G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
Read more
MK-0557
CAS:328232-95-7
MK-0557 is a selective and orally available antagonist of the neuropeptide Y5 receptor (Ki: 1.6 …
Formula:
C22H19FN4O3
Purity:
99.88%
Color and Shape:
Solid
Molecular weight:
406.41
Ref: TM-TQ0286
| 1mg | 35.00 € | ||
| 1ml | 78.00 € | ||
| 5mg | 69.00 € | ||
| 10mg | 93.00 € | ||
| 25mg | 169.00 € | ||
| 50mg | 269.00 € | ||
| 100mg | 379.00 € | ||
| 200mg | 527.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Linzagolix
CAS:935283-04-8
Linzagolix is a small-molecule, non-peptide, orally active gonadotropin-releasing hormone antagonist (GnRH antagonist) which is under …
Formula:
C22H15F3N2O7S
Purity:
99.68%
Color and Shape:
Solid
Molecular weight:
508.42
Ref: TM-T27837
| 1mg | 52.00 € | ||
| 1ml | 115.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 157.00 € | ||
| 25mg | 297.00 € | ||
| 50mg | 537.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
PW0787
CAS:2624131-45-7
PW0787 is a potent, selective, orally active, and brain-penetrant GPR52 agonist (EC50=135 nM).
Formula:
C23H20F4N4O2
Purity:
98.42%
Color and Shape:
Solid
Molecular weight:
460.42
Ref: TM-T9452
| 1mg | 36.00 € | ||
| 1ml | 93.00 € | ||
| 5mg | 77.00 € | ||
| 10mg | 112.00 € | ||
| 25mg | 226.00 € | ||
| 50mg | 338.00 € | ||
| 100mg | 480.00 € | ||
| 200mg | 661.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
ACH-000143
CAS:2225836-30-4
ACH-000143 have been identified as a novel agonist of the melatonin receptors MT1 and MT2.
Formula:
C13H16ClN3O3
Purity:
98.15%
Color and Shape:
Solid
Molecular weight:
297.74
Ref: TM-T9193
| 1mg | 51.00 € | ||
| 1ml | 123.00 € | ||
| 5mg | 112.00 € | ||
| 10mg | 174.00 € | ||
| 25mg | 307.00 € | ||
| 50mg | 430.00 € | ||
| 100mg | 590.00 € | ||
| 200mg | 795.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
ML-193
CAS:713121-80-3
ML-193: GPR55 antagonist, IC50 221nM, 27x selective over GPR35/CB1/CB2, may aid Parkinson's symptoms.
Formula:
C28H25N5O4S
Purity:
97.74%
Color and Shape:
Solid
Molecular weight:
527.59
Ref: TM-T22103
| 1ml | 63.00 € | ||
| 5mg | 46.00 € | ||
| 10mg | 72.00 € | ||
| 25mg | 108.00 € | ||
| 50mg | 163.00 € | ||
| 100mg | To inquire |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Neuropeptide Y (29-64), amide, human acetate
Neuropeptide Y (29-64), amide, human acetate is involved in Alzheimer's disease (AD) and protects rat …
Purity:
98.42%
Molecular weight:
N/A
Ref: TM-TP1140L
| 1mg | 95.00 € | ||
| 5mg | 228.00 € | ||
| 10mg | 337.00 € | ||
| 25mg | 538.00 € | ||
| 50mg | 726.00 € | ||
| 100mg | 971.00 € | ||
| 200mg | 1,310.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
NAN-190 hydrobromide
CAS:115338-32-4
NAN-190 hydrobromide is an antagonist of serotonin receptor 5-HT.
Formula:
C23H28BrN3O3
Purity:
95.92%
Color and Shape:
Solid
Molecular weight:
474.39
Ref: TM-T12172
| 1ml | 34.00 € | ||
| 10mg | 34.00 € | ||
| 25mg | 42.00 € | ||
| 50mg | 51.00 € | ||
| 100mg | 66.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
ONO-7300243
CAS:638132-34-0
ONO-7300243 is an antagonist of lysophosphatidic acid receptor 1 (LPA1; IC50 : 0.16 μM).
Formula:
C28H31NO5
Purity:
99.66%
Color and Shape:
Solid
Molecular weight:
461.55
Ref: TM-T7393
| 1mg | 45.00 € | ||
| 1ml | 88.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 130.00 € | ||
| 25mg | 253.00 € | ||
| 50mg | 407.00 € | ||
| 100mg | 640.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Pancreatic Polypeptide (human) acetate
Pancreatic Polypeptide (human) acetate is a C-terminally amidated 36 amino acid peptide, which acts as …
Purity:
97.26%
Molecular weight:
N/A
Ref: TM-TP1137L
| 1mg | 185.00 € | ||
| 5mg | 460.00 € | ||
| 10mg | 651.00 € | ||
| 25mg | 922.00 € | ||
| 50mg | 1,299.00 € | ||
| 100mg | 1,747.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
HAEGTFT acetate(926018-95-3 free base)
HAEGTFT acetate is the first N-terminal 1-7 residues of GLP-1 peptide.
Formula:
C35H51N9O14
Purity:
100%
Color and Shape:
Solid
Molecular weight:
821.84
Ref: TM-TP1419L
| 1mg | 98.00 € | ||
| 5mg | 299.00 € | ||
| 10mg | 431.00 € | ||
| 25mg | 649.00 € | ||
| 50mg | 891.00 € | ||
| 100mg | 1,200.00 € | ||
| 200mg | 1,621.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Dapiprazole Hydrochloride
CAS:72822-13-0
Dapiprazole Hydrochloride (Glamidolo Hydrochloride) is an alpha-1-adrenergic antagonist that acts by blocking alpha-adrenergic receptors.
