G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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PF-610355
CAS:862541-45-5
PF-610355 is a long-acting and potent β2-adrenergic receptor agonist (EC50: 0.26 nM).PF-610355 can be used …
Formula:
C34H39N3O6S
Purity:
99.90%
Color and Shape:
Solid
Molecular weight:
617.76
Ref: TM-T16509
| 1mg | 627.00 € | ||
| 5mg | 1,347.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Escitalopram
CAS:128196-01-0
Escitalopram (Seroplex), a serotonin inhibitor for depression, curbs alcohol intake and is favored over tricyclics …
Formula:
C20H21FN2O
Purity:
99.82%
Color and Shape:
White Or White Crystalline Powder
Molecular weight:
324.39
Ref: TM-T0185
| 2mg | 35.00 € | ||
| 5mg | 47.00 € | ||
| 10mg | 61.00 € | ||
| 25mg | 110.00 € | ||
| 50mg | 168.00 € | ||
| 100mg | 256.00 € | ||
| 200mg | 372.00 € | ||
| 1mL*10mM (DMSO) | 50.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
YE 120
CAS:383124-82-1
YE 120 is a GPR35 agonist.
Formula:
C16H9Cl2N3O
Purity:
99.67%
Color and Shape:
Solid
Molecular weight:
330.17
Ref: TM-T23542
| 1mg | 95.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
Diclofensine
CAS:67165-56-4
Diclofensine (Ro 8-4650) inhibits the uptake of serotonin, noradrenaline and dopamine.
Formula:
C17H17Cl2NO
Purity:
98.08%
Color and Shape:
Solid
Molecular weight:
322.23
Ref: TM-T7341
| 5mg | 52.00 € | ||
| 10mg | 87.00 € | ||
| 25mg | 142.00 € | ||
| 50mg | 207.00 € | ||
| 100mg | 312.00 € |
Estimated delivery in United States, on Thursday 2 Jan 2025
Paroxetine hydrochloride hemihydrate
CAS:110429-35-1
Paroxetine hydrochloride hemihydrate (Paxil) is an effective and selective serotonin reuptake inhibitor (SSRI).
Formula:
C38H44Cl2F2N2O7
Purity:
100%
Color and Shape:
Solid
Molecular weight:
749.67
Ref: TM-T1636L
| 10mg | 35.00 € | ||
| 25mg | 49.00 € | ||
| 50mg | 69.00 € | ||
| 100mg | 90.00 € | ||
| 500mg | 154.00 € | ||
| 1mL*10mM (DMSO) | 45.00 € |
Estimated delivery in United States, on Thursday 2 Jan 2025
XL413
CAS:1169558-38-6
XL-413 is an oral CDC7 kinase inhibitor, potentially blocking DNA replication, mitosis, and cancer cell …
Formula:
C14H12ClN3O2
Purity:
100% - 99.38%
Color and Shape:
Solid
Molecular weight:
289.72
Ref: TM-T3352
| 1mg | 52.00 € | ||
| 5mg | 114.00 € | ||
| 10mg | 157.00 € | ||
| 25mg | 276.00 € | ||
| 50mg | 461.00 € | ||
| 100mg | 643.00 € |
Estimated delivery in United States, on Thursday 2 Jan 2025
(RS)-ICI-118551 Hydrochloride
CAS:1217094-53-5
ICI-118551 Hydrochloride (ICI-118,551) is a highly selective β2-adrenergic receptor antagonist with Ki values of 0.7, …
Formula:
C17H27NO2·HCl
Purity:
98.02%
Color and Shape:
Solid
Molecular weight:
313.86
Ref: TM-T6860
| 1mg | 183.00 € | ||
| 5mg | 452.00 € | ||
| 10mg | 647.00 € | ||
| 25mg | 1,009.00 € | ||
| 50mg | 1,389.00 € | ||
| 100mg | 1,837.00 € |
Estimated delivery in United States, on Thursday 2 Jan 2025
Ciproxifan
CAS:184025-18-1
Ciproxifan (FUB-359) is a highly effective and specific histamin H3-receptor antagonist (IC50: 9.2 nM).
Formula:
C16H18N2O2
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
270.33
Ref: TM-T6164
| 1mg | 43.00 € | ||
| 2mg | 54.00 € | ||
| 5mg | 80.00 € | ||
| 10mg | 109.00 € | ||
| 25mg | 220.00 € | ||
| 50mg | 393.00 € |
Estimated delivery in United States, on Thursday 2 Jan 2025
Penbutolol sulfate
CAS:38363-32-5
Penbutolol sulfate ((-)-Terbuclomine) is able to bind to both β2-adrenergic receptor and β1-adrenergic receptor, thus …
Formula:
C18H29NO2H2O4S
Purity:
100%
Color and Shape:
Solid
Molecular weight:
340.47
Ref: TM-T12402
| 10mg | 41.00 € | ||
| 50mg | To inquire | ||
| 100mg | To inquire |
Estimated delivery in United States, on Thursday 2 Jan 2025
MK-5046
CAS:1022152-70-0
MK-5046 is a novel BRS-3 agonist, binding to BRS-3 with high affinity (mouse Ki = …
Formula:
C20H18F6N4O
Purity:
98.56%
Color and Shape:
Solid
Molecular weight:
444.37
Ref: TM-T2126
| 1mg | 82.00 € | ||
| 5mg | 172.00 € | ||
| 10mg | 246.00 € |
Estimated delivery in United States, on Thursday 2 Jan 2025
Palosuran
CAS:540769-28-6
Palosuran (ACT-058362) (ACT-058362) is a new potent and specific antagonist of the human UT receptor.
