G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Rec 15/2615 dihydrochloride
CAS:173059-17-1
Rec 15/2615 dihydrochloride is an antagonist of α1B-adrenergic receptor.
Formula:
C26H35Cl2N5O5
Purity:
98.97% - 99.81%
Color and Shape:
Solid
Molecular weight:
568.49
Ref: TM-T23230
| 1mg | 82.00 € | ||
| 5mg | 172.00 € | ||
| 10mg | 254.00 € | ||
| 25mg | 419.00 € | ||
| 50mg | 589.00 € | ||
| 100mg | 796.00 € | ||
| 500mg | To inquire |
Estimated delivery in United States, on Tuesday 26 Nov 2024
SB 611812
CAS:345892-71-9
SB 611812 is an antagonist of urotensin-II (UT) and can be used in studies about …
Formula:
C17H16Cl3F3N2O3S
Purity:
99.34%
Color and Shape:
Solid
Molecular weight:
491.74
Ref: TM-T23323
| 1mg | 45.00 € | ||
| 1ml | 96.00 € | ||
| 5mg | 89.00 € | ||
| 10mg | 143.00 € | ||
| 25mg | 300.00 € | ||
| 50mg | 434.00 € | ||
| 100mg | 609.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
Felypressin acetate
CAS:914453-97-7
Felypressin acetate (PLV-2) is an agonist of vasopressin 1 and acts on all arginine vasopressin …
Formula:
C48H69N13O13S2
Purity:
97.06%
Color and Shape:
Solid
Molecular weight:
1100.27
Ref: TM-T2568L
| 5mg | 46.00 € | ||
| 10mg | 69.00 € | ||
| 25mg | 123.00 € | ||
| 50mg | 183.00 € | ||
| 100mg | 291.00 € | ||
| 200mg | 435.00 € | ||
| 500mg | 700.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
Remogliflozin etabonate
CAS:442201-24-3
Remogliflozin etabonate is a prodrug SGLT2 inhibitor; Ki for hSGLT2: 1.95μM, rSGLT2: 2.14μM, rSGLT1: 8.57μM, …
Formula:
C26H38N2O9
Purity:
99%
Color and Shape:
Solid
Molecular weight:
522.59
Ref: TM-T34286
| 1mg | 37.00 € | ||
| 1ml | 91.00 € | ||
| 2mg | 51.00 € | ||
| 5mg | 89.00 € | ||
| 10mg | 144.00 € | ||
| 25mg | 263.00 € | ||
| 50mg | 404.00 € | ||
| 100mg | 562.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
SB-209670
CAS:157659-79-5
SB-209670 is a selective endothelin receptor antagonist that inhibits the activity of ET(B) receptors in …
Formula:
C29H28O9
Purity:
97.39% - 99.24%
Color and Shape:
Solid
Molecular weight:
520.53
Ref: TM-T34541
| 1mg | 325.00 € | ||
| 1ml | 791.00 € | ||
| 5mg | 769.00 € | ||
| 10mg | 1,054.00 € | ||
| 25mg | 1,476.00 € | ||
| 50mg | 1,846.00 € | ||
| 100mg | 2,320.00 € | ||
| 500mg | 4,577.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
Neldazosin
CAS:109713-79-3
Neldazosin is used as a potent α1-adrenoceptor antagonist.
Formula:
C18H25N5O4
Purity:
100% - 99.87%
Color and Shape:
Solid
Molecular weight:
375.42
Ref: TM-T61535
| 1mg | 196.00 € | ||
| 1ml | 520.00 € | ||
| 5mg | 496.00 € | ||
| 10mg | 711.00 € | ||
| 25mg | 1,096.00 € | ||
| 50mg | 1,476.00 € | ||
| 100mg | 2,004.00 € | ||
| 500mg | 3,999.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
Rolapitant
CAS:552292-08-7
Rolapitant Hydrochloride is an oral NK1-receptor blocker that prevents nausea and has a fast onset …
Formula:
C25H26F6N2O2
Purity:
98.34%
Color and Shape:
Solid
Molecular weight:
500.48
Ref: TM-T3716
| 1mg | 51.00 € | ||
| 1ml | 91.00 € | ||
| 2mg | 65.00 € | ||
| 5mg | 92.00 € | ||
| 10mg | 121.00 € | ||
| 25mg | 184.00 € | ||
| 50mg | 305.00 € | ||
| 100mg | 456.00 € | ||
| 500mg | 1,013.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
SLV-310
CAS:264869-71-8
SLV-310 is a D2 receptor antagonist and 5-HT reuptake receptor inhibitor for the study of …
Formula:
C25H24FN3O2
Purity:
98.91%
Color and Shape:
Solid
Molecular weight:
417.48
Ref: TM-T28809
| 1mg | 278.00 € | ||
| 5mg | 684.00 € | ||
| 10mg | 935.00 € | ||
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
L-168049
CAS:191034-25-0
L-168049: Human glucagon receptor antagonist, IC50 - 3.7 nM human, 63 nM murine, 60 nM …
Formula:
C24H20BrClN2O
Purity:
100%
Color and Shape:
Solid
Molecular weight:
467.79
Ref: TM-T22893
| 1mg | 52.00 € | ||
| 1ml | 123.00 € | ||
| 5mg | 110.00 € | ||
| 10mg | 176.00 € | ||
| 25mg | 369.00 € | ||
| 50mg | 551.00 € | ||
| 100mg | 783.00 € | ||
| 500mg | 1,613.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
SC 51089
CAS:146033-02-5
SC 51089 is a somatic PGE2 antagonist with anti-injurious activity and may rescue memory loss.
