G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Niaprazine
CAS:27367-90-4
Niaprazine is a histamine H1-receptor antagonist with marked sedative properties.
Formula:
C20H25FN4O
Purity:
99.5%
Color and Shape:
Solid
Molecular weight:
356.44
Ref: TM-T36949
| 1ml | 62.00 € | ||
| 2mg | 39.00 € | ||
| 5mg | 56.00 € | ||
| 10mg | 93.00 € | ||
| 25mg | 140.00 € | ||
| 50mg | 203.00 € | ||
| 100mg | 299.00 € | ||
| 200mg | 429.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Perospirone hydrochloride
CAS:129273-38-7
Perospirone hydrochloride (Perospirone HCl) is an atypical antipsychotic agent for the treatment of schizophrenia.
Formula:
C23H31ClN4O2S
Purity:
99.37%
Color and Shape:
White Solid
Molecular weight:
463
Ref: TM-T8136
| 1ml | 34.00 € | ||
| 25mg | 44.00 € | ||
| 50mg | 60.00 € | ||
| 100mg | 87.00 € | ||
| 200mg | 112.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Ablukast
CAS:96566-25-5
Ablukast (Ro 23-3544) is a leuktriene receptor antagonist. Ablukast acts as an anti-asthmatic.
Formula:
C28H34O8
Purity:
99.18%
Color and Shape:
Solid
Molecular weight:
498.56
Ref: TM-T26519
| 1mg | 73.00 € | ||
| 1ml | 198.00 € | ||
| 5mg | 180.00 € | ||
| 10mg | 291.00 € | ||
| 25mg | 575.00 € | ||
| 50mg | 806.00 € | ||
| 100mg | 1,095.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
5,7-Dimethoxyluteolin
CAS:90363-40-9
5,7-Dimethoxyluteolin is a natural product from Hovenia acerba. 5,7-Dimethoxyluteolin is a dopamine transporter (DAT) activator …
Formula:
C17H14O6
Purity:
99.56%
Color and Shape:
Solid
Molecular weight:
314.29
Ref: TM-TN6552
| 1mg | 63.00 € | ||
| 2mg | 94.00 € | ||
| 5mg | 143.00 € | ||
| 10mg | 205.00 € | ||
| 25mg | To inquire |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Atipamezole hydrochloride
CAS:104075-48-1
Atipamezole is a synthetic α2 adrenergic receptor antagonist.
Formula:
C14H16N2·HCl
Purity:
96.71%
Color and Shape:
Solid
Molecular weight:
248.75
Ref: TM-T6765
| 1ml | 57.00 € | ||
| 5mg | 56.00 € | ||
| 10mg | 78.00 € | ||
| 25mg | 135.00 € | ||
| 50mg | 231.00 € | ||
| 100mg | 341.00 € | ||
| 200mg | 528.00 € | ||
| 500mg | 824.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
TG4-155
CAS:1164462-05-8
TG4-155: brain-penetrant EP2 inhibitor, KB 2.4 nM; >1000x weaker at EP4, KB 11.4 μM; selective …
Formula:
C23H26N2O4
Purity:
97.20%
Color and Shape:
Solid
Molecular weight:
394.46
Ref: TM-T5482
| 1mg | 36.00 € | ||
| 1ml | 82.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 74.00 € | ||
| 10mg | 106.00 € | ||
| 25mg | 216.00 € | ||
| 50mg | 373.00 € | ||
| 100mg | 554.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Nociceptin
CAS:170713-75-4
Nociceptin (Orphanin FQ) is a 17-amino-acid polypeptide that is structurally related to the opioid peptide …
Formula:
C79H129N27O22
Purity:
99.35%
Color and Shape:
Solid
Molecular weight:
1809.04
Ref: TM-TP1071
| 1mg | 80.00 € | ||
| 5mg | 222.00 € | ||
| 10mg | 360.00 € | ||
| 25mg | 603.00 € | ||
| 50mg | 861.00 € | ||
| 100mg | 1,170.00 € | ||
| 500mg | 2,341.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
LML134
CAS:1542135-76-1
LML134 (LML-134) is an inverse agonist of Histamine 3 receptor (H3R)(hH3R cAMP and hH3R bdg …
Formula:
C19H29N5O3
Purity:
99.36%
Color and Shape:
Solid
Molecular weight:
375.47
Ref: TM-T8514
| 1mg | 79.00 € | ||
| 1ml | 182.00 € | ||
| 5mg | 170.00 € | ||
| 10mg | 265.00 € | ||
| 25mg | 493.00 € | ||
| 50mg | 726.00 € | ||
| 100mg | 1,081.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Olcegepant
CAS:204697-65-4
Olcegepant (BIBN-4096) is an effective and selective non-peptide calcitonin gene-related peptide 1 (CGRP1) receptor antagonist …
Formula:
C38H47Br2N9O5
Purity:
96.08%
Color and Shape:
Solid
Molecular weight:
869.65
Ref: TM-T12293L
| 1mg | 37.00 € | ||
| 1ml | 188.00 € | ||
| 2mg | 51.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Talinolol
CAS:57460-41-0
(±)-Talinolol is a selective β1 adrenoceptor antagonist well known for its cardioprotective and antihypertensive activity.
