G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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ICI 89406
CAS:53671-71-9
ICI 89406 (1-[2-[[3-(2-cyanophenoxy)-2-hydroxypropyl]amino]ethyl]-3-phenylurea) is a β-adrenergic antagonist.
Formula:
C19H22N4O3
Purity:
99.62%
Color and Shape:
Solid
Molecular weight:
354.4
Ref: TM-T22852
| 1mg | 79.00 € | ||
| 1ml | 153.00 € | ||
| 5mg | 143.00 € | ||
| 10mg | 198.00 € | ||
| 25mg | 452.00 € | ||
| 50mg | 649.00 € | ||
| 100mg | 920.00 € | ||
| 500mg | 1,840.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Adenosine amine congener
CAS:96760-69-9
Adenosine amine congener (ADAC) (ADAC) is an agonist of selective A1 adenosine receptor,.
Formula:
C28H32N8O6
Purity:
97.86%
Color and Shape:
Solid
Molecular weight:
576.6
Ref: TM-T7683
| 1mg | 73.00 € | ||
| 1ml | 245.00 € | ||
| 5mg | 158.00 € | ||
| 10mg | 230.00 € | ||
| 25mg | 416.00 € | ||
| 50mg | 612.00 € | ||
| 100mg | 873.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
USL311
CAS:1373268-67-7
USL311 blocks CXCR4/SDF-1 interaction, inhibits tumor cell growth and migration.
Formula:
C24H34N6O
Purity:
99.56% - 99.73%
Color and Shape:
Solid
Molecular weight:
422.57
Ref: TM-T17208
| 1mg | 90.00 € | ||
| 2mg | 114.00 € | ||
| 5mg | 185.00 € | ||
| 10mg | 268.00 € | ||
| 25mg | 451.00 € | ||
| 50mg | 647.00 € | ||
| 100mg | 922.00 € | ||
| 500mg | 1,846.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Treprostinil
CAS:81846-19-7
Treprostinil (Orenitram) is a potent DP1, IP and EP2 agonist (EC50: 0.6/1.9/6.2 nM).
Formula:
C23H34O5
Purity:
99.71%
Color and Shape:
Solid
Molecular weight:
390.51
Ref: TM-T5150
| 1ml | 67.00 € | ||
| 2mg | 46.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 118.00 € | ||
| 25mg | 268.00 € | ||
| 50mg | 448.00 € | ||
| 100mg | 640.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
BA 1 acetate(183241-31-8 free base)
BA 1 acetate: bombesin agonist, IC50s: 0.26/1.55/2.52 nM (BB1/BB2/BB3), boosts glucose transport, promotes lung cancer …
Formula:
C59H80N14O13
Purity:
95.3%
Color and Shape:
Solid
Molecular weight:
1193.35
Ref: TM-TP1913L1
| 1mg | 94.00 € | ||
| 5mg | 182.00 € | ||
| 10mg | 274.00 € | ||
| 25mg | 495.00 € | ||
| 50mg | 716.00 € | ||
| 100mg | 994.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Binodenoson
CAS:144348-08-3
Binodenoson (WRC 0470), a selective A2A adenosine receptor agonist, aids in coronary imaging.
Formula:
C17H25N7O4
Purity:
99.84%
Color and Shape:
Solid
Molecular weight:
391.42
Ref: TM-T9516
| 1mg | 134.00 € | ||
| 1ml | 309.00 € | ||
| 5mg | 277.00 € | ||
| 10mg | 415.00 € | ||
| 25mg | 689.00 € | ||
| 50mg | 917.00 € | ||
| 100mg | 1,291.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
ML401
CAS:1597489-14-9
ML401 is a selectively EBI2(GPR183) receptor antagonist(IC50 of 1.03 nM) .
Formula:
C20H20BrClN2O
Purity:
99.13%
Color and Shape:
Solid
Molecular weight:
419.74
Ref: TM-T8234
| 1mg | 130.00 € | ||
| 1ml | 205.00 € | ||
| 2mg | 155.00 € | ||
| 5mg | 186.00 € | ||
| 10mg | 304.00 € | ||
| 25mg | 484.00 € | ||
| 50mg | 650.00 € | ||
| 100mg | 841.00 € | ||
| 500mg | 1,715.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Rimegepant
CAS:1289023-67-1
View and buy Rimegepant from TargetMol.BMS-927711 is a highly potent, oral calcitonin gene-related peptide (CGRP) …
Formula:
C28H28F2N6O3
Purity:
99.1% - 99.33%
Color and Shape:
Solid
Molecular weight:
534.56
Ref: TM-T4610
| 1mg | 54.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 157.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Siramesine
CAS:147817-50-3
Siramesine (Lu 28-179)(Lu 28-179) is a selective sigma-2 receptor agonist, which has been shown to …
Formula:
C30H31FN2O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
454.58
Ref: TM-T4620
| 5mg | 193.00 € | ||
| 10mg | 293.00 € | ||
| 25mg | 447.00 € | ||
| 50mg | 688.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
ML-031
CAS:852230-33-2
ML-031 activated S1P2 with an EC50 value of 1 μM in an S1P reporter assay.
Formula:
C19H20N2O3
Purity:
99.21%
Color and Shape:
Solid
Molecular weight:
324.37
Ref: TM-T22101
| 1mg | 62.00 € | ||
| 2mg | 91.00 € | ||
| 5mg | 111.00 € | ||
| 10mg | 184.00 € | ||
| 25mg | 356.00 € | ||
| 50mg | 465.00 € | ||
| 100mg | 677.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Dynorphin A acetate(80448-90-4 free base)
Dynorphin A acetate is an Endogenous kappa receptor agonist.
