G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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VUF10460
CAS:1028327-66-3
VUF10460 is a non-imidazole histamine H4 receptor agonist.
Formula:
C15H19N5
Purity:
98.68% - 99.53%
Color and Shape:
Solid
Molecular weight:
269.34
Ref: TM-T3963
| 5mg | 34.00 € | ||
| 10mg | 52.00 € | ||
| 25mg | 93.00 € | ||
| 50mg | 164.00 € | ||
| 100mg | 247.00 € | ||
| 200mg | 365.00 € | ||
| 1mL*10mM (DMSO) | 39.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
SRT3109
CAS:1204707-71-0
SRT3109 is a CXCR2 ligand used in the treatment of chemokine mediated diseases and conditions.
Formula:
C18H23F2N5O4S2
Purity:
99.65% - 99.92%
Color and Shape:
Solid
Molecular weight:
475.53
Ref: TM-T3047
| 2mg | 41.00 € | ||
| 5mg | 60.00 € | ||
| 10mg | 96.00 € | ||
| 25mg | 170.00 € | ||
| 50mg | 299.00 € | ||
| 1mL*10mM (DMSO) | 64.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
2-(pentylsulfanyl)pyrimidine-4,6-diol
CAS:489403-70-5
2-(pentylsulfanyl)pyrimidine-4,6-diol is a novel GRP84 agonist.
Formula:
C9H14N2O2S
Purity:
97.58%
Color and Shape:
Solid
Molecular weight:
214.28
Ref: TM-T50078
| 1mg | 81.00 € | ||
| 5mg | 166.00 € | ||
| 10mg | 240.00 € | ||
| 25mg | 394.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
L-(R,S)-Tetrahydropalmatine
CAS:10097-84-4
L-(R,S)-Tetrahydropalmatine (Rotundine) is extracted from Corydalis yanhusuo W. T. Wang.
Formula:
C21H25NO4
Purity:
99% - 99.97%
Color and Shape:
Solid
Molecular weight:
355.43
Ref: TM-T2714
| 1g | 137.00 € | ||
| 50mg | 33.00 € | ||
| 100mg | 48.00 € | ||
| 200mg | 61.00 € | ||
| 500mg | 93.00 € | ||
| 1mL*10mM (DMSO) | 33.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Leuphasyl TFA
CAS:67586-27-0
Leuphasyl TFA: a long-lasting, degradation-resistant peptide & δ-opioid receptor agonist for signaling research.
Formula:
C31H40F3N5O9
Purity:
98.79%
Color and Shape:
Solid
Molecular weight:
683.67
Ref: TM-T20435L
| 1mg | 83.00 € | ||
| 2mg | 107.00 € | ||
| 5mg | 172.00 € | ||
| 10mg | 249.00 € | ||
| 25mg | 410.00 € | ||
| 50mg | 577.00 € | ||
| 100mg | 780.00 € | ||
| 200mg | 1,034.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Ansofaxine hydrochloride
CAS:916918-84-8
Ansofaxine hydrochloride (LY03005) is a serotonin-norepinephrine-dopamine reuptake inhibitor (IC50s: 723, 763 and 491 nM, respectively).
Formula:
C24H32ClNO3
Purity:
99.57% - 99.77%
Color and Shape:
Solid
Molecular weight:
417.97
Ref: TM-T5380
| 1mg | 76.00 € | ||
| 5mg | 166.00 € | ||
| 10mg | 258.00 € | ||
| 25mg | 500.00 € | ||
| 50mg | 707.00 € | ||
| 100mg | 916.00 € | ||
| 1mL*10mM (DMSO) | 175.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Tropisetron
CAS:89565-68-4
Tropisetron (ICS 205-930) is an α7-nicotinic receptor agonist and 5-HT3 receptor antagonist with Kis of …
Formula:
C17H20N2O2
Purity:
99.95%
Color and Shape:
White Solid
Molecular weight:
284.35
Ref: TM-T22448
| 10mg | 46.00 € | ||
| 25mg | 79.00 € | ||
| 50mg | 126.00 € | ||
| 100mg | 188.00 € | ||
| 500mg | 478.00 € | ||
| 1mL*10mM (DMSO) | 50.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Taminadenant
CAS:1337962-47-6
Taminadenant is an adenosine receptor antagonist.
