tecadenoson
CAS:204512-90-3
Tecadenoson (CVT-510) is a selective agonist of A1 adenosine receptor.
Formula:
C14H19N5O5
Purity:
99.76%
Color and Shape:
Solid
Molecular weight:
337.33
Ref: TM-T17023
| 1mg | 49.00 € | ||
| 1ml | 124.00 € | ||
| 5mg | 112.00 € | ||
| 10mg | 172.00 € | ||
| 25mg | 296.00 € | ||
| 50mg | 419.00 € | ||
| 100mg | 542.00 € | ||
| 200mg | 717.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
SB-200646
CAS:143797-63-1
SB-200646 is a selective and potent antagonist of 5-HT2B/5-HT2C receptor
Formula:
C15H14N4O
Purity:
99.61%
Color and Shape:
Solid
Molecular weight:
266.3
Ref: TM-T8357
| 1mg | 63.00 € | ||
| 1ml | 130.00 € | ||
| 5mg | 124.00 € | ||
| 10mg | 181.00 € | ||
| 25mg | 304.00 € | ||
| 50mg | 438.00 € | ||
| 100mg | 598.00 € | ||
| 200mg | 805.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Naftopidil hydrochloride
CAS:1164469-60-6
Naftopidil HCl (BM-15275) is a selective alpha1 blocker with Ki: α1a-3.7 nM, α1b-20 nM, α1d-1.2 …
Formula:
C24H29ClN2O3
Purity:
99.50%
Color and Shape:
Solid
Molecular weight:
428.95
Ref: TM-T9220
| 1mg | 66.00 € | ||
| 1ml | 160.00 € | ||
| 2mg | 94.00 € | ||
| 5mg | 126.00 € | ||
| 10mg | 184.00 € | ||
| 25mg | 333.00 € | ||
| 50mg | 495.00 € | ||
| 100mg | 714.00 € | ||
| 500mg | 1,473.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
AM095
CAS:1345614-59-6
AM095 is a potent LPA1 receptor antagonist with IC50 values of 0.98 and 0.73 μM …
Formula:
C27H23N2NaO5
Purity:
99.62%
Color and Shape:
Solid
Molecular weight:
478.47
Ref: TM-T2000
| 1mg | 48.00 € | ||
| 2mg | 64.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 132.00 € | ||
| 25mg | 240.00 € | ||
| 50mg | 417.00 € | ||
| 100mg | 601.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Levobetaxolol hydrochloride
CAS:116209-55-3
Levobetaxolol hydrochloride ((S)-Betaxolol hydrochloride) is a beta blocker, used to lower the pressure in the …
Formula:
C18H29NO3·HCl
Purity:
99.57% - 99.69%
Color and Shape:
Solid
Molecular weight:
343.89
Ref: TM-T6565
| 1ml | 35.00 € | ||
| 25mg | 35.00 € | ||
| 50mg | 51.00 € | ||
| 100mg | 79.00 € | ||
| 500mg | 181.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Desvenlafaxine succinate hydrate
CAS:386750-22-7
Desvenlafaxine succinate hydrate (WY 45233 Succinate) is an antidepressant of the serotonin-norepinephrine reuptake inhibitor (SNRI).
Formula:
C20H33NO7
Purity:
99.39%
Color and Shape:
White Crystalline Powde
Molecular weight:
399.48
Ref: TM-T6188
| 1ml | 49.00 € | ||
| 5mg | 41.00 € | ||
| 10mg | 54.00 € | ||
| 25mg | 95.00 € | ||
| 50mg | 111.00 € | ||
| 100mg | 182.00 € | ||
| 500mg | 452.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Afamelanotide acetate
CAS:1566590-77-9
Afamelanotide acetate is a synthetic α-melanocyte stimulating hormone analogue and first-in-class melanocortin-1 receptor agonist.
Formula:
C80H115N21O21
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1706.9
Ref: TM-T7589
| 1mg | 72.00 € | ||
| 1ml | 336.00 € | ||
| 5mg | 158.00 € | ||
| 10mg | 225.00 € | ||
| 25mg | 371.00 € | ||
| 50mg | 555.00 € | ||
| 100mg | 786.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Bupranolol
CAS:14556-46-8
Bupranolol blocks β2-adrenergic receptor; treats angina, hypertension, glaucoma, arrhythmia, and prevents clots.
Formula:
C14H22ClNO2
Purity:
95.85%
Color and Shape:
Solid
Molecular weight:
271.78
Ref: TM-T8580
| 1mg | 49.00 € | ||
| 1ml | 98.00 € | ||
| 5mg | 107.00 € | ||
| 10mg | 161.00 € | ||
| 25mg | 314.00 € | ||
| 50mg | 448.00 € | ||
| 100mg | 593.00 € | ||
| 200mg | 799.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Piperacetazine
CAS:3819-00-9
Piperacetazine (Piperacetazinum), an antipsychotic prodrug, is used forschizophrenia.
Formula:
C24H30N2O2S
Purity:
99.68% - 99.9%
Color and Shape:
Solid
Molecular weight:
410.57
Ref: TM-T3085
| 1ml | 68.00 € | ||
| 2mg | 42.00 € | ||
| 5mg | 61.00 € | ||
| 10mg | 85.00 € | ||
| 25mg | 129.00 € | ||
| 50mg | 186.00 € | ||
| 100mg | 280.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Ondansetron hydrochloride
CAS:99614-01-4
Ondansetron hydrochloride (Zofran) is a serotonin 5-HT3 receptor antagonist, used to prevent nausea and vomiting …
Formula:
C18H19N3O·HCl
Purity:
98.66%
Color and Shape:
White Powder
Molecular weight:
329.82
Ref: TM-T6616
| 1ml | 46.00 € | ||
| 25mg | 43.00 € | ||
| 50mg | 57.00 € | ||
| 100mg | To inquire |
Estimated delivery in United States, on Tuesday 15 Oct 2024
