G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Rimegepant
CAS:1289023-67-1
View and buy Rimegepant from TargetMol.BMS-927711 is a highly potent, oral calcitonin gene-related peptide (CGRP) …
Formula:
C28H28F2N6O3
Purity:
99.1% - 99.84%
Color and Shape:
Solid
Molecular weight:
534.56
Ref: TM-T4610
| 1mg | 54.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 157.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
ML-031
CAS:852230-33-2
ML-031 activated S1P2 with an EC50 value of 1 μM in an S1P reporter assay.
Formula:
C19H20N2O3
Purity:
99.21%
Color and Shape:
Solid
Molecular weight:
324.37
Ref: TM-T22101
| 1mg | 62.00 € | ||
| 2mg | 91.00 € | ||
| 5mg | 111.00 € | ||
| 10mg | 184.00 € | ||
| 25mg | 356.00 € | ||
| 50mg | 465.00 € | ||
| 100mg | 677.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
Dynorphin A 1-10 acetate(79994-24-4 free base)
Dynorphin A (1-10) acetate is an endogenous opioid neuropeptide, binds to extracellular loop 2 of …
Formula:
C59H95N19O14
Purity:
99.88%
Color and Shape:
Solid
Molecular weight:
1294.53
Ref: TM-TP1813L
| 1mg | 97.00 € | ||
| 5mg | 316.00 € | ||
| 10mg | 478.00 € | ||
| 25mg | 777.00 € | ||
| 50mg | 1,077.00 € | ||
| 100mg | 1,448.00 € | ||
| 500mg | 2,897.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
JNJ-31020028
CAS:1094873-14-9
JNJ-31020028 is a selective brain penetrant antagonist of neuropeptide Y2 receptor with high affinity (pIC50=8.07, …
Formula:
C34H36FN5O2
Purity:
95.92% - 96.24%
Color and Shape:
Solid
Molecular weight:
565.68
Ref: TM-T1997
| 5mg | 50.00 € | ||
| 10mg | 75.00 € | ||
| 25mg | 125.00 € | ||
| 50mg | 206.00 € | ||
| 100mg | 308.00 € | ||
| 200mg | 442.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
Senktide
CAS:106128-89-6
Senktide is an agonist of tachykinin NK3 receptor.
Formula:
C40H55N7O11S
Purity:
100%
Color and Shape:
White Powder
Molecular weight:
841.97
Ref: TM-T7633
| 1mg | 62.00 € | ||
| 5mg | 128.00 € | ||
| 10mg | 183.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
Sarpogrelate hydrochloride
CAS:135159-51-2
Sarpogrelate hydrochloride (MCI-9042), a 5-HT2 antagonist with high affinity (Ki=8.39nM), is used as an anti-platelet …
Formula:
C24H32ClNO6
Purity:
99.42%
Color and Shape:
Colorless Liquid
Molecular weight:
465.97
Ref: TM-T4978
| 5mg | 48.00 € | ||
| 10mg | 72.00 € | ||
| 25mg | 118.00 € | ||
| 50mg | 182.00 € | ||
| 100mg | 270.00 € | ||
| 500mg | 639.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
Lurasidone hydrochloride
CAS:367514-88-3
Lurasidone HCl: Atypical antipsychotic, treats schizophrenia & bipolar, affects dopamine, serotonin & adrenergic receptors.
Formula:
C28H36N4O2S·HCl
Purity:
100%
Color and Shape:
Solid
Molecular weight:
529.14
Ref: TM-T1735
| 5mg | 41.00 € | ||
| 10mg | 62.00 € | ||
| 25mg | 79.00 € | ||
| 50mg | 94.00 € | ||
| 100mg | 142.00 € | ||
| 200mg | 221.00 € | ||
| 500mg | 462.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
Tetrahydrozoline hydrochloride
CAS:522-48-5
Tetrahydrozoline hydrochloride (Murine Plus) is an imidazoline derivative with alpha receptor agonist activity.
Formula:
C13H16N2·HCl
Purity:
99.97%
Color and Shape:
Off-White Solid
Molecular weight:
236.74
Ref: TM-T6703
| 1g | 39.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
Eledoisin Related Peptide 2TFA
Eledoisin Related Peptide 2TFA (Eledoisin Related Peptide 2TFA (2990-43-4(free base))) is a tachykinin receptor ligand.
Formula:
C38H60F6N8O10S
Purity:
99%
Color and Shape:
Solid
Molecular weight:
934.99
Ref: TM-T7631L
| 1mg | 81.00 € | ||
| 5mg | 272.00 € | ||
| 10mg | 427.00 € | ||
| 25mg | 682.00 € | ||
| 50mg | 925.00 € | ||
| 100mg | 1,243.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
PRX-07034 hydrochloride
CAS:903580-39-2
PRX-07034 hydrochloride is a selective antagonist of 5-HT6 receptor. It has cognition and memory-enhancing properties …
Formula:
C21H29Cl2N3O4S
Purity:
98.50%
Color and Shape:
Solid
Molecular weight:
490.44
Ref: TM-T8720
| 1mg | 35.00 € | ||
| 2mg | 47.00 € | ||
| 5mg | 70.00 € | ||
| 10mg | 102.00 € | ||
| 25mg | 186.00 € | ||
| 50mg | 308.00 € | ||
| 100mg | 498.00 € | ||
| 1mL*10mM (DMSO) | 74.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
Cinitapride
CAS:66564-14-5
Cinitapride (Blaston) treats acid reflux and gastric issues, targeting 5-HT2, 5-HT1, and 5-HT4 receptors.
