G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Propionylpromazine hydrochloride
CAS:7681-67-6
Propionylpromazine hydrochloride (Propiopromazine hydrochloride) is a dopamine receptor D2 (DRD2) antagonist.
Formula:
C20H25ClN2OS
Purity:
99.17%
Color and Shape:
Solid
Molecular weight:
376.94
Ref: TM-T9228
| 1mg | 38.00 € | ||
| 5mg | 80.00 € | ||
| 10mg | 118.00 € | ||
| 25mg | 184.00 € | ||
| 50mg | 276.00 € | ||
| 1mL*10mM (DMSO) | 92.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Spinorphin
CAS:137201-62-8
Spinorphin is a heptapeptide, and is a potent enkephalin-degrading enzymes inhibitor.
Formula:
C45H64N8O10
Purity:
99.68%
Color and Shape:
Solid
Molecular weight:
877
Ref: TM-T8455
| 1mg | 129.00 € | ||
| 5mg | 241.00 € | ||
| 10mg | 373.00 € | ||
| 25mg | 622.00 € | ||
| 50mg | 887.00 € | ||
| 100mg | 1,201.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
H2L 5765834
CAS:420841-84-5
H2L 5765834 is a lysophosphatidic acid receptors antagonist
Formula:
C21H12N2O7
Purity:
99.47% - ≥98%
Color and Shape:
Solid
Molecular weight:
404.33
Ref: TM-T22834
| 1mg | 60.00 € | ||
| 5mg | 118.00 € | ||
| 10mg | 184.00 € | ||
| 25mg | 346.00 € | ||
| 50mg | 513.00 € | ||
| 100mg | 730.00 € | ||
| 1mL*10mM (DMSO) | 130.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Ebastine
CAS:90729-43-4
Ebastine (Kestine) (trade names Evastin, Kestine, Ebastel, Aleva) is a non-sedating H1 antihistamine.
Formula:
C32H39NO2
Purity:
100% - 99.93%
Color and Shape:
White To Off-White Powder
Molecular weight:
469.66
Ref: TM-T2335
| 500mg | 56.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Adrenorphin 3TFA(88377-68-8(free base))
Adrenorphin 3TFA(88377-68-8(free base)) (Metorphamide) is an agonist of μ-opioid receptor(Ki :12 nM).
Formula:
C50H72N15O15S
Purity:
100%
Color and Shape:
Solid
Molecular weight:
1326.26
Ref: TM-T7567L
| 1mg | 47.00 € | ||
| 5mg | 121.00 € | ||
| 10mg | 174.00 € | ||
| 25mg | 314.00 € | ||
| 50mg | 450.00 € | ||
| 100mg | 621.00 € | ||
| 200mg | 836.00 € | ||
| 1mL*10mM (DMSO) | 180.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
S1RA hydrochloride
CAS:1265917-14-3
S1RA hydrochloride (E-52862 hydrochloride) is an effective and specific sigma-1 receptor(σ1R, Ki: 17 nM) antagonist, …
Formula:
C20H24ClN3O2
Purity:
98% - 99.78%
Color and Shape:
Solid
Molecular weight:
373.87
Ref: TM-T4229
| 1mg | 38.00 € | ||
| 5mg | 80.00 € | ||
| 10mg | 111.00 € | ||
| 25mg | 217.00 € | ||
| 50mg | 353.00 € | ||
| 100mg | 518.00 € | ||
| 500mg | 1,004.00 € | ||
| 1mL*10mM (DMSO) | 88.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Capadenoson
CAS:544417-40-5
Capadenoson (BAY 68-4986) is a selective adenosine-A1 receptor agonist.
Formula:
C25H18ClN5O2S2
Purity:
98.85% - 99.62%
Color and Shape:
Solid
Molecular weight:
520.03
Ref: TM-TQ0125
| 5mg | 41.00 € | ||
| 10mg | 56.00 € | ||
| 25mg | 104.00 € | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
![[D-Ala2]leucine-enkephalin](https://static.cymitquimica.com/products/TM/thumb/TP1367.jpg)
[D-Ala2]leucine-enkephalin
CAS:64963-01-5
[D-Ala2]-Leucine enkephalin is a delta opioid agonist used to study the signaling pathway of delta …
Formula:
C29H39N5O7
Purity:
98.06%
Color and Shape:
Solid
Molecular weight:
569.65
Ref: TM-TP1367
| 2mg | 41.00 € | ||
| 5mg | 62.00 € | ||
| 10mg | 95.00 € | ||
| 25mg | 167.00 € | ||
| 50mg | 326.00 € | ||
| 100mg | 460.00 € | ||
| 200mg | 643.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
BWX 46 Acetate
BWX 46 Acetate is a potent, highly selective neuropeptide Y (NPY) receptor agonist with IC50 …
Formula:
C118H190N36O30S2
Purity:
96.86%
Color and Shape:
Solid
Molecular weight:
2657.12
Ref: TM-T21611L
| 1mg | 235.00 € | ||
| 2mg | 328.00 € | ||
| 5mg | 489.00 € | ||
| 10mg | 705.00 € | ||
| 25mg | 1,095.00 € | ||
| 50mg | 1,467.00 € | ||
| 100mg | 1,990.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
9-FLUORENOL
CAS:1689-64-1
9-FLUORENOL is a dopamine reuptake inhibitor with IC50 of 9 μM, and a major metabolite …
Formula:
C13H10O
Purity:
99.98%
Color and Shape:
Off-White Crystalline Powder
Molecular weight:
182.22
Ref: TM-T8633
| 1g | 34.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Pitolisant hydrochloride
CAS:903576-44-3
Pitolisant hydrochloride (Ciproxidine) is a potent and selective inverse agonist of the histamine H3 receptor(Ki …
Formula:
C17H27Cl2NO
Purity:
99.26% - 99.72%
Color and Shape:
Solid
Molecular weight:
332.31
Ref: TM-T7176
| 5mg | 51.00 € | ||
| 10mg | 73.00 € | ||
| 25mg | 122.00 € | ||
| 50mg | 193.00 € | ||
| 100mg | 305.00 € | ||
| 200mg | 460.00 € | ||
| 500mg | 731.00 € | ||
| 1mL*10mM (DMSO) | 53.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Ozanimod
CAS:1306760-87-1
Ozanimod (RPC-1063) (RPC1063) is a specific oral S1P Receptor 1 modulator.
