G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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ICI 89406
CAS:53671-71-9
ICI 89406 (1-[2-[[3-(2-cyanophenoxy)-2-hydroxypropyl]amino]ethyl]-3-phenylurea) is a β-adrenergic antagonist.
Formula:
C19H22N4O3
Purity:
99.62%
Color and Shape:
Solid
Molecular weight:
354.4
Ref: TM-T22852
| 1mg | 79.00 € | ||
| 5mg | 144.00 € | ||
| 10mg | 199.00 € | ||
| 25mg | 457.00 € | ||
| 50mg | 653.00 € | ||
| 100mg | 926.00 € | ||
| 500mg | 1,840.00 € | ||
| 1mL*10mM (DMSO) | 152.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Adenosine amine congener
CAS:96760-69-9
Adenosine amine congener (ADAC) (ADAC) is an agonist of selective A1 adenosine receptor,.
Formula:
C28H32N8O6
Purity:
97.86%
Color and Shape:
Solid
Molecular weight:
576.6
Ref: TM-T7683
| 1mg | 73.00 € | ||
| 5mg | 158.00 € | ||
| 10mg | 230.00 € | ||
| 25mg | 416.00 € | ||
| 50mg | 612.00 € | ||
| 100mg | 873.00 € | ||
| 1mL*10mM (DMSO) | 245.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
USL311
CAS:1373268-67-7
USL311 blocks CXCR4/SDF-1 interaction, inhibits tumor cell growth and migration.
Formula:
C24H34N6O
Purity:
99.56% - 99.73%
Color and Shape:
Solid
Molecular weight:
422.57
Ref: TM-T17208
| 1mg | 42.00 € | ||
| 5mg | 88.00 € | ||
| 10mg | 126.00 € | ||
| 25mg | 247.00 € | ||
| 50mg | 388.00 € | ||
| 100mg | 621.00 € | ||
| 500mg | 1,288.00 € | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Treprostinil
CAS:81846-19-7
Treprostinil (Orenitram) is a potent DP1, IP and EP2 agonist (EC50: 0.6/1.9/6.2 nM).
Formula:
C23H34O5
Purity:
99.71%
Color and Shape:
Solid
Molecular weight:
390.51
Ref: TM-T5150
| 2mg | 46.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 118.00 € | ||
| 25mg | 268.00 € | ||
| 50mg | 448.00 € | ||
| 100mg | 640.00 € | ||
| 1mL*10mM (DMSO) | 67.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
BA 1 acetate(183241-31-8 free base)
BA 1 acetate: bombesin agonist, IC50s: 0.26/1.55/2.52 nM (BB1/BB2/BB3), boosts glucose transport, promotes lung cancer …
Formula:
C59H80N14O13
Purity:
95.3%
Color and Shape:
Solid
Molecular weight:
1193.35
Ref: TM-TP1913L1
| 1mg | 94.00 € | ||
| 5mg | 182.00 € | ||
| 10mg | 274.00 € | ||
| 25mg | 495.00 € | ||
| 50mg | 716.00 € | ||
| 100mg | 994.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Binodenoson
CAS:144348-08-3
Binodenoson (WRC 0470), a selective A2A adenosine receptor agonist, aids in coronary imaging.
Formula:
C17H25N7O4
Purity:
99.84%
Color and Shape:
Solid
Molecular weight:
391.42
Ref: TM-T9516
| 1mg | 137.00 € | ||
| 5mg | 282.00 € | ||
| 10mg | 424.00 € | ||
| 25mg | 701.00 € | ||
| 50mg | 937.00 € | ||
| 100mg | 1,319.00 € | ||
| 1mL*10mM (DMSO) | 311.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Dynorphin A acetate(80448-90-4 free base)
Dynorphin A acetate is an Endogenous kappa receptor agonist.