Formula:
C21H30N4O4
Purity:
98.99%
Color and Shape:
Solid
Molecular weight:
402.49
Ref: TM-T21385
| 1mg | 77.00 € | ||
| 5mg | 162.00 € | ||
| 10mg | 250.00 € | ||
| 25mg | 499.00 € | ||
| 50mg | 722.00 € | ||
| 100mg | 1,013.00 € | ||
| 1mL*10mM (DMSO) | 185.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
Bombesin acetate(31362-50-2 free base)
CAS:1222319-87-0
Bombesin acetate is a 14-amino acid peptide originally isolated from the skin of the European …
Formula:
C73H114N24O20S
Purity:
98.44%
Color and Shape:
Solid
Molecular weight:
1679.92
Ref: TM-TP1281L1
| 1mg | 94.00 € | ||
| 5mg | 165.00 € | ||
| 10mg | 286.00 € | ||
| 25mg | 482.00 € | ||
| 50mg | 699.00 € | ||
| 100mg | 991.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
Motilin (26-47), human, porcine
CAS:52906-92-0
Motilin (26-47) binds Motilin receptors in hamster cells; Ki=2.3 nM, EC50=0.3 nM; same for humans, …
Formula:
C120H188N34O35S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
2699.07
Ref: TM-TP1425
| 1mg | 114.00 € | ||
| 5mg | 343.00 € | ||
| 10mg | 516.00 € | ||
| 25mg | 764.00 € | ||
| 50mg | 1,024.00 € | ||
| 100mg | 1,374.00 € | ||
| 200mg | 1,817.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
CB1-IN-1
CAS:1429239-98-4
CB1-IN-1 (DBPR211) is a peripherally restricted CB1R antagonist, for CB1R and CB2R with Ki of …
Formula:
C33H31Cl2F3N6O3S2
Purity:
99.08% - 99.55%
Color and Shape:
Solid
Molecular weight:
751.67
Ref: TM-T5996
| 1mg | 85.00 € | ||
| 2mg | 114.00 € | ||
| 5mg | 186.00 € | ||
| 10mg | 267.00 € | ||
| 25mg | 437.00 € | ||
| 50mg | 609.00 € | ||
| 100mg | 821.00 € | ||
| 500mg | 1,647.00 € | ||
| 1mL*10mM (DMSO) | 225.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
DPCPX
CAS:102146-07-6
DPCPX (PD 116948) is an A1 adenosine receptor antagonist
Formula:
C16H24N4O2
Purity:
99.93%
Color and Shape:
White Solid
Molecular weight:
304.39
Ref: TM-T22744
| 10mg | 48.00 € | ||
| 25mg | 70.00 € | ||
| 50mg | 95.00 € | ||
| 100mg | 139.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
A-836339
CAS:959746-77-1
A-836339: Potent cannabinoid, CB2-focused (Ki=0.64nM), lesser CB1 affinity (Ki=270nM); analgesic, anti-inflammatory in mice.
Formula:
C16H26N2O2S
Purity:
99.94%
Color and Shape:
Solid
Molecular weight:
310.45
Ref: TM-T7375
| 2mg | 47.00 € | ||
| 5mg | 89.00 € | ||
| 10mg | 159.00 € | ||
| 25mg | 258.00 € | ||
| 50mg | 379.00 € | ||
| 100mg | 538.00 € | ||
| 200mg | 727.00 € | ||
| 1mL*10mM (DMSO) | 91.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
ACTH (1-17) acetate
ACTH (1-17) acetate is a potent agonist at the human melanocortin 1 (MC1) receptor with …
Formula:
C97H149N29O25S
Purity:
98.53%
Color and Shape:
Liquid
Molecular weight:
2153.47
Ref: TM-TP1011L
| 1mg | 118.00 € | ||
| 5mg | 382.00 € | ||
| 10mg | 548.00 € | ||
| 25mg | 988.00 € | ||
| 50mg | 1,471.00 € | ||
| 100mg | 2,206.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
Ginsenoside Rb2
CAS:11021-13-9
Ginsenoside Rb2 (Ginsenoside C) found in species of Panax, upregulating GPR120 gene expression.
Formula:
C53H90O22
Purity:
99.01% - 99.66%
Color and Shape:
White Powder
Molecular weight:
1079.27
Ref: TM-T3919
| 20mg | 87.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
RBC8
CAS:361185-42-4
RBC8 is a specific GTPases RalA/RalB inhibitor by inhibiting the binding of Ral to its …
Formula:
C25H20N4O3
Purity:
99.81% - 99.86%
Color and Shape:
Solid
Molecular weight:
424.45
Ref: TM-T6634
| 1mg | 49.00 € | ||
| 2mg | 68.00 € | ||
| 5mg | 108.00 € | ||
| 10mg | 185.00 € | ||
| 25mg | 313.00 € | ||
| 50mg | 467.00 € | ||
| 100mg | 678.00 € | ||
| 1mL*10mM (DMSO) | 115.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
AH-7614
CAS:6326-06-3
AH-7614 (AH 7614) is a selective and potent free fatty acid receptor 4 (FFA4/GPR120) antagonist.
Formula:
C20H17NO3S
Purity:
98.05%
Color and Shape:
Solid
Molecular weight:
351.42
Ref: TM-T22027
| 5mg | 52.00 € | ||
| 10mg | 91.00 € | ||
| 25mg | 174.00 € | ||
| 50mg | 312.00 € | ||
| 100mg | 423.00 € | ||
| 200mg | 551.00 € | ||
| 500mg | 700.00 € | ||
| 1mL*10mM (DMSO) | 64.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