Formula:
C23H24N4O3
Purity:
98.68% - 99.74%
Color and Shape:
Solid
Molecular weight:
404.46
Ref: TM-T6923
| 1mg | 48.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 142.00 € | ||
| 25mg | 276.00 € | ||
| 50mg | 444.00 € | ||
| 100mg | 641.00 € | ||
| 200mg | 907.00 € | ||
| 500mg | 1,346.00 € | ||
| 1mL*10mM (DMSO) | 95.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Almotriptan Malate
CAS:181183-52-8
Almotriptan Malate (PNU180638), a selective 5-HT1B/1D receptor agonist, is used in the therapy of Migraine …
Formula:
C17H25N3O2S·C4H6O5
Purity:
98.66%
Color and Shape:
Pale Yellow Solid
Molecular weight:
469.55
Ref: TM-T2317
| 25mg | 51.00 € | ||
| 50mg | 88.00 € | ||
| 100mg | 126.00 € | ||
| 200mg | 181.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
5'-N-Ethylcarboxamidoadenosine
CAS:35920-39-9
NECA, an adenosine receptor agonist, boosts brain extravasation of fluorescein and dextran without affecting the …
Formula:
C12H16N6O4
Purity:
≥95%
Color and Shape:
Powder
Molecular weight:
308.29
Ref: TM-T7340
| 5mg | 53.00 € | ||
| 10mg | 60.00 € | ||
| 25mg | 99.00 € | ||
| 50mg | 146.00 € | ||
| 100mg | 207.00 € | ||
| 1mL*10mM (DMSO) | 63.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Endothelin 1 (swine, human) acetate
Endothelin 1 acetate is a synthetic vasoconstrictor peptide mimicking human/swine sequences, targeting ETA/ETB receptors.
Formula:
C111H163N25O34S5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
2551.95
Ref: TM-T19309L1
| 1mg | 207.00 € | ||
| 5mg | 514.00 € | ||
| 50mg | 1,538.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
ELA-14(human) acetate
ELA-14(human) acetate, a fragment of ELA, targets APJ, activates Gαi1 and β-arrestin-2, and prompts receptor …
Formula:
C77H123N25O19S2
Purity:
97.20%
Color and Shape:
Solid
Molecular weight:
1767.09
Ref: TM-TP1923L1
| 1mg | 61.00 € | ||
| 5mg | 196.00 € | ||
| 10mg | 294.00 € | ||
| 25mg | 475.00 € | ||
| 50mg | 653.00 € | ||
| 100mg | 869.00 € | ||
| 200mg | 1,163.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Desvenlafaxine succinate hydrate
CAS:386750-22-7
Desvenlafaxine succinate hydrate (WY 45233 Succinate) is an antidepressant of the serotonin-norepinephrine reuptake inhibitor (SNRI).
Formula:
C20H33NO7
Purity:
99.39%
Color and Shape:
White Crystalline Powde
Molecular weight:
399.48
Ref: TM-T6188
| 10mg | 35.00 € | ||
| 25mg | 57.00 € | ||
| 50mg | 73.00 € | ||
| 100mg | 113.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Tyr-Gly-Gly-Phe-Met-OH
CAS:58569-55-4
Tyr-Gly-Gly-Phe-Met-OH (Met-Enkephalin), is a naturally occurring, endogenous opioid peptide that inhibits tumor growth via binding …
Formula:
C27H35N5O7S
Purity:
≥95%
Color and Shape:
White Lyophilised Solid
Molecular weight:
573.66
Ref: TM-T7211
| 10mg | 35.00 € | ||
| 25mg | 55.00 € | ||
| 50mg | 88.00 € | ||
| 100mg | 124.00 € | ||
| 200mg | 177.00 € | ||
| 1mL*10mM (DMSO) | 37.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Cetrorelix diacetate
CAS:130143-01-0
Cetrorelix diacetate (NS-75A) is is a gonadotropin-releasing hormone antagonist.
Formula:
C74H100ClN17O18
Purity:
98.38%
Color and Shape:
Solid
Molecular weight:
1551.17
Ref: TM-T5520L
| 1mg | 52.00 € | ||
| 5mg | 89.00 € | ||
| 10mg | 147.00 € | ||
| 25mg | 287.00 € | ||
| 50mg | 428.00 € | ||
| 100mg | 628.00 € | ||
| 500mg | 1,327.00 € | ||
| 1mL*10mM (DMSO) | 250.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Namodenoson
CAS:163042-96-4
Namodenoson (2-Cl-IB-MECA) is an adenosine A3 receptor agonist.
Formula:
C18H18ClIN6O4
Purity:
99.4%
Color and Shape:
Solid
Molecular weight:
544.73
Ref: TM-T6884
| 1mg | 37.00 € | ||
| 5mg | 79.00 € | ||
| 10mg | 120.00 € | ||
| 25mg | 235.00 € | ||
| 50mg | 377.00 € | ||
| 100mg | 567.00 € | ||
| 1mL*10mM (DMSO) | 96.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