Formula:
C101H159N31O25
Purity:
99.69%
Color and Shape:
Solid
Molecular weight:
2207.58
Ref: TM-TP2040L
| 1mg | 70.00 € | ||
| 5mg | 234.00 € | ||
| 10mg | 321.00 € | ||
| 25mg | 541.00 € | ||
| 50mg | 774.00 € | ||
| 100mg | 1,067.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Nelotanserin
CAS:839713-36-9
Nelotanserin (APD125): strong 5-HT2A inverse agonist (IC50: 1.7 nM), moderate 5-HT2C (79 nM), weak 5-HT2B …
Formula:
C18H15BrF2N4O2
Purity:
98.01% - 98.42%
Color and Shape:
Solid
Molecular weight:
437.24
Ref: TM-T7350
| 1mg | 40.00 € | ||
| 1ml | 84.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 86.00 € | ||
| 10mg | 118.00 € | ||
| 25mg | 185.00 € | ||
| 50mg | 343.00 € | ||
| 100mg | 510.00 € | ||
| 500mg | 1,109.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Dynorphin A 1-10 acetate(79994-24-4 free base)
Dynorphin A (1-10) acetate is an endogenous opioid neuropeptide, binds to extracellular loop 2 of …
Formula:
C59H95N19O14
Purity:
99.88%
Color and Shape:
Solid
Molecular weight:
1294.53
Ref: TM-TP1813L
| 1mg | 97.00 € | ||
| 5mg | 316.00 € | ||
| 10mg | 478.00 € | ||
| 25mg | 777.00 € | ||
| 50mg | 1,077.00 € | ||
| 100mg | 1,448.00 € | ||
| 500mg | 2,897.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
JNJ-31020028
CAS:1094873-14-9
JNJ-31020028 is a selective brain penetrant antagonist of neuropeptide Y2 receptor with high affinity (pIC50=8.07, …
Formula:
C34H36FN5O2
Purity:
95.92% - 96.24%
Color and Shape:
Solid
Molecular weight:
565.68
Ref: TM-T1997
| 1mg | 36.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 113.00 € | ||
| 25mg | 202.00 € | ||
| 50mg | 346.00 € | ||
| 100mg | 516.00 € | ||
| 500mg | 1,137.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
BETP
CAS:1371569-69-5
BETP is an agonist of GLP-1 receptor (EC50s: 0.66 and 0.755 μM for human and …
Formula:
C20H17F3N2O2S
Purity:
97.92%
Color and Shape:
Solid
Molecular weight:
406.42
Ref: TM-TQ0124
| 1mg | 47.00 € | ||
| 1ml | 96.00 € | ||
| 5mg | 91.00 € | ||
| 10mg | 137.00 € | ||
| 25mg | 258.00 € | ||
| 50mg | 414.00 € | ||
| 100mg | 661.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Phenylbiguanide
CAS:102-02-3
Phenylbiguanide (N-Phenylbiguanide) is a 5-HT3 receptor selective agonist(EC50 : 3.0±0.1 μM)
Formula:
C8H11N5
Purity:
99.87%
Color and Shape:
Solid
Molecular weight:
177.21
Ref: TM-T7135
| 1g | 82.00 € | ||
| 1ml | 34.00 € | ||
| 200mg | 38.00 € | ||
| 500mg | 56.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Sotagliflozin
CAS:1018899-04-1
Sotagliflozin (LP-802034) is an orally bioavailable inhibitor of the sodium-glucose co-transporter subtype 1 (SGLT1) and …
Formula:
C21H25ClO5S
Purity:
98% - 99.37%
Color and Shape:
Solid
Molecular weight:
424.94
Ref: TM-T3547
| 1mg | 45.00 € | ||
| 1ml | 88.00 € | ||
| 2mg | 56.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 129.00 € | ||
| 25mg | 244.00 € | ||
| 50mg | 369.00 € | ||
| 100mg | 548.00 € | ||
| 500mg | 1,175.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Secretin (33-59), rat
CAS:121028-49-7
Secretin (33-59), rat (Secretin (rat)) is a classical hormone in the gastrointestinal system and a …
Formula:
C129H216N42O42
Purity:
98.12%
Color and Shape:
Solid
Molecular weight:
3027.35
Ref: TM-TP1039
| 1mg | 100.00 € | ||
| 5mg | 239.00 € | ||
| 10mg | 352.00 € | ||
| 25mg | 539.00 € | ||
| 50mg | 748.00 € | ||
| 100mg | 1,010.00 € | ||
| 200mg | 1,356.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Senktide
CAS:106128-89-6
Senktide is an agonist of tachykinin NK3 receptor.
Formula:
C40H55N7O11S
Purity:
100%
Color and Shape:
White Powder
Molecular weight:
841.97
Ref: TM-T7633
| 1mg | 62.00 € | ||
| 5mg | 128.00 € | ||
| 10mg | 183.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Paltusotine
CAS:2172870-89-0
Paltusotine: nonpeptide SST2 agonist, orally bioavailable, regulates GH/IGF-1 in acromegaly.
Formula:
C27H22F2N4O
Purity:
99.77%
Color and Shape:
Solid
Molecular weight:
456.49
Ref: TM-T9692
| 1mg | 171.00 € | ||
| 5mg | 413.00 € | ||
| 10mg | 597.00 € | ||
| 25mg | 903.00 € | ||
| 50mg | 1,220.00 € | ||
| 100mg | 1,645.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
