G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Afamelanotide acetate
CAS:1566590-77-9
Afamelanotide acetate is a synthetic α-melanocyte stimulating hormone analogue and first-in-class melanocortin-1 receptor agonist.
Formula:
C80H115N21O21
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1706.9
Ref: TM-T7589
| 1mg | 73.00 € | ||
| 5mg | 160.00 € | ||
| 10mg | 230.00 € | ||
| 25mg | 378.00 € | ||
| 50mg | 565.00 € | ||
| 100mg | 805.00 € | ||
| 1mL*10mM (DMSO) | 339.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
Talinolol
CAS:57460-41-0
(±)-Talinolol is a selective β1 adrenoceptor antagonist well known for its cardioprotective and antihypertensive activity.
Formula:
C20H33N3O3
Purity:
98.80%
Color and Shape:
Solid
Molecular weight:
363.49
Ref: TM-T21640
| 1mg | 74.00 € | ||
| 2mg | 99.00 € | ||
| 5mg | 168.00 € | ||
| 10mg | 304.00 € | ||
| 25mg | 547.00 € | ||
| 50mg | 782.00 € | ||
| 100mg | 1,074.00 € | ||
| 1mL*10mM (DMSO) | 170.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
Obestatin (rat) acetate
Obestatin (rat) acetate is an endogenous ligand of G-protein coupled receptor 39 (GPR39).
Formula:
C114H174N34O31
Purity:
99.05%
Color and Shape:
Liquid
Molecular weight:
2516.81
Ref: TM-TP2279L
| 1mg | 115.00 € | ||
| 5mg | 250.00 € | ||
| 10mg | 375.00 € | ||
| 25mg | 627.00 € | ||
| 50mg | 893.00 € | ||
| 100mg | 1,216.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
CS 2100
CAS:913827-99-3
CS 2100 (1-[[4-Ethyl-5-[5-(4-phenoxyphenyl)-1,2,4-oxadiazol-3-yl]-2-thienyl]methyl]-3-azetidinecarboxylic acid) is an S1P1 agonist.
Formula:
C25H23N3O4S
Purity:
98.13%
Color and Shape:
Solid
Molecular weight:
461.53
Ref: TM-T22697
| 2mg | 42.00 € | ||
| 5mg | 64.00 € | ||
| 10mg | 92.00 € | ||
| 25mg | 177.00 € | ||
| 50mg | 281.00 € | ||
| 100mg | 414.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
Clomipramine
CAS:303-49-1
Clomipramine treats OCD, depression, chronic pain, and may lower suicide risk in seniors; works by …
Formula:
C19H23ClN2
Purity:
99.31%
Color and Shape:
Solid
Molecular weight:
314.85
Ref: TM-T21013
| 2mg | 47.00 € | ||
| 5mg | 70.00 € | ||
| 10mg | 96.00 € | ||
| 25mg | 180.00 € | ||
| 50mg | 274.00 € | ||
| 100mg | 406.00 € | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
Bupranolol
CAS:14556-46-8
Bupranolol blocks β2-adrenergic receptor; treats angina, hypertension, glaucoma, arrhythmia, and prevents clots.
Formula:
C14H22ClNO2
Purity:
95.85%
Color and Shape:
Solid
Molecular weight:
271.78
Ref: TM-T8580
| 1mg | 50.00 € | ||
| 5mg | 111.00 € | ||
| 10mg | 167.00 € | ||
| 25mg | 325.00 € | ||
| 50mg | 465.00 € | ||
| 100mg | 615.00 € | ||
| 200mg | 830.00 € | ||
| 1mL*10mM (DMSO) | 101.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
JNJ-37822681
CAS:935776-74-2
JNJ-37822681 is a novel, highly selective dopamine D₂ receptor antagonist characterized by a rapid dissociation …
Formula:
C17H17F5N4
Purity:
99.48%
Color and Shape:
Solid
Molecular weight:
372.34
Ref: TM-T27677
| 1mg | 87.00 € | ||
| 2mg | 124.00 € | ||
| 5mg | 187.00 € | ||
| 10mg | 284.00 € | ||
| 25mg | 462.00 € | ||
| 1mL*10mM (DMSO) | 202.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
Ibutamoren Mesylate
CAS:159752-10-0
Ibutamoren Mesylate (MK-0677) is a potent, non-peptide Growth hormone secretagogue receptor (GHSR) agonist.