Formula:
C19H28ClN5
Purity:
100% - 99.86%
Color and Shape:
Solid
Molecular weight:
361.92
Ref: TM-T3996
| 1ml | 34.00 € | ||
| 25mg | 56.00 € | ||
| 50mg | 87.00 € | ||
| 100mg | 112.00 € | ||
| 200mg | 169.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
ELA-14(human) acetate
ELA-14(human) acetate, a fragment of ELA, targets APJ, activates Gαi1 and β-arrestin-2, and prompts receptor …
Formula:
C77H123N25O19S2
Purity:
97.20%
Color and Shape:
Solid
Molecular weight:
1767.09
Ref: TM-TP1923L1
| 1mg | 61.00 € | ||
| 5mg | 196.00 € | ||
| 10mg | 294.00 € | ||
| 25mg | 475.00 € | ||
| 50mg | 653.00 € | ||
| 100mg | 869.00 € | ||
| 200mg | 1,163.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
AnaMorelin hydrochloride
CAS:861998-00-7
AnaMorelin hydrochloride (RC-1291 hydrochloride) is a novel ghrelin receptor agonist(EC50 : 0.74 nM, in the …
Formula:
C31H43ClN6O3
Purity:
99.18% - ≥98%
Color and Shape:
Solid
Molecular weight:
583.16
Ref: TM-T7225
| 1mg | 35.00 € | ||
| 1ml | 95.00 € | ||
| 2mg | 51.00 € | ||
| 5mg | 72.00 € | ||
| 10mg | 94.00 € | ||
| 25mg | 143.00 € | ||
| 50mg | 175.00 € | ||
| 100mg | 231.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Medetomidine hydrochloride
CAS:86347-15-1
Medetomidine hydrochloride (MPV785) is a selective α2-adrenoceptor agonist, with Ki of 1.08 nM, exhibts 1620-fold …
Formula:
C13H16N2·HCl
Purity:
96.72%
Color and Shape:
White Or Off White Crystalline Powder
Molecular weight:
236.74
Ref: TM-T6579
| 1ml | 55.00 € | ||
| 10mg | 52.00 € | ||
| 25mg | 88.00 € | ||
| 50mg | 144.00 € | ||
| 100mg | 183.00 € | ||
| 200mg | 236.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
SB225002
CAS:182498-32-4
SB225002 is a potent and selective CXCR2 antagonist inhibiting interleukin IL-8 binding to CXCR2.
Formula:
C13H10BrN3O4
Purity:
96.86% - 98.79%
Color and Shape:
Solid
Molecular weight:
352.14
Ref: TM-T1955
| 1ml | 53.00 € | ||
| 5mg | 50.00 € | ||
| 10mg | 66.00 € | ||
| 25mg | 124.00 € | ||
| 50mg | 220.00 € | ||
| 100mg | 395.00 € | ||
| 200mg | 603.00 € | ||
| 500mg | 922.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Melanotan (MT)-II
CAS:121062-08-6
Melanotan (MT)-II, a synthetic melanocortin receptor agonist, is a synthetic analogue of the peptide hormone …
Formula:
C50H69N15O9
Purity:
100%
Color and Shape:
Solid
Molecular weight:
1024.18
Ref: TM-TP1324
| 2mg | 49.00 € | ||
| 5mg | 73.00 € | ||
| 10mg | 97.00 € | ||
| 25mg | 169.00 € | ||
| 50mg | 259.00 € | ||
| 100mg | 434.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Thrombin Receptor Activator for Peptide
Thrombin Receptor Activator (TRAP) or Coagulation Factor II (1-5), used in CHD research.
Formula:
C32H51F3N8O9
Purity:
99.88%
Color and Shape:
Solid
Molecular weight:
748.79
Ref: TM-T7674
| 1mg | 45.00 € | ||
| 5mg | 88.00 € | ||
| 10mg | 141.00 € | ||
| 25mg | 249.00 € | ||
| 50mg | 359.00 € | ||
| 100mg | 516.00 € | ||
| 200mg | 703.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
SDZ WAG 994
CAS:130714-47-5
SDZ WAG 994 is an A1 adenosine receptor agonist.
Formula:
C17H25N5O4
Purity:
99.90%
Color and Shape:
Solid
Molecular weight:
363.41
Ref: TM-T23347
| 1mg | 98.00 € | ||
| 1ml | 203.00 € | ||
| 5mg | 191.00 € | ||
| 10mg | 286.00 € | ||
| 25mg | 516.00 € | ||
| 50mg | 741.00 € | ||
| 100mg | 1,013.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Hypidone hydrochloride
CAS:1339058-04-6
Hypidone hydrochloride (YL0919) is a novel antidepressant candidate with dual activity as a 5-HT1A receptor …
Formula:
C18H23ClN2O2
Purity:
99.82% - 99.93%
Color and Shape:
Solid
Molecular weight:
334.84
Ref: TM-T3648
| 1ml | 81.00 € | ||
| 2mg | 46.00 € | ||
| 5mg | 69.00 € | ||
| 10mg | 87.00 € | ||
| 25mg | 118.00 € | ||
| 50mg | 185.00 € | ||
| 100mg | 343.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Vortioxetine
CAS:508233-74-7
Vortioxetine (Lu AA 21004) is a serotonergic antidepressant used for major depression disorders.
Formula:
C18H22N2S
Purity:
99.34% - 99.82%
Color and Shape:
Solid
Molecular weight:
298.45
Ref: TM-T2395
| 1g | 493.00 € | ||
| 1ml | 48.00 € | ||
| 10mg | 50.00 € | ||
| 25mg | 68.00 € | ||
| 50mg | 94.00 € | ||
| 100mg | 121.00 € | ||
| 200mg | 211.00 € | ||
| 500mg | 345.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
