G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Piperoxan hydrochloride
CAS:135-87-5
Piperoxan hydrochloride (Benodaine hydrochloride) is an α2 adrenoceptor antagonist.
Formula:
C14H20ClNO2
Purity:
99.59%
Color and Shape:
Solid
Molecular weight:
269.77
Ref: TM-T4526
| 1mg | 48.00 € | ||
| 2mg | 64.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 143.00 € | ||
| 25mg | 214.00 € | ||
| 50mg | 279.00 € | ||
| 100mg | 349.00 € | ||
| 200mg | 304.00 € | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Tolvaptan
CAS:150683-30-0
Tolvaptan (OPC-41061) is an orally bioavailable, selective, arginine vasopressin receptor 2 (V2, AVPR2) antagonist that …
Formula:
C26H25ClN2O3
Purity:
97% - 99.78%
Color and Shape:
Solid
Molecular weight:
448.94
Ref: TM-T2326
| 1mg | 38.00 € | ||
| 2mg | 49.00 € | ||
| 5mg | 80.00 € | ||
| 10mg | 113.00 € | ||
| 25mg | 202.00 € | ||
| 50mg | 357.00 € | ||
| 1mL*10mM (DMSO) | 126.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Urantide acetate(669089-53-6 free base)
Urantide acetate: selective UT receptor blocker, doesn't affect other contractions or relaxations, partial agonist in …
Formula:
C53H70N10O14S2
Purity:
99.22%
Color and Shape:
Solid
Molecular weight:
1135.31
Ref: TM-TP2106L
| 1mg | 112.00 € | ||
| 5mg | 217.00 € | ||
| 10mg | 311.00 € | ||
| 25mg | 525.00 € | ||
| 50mg | 757.00 € | ||
| 100mg | 1,056.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
(S)-Amisulpride
CAS:71675-92-8
(S)-Amisulpride ((S) Amisulpride) (Esamisulpride) is a potent dopamine D2/D3 receptor antagonist.
Formula:
C17H27N3O4S
Purity:
98.38%
Color and Shape:
Solid
Molecular weight:
369.48
Ref: TM-T26375
| 1mg | 49.00 € | ||
| 2mg | 69.00 € | ||
| 5mg | 110.00 € | ||
| 10mg | 172.00 € | ||
| 25mg | 326.00 € | ||
| 50mg | 516.00 € | ||
| 100mg | 699.00 € | ||
| 200mg | 898.00 € | ||
| 1mL*10mM (DMSO) | 121.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Procaterol hydrochloride
CAS:81262-93-3
Short-acting β2-adrenergic receptor agonist used to treat asthma.
Formula:
C32H48Cl2N4O7
Purity:
100%
Color and Shape:
Solid
Molecular weight:
671.65
Ref: TM-T4548
| 1mg | 64.00 € | ||
| 5mg | 130.00 € | ||
| 10mg | 184.00 € | ||
| 25mg | 328.00 € | ||
| 50mg | 547.00 € | ||
| 100mg | 777.00 € | ||
| 1mL*10mM (DMSO) | 186.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Mini Gastrin I, human acetate
Mini Gastrin I, human acetate is a shorter version of human gastrin, consists of amino …
Formula:
C76H103N15O28S
Purity:
99.35% - 99.82%
Color and Shape:
Solid
Molecular weight:
1706.78
Ref: TM-TP1821L
| 1mg | 170.00 € | ||
| 5mg | 629.00 € | ||
| 10mg | 1,007.00 € | ||
| 25mg | 1,825.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
ML339
CAS:2579689-83-9
ML339 a selective inhibitor of CXCR6(IC50 = 140 nM) with no response when screened against …
Formula:
C26H32ClN3O5
Purity:
99.46%
Color and Shape:
Solid
Molecular weight:
502
Ref: TM-T9721
| 1mg | 45.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 142.00 € | ||
| 25mg | 276.00 € | ||
| 50mg | 446.00 € | ||
| 100mg | 640.00 € | ||
| 1mL*10mM (DMSO) | 96.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
S 38093
CAS:862896-30-8
S 38093 is a brain-penetrant antagonist of the H3 receptor (Ki: 8.8/1.44/1.2 μM, for rat/mouse/human).
