G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Fexofenadine hydrochloride
CAS:153439-40-8
Fexofenadine hydrochloride (Terfenidine carboxylate hydrochloride) is a second generation antihistamine that is used for the …
Formula:
C32H39NO4·HCl
Purity:
99.39% - ≥95%
Color and Shape:
Solid
Molecular weight:
538.13
Ref: TM-T1470
| 10mg | 49.00 € | ||
| 25mg | 78.00 € | ||
| 50mg | 96.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
PNU 22394 hydrochloride
CAS:15923-42-9
PNU 22394 hydrochloride is a 5-HT2C agonist and partial 5-HT2A/5-HT2B agonist
Formula:
C13H17ClN2
Purity:
97.83%
Color and Shape:
Solid
Molecular weight:
236.74
Ref: TM-T23168
| 1mg | 54.00 € | ||
| 2mg | 74.00 € | ||
| 5mg | 103.00 € | ||
| 10mg | 148.00 € | ||
| 25mg | 258.00 € | ||
| 50mg | 378.00 € | ||
| 100mg | 540.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
Pergolide mesylate
CAS:66104-23-2
Pergolide mesylate (LY127809), a dopamine agonist for Parkinson's and hyperprolactinemia, was withdrawn for heart valve …
Formula:
C20H30N2O3S2
Purity:
99.70%
Color and Shape:
White To Off-White Solid
Molecular weight:
410.59
Ref: TM-T2226
| 5mg | 51.00 € | ||
| 10mg | 73.00 € | ||
| 25mg | 115.00 € | ||
| 50mg | 177.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
Montelukast sodium
CAS:151767-02-1
Montelukast sodium (MK0476), an oral leukotriene antagonist for asthma, can cause rare liver injury.
Formula:
C35H35ClNNaO3S
Purity:
99.35% - 99.89%
Color and Shape:
White To Off-White Crystalline Powder
Molecular weight:
608.17
Ref: TM-T1677L
| 50mg | 48.00 € | ||
| 100mg | 72.00 € | ||
| 500mg | 130.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
MS21570
CAS:65373-29-7
MS21570 as a GPR171 antagonist based on its ability to block,with an IC50 of 220 …
Formula:
C10H11N3S2
Purity:
97.79%
Color and Shape:
Solid
Molecular weight:
237.34
Ref: TM-T5828
| 5mg | 46.00 € | ||
| 10mg | 59.00 € | ||
| 25mg | 97.00 € | ||
| 50mg | 148.00 € | ||
| 100mg | 213.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
Dexmedetomidine
CAS:113775-47-6
Dexmedetomidine: a central alpha-2 adrenergic agonist for general anesthesia.
Formula:
C13H16N2
Purity:
100% - 99.74%
Color and Shape:
Solid
Molecular weight:
200.28
Ref: TM-T2524
| 25mg | 47.00 € | ||
| 50mg | 70.00 € | ||
| 100mg | 96.00 € | ||
| 200mg | 153.00 € | ||
| 500mg | 249.00 € | ||
| 1mL*10mM (DMSO) | 50.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
1-methoxycyclopropanecarboxylic acid
CAS:100683-08-7
1-methoxycyclopropanecarboxylic acid is an agonist of free fatty acid receptor 3 (FFAR3, human).
Formula:
C5H8O3
Purity:
99.44%
Color and Shape:
Light-Yellow To Yellow Solid Or Liquid
Molecular weight:
116.12
Ref: TM-T9437
| 5mg | 35.00 € | ||
| 10mg | 49.00 € | ||
| 25mg | 85.00 € | ||
| 50mg | 113.00 € | ||
| 100mg | 169.00 € | ||
| 200mg | 246.00 € | ||
| 1mL*10mM (DMSO) | 37.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
Oxyntomodulin acetate
Oxyntomodulin acetate, a 37-amino acid peptide hormone, is a glucagon-like peptide 1 (GLP-1) receptor agonist[1].
Purity:
99.24%
Molecular weight:
N/A
Ref: TM-TP1976L
| 1mg | 175.00 € | ||
| 5mg | 517.00 € | ||
| 10mg | 842.00 € | ||
| 25mg | 1,510.00 € | ||
| 50mg | 2,270.00 € | ||
| 100mg | 3,068.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
SB-265610
CAS:211096-49-0
SB-265610 (GSK-CXCR2) is a nonpeptide and allosteric CXCR2 antagonist.
Formula:
C14H9BrN6O
Purity:
97.67%
Color and Shape:
Solid
Molecular weight:
357.16
Ref: TM-T16850
| 1mg | 56.00 € | ||
| 5mg | 119.00 € | ||
| 10mg | 187.00 € | ||
| 25mg | 376.00 € | ||
| 50mg | 560.00 € | ||
| 100mg | 800.00 € | ||
| 500mg | 1,644.00 € | ||
| 1mL*10mM (DMSO) | 131.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
Almorexant
CAS:871224-64-5
Almorexant (ACT 078573), a strong dual orexin receptor antagonist, has Ki of 1.3 nM for …
Formula:
C29H31F3N2O3
Purity:
97.75% - 98.02%
Color and Shape:
Solid
Molecular weight:
512.56
Ref: TM-T2613
| 1mg | 47.00 € | ||
| 5mg | 88.00 € | ||
| 10mg | 143.00 € | ||
| 25mg | 316.00 € | ||
| 50mg | 522.00 € | ||
| 100mg | 758.00 € | ||
| 1mL*10mM (DMSO) | 97.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
Vipadenant
CAS:442908-10-3
Vipadenant (CEB-4520)(BIIB-014) is an adenosine A2a antagonist with Ki of 1.3 nM; less potent for …
Formula:
C16H15N7O
Purity:
97.25% - 97.36%
Color and Shape:
Solid
Molecular weight:
321.34
Ref: TM-T2373
| 1mg | 40.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 119.00 € | ||
| 25mg | 210.00 € | ||
| 50mg | 350.00 € | ||
| 100mg | 522.00 € | ||
| 500mg | 1,130.00 € | ||
| 1mL*10mM (DMSO) | 359.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
ML382
CAS:1646499-97-9
ML382 is a potent and selective MrgX1 positive allosteric modulator(EC50 : 190 nM).
