G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Substance P 1-9 aceate
Substance P 1-9 aceate is nonapeptide, which decreases the inactivation of substance P by the …
Formula:
C54H81N15O14
Purity:
99.01%
Color and Shape:
Liquid
Molecular weight:
1164.31
Ref: TM-TP1819L
| 1mg | 65.00 € | ||
| 5mg | 164.00 € | ||
| 10mg | 244.00 € | ||
| 25mg | 440.00 € | ||
| 50mg | 643.00 € | ||
| 100mg | 919.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
N-terminally acetylated Leu-enkephalin
Leu-enkephalin, an endogenous 5-amino acid peptide, activates opioid receptors; its acetylated form exists.
Formula:
C30H39N5O8
Purity:
100%
Color and Shape:
Solid
Molecular weight:
597.66
Ref: TM-T8557
| 1mg | 79.00 € | ||
| 5mg | 142.00 € | ||
| 10mg | 212.00 € | ||
| 25mg | 368.00 € | ||
| 50mg | 538.00 € | ||
| 100mg | 769.00 € | ||
| 500mg | 1,533.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
WAY-100635 Monomaleate
CAS:1092679-51-0
WAY-100635 maleate is a selective 5-hydroxytryptamine 1A receptor antagonist with an IC50 value of 0.91 …
Formula:
C25H34N4O2·C4H4O4
Purity:
100% - 99.68%
Color and Shape:
Solid
Molecular weight:
538.64
Ref: TM-T2631
| 2mg | 50.00 € | ||
| 5mg | 66.00 € | ||
| 10mg | 94.00 € | ||
| 25mg | 178.00 € | ||
| 50mg | 330.00 € | ||
| 100mg | 490.00 € | ||
| 200mg | 708.00 € | ||
| 500mg | 1,093.00 € | ||
| 1mL*10mM (DMSO) | 78.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Detomidine hydrochloride
CAS:90038-01-0
Detomidine hydrochloride (MPV-253 AII) produce dose-dependent sedative and analgesic effects, mediatated by activation of α2 …
Formula:
C12H14N2·HCl
Purity:
99.89%
Color and Shape:
Solid
Molecular weight:
222.71
Ref: TM-T6464
| 10mg | 35.00 € | ||
| 25mg | 47.00 € | ||
| 50mg | 51.00 € | ||
| 100mg | 69.00 € | ||
| 500mg | 147.00 € | ||
| 1mL*10mM (DMSO) | 35.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
AMD-070 hydrochloride
CAS:880549-30-4
AMD-070 hydrochloride is a CXCR4 antagonist, is useful for Anti HIV.
Formula:
C21H28ClN5
Purity:
98.38% - 98.57%
Color and Shape:
Solid
Molecular weight:
385.93
Ref: TM-T22565
| 1mg | 49.00 € | ||
| 2mg | 68.00 € | ||
| 5mg | 92.00 € | ||
| 10mg | 138.00 € | ||
| 25mg | 267.00 € | ||
| 50mg | 400.00 € | ||
| 100mg | 592.00 € | ||
| 1mL*10mM (DMSO) | 104.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
MCL0020
CAS:475498-26-1
MCL0020 is a potent and selective melanocortin MC4 receptor antagonist, reverses stress-induced anorexia but has …
Formula:
C34H39N7O4
Purity:
99.18%
Color and Shape:
Solid
Molecular weight:
609.72
Ref: TM-TP1889
| 1mg | 112.00 € | ||
| 5mg | 273.00 € | ||
| 10mg | 378.00 € | ||
| 25mg | 582.00 € | ||
| 50mg | 796.00 € | ||
| 100mg | 1,052.00 € | ||
| 200mg | 1,427.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
![[Pyr1]-Apelin-13](https://static.cymitquimica.com/products/TM/thumb/TP1260.jpg)
[Pyr1]-Apelin-13
CAS:217082-60-5
[Pyr1]-Apelin-13 ([pGlu1]-Apelin-13) is a potent and selective endogenous Apelin receptor (APJ) agonist.