Formula:
C17H24N2O2
Purity:
99.98%
Color and Shape:
Solid
Molecular weight:
288.38
Ref: TM-T4099
| 1mg | 46.00 € | ||
| 2mg | 59.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 119.00 € | ||
| 25mg | 209.00 € | ||
| 50mg | 347.00 € | ||
| 100mg | 551.00 € | ||
| 200mg | 451.00 € | ||
| 1mL*10mM (DMSO) | 89.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Etelcalcetide hydrochloride
CAS:1334237-71-6
Etelcalcetide HCl, a synthetic peptide modulator of CaSR, lowers PTH in dialysis patients with secondary …
Formula:
C38H73N21O10S2HCl
Purity:
100%
Color and Shape:
Solid
Molecular weight:
1353.33
Ref: TM-TP1236
| 1mg | 35.00 € | ||
| 5mg | 73.00 € | ||
| 10mg | 101.00 € | ||
| 25mg | 184.00 € | ||
| 50mg | 325.00 € | ||
| 100mg | 535.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Tandospirone citrate
CAS:112457-95-1
Tandospirone citrate (SM-3997 citrate) is a potent and selective 5-HT1A receptor partial agonist (Ki : …
Formula:
C27H37N5O9
Purity:
97.84% - 99.83%
Color and Shape:
Solid
Molecular weight:
575.61
Ref: TM-T7412
| 2mg | 35.00 € | ||
| 5mg | 51.00 € | ||
| 10mg | 82.00 € | ||
| 25mg | 148.00 € | ||
| 50mg | 226.00 € | ||
| 100mg | 362.00 € | ||
| 1mL*10mM (DMSO) | 72.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
MDL 100009
CAS:175673-57-1
MDL 100009, the S-enantiomer of MDL 100151 and the opposite enantiomer of MDL 100907, is …
Formula:
C22H28FNO3
Purity:
98.96%
Color and Shape:
Solid
Molecular weight:
373.46
Ref: TM-T22359
| 1mg | 143.00 € | ||
| 2mg | 182.00 € | ||
| 5mg | 272.00 € | ||
| 10mg | 408.00 € | ||
| 25mg | 632.00 € | ||
| 50mg | 851.00 € | ||
| 100mg | 1,126.00 € | ||
| 200mg | 1,537.00 € | ||
| 1mL*10mM (DMSO) | 323.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
BMY 7378 dihydrochloride
CAS:21102-95-4
BMY 7378 dihydrochloride (BMY7378 HCl) , α1D-adrenergic receptor antagonist, is a weak partial agonist/antagonist of …
Formula:
C22H33Cl2N3O3
Purity:
97.67% - 99.08%
Color and Shape:
Solid
Molecular weight:
458.42
Ref: TM-T3046
| 5mg | 43.00 € | ||
| 10mg | 47.00 € | ||
| 25mg | 84.00 € | ||
| 50mg | 99.00 € | ||
| 1mL*10mM (DMSO) | 46.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
FK962
CAS:283167-06-6
FK962 is an somatostatin release enhancer , exerts cognitive-enhancing actions.
Formula:
C14H17FN2O2
Purity:
99.89%
Color and Shape:
Solid
Molecular weight:
264.3
Ref: TM-T7829
| 1mg | 36.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 108.00 € | ||
| 25mg | 203.00 € | ||
| 50mg | 293.00 € | ||
| 100mg | 403.00 € | ||
| 200mg | 566.00 € | ||
| 1mL*10mM (DMSO) | 84.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
AC 187 Acetate
AC 187 Acetate is a potent antagonist of amylin receptor .AC 187 shows more selective …
Formula:
C129H209N37O42
Purity:
99.71%
Color and Shape:
Solid
Molecular weight:
2950.26
Ref: TM-T21581L
| 1mg | 851.00 € | ||
| 5mg | 1,726.00 € | ||
| 10mg | 2,303.00 € | ||
| 25mg | 3,452.00 € | ||
| 50mg | 4,565.00 € | ||
| 100mg | 6,288.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Landiolol hydrochloride
CAS:144481-98-1
Landiolol hydrochloride (ONO-1101 hydrochloride) is an ultra-short-acting β1 selective adrenoceptor antagonist.