Formula:
C25H30N4O2
Purity:
98.46%
Color and Shape:
Solid
Molecular weight:
418.53
Ref: TM-T2058
| 1mg | 35.00 € | ||
| 2mg | 46.00 € | ||
| 5mg | 73.00 € | ||
| 10mg | 105.00 € | ||
| 25mg | 230.00 € | ||
| 50mg | 384.00 € | ||
| 100mg | 630.00 € | ||
| 200mg | 886.00 € | ||
| 1mL*10mM (DMSO) | 201.00 € |
Estimated delivery in United States, on Thursday 2 Jan 2025
SB 271046 hydrochloride
CAS:209481-24-3
SB 271046 hydrochloride (SB 271046A) is selective, orally active 5-HT6 antagonist and is >200-fold selective …
Formula:
C20H22ClN3O3S2·HCl
Purity:
99.57%
Color and Shape:
Solid
Molecular weight:
488.45
Ref: TM-T4118
| 5mg | 37.00 € | ||
| 10mg | 62.00 € | ||
| 25mg | 126.00 € | ||
| 50mg | 232.00 € | ||
| 100mg | 345.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Thursday 2 Jan 2025
5-Methyltryptamine hydrochloride
CAS:1010-95-3
5-Methyltryptamine hydrochloride is a high-affinity 5-HT1C receptor ligand and a partial agonist of 5-HT. 5-Methyltryptamine …
Formula:
C11H15ClN2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
210.703
Ref: TM-T19813
| 5mg | 36.00 € | ||
| 10mg | 53.00 € | ||
| 25mg | 78.00 € | ||
| 50mg | 101.00 € | ||
| 100mg | 149.00 € | ||
| 200mg | 212.00 € |
Estimated delivery in United States, on Thursday 2 Jan 2025
Lodoxamide tromethamine
CAS:63610-09-3
Lodoxamide tromethamine is a mast cell stabilizer with anti-allergic properties and can be used in …
Formula:
C19H28ClN5O12
Purity:
99.58%
Color and Shape:
Solid
Molecular weight:
553.91
Ref: TM-T15772
| 5mg | 46.00 € | ||
| 10mg | 59.00 € | ||
| 25mg | 93.00 € | ||
| 50mg | 109.00 € | ||
| 100mg | 183.00 € | ||
| 200mg | 273.00 € | ||
| 1mL*10mM (DMSO) | 53.00 € |
Estimated delivery in United States, on Thursday 2 Jan 2025
Pardoprunox
CAS:269718-84-5
Pardoprunox (SLV-308) is a partial dopamine D2 agonist and noradrenergic agonist with serotonin 5-HT1A agonist …
Formula:
C12H15N3O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
233.27
Ref: TM-T1769
| 25mg | 823.00 € |
Estimated delivery in United States, on Thursday 2 Jan 2025
D-Kynurenine
CAS:13441-51-5
D-Kynurenine, ZINC901103, metabolizes from D-tryptophan, activates AhR, changes epithelium to mesenchyme, and tests for D-amino …
Formula:
C10H12N2O3
Purity:
97.08%
Color and Shape:
Solid
Molecular weight:
208.21
Ref: TM-T10938
| 25mg | 52.00 € | ||
| 50mg | 89.00 € | ||
| 100mg | 129.00 € | ||
| 200mg | 183.00 € |
Estimated delivery in United States, on Thursday 2 Jan 2025
NDT 9513727
CAS:439571-48-9
Complement C5a receptor (C5aR) antagonist
Formula:
C36H35N3O4
Purity:
Min. 95%
Molecular weight:
573.68 g/mol
Ref: 3D-BN162458
| 1mg | 213.00 € | ||
| 2mg | 341.00 € | ||
| 5mg | 498.00 € | ||
| 10mg | 746.00 € | ||
| 25mg | 1,276.00 € |
Estimated delivery in United States, on Tuesday 7 Jan 2025
LY 344864
CAS:186544-26-3
LY 344864, a specifc receptor agonist, is an affinity of 6 nM (Ki) at the …
Formula:
C21H22FN3O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
351.42
Ref: TM-T2344
| 2mg | 40.00 € | ||
| 5mg | 59.00 € | ||
| 10mg | 96.00 € | ||
| 25mg | 163.00 € | ||
| 50mg | 290.00 € | ||
| 100mg | 516.00 € | ||
| 1mL*10mM (DMSO) | 67.00 € |
Estimated delivery in United States, on Tuesday 7 Jan 2025
BRL 44408 Maleate Salt
CAS:681806-46-2
BRL 44408 Maleate is an α2A-adrenoceptor antagonist with antidepressant and analgesic activity.
Formula:
C17H21N3O4
Color and Shape:
Solid
Molecular weight:
331.37
Ref: TM-T26904
| 1mg | 74.00 € | ||
| 5mg | 162.00 € | ||
| 10mg | 279.00 € | ||
| 25mg | 462.00 € | ||
| 50mg | 673.00 € | ||
| 100mg | 991.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
CRTh2 antagonist 2
CAS:780763-95-3
CRTh2 antagonist 2 is a selective and potent CRTH2 antagonist, IC50≤10 nM. CRTh2 antagonist 2 …
Formula:
C26H23ClN4O3
Purity:
99.53%
Color and Shape:
Solid
Molecular weight:
474.94
Ref: TM-T10889
| 1mg | 106.00 € | ||
| 5mg | 202.00 € | ||
| 10mg | 328.00 € | ||
| 25mg | 524.00 € | ||
| 50mg | 716.00 € | ||
| 100mg | 920.00 € | ||
| 500mg | 1,845.00 € | ||
| 1mL*10mM (DMSO) | 273.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