Formula:
C69H108N22O16S
Purity:
100%
Color and Shape:
Solid
Molecular weight:
1533.8
Ref: TM-TP1260
| 1mg | 96.00 € | ||
| 5mg | 269.00 € | ||
| 10mg | 424.00 € | ||
| 25mg | 684.00 € | ||
| 50mg | 916.00 € | ||
| 100mg | 1,271.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Indacaterol
CAS:312753-06-3
Indacaterol (Onbrez; Arcapta) is a β2-Adrenergic Agonist. The mechanism of action of indacaterol is as …
Formula:
C24H28N2O3
Purity:
100.00% - 99.63%
Color and Shape:
Solid
Molecular weight:
392.49
Ref: TM-T2320
| 25mg | 50.00 € | ||
| 50mg | 67.00 € | ||
| 1mL*10mM (DMSO) | 96.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Bay 59-3074
CAS:406205-74-1
Bay 59-3074 is a CB1/CB2 receptor partial agonist (Ki: 48.3/45.5 nM).
Formula:
C18H13F6NO4S
Purity:
97.68% - 99.69%
Color and Shape:
Solid
Molecular weight:
453.36
Ref: TM-T3699
| 10mg | 44.00 € | ||
| 25mg | 78.00 € | ||
| 50mg | 113.00 € | ||
| 100mg | 203.00 € | ||
| 200mg | 301.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
SAX-187
CAS:554403-49-5
SAX-187 (SAX-187) has high-affinity binding at the human 5-HT6 receptor.
Formula:
C15H13ClN4O2S2
Purity:
97.82% - 98%
Color and Shape:
Solid
Molecular weight:
380.87
Ref: TM-T3183
| 1mg | 124.00 € | ||
| 2mg | 167.00 € | ||
| 5mg | 256.00 € | ||
| 10mg | 427.00 € | ||
| 25mg | 691.00 € | ||
| 50mg | 926.00 € | ||
| 100mg | 1,276.00 € | ||
| 1mL*10mM (DMSO) | 279.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
(+)-PD 128907 hydrochloride
CAS:300576-59-4
(+)-PD 128907 hydrochloride is an agonist of D3 dopamine receptor .
Formula:
C14H20ClNO3
Purity:
97.76%
Color and Shape:
Solid
Molecular weight:
285.77
Ref: TM-T7553
| 2mg | 39.00 € | ||
| 5mg | 56.00 € | ||
| 10mg | 88.00 € | ||
| 25mg | 159.00 € | ||
| 50mg | 271.00 € | ||
| 100mg | 395.00 € | ||
| 200mg | 560.00 € | ||
| 1mL*10mM (DMSO) | 85.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Fevipiprant
CAS:872365-14-5
Fevipiprant (NVP-QAW039) is a selective, potent, reversible competitive CRTh2 antagonist.
Formula:
C19H17F3N2O4S
Purity:
99.32% - 99.59%
Color and Shape:
Solid
Molecular weight:
426.41
Ref: TM-T3965
| 5mg | 34.00 € | ||
| 10mg | 50.00 € | ||
| 25mg | 93.00 € | ||
| 50mg | 130.00 € | ||
| 100mg | 204.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Calcitonin(salmon) Acetate(47931-85-1(free base))
Calcitonin(salmon)Acetate(47931-85-1(free base))(Salmon calcitonin) , a calcium regulating hormone, is used to treat osteoporosis in women …
Formula:
C145H240N44O48S2
Purity:
99.29%
Color and Shape:
Solid
Molecular weight:
3431.85
Ref: TM-TP1040L
| 1mg | 93.00 € | ||
| 2mg | 119.00 € | ||
| 5mg | 176.00 € | ||
| 10mg | 253.00 € | ||
| 25mg | 395.00 € | ||
| 50mg | 582.00 € | ||
| 100mg | 826.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
GRA Ex-25
CAS:307983-31-9
GRA Ex-25 (GRA-Ex-25) is an inhibitor of glucagon receptor.
