G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Cloprostenol sodium salt
CAS:55028-72-3
Cloprostenol sodium salt (ICI 80996 sodium salt) is a synthetic prostaglandin analogue, an agonist at …
Formula:
C22H28ClNaO6
Purity:
97.17% - 98.47%
Color and Shape:
White To Almost White Hygroscopic Powder
Molecular weight:
446.9
Ref: TM-T5847
| 1mg | 52.00 € | ||
| 5mg | 101.00 € | ||
| 10mg | 163.00 € | ||
| 25mg | 318.00 € | ||
| 50mg | 470.00 € | ||
| 100mg | 675.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
BAM 22P acetate
BAM 22P acetate is a potent opioid agonist.
Formula:
C132H188N38O33S2
Purity:
99.87%
Color and Shape:
Soild
Molecular weight:
2899.27
Ref: TM-TP1211L
| 1mg | 240.00 € | ||
| 5mg | 924.00 € | ||
| 10mg | 1,392.00 € | ||
| 25mg | 2,494.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Formoterol fumarate
CAS:43229-80-7
Formoterol fumarate (Eformoterol Hemifumarate), an effective, specific and long-acting β2-adrenoceptor agonist, is utilized in the …
Formula:
C19H24N2O4C4H4O4
Purity:
100% - 99.86%
Color and Shape:
White Powder
Molecular weight:
402.4
Ref: TM-T6505
| 5mg | 53.00 € | ||
| 10mg | 74.00 € | ||
| 25mg | 143.00 € | ||
| 50mg | 254.00 € | ||
| 100mg | 383.00 € | ||
| 200mg | 552.00 € | ||
| 1mL*10mM (DMSO) | 49.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
![[D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate](https://static.cymitquimica.com/products/TM/thumb/TP1931L1.jpg)
[D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate
Broad-spectrum neuropeptide inverse agonist/antagonist; potent at ghrelin receptor (EC50 = 5.2 nM); inhibits cancer growth, …
Formula:
C81H113N19O14
Purity:
97.68%
Color and Shape:
Solid
Molecular weight:
1576.91
Ref: TM-TP1931L1
| 1mg | 141.00 € | ||
| 5mg | 308.00 € | ||
| 10mg | 462.00 € | ||
| 25mg | 755.00 € | ||
| 50mg | 1,038.00 € | ||
| 100mg | 1,418.00 € | ||
| 500mg | 2,793.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Methylnaltrexone bromide
CAS:73232-52-7
Methylnaltrexone bromide (MOA-728) is one of the newer agents of peripherally-acting μ-opioid antagonists, acts to …
Formula:
C21H26BrNO4
Purity:
99.02%
Color and Shape:
Solid
Molecular weight:
436.35
Ref: TM-T21422
| 2mg | 51.00 € | ||
| 5mg | 83.00 € | ||
| 10mg | 114.00 € | ||
| 25mg | 187.00 € | ||
| 50mg | 266.00 € | ||
| 100mg | 462.00 € | ||
| 1mL*10mM (DMSO) | 89.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
CTAP(TFA) (103429-32-9 free base)
CTAP(TFA) (103429-32-9 free base) is a potent, highly selective, and brain-penetrant antagonist of the μ-opioid …
Formula:
C53H70F3N13O13S2
Purity:
99.62%
Color and Shape:
Solid
Molecular weight:
1218.33
Ref: TM-TP2050L
| 1mg | 191.00 € | ||
| 5mg | 477.00 € | ||
| 10mg | 690.00 € | ||
| 25mg | 1,072.00 € | ||
| 50mg | 1,439.00 € | ||
| 100mg | 1,939.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Atosiban acetate
CAS:914453-95-5
Atosiban acetate (RW22164) is an inhibitor of the hormones oxytocin and vasopressin.
Formula:
C45H71N11O14S2
Purity:
99.15% - 99.84%
Color and Shape:
Solid
Molecular weight:
1054.24
Ref: TM-T5148
| 5mg | 72.00 € | ||
| 10mg | 113.00 € | ||
| 25mg | 171.00 € | ||
| 50mg | 202.00 € | ||
| 100mg | 262.00 € | ||
| 500mg | 648.00 € | ||
| 1mL*10mM (DMSO) | 133.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Neuropeptide S (Rat) acetate
Neuropeptide S (Rat) acetate is an endogenous ligand of a previously orphan G-protein-coupled receptor now …
Formula:
C97H164N34O29
Purity:
95.36%
Color and Shape:
Solid
Molecular weight:
2270.59
Ref: TM-TP1982L
| 1mg | 144.00 € | ||
| 5mg | 316.00 € | ||
| 10mg | 467.00 € | ||
| 25mg | 744.00 € | ||
| 50mg | 1,060.00 € | ||
| 100mg | 1,426.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
BRL-15572 dihydrochloride
CAS:193611-72-2
BRL-15572 dihydrochloride: 5-HT1D antagonist, pKi 7.9, also binds 5-HT1A/2B, 60x selective over 5-HT1B.
Formula:
C25H27ClN2O·2HCl
Purity:
99.8%
Color and Shape:
Solid
Molecular weight:
479.87
Ref: TM-T6423
| 5mg | 48.00 € | ||
| 10mg | 72.00 € | ||
| 25mg | 105.00 € | ||
| 50mg | 162.00 € | ||
| 100mg | 233.00 € | ||
| 200mg | 347.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
(D-Ser2)-Leu-Enkephalin-Thr
(D-Ser2)-Leu-Enkephalin-Thr is a delta selective agent of opioid receptor and shows analgesic effects.