Formula:
C28H40N4O8S2
Purity:
97.98% - ≥98%
Color and Shape:
Solid
Molecular weight:
624.77
Ref: TM-T7112
| 5mg | 63.00 € | ||
| 10mg | 85.00 € | ||
| 50mg | 105.00 € | ||
| 100mg | 125.00 € | ||
| 500mg | 168.00 € | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
Ondansetron hydrochloride
CAS:99614-01-4
Ondansetron hydrochloride (Zofran) is a serotonin 5-HT3 receptor antagonist, used to prevent nausea and vomiting …
Formula:
C18H19N3O·HCl
Purity:
99.78%
Color and Shape:
White Powder
Molecular weight:
329.82
Ref: TM-T6616
| 25mg | 44.00 € | ||
| 50mg | 58.00 € | ||
| 100mg | To inquire | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
Relugolix
CAS:737789-87-6
Relugolix (RVT-601) is an orally available, non-peptide gonadotropin-releasing hormone (GnRH or luteinizing hormone-releasing hormone (LHRH)) …
Formula:
C29H27F2N7O5S
Purity:
98.64% - 99.67%
Color and Shape:
Solid
Molecular weight:
623.63
Ref: TM-T3630
| 1mg | 37.00 € | ||
| 5mg | 79.00 € | ||
| 10mg | 116.00 € | ||
| 25mg | 198.00 € | ||
| 50mg | 329.00 € | ||
| 100mg | 512.00 € | ||
| 500mg | 1,093.00 € | ||
| 1mL*10mM (DMSO) | 96.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
Dapiprazole Hydrochloride
CAS:72822-13-0
Dapiprazole Hydrochloride (Glamidolo Hydrochloride) is an alpha-1-adrenergic antagonist that acts by blocking alpha-adrenergic receptors.
Formula:
C19H28ClN5
Purity:
100% - 99.86%
Color and Shape:
Solid
Molecular weight:
361.92
Ref: TM-T3996
| 10mg | 50.00 € | ||
| 25mg | 87.00 € | ||
| 50mg | 135.00 € | ||
| 100mg | 187.00 € | ||
| 200mg | 283.00 € | ||
| 1mL*10mM (DMSO) | 35.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
BAY-545
CAS:1699717-32-2
BAY-545 is an antagonist of A2B adenosine receptor(IC50 : 59 nM).
Formula:
C18H22F3N3O4S
Purity:
98.05%
Color and Shape:
Solid
Molecular weight:
433.45
Ref: TM-T8512
| 1mg | 88.00 € | ||
| 5mg | 170.00 € | ||
| 10mg | 248.00 € | ||
| 25mg | 444.00 € | ||
| 50mg | 638.00 € | ||
| 100mg | 889.00 € | ||
| 200mg | 1,198.00 € | ||
| 1mL*10mM (DMSO) | 182.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
GR-73632
CAS:133156-06-6
Potent and selective tachykinin NK1 receptor agonist (EC50 = 2 nM in guinea pig vas …
Formula:
C40H59N7O6S
Purity:
99.68%
Color and Shape:
Solid
Molecular weight:
766
Ref: TM-TP1572
| 1mg | 52.00 € | ||
| 5mg | 111.00 € | ||
| 10mg | 170.00 € | ||
| 25mg | 283.00 € | ||
| 50mg | 430.00 € | ||
| 100mg | 620.00 € | ||
| 200mg | 870.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
SB-334867 free base
CAS:792173-99-0
SB-334867 free base (SB334867A free base) is a selective orexin-1 (OX1) receptor antagonist.
