G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Carbetocin
CAS:37025-55-1
Carbetocin is an obstetric drug used to control postpartum hemorrhage and bleeding after giving birth.
Formula:
C45H69N11O12S
Purity:
99.96%
Color and Shape:
Solid
Molecular weight:
988.16
Ref: TM-T7601
| 10mg | 513.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
![[Lys8, Lys9]-Neurotensin (8-13) acetate](https://static.cymitquimica.com/products/TM/thumb/T38807L.jpg)
[Lys8, Lys9]-Neurotensin (8-13) acetate
[Lys8, Lys9]-Neurotensin (8-13) acetate, a Neurotensin analog, exerts its analgesic effects through activation of the …
Formula:
C40H68N8O10
Purity:
98%
Color and Shape:
Solid
Molecular weight:
821.02
Ref: TM-T38807L
| 1mg | 143.00 € | ||
| 5mg | 312.00 € | ||
| 10mg | 464.00 € | ||
| 25mg | 739.00 € | ||
| 50mg | 1,049.00 € | ||
| 100mg | 1,420.00 € | ||
| 1ml*10 (DMSO) | 491.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Betahistine dihydrochloride
CAS:5579-84-0
Betahistine dihydrochloride (Betahistine 2HCl) is a histamine analog and H1 receptor agonist that serves as …
Formula:
C8H14Cl2N2
Purity:
99.34% - 99.88%
Color and Shape:
White To Light Yellow Crystalline Powder
Molecular weight:
209.12
Ref: TM-T0246
| 1g | 34.00 € | ||
| 1ml | 34.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Ritanserin
CAS:87051-43-2
Ritanserin (R 55667) is a highly effective, relatively selective, long-acting antagonist of 5-HT2 receptor (IC50: …
Formula:
C27H25F2N3OS
Purity:
99.45% - 99.89%
Color and Shape:
Solid
Molecular weight:
477.57
Ref: TM-T16759
| 1mg | 40.00 € | ||
| 1ml | 96.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 83.00 € | ||
| 10mg | 113.00 € | ||
| 25mg | 182.00 € | ||
| 50mg | 268.00 € | ||
| 100mg | 403.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Zafirlukast
CAS:107753-78-6
Zafirlukast (ICI 204219) is an orally available leukotriene receptor antagonist which is widely used for …
Formula:
C31H33N3O6S
Purity:
99% - 99.31%
Color and Shape:
Solid
Molecular weight:
575.68
Ref: TM-T6736
| 1ml | 65.00 € | ||
| 25mg | 48.00 € | ||
| 50mg | 63.00 € | ||
| 100mg | 91.00 € | ||
| 200mg | 145.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
KH7
CAS:330676-02-3
KH7 is a soluble inhibitor of adenylyl cyclase (sAC)-specific.
Formula:
C17H15BrN4O2S
Purity:
98.43%
Color and Shape:
Solid
Molecular weight:
419.3
Ref: TM-T15658
| 1mg | 43.00 € | ||
| 1ml | 89.00 € | ||
| 2mg | 54.00 € | ||
| 5mg | 89.00 € | ||
| 10mg | 128.00 € | ||
| 25mg | 246.00 € | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 15 Oct 2024
JNJ-7777120
CAS:459168-41-3
JNJ-7777120 is the first potent and selective non-imidazole histamine H4 receptor antagonist, exhibits >1000-fold selectivity …
Formula:
C14H16ClN3O
Purity:
99.71% - 99.93%
Color and Shape:
Solid
Molecular weight:
277.75
Ref: TM-T2232
| 1ml | 73.00 € | ||
| 5mg | 69.00 € | ||
| 10mg | 94.00 € | ||
| 25mg | 167.00 € | ||
| 50mg | 268.00 € | ||
| 100mg | 430.00 € | ||
| 500mg | 920.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
PRX-08066
CAS:866206-54-4
PRX-08066 is a selective 5-hydroxytryptamine receptor 2B (5-HT2BR, IC50= 3.4 nM) antagonist that induces selective …
Formula:
C19H17ClFN5S
Purity:
98.04% - 98.07%
Color and Shape:
Solid
Molecular weight:
401.89
Ref: TM-T16669
| 1mg | 59.00 € | ||
| 1ml | 140.00 € | ||
| 5mg | 118.00 € | ||
| 10mg | 171.00 € | ||
| 25mg | 343.00 € | ||
| 50mg | 510.00 € | ||
| 100mg | 732.00 € | ||
| 500mg | 1,514.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Zuclopenthixol
CAS:53772-83-1
Zuclopenthixol (cis-Clopenthixol) is a thioxanthene with therapeutic actions similar to the phenothiazine antipsychotics.
Formula:
C22H25ClN2OS
Purity:
98.90% - 99.82%
Color and Shape:
Solid
Molecular weight:
400.96
Ref: TM-T4117
| 1ml | 51.00 € | ||
| 25mg | 36.00 € | ||
| 50mg | 46.00 € | ||
| 100mg | 59.00 € | ||
| 200mg | 86.00 € | ||
| 500mg | 128.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
CLOZAPINE N-OXIDE
CAS:34233-69-7
View and buy CLOZAPINE N-OXIDE from TargetMol.Clozapine N-oxide is a major metabolite of clozapine also …
Formula:
C18H19ClN4O
Purity:
98.43% - 99.94%
Color and Shape:
Solid
Molecular weight:
342.82
Ref: TM-T4494
| 2mg | 40.00 € | ||
| 5mg | 54.00 € | ||
| 10mg | 87.00 € | ||
| 25mg | 126.00 € | ||
| 50mg | 179.00 € | ||
| 100mg | 264.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
R 396 acetate
R 396 acetate is an NK-2 Tachykinin Receptor Antagonist.