Formula:
C101H159N31O25
Purity:
99.69%
Color and Shape:
Solid
Molecular weight:
2207.58
Ref: TM-TP2040L
| 1mg | 70.00 € | ||
| 5mg | 234.00 € | ||
| 10mg | 321.00 € | ||
| 25mg | 541.00 € | ||
| 50mg | 774.00 € | ||
| 100mg | 1,067.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Nelotanserin
CAS:839713-36-9
Nelotanserin (APD125): strong 5-HT2A inverse agonist (IC50: 1.7 nM), moderate 5-HT2C (79 nM), weak 5-HT2B …
Formula:
C18H15BrF2N4O2
Purity:
98.01% - 98.42%
Color and Shape:
Solid
Molecular weight:
437.24
Ref: TM-T7350
| 1mg | 40.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 86.00 € | ||
| 10mg | 118.00 € | ||
| 25mg | 185.00 € | ||
| 50mg | 343.00 € | ||
| 100mg | 510.00 € | ||
| 500mg | 1,109.00 € | ||
| 1mL*10mM (DMSO) | 84.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
BETP
CAS:1371569-69-5
BETP is an agonist of GLP-1 receptor (EC50s: 0.66 and 0.755 μM for human and …
Formula:
C20H17F3N2O2S
Purity:
97.92%
Color and Shape:
Solid
Molecular weight:
406.42
Ref: TM-TQ0124
| 1mg | 47.00 € | ||
| 5mg | 91.00 € | ||
| 10mg | 137.00 € | ||
| 25mg | 258.00 € | ||
| 50mg | 414.00 € | ||
| 100mg | 661.00 € | ||
| 1mL*10mM (DMSO) | 96.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Phenylbiguanide
CAS:102-02-3
Phenylbiguanide (N-Phenylbiguanide) is a 5-HT3 receptor selective agonist(EC50 : 3.0±0.1 μM)
Formula:
C8H11N5
Purity:
99.87%
Color and Shape:
Solid
Molecular weight:
177.21
Ref: TM-T7135
| 50mg | 35.00 € | ||
| 100mg | 46.00 € | ||
| 500mg | 87.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
TUG-1375
CAS:2247372-59-2
TUG-1375 is an Agonist of Thiazolidine Free Fatty Acid Receptor 2
Formula:
C22H19ClN2O4S
Purity:
97.72% - 99.41%
Color and Shape:
Solid
Molecular weight:
442.92
Ref: TM-T7796
| 1mg | 131.00 € | ||
| 5mg | 318.00 € | ||
| 10mg | 521.00 € | ||
| 25mg | 812.00 € | ||
| 50mg | 1,088.00 € | ||
| 100mg | 1,463.00 € | ||
| 500mg | 2,895.00 € | ||
| 1mL*10mM (DMSO) | 350.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
AM1241
CAS:444912-48-5
AM-1241 is a selective cannabinoid CB2 receptor agonist with Ki of 3.4 nM, exhibits 82-fold …
Formula:
C22H22IN3O3
Purity:
98.82% - 99.10%
Color and Shape:
Solid
Molecular weight:
503.33
Ref: TM-T6755
| 2mg | 38.00 € | ||
| 5mg | 51.00 € | ||
| 10mg | 88.00 € | ||
| 25mg | 168.00 € | ||
| 50mg | 284.00 € | ||
| 100mg | 512.00 € | ||
| 500mg | 1,112.00 € | ||
| 1mL*10mM (DMSO) | 92.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Ponesimod
CAS:854107-55-4
Ponesimod (ACT-128800) is an orally available sphingosine-1-phosphate receptor 1 (S1PR1, S1P1) agonist with potential immunomodulating …
Formula:
C23H25ClN2O4S
Purity:
98.22% - 99.42%
Color and Shape:
Solid
Molecular weight:
460.97
Ref: TM-T3258
| 1mg | 45.00 € | ||
| 2mg | 58.00 € | ||
| 5mg | 92.00 € | ||
| 10mg | 128.00 € | ||
| 25mg | 229.00 € | ||
| 50mg | 397.00 € | ||
| 100mg | 583.00 € | ||
| 500mg | 1,254.00 € | ||
| 1mL*10mM (DMSO) | 96.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
![Lys-[Des-Arg9]Bradykinin acetate](https://static.cymitquimica.com/products/TM/thumb/TP1918L1.jpg)