Formula:
C20H33N3O3
Purity:
98.80%
Color and Shape:
Solid
Molecular weight:
363.49
Ref: TM-T21640
| 1mg | 73.00 € | ||
| 1ml | 168.00 € | ||
| 2mg | 97.00 € | ||
| 5mg | 165.00 € | ||
| 10mg | 296.00 € | ||
| 25mg | 534.00 € | ||
| 50mg | 768.00 € | ||
| 100mg | 1,054.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Spexin acetate(1370290-58-6 free base)
Spexin acetate: GAL2/GAL3 agonist. EC50: 45.7/112.2 nM. Inactive at GAL1. Reduces appetite, fat uptake, and …
Formula:
C76H117N19O22S
Purity:
95.43%
Color and Shape:
Solid
Molecular weight:
1680.94
Ref: TM-TP1930L1
| 1mg | 110.00 € | ||
| 5mg | 246.00 € | ||
| 10mg | 362.00 € | ||
| 25mg | 543.00 € | ||
| 50mg | 759.00 € | ||
| 100mg | 1,035.00 € | ||
| 200mg | 1,392.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Cinacalcet hydrochloride
CAS:364782-34-3
Cinacalcet hydrochloride (AMG-073 hydrochloride) is a naphthalene derivative and CALCIMIMETIC AGENT that increases the sensitivity …
Formula:
C22H23ClF3N
Purity:
99.9% - 99.94%
Color and Shape:
Off-White To Tan Solid
Molecular weight:
393.87
Ref: TM-T2406
| 1ml | 53.00 € | ||
| 10mg | 51.00 € | ||
| 25mg | 69.00 € | ||
| 50mg | 86.00 € | ||
| 100mg | 143.00 € | ||
| 200mg | 182.00 € | ||
| 500mg | 304.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Benorilate
CAS:5003-48-5
Benorilate (Salipran) is the esterification product of paracetamol and acetylsalicylic acid with anti-inflammatory, analgesic and …
Formula:
C17H15NO5
Purity:
98.39% - 99.56%
Color and Shape:
Solid
Molecular weight:
313.3
Ref: TM-T3276
| 1g | 38.00 € | ||
| 1ml | 34.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
SB 242084
CAS:181632-25-7
SB 242084 dihydrochloride hydrate is a psychoactive drug and research chemical which acts as a …
Formula:
C21H19ClN4O2
Purity:
99.77% - ≥98%
Color and Shape:
Solid
Molecular weight:
394.85
Ref: TM-T7277
| 1mg | 41.00 € | ||
| 1ml | 89.00 € | ||
| 2mg | 54.00 € | ||
| 5mg | 90.00 € | ||
| 10mg | 113.00 € | ||
| 25mg | 241.00 € | ||
| 50mg | 462.00 € | ||
| 100mg | 704.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Obestatin (rat) acetate
Obestatin (rat) acetate is an endogenous ligand of G-protein coupled receptor 39 (GPR39).
Formula:
C114H174N34O31
Purity:
99.05%
Color and Shape:
Solid
Molecular weight:
2516.81
Ref: TM-TP2279L
| 1mg | 74.00 € | ||
| 5mg | 150.00 € | ||
| 10mg | 217.00 € | ||
| 25mg | 362.00 € | ||
| 50mg | 515.00 € | ||
| 100mg | 703.00 € | ||
| 200mg | 903.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
BRL 54443
CAS:57477-39-1
BRL 54443 is a potent 5-HT1E/1F receptor agonist (pKi values are 8.7 and 8.9 respectively).
Formula:
C14H18N2O
Purity:
99.95%
Color and Shape:
Solid
Molecular weight:
230.31
Ref: TM-T2459
| 1ml | 59.00 € | ||
| 5mg | 52.00 € | ||
| 10mg | 82.00 € | ||
| 25mg | 154.00 € | ||
| 50mg | 234.00 € | ||
| 100mg | 393.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Lodoxamide
CAS:53882-12-5
Lodoxamide (Lodoxamidum) is an antiallergic drug acting as a mast-cell stabilizer. It is effective in …
Formula:
C11H6ClN3O6
Purity:
99.13% - 99.81%
Color and Shape:
Solid
Molecular weight:
311.63
Ref: TM-T4566
| 1ml | 51.00 € | ||
| 5mg | 46.00 € | ||
| 10mg | 59.00 € | ||
| 25mg | 93.00 € | ||
| 50mg | 110.00 € | ||
| 100mg | 183.00 € | ||
| 200mg | 319.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Fenoldopam mesylate
CAS:67227-57-0
Fenoldopam mesylate (Corlopam mesylate) is a selective dopamine-1 receptor (DA1) agonist with natriuretic/diuretic properties.
Formula:
C16H16ClNO3·CH4O3S
Purity:
99.19%
Color and Shape:
Solid
Molecular weight:
401.86
Ref: TM-T6835
| 1ml | 53.00 € | ||
| 10mg | 50.00 € | ||
| 25mg | 88.00 € | ||
| 50mg | 147.00 € | ||
| 100mg | 206.00 € | ||
| 200mg | 315.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
VUF10460
CAS:1028327-66-3
VUF10460 is a non-imidazole histamine H4 receptor agonist.
Formula:
C15H19N5
Purity:
98.68% - 99.53%
Color and Shape:
Solid
Molecular weight:
269.34
Ref: TM-T3963
| 1ml | 39.00 € | ||
| 5mg | 34.00 € | ||
| 10mg | 52.00 € | ||
| 25mg | 93.00 € | ||
| 50mg | 164.00 € | ||
| 100mg | 247.00 € | ||
| 200mg | 365.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
HS024
CAS:212370-59-7
HS024 is a highly potent melanocortin MC4 receptor antagonist, increases food intake, and blocks α-MSH- …
Formula:
C58H79N19O10S2
Purity:
100%
Color and Shape:
Solid
Molecular weight:
1266.5
Ref: TM-TP1898
| 1mg | 322.00 € | ||
| 5mg | 780.00 € | ||
| 10mg | 1,067.00 € | ||
| 25mg | 1,576.00 € | ||
| 50mg | 2,127.00 € | ||
| 100mg | 2,915.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