Formula:
C41H55N9O12
Purity:
99.52%
Color and Shape:
Solid
Molecular weight:
865.93
Ref: TM-T24697L
| 1mg | 111.00 € | ||
| 2mg | 157.00 € | ||
| 5mg | 240.00 € | ||
| 10mg | 356.00 € | ||
| 25mg | 543.00 € | ||
| 50mg | 759.00 € | ||
| 100mg | 1,017.00 € | ||
| 200mg | 1,356.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Dolasetron Mesylate hydrate
CAS:878143-33-0
Dolasetron Mesylate hydrate blocks 5HT3 to prevent chemo and radiotherapy nausea.
Formula:
C20H26N2O7S
Purity:
99.86% - 99.9%
Color and Shape:
Solid
Molecular weight:
438.49
Ref: TM-T2589
| 1ml | 51.00 € | ||
| 5mg | 34.00 € | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Aticaprant
CAS:1174130-61-0
Aticaprant (LY-2456302) (CERC-501) is a potent and centrally-penetrant antagonist of the kappa-opioid receptor (Ki: 0.807 …
Formula:
C26H27FN2O2
Purity:
99.53% - 99.93%
Color and Shape:
Solid
Molecular weight:
418.5
Ref: TM-TQ0082
| 1mg | 40.00 € | ||
| 1ml | 87.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 124.00 € | ||
| 25mg | 254.00 € | ||
| 50mg | 398.00 € | ||
| 100mg | 593.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
SB-203186 hydrochloride
CAS:207572-69-8
SB 203186 hydrochloride is a potent 5-HT4 receptor antagonist
Formula:
C16H20N2O2·HCl
Purity:
99.64%
Color and Shape:
Solid
Molecular weight:
308.81
Ref: TM-T23310
| 5mg | 39.00 € | ||
| 10mg | 63.00 € | ||
| 25mg | 114.00 € | ||
| 50mg | 183.00 € | ||
| 100mg | 274.00 € | ||
| 500mg | 603.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Ivabradine hydrochloride
CAS:148849-67-6
Ivabradine HCl (S 16257-2) is an If inhibitor (IC50: 2.9 μM) and SA node HCN …
Formula:
C27H37ClN2O5
Purity:
98.6% - 99.73%
Color and Shape:
Solid
Molecular weight:
505.05
Ref: TM-T2535
| 1ml | 47.00 € | ||
| 10mg | 39.00 € | ||
| 25mg | 54.00 € | ||
| 50mg | 73.00 € | ||
| 100mg | 95.00 € | ||
| 200mg | 143.00 € | ||
| 500mg | 246.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
LY255283
CAS:117690-79-6
LY255283 is a specific antagonit of leukotriene B4 (LTB4) receptor. It inhibits the production of …
Formula:
C19H28N4O3
Purity:
99.18%
Color and Shape:
Solid
Molecular weight:
360.45
Ref: TM-T22946
| 1mg | 41.00 € | ||
| 1ml | 96.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 124.00 € | ||
| 25mg | 244.00 € | ||
| 50mg | 393.00 € | ||
| 100mg | 630.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
PACAP (1-27), human, ovine, rat acetate
PACAP (1-27), human, ovine, rat acetate (PACAP 1-27 acetate) is a novel neuropeptides originally isolated …
Formula:
C144H228N40O41S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
3207.71
Ref: TM-TP1070L
| 1mg | 148.00 € | ||
| 5mg | 418.00 € | ||
| 10mg | 618.00 € | ||
| 25mg | 917.00 € | ||
| 50mg | 1,299.00 € | ||
| 100mg | 1,746.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
AVN-492
CAS:1220646-23-0
AVN-49 is a potent and selective 5-HT6R Antagonist (Ki: 91 pM).
Formula:
C17H21N5O2S
Purity:
99.29%
Color and Shape:
Solid
Molecular weight:
359.45
Ref: TM-T5179
| 1mg | 39.00 € | ||
| 1ml | 90.00 € | ||
| 2mg | 49.00 € | ||
| 5mg | 80.00 € | ||
| 10mg | 119.00 € | ||
| 25mg | 232.00 € | ||
| 50mg | 347.00 € | ||
| 100mg | 501.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
FAUC-365
CAS:474432-66-1
FAUC-365 is a D3 dopamine receptor agonist.
Formula:
C23H25Cl2N3OS
Purity:
98.09%
Color and Shape:
Solid
Molecular weight:
462.44
Ref: TM-T21667
| 1mg | 34.00 € | ||
| 1ml | 80.00 € | ||
| 2mg | 45.00 € | ||
| 5mg | 72.00 € | ||
| 10mg | 93.00 € | ||
| 25mg | 182.00 € | ||
| 50mg | 296.00 € | ||
| 100mg | 428.00 € | ||
| 200mg | 600.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
OXA (17-33) acetate
OXA (17-33) acetate is a more potent agonist of orexin-1 receptor (OX1, EC50 = 8.29 …
Formula:
C79H125N23O22
Purity:
98.52%
Color and Shape:
Solid
Molecular weight:
1748.98
Ref: TM-TP1973L
| 1mg | 269.00 € | ||
| 5mg | 598.00 € | ||
| 10mg | 813.00 € | ||
| 25mg | 1,217.00 € | ||
| 50mg | 1,601.00 € | ||
| 100mg | 2,177.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
