G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Bilastine
CAS:202189-78-4
Bilastine (Bilaxten) is a novel new-generation antihistamine that is highly selective for the H1 histamine …
Formula:
C28H37N3O3
Purity:
99.59% - 99.61%
Color and Shape:
Solid
Molecular weight:
463.61
Ref: TM-T4250
| 25mg | 46.00 € | ||
| 50mg | 69.00 € | ||
| 100mg | 101.00 € | ||
| 200mg | 149.00 € | ||
| 500mg | 244.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
ML 154
CAS:1345964-89-7
ML 154 is a potent neuropeptide S receptor (NPSR) antagonist.
Formula:
C29H26BrN2PS
Purity:
99.44%
Color and Shape:
Solid
Molecular weight:
545.47
Ref: TM-T22994
| 1mg | 56.00 € | ||
| 2mg | 78.00 € | ||
| 5mg | 108.00 € | ||
| 10mg | 151.00 € | ||
| 25mg | 269.00 € | ||
| 50mg | 384.00 € | ||
| 100mg | 532.00 € | ||
| 200mg | 717.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
LY2828360
CAS:1231220-79-3
LY2828360: CB2 agonist, Ki=40.3 nM; biases CB2 over CB1 with EC50s of 20.1 nM and …
Formula:
C22H27ClN6O
Purity:
98.45% - 99.51%
Color and Shape:
Solid
Molecular weight:
426.94
Ref: TM-T7316
| 2mg | 43.00 € | ||
| 5mg | 51.00 € | ||
| 10mg | 83.00 € | ||
| 25mg | 142.00 € | ||
| 50mg | 198.00 € | ||
| 100mg | 291.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
MK 212 hydrochloride
CAS:61655-58-1
MK 212 hydrochloride is a 5-HT2C receptor agonist
Formula:
C8H11ClN4·HCl
Purity:
99.88%
Color and Shape:
Solid
Molecular weight:
235.12
Ref: TM-T22987
| 5mg | 44.00 € | ||
| 10mg | 56.00 € | ||
| 25mg | 102.00 € | ||
| 50mg | 164.00 € | ||
| 100mg | 250.00 € | ||
| 200mg | 359.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
IMM-01
CAS:218795-74-5
IMM-01 is a novel class of small-molecule agonists of the mammalian Diaphanous (mDia)-related formins, which …
Formula:
C12H17N3O2S
Purity:
98.87%
Color and Shape:
Solid
Molecular weight:
267.35
Ref: TM-T25529
| 1mg | 88.00 € | ||
| 5mg | 185.00 € | ||
| 10mg | 271.00 € | ||
| 25mg | 462.00 € | ||
| 50mg | 647.00 € | ||
| 100mg | 894.00 € | ||
| 500mg | 1,743.00 € | ||
| 1mL*10mM (DMSO) | 204.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
carfenazine
CAS:2622-30-2
carfenazine targets the Dopamine receptor and is used for schizophrenia research.
Formula:
C24H31N3O2S
Purity:
98.15%
Color and Shape:
Solid
Molecular weight:
425.59
Ref: TM-T9827
| 1mg | 178.00 € | ||
| 5mg | 364.00 € | ||
| 10mg | 539.00 € | ||
| 25mg | 868.00 € | ||
| 50mg | 1,186.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
FSLLRY-NH2 TFA(245329-02-6 free base)
FSLLRY-NH2 TFA inhibits PAR2, reverses taxol-induced pain, and reduces itch in mice; blocks ERK and …
Formula:
C41H61F3N10O10
Purity:
99.32%
Color and Shape:
Solid
Molecular weight:
910.99
Ref: TM-TP1904L
| 1mg | 95.00 € | ||
| 5mg | 170.00 € | ||
| 10mg | 258.00 € | ||
| 25mg | 466.00 € | ||
| 50mg | 673.00 € | ||
| 100mg | 917.00 € | ||
| 500mg | 1,839.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
PF-04418948
CAS:1078166-57-0
PF-04418948 is a potent EP2 receptor antagonist. Displays over 2000-fold selectivity for EP2 receptors over …
Formula:
C23H20FNO5
Purity:
97.61% - 99.45%
Color and Shape:
Solid
Molecular weight:
409.41
Ref: TM-T3306
| 2mg | 47.00 € | ||
| 5mg | 68.00 € | ||
| 10mg | 87.00 € | ||
| 25mg | 183.00 € | ||
| 50mg | 315.00 € | ||
| 100mg | 348.00 € | ||
| 1mL*10mM (DMSO) | 75.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
![d[Cha4]-AVP acetate(500170-27-4 free base)](https://static.cymitquimica.com/products/TM/thumb/TP2082L.jpg)
d[Cha4]-AVP acetate(500170-27-4 free base)
'd[Cha4]-AVP acetate: strong V1B agonist, weak on V1A/Oxytocin/V2. Boosts ACTH, corticosterone; low blood pressure effect.'
