G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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SCH 58261
CAS:160098-96-4
SCH 58261 is a potent and selective A2a adenosine receptor antagonist.The Ki =2.3 nM for …
Formula:
C18H15N7O
Purity:
99.75%
Color and Shape:
Solid
Molecular weight:
345.36
Ref: TM-T6979
| 1mg | 40.00 € | ||
| 2mg | 51.00 € | ||
| 5mg | 83.00 € | ||
| 10mg | 124.00 € | ||
| 25mg | 224.00 € | ||
| 50mg | 361.00 € | ||
| 100mg | 577.00 € | ||
| 1mL*10mM (DMSO) | 85.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Histamine Phosphate
CAS:51-74-1
Histamine Phosphate (Histamine acid phosphate) acts directly on the blood vessels to dilate arteries and …
Formula:
C5H9N·2H3O4P
Purity:
100%
Color and Shape:
White Crystal Powder
Molecular weight:
307.14
Ref: TM-T6535
| 1g | 53.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
ACEPROMAZINE MALEATE
CAS:3598-37-6
ACEPROMAZINE MALEATE is a dopamine receptor antagonist
Formula:
C23H26N2O5S
Purity:
98.87% - 99.30%
Color and Shape:
Off White Or Yellow Crystalline Powder
Molecular weight:
442.53
Ref: TM-T7728
| 5mg | 48.00 € | ||
| 10mg | 74.00 € | ||
| 25mg | 96.00 € | ||
| 50mg | 115.00 € | ||
| 100mg | 167.00 € | ||
| 500mg | 412.00 € | ||
| 1mL*10mM (DMSO) | 58.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Tozadenant
CAS:870070-55-6
Tozadenant (SYN115) is an adenosine A2A receptor antagonist(Ki of 11.5 nM and 6 nM on …
Formula:
C19H26N4O4S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
406.5
Ref: TM-T7320
| 2mg | 37.00 € | ||
| 5mg | 56.00 € | ||
| 10mg | 93.00 € | ||
| 25mg | 157.00 € | ||
| 50mg | 263.00 € | ||
| 100mg | 378.00 € | ||
| 200mg | 543.00 € | ||
| 1mL*10mM (DMSO) | 62.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
L-745870 trihydrochloride
CAS:866021-03-6
L-745870 trihydrochloride is a highly potent and selective D4 dopamine receptor antagonist.
Formula:
C18H22Cl4N4
Purity:
97.52%
Color and Shape:
Solid
Molecular weight:
436.21
Ref: TM-T22904
| 1mg | 74.00 € | ||
| 2mg | 96.00 € | ||
| 5mg | 144.00 € | ||
| 10mg | 199.00 € | ||
| 25mg | 457.00 € | ||
| 50mg | 653.00 € | ||
| 100mg | 926.00 € | ||
| 500mg | 1,839.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Ramosetron
CAS:132036-88-5
Ramosetron is a serotonin 5-HT3 receptor antagonist for the treatment of nausea and vomiting.
Formula:
C17H17N3O
Purity:
98.98%
Color and Shape:
Solid
Molecular weight:
279.34
Ref: TM-T4562
| 10mg | 55.00 € | ||
| 25mg | 72.00 € | ||
| 50mg | 111.00 € | ||
| 100mg | 162.00 € | ||
| 200mg | 240.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Navarixin
CAS:473727-83-2
Navarixin (MK-7123)(SCH527123) is a novel, selective CXC chemokine receptor 2(CXCR2) antagonist that inhibits neutrophil activation …
Formula:
C21H23N3O5
Purity:
98% - 98.63%
Color and Shape:
Solid
Molecular weight:
397.42
Ref: TM-T7130
| 1mg | 40.00 € | ||
| 5mg | 83.00 € | ||
| 10mg | 119.00 € | ||
| 25mg | 207.00 € | ||
| 50mg | 310.00 € | ||
| 100mg | 458.00 € | ||
| 500mg | 1,005.00 € | ||
| 1mL*10mM (DMSO) | 93.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
4i
CAS:930478-88-9
4i (CHEMBL1269981) is a 5-HT3 receptor antagonist,It modulates the serotonergic system.
Formula:
C16H12ClN3O
Purity:
99.49%
Color and Shape:
Solid
Molecular weight:
297.74
Ref: TM-T8438
| 1mg | 84.00 € | ||
| 5mg | 168.00 € | ||
| 10mg | 248.00 € | ||
| 25mg | 408.00 € | ||
| 50mg | 574.00 € | ||
| 100mg | 776.00 € | ||
| 200mg | 1,029.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Neurokinin A(4-10) TFA(97559-35-8 free base)
Neurokinin A(4-10) TFA(97559-35-8 free base) is a tachykinin NK2 receptor agonist[1].
Formula:
C36H55F3N8O12S
Purity:
100%
Color and Shape:
Solid
Molecular weight:
880.93
Ref: TM-TP1385
| 1mg | 47.00 € | ||
| 5mg | 150.00 € | ||
| 10mg | 252.00 € | ||
| 25mg | 415.00 € | ||
| 50mg | 582.00 € | ||
| 100mg | 785.00 € | ||
| 200mg | 1,052.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
NPY 5RA972
CAS:439861-56-0
NPY 5RA972 is a neuropeptide Y Y5 receptor antagonist
Formula:
C21H25N3O2
Purity:
99.02%
Color and Shape:
Solid
Molecular weight:
351.44
Ref: TM-T23087
| 1mg | 46.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 135.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Alloxazine
CAS:490-59-5
Alloxazine (Isoalloxazine) is an A2 receptor antagonist, which is approximately 10-fold more selective for the …
Formula:
C10H6N4O2
Purity:
99.75%
Color and Shape:
Solid
Molecular weight:
214.18
Ref: TM-T22234
| 50mg | 36.00 € | ||
| 100mg | 51.00 € | ||
| 200mg | 72.00 € | ||
| 1mL*10mM (DMSO) | 45.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Litorin acetate(55749-97-8 Free base)
Litorin acetate, an amphibian bombesin peptide derivative, is an bombesin receptor agonist.