Formula:
C10H8BrN7
Purity:
99.11%
Color and Shape:
Solid
Molecular weight:
306.12
Ref: TM-T16980
| 5mg | 51.00 € | ||
| 10mg | 87.00 € | ||
| 25mg | 126.00 € | ||
| 50mg | 167.00 € | ||
| 100mg | 247.00 € | ||
| 200mg | 369.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Riociguat
CAS:625115-55-1
Riociguat (BAY 632521) is a stimulator of guanylate cyclase which causes relaxation of vascular smooth …
Formula:
C20H19FN8O2
Purity:
99.91% - 99.95%
Color and Shape:
Solid
Molecular weight:
422.42
Ref: TM-T6968
| 5mg | 42.00 € | ||
| 10mg | 62.00 € | ||
| 25mg | 96.00 € | ||
| 50mg | 145.00 € | ||
| 100mg | 240.00 € | ||
| 200mg | 349.00 € | ||
| 1mL*10mM (DMSO) | 44.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Etrasimod
CAS:1206123-37-6
Etrasimod (APD334) is a specific and orally available antagonist of the sphingosine-1-phosphate-1 (S1P1) receptor (IC50: …
Formula:
C26H26F3NO3
Purity:
99.17% - 99.77%
Color and Shape:
Solid
Molecular weight:
457.48
Ref: TM-TQ0227
| 1mg | 52.00 € | ||
| 5mg | 109.00 € | ||
| 10mg | 176.00 € | ||
| 25mg | 237.00 € | ||
| 50mg | 299.00 € | ||
| 100mg | 414.00 € | ||
| 1mL*10mM (DMSO) | 111.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Asapiprant
CAS:932372-01-5
Asapiprant (S-555739) is a potent and selective DP1 receptor antagonist (Ki: 0.44 nM). It exhibited …
Formula:
C24H27N3O7S
Purity:
99.64%
Color and Shape:
Solid
Molecular weight:
501.55
Ref: TM-T5386
| 1mg | 41.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 155.00 € | ||
| 25mg | 282.00 € | ||
| 50mg | 446.00 € | ||
| 100mg | 726.00 € | ||
| 200mg | 933.00 € | ||
| 1mL*10mM (DMSO) | 105.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Lecirelin acetate(61012-19-9 free base)
Lecirelin acetate is a synthetic GnRH (gonadotropin releasing hormone) analogue which shows a great efficacy …
Formula:
C61H88N16O14
Purity:
98.1%
Color and Shape:
Solid
Molecular weight:
1269.45
Ref: TM-TP1434L
| 1mg | 75.00 € | ||
| 5mg | 131.00 € | ||
| 10mg | 180.00 € | ||
| 25mg | 269.00 € | ||
| 50mg | 322.00 € | ||
| 100mg | 487.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Flupentixol dihydrochloride
CAS:2413-38-9
Flupentixol dihydrochloride is used in therapy of schizophrenia as well as in anxiolytic and depressive …
Formula:
C23H27Cl2F3N2OS
Purity:
100% - ≥95%
Color and Shape:
White Or Off-White Solid
Molecular weight:
507.43
Ref: TM-T5135
| 5mg | 51.00 € | ||
| 10mg | 64.00 € | ||
| 25mg | 92.00 € | ||
| 50mg | 132.00 € | ||
| 100mg | 182.00 € | ||
| 500mg | 467.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Nelociguat
CAS:625115-52-8
Nelociguat (BAY60-4552) is an sGC stimulator, crucial in NO signal pathways.
