G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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VPC171
CAS:1018830-99-3
VPC171 is a novel adenosine A1 receptor positive allosteric modulator (PAM).
Formula:
C18H12F3NOS
Purity:
99.52%
Color and Shape:
Solid
Molecular weight:
347.35
Ref: TM-T29112
| 1mg | 71.00 € | ||
| 2mg | 93.00 € | ||
| 5mg | 126.00 € | ||
| 10mg | 175.00 € | ||
| 25mg | 324.00 € | ||
| 50mg | 451.00 € | ||
| 100mg | 638.00 € | ||
| 200mg | 859.00 € | ||
| 1mL*10mM (DMSO) | 129.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Diphenhydramine
CAS:58-73-1
Diphenhydramine (Syntedril): first-gen antihistamine for allergies, antiemetic, antitussive, anticholinergic, sedative, treats drug-induced parkinsonism.
Formula:
C17H21NO
Purity:
99.49%
Color and Shape:
Solid
Molecular weight:
255.35
Ref: TM-T21419
| 200mg | 40.00 € | ||
| 500mg | 60.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
6-OAU
CAS:83797-69-7
6-OAU is a GPR84 agonist, activates it in HEK293 cells with a 105 nM EC50.
Formula:
C12H21N3O2
Purity:
99.01% - 99.68%
Color and Shape:
Solid
Molecular weight:
239.31
Ref: TM-T2036
| 1mg | 157.00 € | ||
| 2mg | 210.00 € | ||
| 5mg | 322.00 € | ||
| 10mg | 462.00 € | ||
| 25mg | 737.00 € | ||
| 50mg | 1,056.00 € | ||
| 100mg | 1,417.00 € | ||
| 1mL*10mM (DMSO) | 300.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
SB 242084
CAS:181632-25-7
SB 242084 dihydrochloride hydrate is a psychoactive drug and research chemical which acts as a …
Formula:
C21H19ClN4O2
Purity:
99.77% - ≥98%
Color and Shape:
Solid
Molecular weight:
394.85
Ref: TM-T7277
| 1mg | 41.00 € | ||
| 2mg | 54.00 € | ||
| 5mg | 90.00 € | ||
| 10mg | 113.00 € | ||
| 25mg | 241.00 € | ||
| 50mg | 462.00 € | ||
| 100mg | 704.00 € | ||
| 1mL*10mM (DMSO) | 89.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
AnaMorelin hydrochloride
CAS:861998-00-7
AnaMorelin hydrochloride (RC-1291 hydrochloride) is a novel ghrelin receptor agonist(EC50 : 0.74 nM, in the …
Formula:
C31H43ClN6O3
Purity:
99.18% - ≥98%
Color and Shape:
Solid
Molecular weight:
583.16
Ref: TM-T7225
| 1mg | 35.00 € | ||
| 2mg | 51.00 € | ||
| 5mg | 72.00 € | ||
| 10mg | 94.00 € | ||
| 25mg | 143.00 € | ||
| 50mg | 175.00 € | ||
| 100mg | 231.00 € | ||
| 1mL*10mM (DMSO) | 95.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Zuclopenthixol
CAS:53772-83-1
Zuclopenthixol (cis-Clopenthixol) is a thioxanthene with therapeutic actions similar to the phenothiazine antipsychotics.
Formula:
C22H25ClN2OS
Purity:
98.90% - 99.82%
Color and Shape:
Solid
Molecular weight:
400.96
Ref: TM-T4117
| 1g | 181.00 € | ||
| 25mg | 36.00 € | ||
| 50mg | 46.00 € | ||
| 100mg | 59.00 € | ||
| 500mg | 128.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
BAY-545
CAS:1699717-32-2
BAY-545 is an antagonist of A2B adenosine receptor(IC50 : 59 nM).