Formula:
C53H72N14O13S
Purity:
97.64%
Color and Shape:
Liquid
Molecular weight:
1145.29
Ref: TM-T20604L
| 1mg | 83.00 € | ||
| 5mg | 207.00 € | ||
| 10mg | 332.00 € | ||
| 25mg | 546.00 € | ||
| 50mg | 801.00 € | ||
| 100mg | 1,100.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Chlorprothixene
CAS:113-59-7
Chlorprothixene (Truxal) is a typical antipsychotic drug of the thioxanthene class, which was the first …
Formula:
C18H18ClNS
Purity:
98.77% - 99.69%
Color and Shape:
Pale Yellow Crystals Solid
Molecular weight:
315.86
Ref: TM-T0074
| 1g | 140.00 € | ||
| 100mg | 37.00 € | ||
| 200mg | 53.00 € | ||
| 500mg | 96.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
TC-G-1008
CAS:1621175-65-2
TC-G-1008 (GPR39-C3) is a GPR39 (zinc receptor) agonist (EC50 values are 0.4 and 0.8 nM …
Formula:
C18H19ClN6O2S
Purity:
97.37% - 99%
Color and Shape:
Solid
Molecular weight:
418.9
Ref: TM-T4648
| 1mg | 48.00 € | ||
| 2mg | 64.00 € | ||
| 5mg | 89.00 € | ||
| 10mg | 154.00 € | ||
| 25mg | 313.00 € | ||
| 50mg | 536.00 € | ||
| 100mg | 770.00 € | ||
| 500mg | 1,559.00 € | ||
| 1mL*10mM (DMSO) | 90.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Sevoflurane
CAS:28523-86-6
Sevoflurane (Fluoromethyl), a noncompetitive inhibitor of 5-HT3 receptor, acts as a low-soluble inhalation anesthetics.
Formula:
C4H3F7O
Purity:
99.78%
Color and Shape:
Less Oil Colorless Oil
Molecular weight:
200.05
Ref: TM-T22425
| 5mg | 50.00 € | ||
| 10mg | 74.00 € | ||
| 25mg | 115.00 € | ||
| 50mg | 162.00 € | ||
| 100mg | 234.00 € | ||
| 200mg | 350.00 € | ||
| 500mg | 588.00 € | ||
| 1mL*10mM (DMSO) | 59.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Neuropeptide FF acetate(99566-27-5 free base)
Neuropeptide FF acetate(99566-27-5 free base) (NPFF acetate) is an octapeptide belonging to the RF amide …
Formula:
C56H80N14O12
Purity:
98.03%
Color and Shape:
Solid
Molecular weight:
1141.32
Ref: TM-TP1074L
| 1mg | 142.00 € | ||
| 5mg | 310.00 € | ||
| 10mg | 463.00 € | ||
| 25mg | 757.00 € | ||
| 50mg | 1,054.00 € | ||
| 100mg | 1,417.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Felypressin
CAS:56-59-7
Felypressin, a Lypressin analog with a phenylalanine substitution, acts as a vasoconstrictor with less antidiuretic …
Formula:
C46H65N13O11S2
Purity:
99.65%
Color and Shape:
Solid
Molecular weight:
1040.22
Ref: TM-T2568
| 2mg | 37.00 € | ||
| 5mg | 54.00 € | ||
| 10mg | 78.00 € | ||
| 25mg | 114.00 € | ||
| 50mg | 169.00 € | ||
| 1mL*10mM (DMSO) | 93.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
MK-571 sodium
CAS:115103-85-0
MK-571 sodium, a CysLT1 antagonist and MRP2 inhibitor, obstructs drug efflux and hampers enterocyte phase-2 …
Formula:
C26H27ClN2O3S2·Na
Purity:
97% - 98.69%
Color and Shape:
Solid
Molecular weight:
537.07
Ref: TM-T3148
| 5mg | 51.00 € | ||
| 10mg | 83.00 € | ||
| 25mg | 170.00 € | ||
| 50mg | 295.00 € | ||
| 100mg | 440.00 € | ||
| 1mL*10mM (DMSO) | 69.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
NPS-2143 hydrochloride
CAS:324523-20-8
NPS-2143 hydrochloride (NPS-2143 HCL) is a selective potent calcium ion-sensing receptor antagonist.
Formula:
C24H25ClN2O2·HCl
Purity:
99.22% - 99.38%
Color and Shape:
Solid
Molecular weight:
445.38
Ref: TM-T4967
| 1mg | 45.00 € | ||
| 2mg | 59.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 128.00 € | ||
| 25mg | 216.00 € | ||
| 50mg | 337.00 € | ||
| 100mg | 493.00 € | ||
| 1mL*10mM (DMSO) | 90.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Pirenperone
CAS:75444-65-4
Pirenperone is a putative 5-HT2 receptor antagonist with the central antiserotonergic and antidopaminergic action.
Formula:
C23H24FN3O2
Purity:
99.20%
Color and Shape:
Solid
Molecular weight:
393.45
Ref: TM-T2599
| 1mg | 40.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 113.00 € | ||
| 25mg | 225.00 € | ||
| 50mg | 355.00 € | ||
| 100mg | 524.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