Formula:
C25H40ClN3O8
Purity:
100%
Color and Shape:
White Crystalline Powder
Molecular weight:
546.05
Ref: TM-T5028
| 5mg | 35.00 € | ||
| 10mg | 47.00 € | ||
| 25mg | 79.00 € | ||
| 50mg | 102.00 € | ||
| 100mg | 141.00 € | ||
| 200mg | 203.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Substance P 1-9 aceate
Substance P 1-9 aceate is nonapeptide, which decreases the inactivation of substance P by the …
Formula:
C54H81N15O14
Purity:
99.01%
Color and Shape:
Solid
Molecular weight:
1164.31
Ref: TM-TP1819L
| 1mg | 41.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 147.00 € | ||
| 25mg | 258.00 € | ||
| 50mg | 377.00 € | ||
| 100mg | 538.00 € | ||
| 200mg | 729.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
N-terminally acetylated Leu-enkephalin
Leu-enkephalin, an endogenous 5-amino acid peptide, activates opioid receptors; its acetylated form exists.
Formula:
C30H39N5O8
Purity:
100%
Color and Shape:
Solid
Molecular weight:
597.66
Ref: TM-T8557
| 1mg | 79.00 € | ||
| 5mg | 142.00 € | ||
| 10mg | 212.00 € | ||
| 25mg | 368.00 € | ||
| 50mg | 538.00 € | ||
| 100mg | 769.00 € | ||
| 500mg | 1,533.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
WAY-100635 Monomaleate
CAS:1092679-51-0
WAY-100635 maleate is a selective 5-hydroxytryptamine 1A receptor antagonist with an IC50 value of 0.91 …
Formula:
C25H34N4O2·C4H4O4
Purity:
100% - 99.68%
Color and Shape:
Solid
Molecular weight:
538.64
Ref: TM-T2631
| 2mg | 50.00 € | ||
| 5mg | 66.00 € | ||
| 10mg | 94.00 € | ||
| 25mg | 178.00 € | ||
| 50mg | 330.00 € | ||
| 100mg | 490.00 € | ||
| 200mg | 708.00 € | ||
| 500mg | 1,093.00 € | ||
| 1mL*10mM (DMSO) | 78.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Detomidine hydrochloride
CAS:90038-01-0
Detomidine hydrochloride (MPV-253 AII) produce dose-dependent sedative and analgesic effects, mediatated by activation of α2 …
Formula:
C12H14N2·HCl
Purity:
99.89%
Color and Shape:
Solid
Molecular weight:
222.71
Ref: TM-T6464
| 10mg | 35.00 € | ||
| 25mg | 47.00 € | ||
| 50mg | 51.00 € | ||
| 100mg | 69.00 € | ||
| 500mg | 147.00 € | ||
| 1mL*10mM (DMSO) | 35.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
AMD-070 hydrochloride
CAS:880549-30-4
AMD-070 hydrochloride is a CXCR4 antagonist, is useful for Anti HIV.
Formula:
C21H28ClN5
Purity:
98.38% - 98.57%
Color and Shape:
Solid
Molecular weight:
385.93
Ref: TM-T22565
| 1mg | 49.00 € | ||
| 2mg | 68.00 € | ||
| 5mg | 92.00 € | ||
| 10mg | 138.00 € | ||
| 25mg | 267.00 € | ||
| 50mg | 400.00 € | ||
| 100mg | 592.00 € | ||
| 1mL*10mM (DMSO) | 104.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