Formula:
C18H22F3N3O4S
Purity:
98.05%
Color and Shape:
Solid
Molecular weight:
433.45
Ref: TM-T8512
| 1mg | 86.00 € | ||
| 5mg | 164.00 € | ||
| 10mg | 238.00 € | ||
| 25mg | 428.00 € | ||
| 50mg | 615.00 € | ||
| 100mg | 857.00 € | ||
| 200mg | 1,153.00 € | ||
| 1mL*10mM (DMSO) | 175.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
CS 2100
CAS:913827-99-3
CS 2100 (1-[[4-Ethyl-5-[5-(4-phenoxyphenyl)-1,2,4-oxadiazol-3-yl]-2-thienyl]methyl]-3-azetidinecarboxylic acid) is an S1P1 agonist.
Formula:
C25H23N3O4S
Purity:
98.13%
Color and Shape:
Solid
Molecular weight:
461.53
Ref: TM-T22697
| 2mg | 41.00 € | ||
| 5mg | 62.00 € | ||
| 10mg | 88.00 € | ||
| 25mg | 172.00 € | ||
| 50mg | 271.00 € | ||
| 100mg | 398.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
cangrelor tetrasodium
CAS:163706-36-3
Cangrelor tetrasodium is a reversible and selective antagonist of platelet P2Y12, with prompt and potent …
Formula:
C17H21Cl2F3N5Na4O12P3S2
Purity:
100% - 99.15%
Color and Shape:
Solid
Molecular weight:
864.29
Ref: TM-T5036
| 1mg | 46.00 € | ||
| 2mg | 60.00 € | ||
| 5mg | 90.00 € | ||
| 10mg | 138.00 € | ||
| 25mg | 245.00 € | ||
| 50mg | 425.00 € | ||
| 100mg | 611.00 € | ||
| 500mg | 1,262.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
F-15599
CAS:635323-95-4
F-15599 is a highly selective G-protein biased 5-HT1A receptor agonist(Ki : 3.4 nM).
Formula:
C19H21ClF2N4O
Purity:
98.72%
Color and Shape:
Solid
Molecular weight:
394.85
Ref: TM-T7281
| 1mg | 51.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 156.00 € | ||
| 25mg | 304.00 € | ||
| 50mg | 489.00 € | ||
| 100mg | 735.00 € | ||
| 1mL*10mM (DMSO) | 131.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
1-Ethyl-6-aminouracil
CAS:41862-09-3
1-Ethyl-6-aminouracil (6-AMINO-1-ETHYL-1H-PYRIMIDINE-2,4-DIONE) is an intermediate in the synthesis of a series of new substituted Xanthines …
Formula:
C6H9N3O2
Purity:
99.29%
Color and Shape:
Solid
Molecular weight:
155.15
Ref: TM-T8613
| 2mg | 55.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 98.00 € | ||
| 25mg | 172.00 € | ||
| 50mg | 258.00 € | ||
| 100mg | 388.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
DAMGO
CAS:78123-71-4
DAMGO (DAGO) is an opioid receptor agonist with the ability to affect the locomotive activity …
Formula:
C26H35N5O6
Purity:
98.83% - 99.92%
Color and Shape:
Solid
Molecular weight:
513.59
Ref: TM-T4351
| 1mg | 50.00 € | ||
| 2mg | 59.00 € | ||
| 5mg | 85.00 € | ||
| 10mg | 138.00 € | ||
| 25mg | 276.00 € | ||
| 50mg | 416.00 € | ||
| 100mg | 609.00 € | ||
| 1mL*10mM (DMSO) | 88.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Pimavanserin tartrate
CAS:706782-28-7
Pimavanserin tartrate is a potent 5-HT 2A receptor inverse agonist used to treat Parkinson's disease-related …
Formula:
C50H68F2N6O4·C4H6O6
Purity:
100% - 99.98%
Color and Shape:
Solid
Molecular weight:
1005.2
Ref: TM-T6946
| 25mg | 50.00 € | ||
| 50mg | 73.00 € | ||
| 100mg | 104.00 € | ||
| 200mg | 141.00 € | ||
| 500mg | 227.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
ELA-11 (human) acetate(1784687-32-6 free base)
ELA-11: potent apelin receptor agonist, Ki=14 nM. Blocks cAMP, boosts β-arrestin. Part of ELA-32.