Formula:
C52H75N13O13S2
Purity:
99.86%
Color and Shape:
Solid
Molecular weight:
1154.37
Ref: TM-TP2082L
| 1mg | 99.00 € | ||
| 5mg | 195.00 € | ||
| 10mg | 234.00 € | ||
| 25mg | 350.00 € | ||
| 50mg | 421.00 € | ||
| 100mg | 547.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Taprenepag
CAS:752187-80-7
Taprenepag (CP-544326) (CP-544326) is a potent and selective prostaglandin E2 receptor agonist (EC50 = 2.8 …
Formula:
C24H22N4O5S
Purity:
99.15% - 99.41%
Color and Shape:
Solid
Molecular weight:
478.52
Ref: TM-T3174
| 2mg | 43.00 € | ||
| 5mg | 63.00 € | ||
| 10mg | 94.00 € | ||
| 25mg | 193.00 € | ||
| 50mg | 303.00 € | ||
| 100mg | 437.00 € | ||
| 200mg | 612.00 € | ||
| 1mL*10mM (DMSO) | 75.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Urapidil
CAS:34661-75-1
Urapidil (Ebrantil), a sympatholytic antihypertensive drug, acts as a 5-HT1A receptor agonist and as an …
Formula:
C20H29N5O3
Purity:
100%
Color and Shape:
Solid
Molecular weight:
387.48
Ref: TM-T0165
| 25mg | 39.00 € | ||
| 50mg | 56.00 € | ||
| 100mg | 79.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
ELN-441958
CAS:913064-47-8
ELN-441958 is a potent, neutral antagonist of B1 receptor, inhibits the binding of the B1 …
Formula:
C29H29ClN4O2
Purity:
98.9%
Color and Shape:
Solid
Molecular weight:
501.02
Ref: TM-T2086
| 1mg | 60.00 € | ||
| 5mg | 131.00 € | ||
| 10mg | 206.00 € | ||
| 25mg | 349.00 € | ||
| 50mg | 497.00 € | ||
| 100mg | 676.00 € | ||
| 200mg | 913.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
SEW2871
CAS:256414-75-2
SEW 2871 is an orally available, highly selective S1P1 agonist. It activates ERK, Akt and …
Formula:
C20H10F6N2OS
Purity:
99.62%
Color and Shape:
White Solid
Molecular weight:
440.36
Ref: TM-T2171
| 1mg | 57.00 € | ||
| 2mg | 82.00 € | ||
| 5mg | 152.00 € | ||
| 10mg | 250.00 € | ||
| 25mg | 405.00 € | ||
| 50mg | 597.00 € | ||
| 1mL*10mM (DMSO) | 145.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Olivetol
CAS:500-66-3
Olivetol, found in lichens, is an organic antioxidant and THC synthesis precursor.
Formula:
C11H16O2
Purity:
99.74%
Color and Shape:
(Melting Point 102-106°F) (Ntp 1992)
Molecular weight:
180.24
Ref: TM-T3736
| 500mg | 54.00 € | ||
| 1mL*10mM (DMSO) | 36.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Atrasentan
CAS:173937-91-2
Atrasentan (ABT-627) is an endothelin receptor antagonist that can inhibit the activity of ETA.Cost-effective and …
Formula:
C29H38N2O6
Purity:
99.08% - 99.08%
Color and Shape:
Solid
Molecular weight:
510.62
Ref: TM-TQ0259
| 1mg | 48.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 134.00 € | ||
| 25mg | 260.00 € | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 120.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Grapiprant
CAS:415903-37-6
Grapiprant (AAT-007) is a selective EP4 receptor antagonist.
Formula:
C26H29N5O3S
Purity:
99.49%
Color and Shape:
Solid
Molecular weight:
491.61
Ref: TM-TQ0292
| 1mg | 36.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 118.00 € | ||
| 25mg | 183.00 € | ||
| 50mg | 347.00 € | ||
| 100mg | 524.00 € | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Scyliorhinin II acetate
Scyliorhinin II acetate is a selective agonist of the neurokinin-3 (NK3) receptor (Ki = 2.5 …
Formula:
C79H123N21O28S3
Purity:
99.06%
Color and Shape:
Solid
Molecular weight:
1911.14
Ref: TM-TP1851L
| 1mg | 72.00 € | ||
| 5mg | 136.00 € | ||
| 10mg | 211.00 € | ||
| 25mg | 354.00 € | ||
| 50mg | 503.00 € | ||
| 100mg | 687.00 € | ||
| 200mg | 903.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Otenabant
CAS:686344-29-6
Otenabant (CP-945598) has been investigated for the treatment of Obesity.
Formula:
C25H25Cl2N7O
Purity:
100%
Color and Shape:
Solid
Molecular weight:
510.42
Ref: TM-T3530
| 2mg | 48.00 € | ||
| 5mg | 73.00 € | ||
| 10mg | 93.00 € | ||
| 25mg | 171.00 € | ||
| 50mg | 304.00 € | ||
| 100mg | 456.00 € | ||
| 1mL*10mM (DMSO) | 82.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
SB-649868
CAS:380899-24-1
SB-649868 (GSK649868) is a potent and selective orally active antagonist of orexin(pKi =9.4 and 9.5 …
Formula:
C26H24FN3O3S
Purity:
99.53%
Color and Shape:
Solid
Molecular weight:
477.55
Ref: TM-T5498
| 1mg | 37.00 € | ||
| 5mg | 109.00 € | ||
| 10mg | 184.00 € | ||
| 25mg | 390.00 € | ||
| 50mg | 632.00 € | ||
| 100mg | 1,014.00 € | ||
| 200mg | 1,368.00 € | ||
| 1mL*10mM (DMSO) | 135.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Takeda103A
CAS:865609-72-9
Takeda103A (CMPD103A) is the GRK2-dependent bovine tubulin oxidation effective inhibitor.
Formula:
C24H23F2N7O
Purity:
97.17%
Color and Shape:
Solid
Molecular weight:
463.48
Ref: TM-T24850
| 1mg | 82.00 € | ||
| 2mg | 102.00 € | ||
| 5mg | 159.00 € | ||
| 10mg | 249.00 € | ||
| 25mg | 409.00 € | ||
| 50mg | 543.00 € | ||
| 100mg | 759.00 € | ||
| 200mg | 999.00 € | ||
| 1mL*10mM (DMSO) | 180.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