Formula:
C29H36F3N3O5
Purity:
98.2% - 98.88%
Color and Shape:
Solid
Molecular weight:
563.61
Ref: TM-T3422
| 1mg | 62.00 € | ||
| 2mg | 88.00 € | ||
| 5mg | 138.00 € | ||
| 10mg | 203.00 € | ||
| 25mg | 414.00 € | ||
| 50mg | 609.00 € | ||
| 100mg | 869.00 € | ||
| 1mL*10mM (DMSO) | 184.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Mequitazine
CAS:29216-28-2
Mequitazine (Virginan) is an effective, nonsedative and long-acting histamine H1 antagonist.
Formula:
C20H22N2S
Purity:
99.95%
Color and Shape:
Solid
Molecular weight:
322.47
Ref: TM-T4499
| 5mg | 55.00 € | ||
| 10mg | 63.00 € | ||
| 25mg | 89.00 € | ||
| 50mg | 121.00 € | ||
| 100mg | 152.00 € | ||
| 1mL*10mM (DMSO) | 50.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
A2B receptor antagonist 2
CAS:784-90-7
A2B receptor antagonist 2 is an antagonist of adenosine receptor A2B (Ki = 2.30 μM …
Formula:
C12H15N5
Purity:
100%
Color and Shape:
Liquid
Molecular weight:
229.28
Ref: TM-T37793
| 10mg | 45.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Lixisenatide acetate (320367-13-3 free base)
CAS:1997361-87-1
Lixisenatide acetate is a receptor agonist similar to glucagon-like peptide-1 (glp-1) for the treatment of …
Formula:
C215H347N61O65S·6C2H4O2
Purity:
98% - 99.9%
Color and Shape:
Solid
Molecular weight:
5218.88
Ref: TM-TP1469
| 1mg | 62.00 € | ||
| 5mg | 113.00 € | ||
| 10mg | 179.00 € | ||
| 25mg | 299.00 € | ||
| 50mg | 428.00 € | ||
| 100mg | 582.00 € | ||
| 200mg | 784.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Ondansetron
CAS:99614-02-5
Ondansetron (GR 38032) is a serotonin 5-HT3 receptor antagonist used mainly as an antiemetic.
Formula:
C18H19N3O
Purity:
98.9%
Color and Shape:
White To Yellow Crystals
Molecular weight:
293.36
Ref: TM-T6615
| 25mg | 55.00 € | ||
| 100mg | 78.00 € | ||
| 200mg | 102.00 € | ||
| 1mL*10mM (DMSO) | 60.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Darbufelone mesylate
CAS:139340-56-0
Darbufelone mesylate blocks PGF2α, LTB4, PGHS-2 (IC50: 0.19 μM), and PGHS-1 (IC50: 20 μM).
Formula:
C19H28N2O5S2
Purity:
96.81%
Color and Shape:
Solid
Molecular weight:
428.57
Ref: TM-T10960L
| 5mg | 118.00 € | ||
| 25mg | 423.00 € | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 16 Dec 2024
MF-766
CAS:1050656-06-8
MF-766: potent, selective oral EP4 antagonist, Ki=0.23 nM, IC50=1.4 nM; shifts to 1.8 nM with …
Formula:
C27H21F3N2O3
Purity:
98% - 98.06%
Color and Shape:
Solid
Molecular weight:
478.46
Ref: TM-T9622
| 1mg | 81.00 € | ||
| 5mg | 167.00 € | ||
| 10mg | 271.00 € | ||
| 25mg | 537.00 € | ||
| 50mg | 771.00 € | ||
| 100mg | 1,060.00 € | ||
| 500mg | 2,118.00 € | ||
| 1mL*10mM (DMSO) | 181.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