Lys-[Des-Arg9]Bradykinin acetate
Lys-[Des-Arg9]Bradykinin acetate is an endogenous potent and highly selective bradykinin B1 receptor agonist (Ki values …
Formula:
C52H77N13O13
Purity:
99.93%
Color and Shape:
Solid
Molecular weight:
1092.27
Ref: TM-TP1918L1
| 1mg | 88.00 € | ||
| 5mg | 172.00 € | ||
| 10mg | 258.00 € | ||
| 25mg | 472.00 € | ||
| 50mg | 683.00 € | ||
| 100mg | 966.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
HCGRP-(8-37) acetate
HCGRP-(8-37) acetate is a human calcitonin gene-related peptide (hCGRP) fragment acetate and also an antagonist …
Formula:
C141H234N44O40
Purity:
99.29%
Color and Shape:
Solid
Molecular weight:
3185.64
Ref: TM-TP1134L
| 1mg | 164.00 € | ||
| 5mg | 379.00 € | ||
| 10mg | 541.00 € | ||
| 25mg | 815.00 € | ||
| 50mg | 1,073.00 € | ||
| 100mg | 1,468.00 € | ||
| 200mg | 1,981.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
GSK137647A
CAS:349085-82-1
GSK137647A (GSK 137647) is a selective FFA4 agonist.
Formula:
C16H19NO3S
Purity:
99.15% - 99.87%
Color and Shape:
Solid
Molecular weight:
305.39
Ref: TM-T3171
| 2mg | 35.00 € | ||
| 5mg | 51.00 € | ||
| 10mg | 83.00 € | ||
| 25mg | 151.00 € | ||
| 50mg | 241.00 € | ||
| 100mg | 416.00 € | ||
| 200mg | 604.00 € | ||
| 500mg | 916.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
M40 acetate(143896-17-7 free base)
M40 acetate is a potent, non-selective galanin receptor antagonist (Ki values are 1.82 and 5.1 …
Formula:
C96H149N23O26
Purity:
99.88%
Color and Shape:
Solid
Molecular weight:
2041.38
Ref: TM-TP1992L
| 1mg | 112.00 € | ||
| 5mg | 268.00 € | ||
| 10mg | 383.00 € | ||
| 25mg | 598.00 € | ||
| 50mg | 818.00 € | ||
| 100mg | 1,081.00 € | ||
| 200mg | 1,447.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Salbutamol hemisulfate
CAS:51022-70-9
Salbutamol hemisulfate (Albuterol Sulfate) is a short-acting β2-adrenergic receptor agonist with an IC50 of 8.93 …
Formula:
C13H21NO3H2O4S
Purity:
99.35%
Color and Shape:
White Or Almost White Odourless Powder
Molecular weight:
576.7
Ref: TM-T6652
| 100mg | 54.00 € | ||
| 200mg | 64.00 € | ||
| 500mg | 95.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
PHA-767491
CAS:845714-00-3
PHA-767491 (CAY10572) is a potent ATP-competitive dual Cdc7/CDK9 inhibitor with IC50 of 10 nM and …
Formula:
C12H11N3O
Purity:
100.00% - 99.49%
Color and Shape:
Solid
Molecular weight:
213.24
Ref: TM-T6206
| 2mg | 35.00 € | ||
| 5mg | 49.00 € | ||
| 10mg | 68.00 € | ||
| 25mg | 130.00 € | ||
| 50mg | 220.00 € | ||
| 100mg | 396.00 € | ||
| 1mL*10mM (DMSO) | 49.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Kisspeptin 234 acetate(1145998-81-7 free base)
Kisspeptin receptor (KISS1/GPR54) blocker; analog to kisspeptin-10. Curbs IP activation (IC50=7nM) & GnRH release.
Formula:
C65H82N18O15
Purity:
99.34%
Color and Shape:
Solid
Molecular weight:
1355.46
Ref: TM-TP1896L1
| 1mg | 143.00 € | ||
| 5mg | 303.00 € | ||
| 10mg | 468.00 € | ||
| 25mg | 761.00 € | ||
| 50mg | 1,049.00 € | ||
| 100mg | 1,421.00 € | ||
| 500mg | 2,769.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