Formula:
C60H94N16O15S2
Purity:
99.53%
Color and Shape:
Solid
Molecular weight:
1343.61
Ref: TM-TP1922L1
| 1mg | 130.00 € | ||
| 5mg | 284.00 € | ||
| 10mg | 425.00 € | ||
| 25mg | 702.00 € | ||
| 50mg | 985.00 € | ||
| 100mg | 1,332.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
![[D-Phe12,Leu14]-Bombesin acetate](https://static.cymitquimica.com/products/TM/thumb/TP1916L1.jpg)
[D-Phe12,Leu14]-Bombesin acetate
[D-Phe12,Leu14]-Bombesin acetate inhibits bombesin-stimulated secretion.
Formula:
C77H118N22O20
Purity:
98.41% - 99.14%
Color and Shape:
Solid
Molecular weight:
1671.9
Ref: TM-TP1916L1
| 1mg | 95.00 € | ||
| 5mg | 207.00 € | ||
| 10mg | 310.00 € | ||
| 25mg | 488.00 € | ||
| 50mg | 676.00 € | ||
| 100mg | 915.00 € | ||
| 200mg | 1,235.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Gadolinium chloride
CAS:10138-52-0
Gadolinium chloride is a calcium-sensing receptor (CaSR) agonist
Formula:
Cl3Gd
Purity:
98%
Color and Shape:
White Crystalline Solid
Molecular weight:
263.61
Ref: TM-T22795
| 25mg | 48.00 € | ||
| 50mg | 58.00 € | ||
| 100mg | 90.00 € | ||
| 200mg | 124.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
RS-127445
CAS:199864-87-4
RS-127445 (MT500) is a selective 5-HT2B receptor antagonist with pKi of 9.5 and pIC50 of …
Formula:
C17H16FN3
Purity:
98.81%
Color and Shape:
Solid
Molecular weight:
281.33
Ref: TM-T6973
| 2mg | 35.00 € | ||
| 5mg | 49.00 € | ||
| 10mg | 74.00 € | ||
| 25mg | 135.00 € | ||
| 50mg | 197.00 € | ||
| 100mg | 292.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Regadenoson
CAS:313348-27-5
Regadenoson (CVT-3146) is a selective A2A receptor agonist that increases coronary blood flow with a …
Formula:
C15H18N8O5
Purity:
100% - 99.78%
Color and Shape:
Off-White Solid
Molecular weight:
390.35
Ref: TM-T2671
| 2mg | 46.00 € | ||
| 5mg | 64.00 € | ||
| 10mg | 90.00 € | ||
| 25mg | 170.00 € | ||
| 50mg | 269.00 € | ||
| 100mg | 407.00 € | ||
| 500mg | 914.00 € | ||
| 1mL*10mM (DMSO) | 72.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
RFRP-1 (human) acetate(311309-25-8 free base)
RFRP-1 (human) acetate: potent NPFF2/1 agonist, alters rat/rabbit cardiac functions, and regulates rat prolactin.
Formula:
C69H105N19O16S
Purity:
96.84%
Color and Shape:
Solid
Molecular weight:
1488.77
Ref: TM-TP1937L1
| 1mg | 130.00 € | ||
| 5mg | 284.00 € | ||
| 10mg | 425.00 € | ||
| 25mg | 702.00 € | ||
| 50mg | 985.00 € | ||
| 100mg | 1,332.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Cariprazine
CAS:839712-12-8
Cariprazine (RGH-188) is a novel antipsychotic drug candidate that exhibits high affinity for the D3 …
Formula:
C21H32Cl2N4O
Purity:
99.68% - 99.75%
Color and Shape:
Solid
Molecular weight:
427.41
Ref: TM-T4577
| 1mg | 51.00 € | ||
| 2mg | 78.00 € | ||
| 5mg | 107.00 € | ||
| 10mg | 176.00 € | ||
| 25mg | 312.00 € | ||
| 50mg | 462.00 € | ||
| 100mg | 646.00 € | ||
| 1mL*10mM (DMSO) | 108.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