Formula:
C17H13N5O2
Purity:
100% - 99.91%
Color and Shape:
Solid
Molecular weight:
319.32
Ref: TM-T6140
| 2mg | 42.00 € | ||
| 5mg | 70.00 € | ||
| 10mg | 99.00 € | ||
| 25mg | 160.00 € | ||
| 50mg | 226.00 € | ||
| 100mg | 338.00 € | ||
| 200mg | 502.00 € | ||
| 1mL*10mM (DMSO) | 78.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
Nastorazepide
CAS:209219-38-5
Nastorazepide is a selective, orally available antagonist of gastrin/cholecystokinin 2 (CCK-2) receptor with potential antineoplastic …
Formula:
C29H36N4O5
Purity:
99.60%
Color and Shape:
Solid
Molecular weight:
520.62
Ref: TM-TQ0062
| 1mg | 52.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 180.00 € | ||
| 25mg | 344.00 € | ||
| 50mg | 525.00 € | ||
| 100mg | 758.00 € | ||
| 1mL*10mM (DMSO) | 120.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
Avexitide
CAS:133514-43-9
Avexitide (Exendin-3 (9-39) amide) (Exendin (9-39)) is a specific and competitive antagonist of glucagon-like peptide-1 …
Formula:
C149H234N40O47S
Purity:
98% - 99.65%
Color and Shape:
Solid
Molecular weight:
3369.76
Ref: TM-TP2100
| 1mg | 188.00 € | ||
| 5mg | 502.00 € | ||
| 10mg | 715.00 € | ||
| 25mg | 1,074.00 € | ||
| 50mg | 1,454.00 € | ||
| 100mg | 1,882.00 € | ||
| 500µg | 133.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
Questiomycin A
CAS:1916-59-2
Questiomycin A: crème fraiche antibiotic with antibacterial, anticancer effects; inhibits GRP78.
Formula:
C12H8N2O2
Purity:
98% - 99.07%
Color and Shape:
Solid
Molecular weight:
212.2
Ref: TM-T36818
| 10mg | 55.00 € | ||
| 25mg | 87.00 € | ||
| 50mg | 127.00 € | ||
| 100mg | 175.00 € | ||
| 200mg | 250.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
Exendin-4 acetate
CAS:914454-01-6
Exendin-4 acetate is a 39 amino acid peptide.Exendin-4 acetate is a long-acting GLP-1 receptor agonist(IC50 …
Formula:
C186H286N50O62S
Purity:
98.65%
Color and Shape:
Solid
Molecular weight:
4247
Ref: TM-T8748
| 1mg | 67.00 € | ||
| 5mg | 138.00 € | ||
| 10mg | 197.00 € | ||
| 25mg | 281.00 € | ||
| 50mg | 420.00 € | ||
| 100mg | 620.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
Clebopride malate
CAS:57645-91-7
Clebopride malate is a dopamine antagonist drug Used to treat functional gastrointestinal disorders such as …
Formula:
C24H30ClN3O7
Purity:
99.52%
Color and Shape:
Solid
Molecular weight:
507.96
Ref: TM-T7569
| 5mg | 35.00 € | ||
| 10mg | 48.00 € | ||
| 25mg | 70.00 € | ||
| 50mg | 96.00 € | ||
| 100mg | 145.00 € | ||
| 200mg | 210.00 € | ||
| 1mL*10mM (DMSO) | 38.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
![[Sar9,Met(O2)11]-Substance P](https://static.cymitquimica.com/products/TM/thumb/T7828.jpg)
[Sar9,Met(O2)11]-Substance P
CAS:110880-55-2
[Sar9,Met(O2)11]-Substance P (NA) is an agonist of NK1 receptor.
Formula:
C64H100N18O15S
Purity:
100%
Color and Shape:
Solid
Molecular weight:
1393.66
Ref: TM-T7828
| 1mg | 85.00 € | ||
| 5mg | 273.00 € | ||
| 10mg | 492.00 € | ||
| 25mg | 800.00 € | ||
| 50mg | 1,103.00 € | ||
| 100mg | 1,491.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