Formula:
C33H46N6O10
Purity:
94.17%
Color and Shape:
Soild
Molecular weight:
686.75
Ref: TM-T22752L
| 1mg | 74.00 € | ||
| 5mg | 149.00 € | ||
| 10mg | 215.00 € | ||
| 25mg | 388.00 € | ||
| 50mg | 577.00 € | ||
| 100mg | 822.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Difelikefalin acetate
Difelikefalin acetate (CR 845 acetate) is a peripherally restricted kappa opioid receptor agonist.
Formula:
C38H57N7O8
Purity:
99.55%
Color and Shape:
Liquid
Molecular weight:
739.9
Ref: TM-TP2501
| 1mg | 95.00 € | ||
| 5mg | 191.00 € | ||
| 10mg | 300.00 € | ||
| 25mg | 483.00 € | ||
| 50mg | 653.00 € | ||
| 100mg | 895.00 € | ||
| 200mg | 1,180.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
BisfluoroModafinil
CAS:90280-13-0
CRL-40940 is a selective dopaminergic reuptake inhibitor
Formula:
C15H13F2NO2S
Purity:
97.61%
Color and Shape:
Solid
Molecular weight:
309.33
Ref: TM-T4262
| 1mg | 47.00 € | ||
| 2mg | 63.00 € | ||
| 5mg | 93.00 € | ||
| 10mg | 138.00 € | ||
| 25mg | 234.00 € | ||
| 50mg | 355.00 € | ||
| 100mg | 534.00 € | ||
| 500mg | 1,106.00 € | ||
| 1mL*10mM (DMSO) | 103.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
GSK189254A
CAS:720690-73-3
GSK189254A (GSK189254) is a potent and specific histamine H3 receptor antagonist (pKi values: 9.59-9.90 and …
Formula:
C21H25N3O2
Purity:
98.04% - 98.71%
Color and Shape:
Solid
Molecular weight:
351.44
Ref: TM-TQ0066
| 1mg | 52.00 € | ||
| 5mg | 92.00 € | ||
| 10mg | 122.00 € | ||
| 50mg | 343.00 € | ||
| 100mg | 495.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Ref: 4Z-G-053001
| 10mg | To inquire | ||
| 25mg | To inquire | ||
| 50mg | To inquire | ||
| 100mg | To inquire |
Estimated delivery in United States, on Monday 16 Dec 2024
RS-127445 hydrochloride
CAS:199864-86-3
RS-127445 hydrochloride (MT 500) is a selective, high affinity, orally bioavailable 5-HT2B receptor antagonist(pKi : …
Formula:
C17H17ClFN3
Purity:
99.48%
Color and Shape:
Solid
Molecular weight:
317.79
Ref: TM-T7519
| 5mg | 35.00 € | ||
| 10mg | 49.00 € | ||
| 25mg | 90.00 € | ||
| 50mg | 123.00 € | ||
| 100mg | 177.00 € | ||
| 200mg | 264.00 € | ||
| 1mL*10mM (DMSO) | 35.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
R715 TFA(185052-09-9 free base)
R715 TFA(185052-09-9 free base) is a potent and selective bradykinin B1 receptor antagonist (pA2 = …
Formula:
C59H82F3N13O14
Purity:
100%
Color and Shape:
Solid
Molecular weight:
1254.36
Ref: TM-TP1933
| 1mg | 147.00 € | ||
| 5mg | 305.00 € | ||
| 10mg | 455.00 € | ||
| 25mg | 728.00 € | ||
| 50mg | 1,013.00 € | ||
| 100mg | 1,380.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
ML-097
CAS:743456-83-9
ML-097 (CID-2160985) is a pan activator of Ras-related GTPases
Formula:
C14H11BrO3
Purity:
99.12%
Color and Shape:
Solid
Molecular weight:
307.139
Ref: TM-T21970
| 5mg | 64.00 € | ||
| 10mg | 95.00 € | ||
| 25mg | 139.00 € | ||
| 50mg | 200.00 € | ||
| 100mg | 299.00 € | ||
| 500mg | 711.00 € | ||
| 1mL*10mM (DMSO) | 71.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
MCH(human, mouse, rat)
CAS:128315-56-0
MCH(human, mouse, rat) is a potent endogenous agonist at melanin-concentration hormone (MCH) receptors. MCH increases …
Formula:
C105H160N30O26S4
Purity:
99.55% - 99.55%
Color and Shape:
White Powder
Molecular weight:
2386.84
Ref: TM-TP1996
| 1mg | 212.00 € | ||
| 5mg | 527.00 € | ||
| 10mg | 731.00 € | ||
| 25mg | 1,096.00 € | ||
| 50mg | 1,448.00 € | ||
| 100mg | 1,953.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Nitroprusside disodium dihydrate
CAS:13755-38-9
Nitroprusside disodium dihydrate (Sodium Nitroprusside Dihydrate) is a potent vasodilator working through releasing NO spontaneously …
Formula:
C5H4FeN6Na2O3
Purity:
98%
Color and Shape:
Bright Red
Molecular weight:
297.95
Ref: TM-T6991
| 500mg | 49.00 € | ||
| 1mL*10mM (DMSO) | 53.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
![[Lys8, Lys9]-Neurotensin (8-13) acetate](https://static.cymitquimica.com/products/TM/thumb/T38807L.jpg)
[Lys8, Lys9]-Neurotensin (8-13) acetate
[Lys8, Lys9]-Neurotensin (8-13) acetate, a Neurotensin analog, exerts its analgesic effects through activation of the …
Formula:
C40H68N8O10
Purity:
98%
Color and Shape:
Solid
Molecular weight:
821.02
Ref: TM-T38807L
| 1mg | 143.00 € | ||
| 5mg | 312.00 € | ||
| 10mg | 464.00 € | ||
| 25mg | 739.00 € | ||
| 50mg | 1,049.00 € | ||
| 100mg | 1,420.00 € | ||
| 1ml*10 (DMSO) | 491.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