Formula:
C18H20N2O4S
Purity:
99.79%
Color and Shape:
Solid
Molecular weight:
360.43
Ref: TM-T8538
| 5mg | 48.00 € | ||
| 10mg | 74.00 € | ||
| 25mg | 129.00 € | ||
| 50mg | 226.00 € | ||
| 100mg | 335.00 € | ||
| 200mg | 469.00 € | ||
| 1mL*10mM (DMSO) | 50.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
Protease-Activated Receptor-4 diTFA
Protease-Activated Receptor-4 diTFA,2454 is the proteinase-activated receptor-4 (PAR4)agonist
Formula:
C37H48F6N8O11
Purity:
98.54%
Color and Shape:
Solid
Molecular weight:
894.81
Ref: TM-T7740
| 1mg | 48.00 € | ||
| 2mg | 60.00 € | ||
| 5mg | 86.00 € | ||
| 10mg | 138.00 € | ||
| 25mg | 274.00 € | ||
| 50mg | 411.00 € | ||
| 100mg | 607.00 € | ||
| 1mL*10mM (DMSO) | 170.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
GR 94800 acetate
GR 94800 acetate is a potent and selective neurokinin 2(NK-2) antagonist.
Formula:
C51H65N9O10
Purity:
97.86%
Color and Shape:
Liquid
Molecular weight:
964.12
Ref: TM-T22811L
| 1mg | 363.00 € | ||
| 2mg | 515.00 € | ||
| 5mg | 775.00 € | ||
| 10mg | 1,035.00 € | ||
| 25mg | 1,549.00 € | ||
| 50mg | 2,090.00 € | ||
| 100mg | 2,822.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
Glucagon-like peptide 1 (1-37), human acetate
Glucagon-like peptide 1 (1-37), human acetate is a highly potent the GLP-1 receptor agonist.
Purity:
98%
Molecular weight:
N/A
Ref: TM-TP1148L
| 1mg | 378.00 € | ||
| 5mg | 850.00 € | ||
| 10mg | 1,273.00 € | ||
| 25mg | 2,292.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
Cyproheptadine hydrochloride
CAS:969-33-5
Cyproheptadine hydrochloride (Periactin hydrochloride) is a hydrochloride salt form of cyproheptadine which is a histamine …
Formula:
C21H21N·HCl
Purity:
99.97%
Color and Shape:
Solid
Molecular weight:
323.86
Ref: TM-T6814
| 100mg | 34.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
VER-155008
CAS:1134156-31-2
VER-155008 is a potent Hsp70 family inhibitor with IC50 of 0.5 μM, 2.6 μM, and …
Formula:
C25H23Cl2N7O4
Purity:
98.88% - 99.55%
Color and Shape:
Solid
Molecular weight:
556.4
Ref: TM-T7010
| 2mg | 47.00 € | ||
| 5mg | 69.00 € | ||
| 10mg | 93.00 € | ||
| 25mg | 163.00 € | ||
| 50mg | 283.00 € | ||
| 100mg | 467.00 € | ||
| 200mg | 653.00 € | ||
| 1mL*10mM (DMSO) | 85.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
Orphanin FQ(1-11) acetate(178249-41-7 free base)
Nociceptin peptide fragment (1-11 aa), potent ORL1/KOR-3 agonist (Ki=55 nM), non-opioid, analgesic in mice.
Formula:
C51H79N15O16
Purity:
95.54%
Color and Shape:
Solid
Molecular weight:
1158.26
Ref: TM-TP1882L1
| 1mg | 159.00 € | ||
| 5mg | 346.00 € | ||
| 10mg | 520.00 € | ||
| 25mg | 838.00 € | ||
| 50mg | 1,130.00 € | ||
| 100mg | 1,549.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
Brimonidine Tartrate
CAS:70359-46-5
Brimonidine Tartrate (AGN190342 tartrate) is a quinoxaline derivative and adrenergic α-2 receptor agonist (EC50: 0.45 …
Formula:
C15H16BrN5O6
Purity:
99.83%
Color and Shape:
Off-White Crystalline Solid
Molecular weight:
442.22
Ref: TM-T6422
| 100mg | 48.00 € | ||
| 500mg | 124.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
(±)-Ibipinabant
CAS:362519-49-1
(±)-Ibipinabant ((±)-SLV319) has been used in trials studying the treatment of Obesity and Obesity and …
Formula:
C23H20Cl2N4O2S
Purity:
99.28% - 99.83%
Color and Shape:
Solid
Molecular weight:
487.4
Ref: TM-T4654
| 5mg | 50.00 € | ||
| 10mg | 90.00 € | ||
| 25mg | 164.00 € | ||
| 50mg | 293.00 € | ||
| 100mg | 424.00 € | ||
| 200mg | 588.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