Formula:
C19H17FN8O2
Purity:
99.19%
Color and Shape:
Solid
Molecular weight:
408.39
Ref: TM-T7201
| 1mg | 36.00 € | ||
| 5mg | 73.00 € | ||
| 10mg | 105.00 € | ||
| 25mg | 156.00 € | ||
| 50mg | 203.00 € | ||
| 100mg | 331.00 € | ||
| 200mg | 422.00 € | ||
| 500mg | 554.00 € | ||
| 1mL*10mM (DMSO) | 84.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Cinacalcet hydrochloride
CAS:364782-34-3
Cinacalcet hydrochloride (AMG-073 hydrochloride) is a naphthalene derivative and CALCIMIMETIC AGENT that increases the sensitivity …
Formula:
C22H23ClF3N
Purity:
99.9% - 99.94%
Color and Shape:
Off-White To Tan Solid
Molecular weight:
393.87
Ref: TM-T2406
| 10mg | 51.00 € | ||
| 25mg | 69.00 € | ||
| 50mg | 86.00 € | ||
| 100mg | 143.00 € | ||
| 200mg | 182.00 € | ||
| 500mg | 304.00 € | ||
| 1mL*10mM (DMSO) | 53.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
THIQ
CAS:312637-48-2
THIQ is a selective melanocortin-4 receptor (MC4R) agonist (hMC4R and rMC4R with IC50 of 1.2 …
Formula:
C33H41ClN6O2
Purity:
98.93%
Color and Shape:
Solid
Molecular weight:
589.17
Ref: TM-T8485
| 1mg | 52.00 € | ||
| 2mg | 72.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 176.00 € | ||
| 25mg | 365.00 € | ||
| 50mg | 557.00 € | ||
| 100mg | 829.00 € | ||
| 1mL*10mM (DMSO) | 133.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
PF3274167
CAS:900510-03-4
PF3274167 (Cligosiban) is a potent and selective, high-affinity nonpeptide oxytocin receptor antagonist.
Formula:
C19H19ClFN5O3
Purity:
99.67% - 99.88%
Color and Shape:
Solid
Molecular weight:
419.84
Ref: TM-T3347
| 5mg | 35.00 € | ||
| 10mg | 50.00 € | ||
| 25mg | 91.00 € | ||
| 50mg | 147.00 € | ||
| 100mg | 229.00 € | ||
| 1mL*10mM (DMSO) | 36.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
MCOPPB triHydrochloride
CAS:1108147-88-1
MCOPPB triHydrochloride (MCOPPB 3HCl) is a nociceptin receptor agonist.
Formula:
C26H43Cl3N4
Purity:
99.89% - 99.91%
Color and Shape:
Solid
Molecular weight:
518.01
Ref: TM-T2071
| 2mg | 34.00 € | ||
| 5mg | 49.00 € | ||
| 10mg | 84.00 € | ||
| 25mg | 158.00 € | ||
| 50mg | 246.00 € | ||
| 100mg | 362.00 € | ||
| 200mg | 516.00 € | ||
| 1mL*10mM (DMSO) | 56.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
LIT927
CAS:2172879-52-4
LIT927 (LIT-927) is an orally active CXCL12 neutraligand (Ki: 267 nM for CXCL12 binding to …
Formula:
C17H13ClN2O3
Purity:
99.57% - 99.73%
Color and Shape:
Solid
Molecular weight:
328.75
Ref: TM-T5207
| 2mg | 41.00 € | ||
| 5mg | 61.00 € | ||
| 10mg | 96.00 € | ||
| 25mg | 152.00 € | ||
| 50mg | 226.00 € | ||
| 100mg | 330.00 € | ||
| 500mg | 779.00 € | ||
| 1mL*10mM (DMSO) | 68.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Neurokinin A
CAS:86933-74-6
Neurokinin A (NKA), formerly known as Substance K, is a neurologically active peptide translated from …
Formula:
C50H80N14O14S
Purity:
100%
Color and Shape:
White To Off-White Lyophilized Solid
Molecular weight:
1133.32
Ref: TM-TP1008
| 1mg | 60.00 € | ||
| 5mg | 117.00 € | ||
| 10mg | 195.00 € | ||
| 25mg | 329.00 € | ||
| 50mg | 488.00 € | ||
| 100mg | 694.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