Formula:
C22H20Cl2N4O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
459.33
Ref: TM-T23331
| 1mg | 278.00 € | ||
| 5mg | 684.00 € | ||
| 10mg | 935.00 € | ||
| 25mg | 1,410.00 € | ||
| 50mg | 1,845.00 € | ||
| 100mg | 2,329.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
PGD2-IN-1
CAS:885066-67-1
PGD2-IN-1 (PGD2-inhibitor) is an effective DP receptor antagonist (IC50:0.3 nM), a compound that can inhibit …
Formula:
C23H23Cl2N3O3
Purity:
99%
Color and Shape:
Solid
Molecular weight:
460.35
Ref: TM-T4624
| 1mg | 69.00 € | ||
| 1ml | 167.00 € | ||
| 5mg | 156.00 € | ||
| 10mg | 255.00 € | ||
| 25mg | 428.00 € | ||
| 50mg | 631.00 € | ||
| 100mg | 895.00 € | ||
| 500mg | 1,791.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
Arbutamine
CAS:128470-16-6
Arbutamine (GP 21213) is a β-adrenoceptor agonist with alpha-1-sympathomimetic activity that can be used to …
Formula:
C18H23NO4
Purity:
95.06%
Color and Shape:
Solid
Molecular weight:
317.38
Ref: TM-T10364
| 1mg | 378.00 € | ||
| 5mg | 905.00 € | ||
| 10mg | 1,122.00 € | ||
| 25mg | 1,502.00 € | ||
| 50mg | 1,846.00 € | ||
| 100mg | 2,331.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
(Iso)-FK-480
CAS:167820-10-2
(Iso)-FK-480 is a novel orally available cholecystokinin A (CCK-A) antagonist for investigational treatment of chronic …
Formula:
C26H19FN4O2
Purity:
99.68%
Color and Shape:
Solid
Molecular weight:
438.45
Ref: TM-T10055
| 25mg | 1,410.00 € | ||
| 50mg | 1,845.00 € | ||
| 100mg | 2,329.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
ANR 94
CAS:634924-89-3
ANR94 is a potent hAA2AR antagonist (Ki 46 nM) with potential for Parkinson's research.
Formula:
C9H13N5O
Purity:
98.21%
Color and Shape:
Solid
Molecular weight:
207.23
Ref: TM-T22031
| 1ml | 61.00 € | ||
| 2mg | 41.00 € | ||
| 5mg | 62.00 € | ||
| 10mg | 93.00 € | ||
| 25mg | 182.00 € | ||
| 50mg | 318.00 € | ||
| 100mg | 449.00 € | ||
| 200mg | 631.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
BMY-25271
CAS:78441-82-4
BMY-25271 is an antagonist of histamine H2 receptor.
Formula:
C12H19N5O2S2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
329.44
Ref: TM-T10575
| 25mg | 1,410.00 € | ||
| 50mg | 1,845.00 € | ||
| 100mg | 2,329.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
LY377604
CAS:204592-94-9
LY377604 is a human β3-adrenergic receptor agonist (EC50: 2.4 nM) and β1/2-adrenergic receptor antagonist for …
Formula:
C31H32N4O4
Purity:
100% - 99.72%
Color and Shape:
Solid
Molecular weight:
524.61
Ref: TM-T15819
| 1mg | 123.00 € | ||
| 5mg | 298.00 € | ||
| 10mg | 441.00 € | ||
| 25mg | 722.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
Itriglumide
CAS:201605-51-8
Itriglumide, a CCK2 receptor antagonist, is used potentially for the treatment of peptic ulcers, dyspepsia, …
Formula:
C33H38N2O4
Purity:
99.95%
Color and Shape:
Solid
Molecular weight:
526.67
Ref: TM-T27640
| 1mg | 272.00 € | ||
| 2mg | 405.00 € | ||
| 5mg | 670.00 € | ||
| 10mg | 915.00 € | ||
| 25mg | 1,409.00 € | ||
| 50mg | 1,836.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
AZD1940
CAS:881413-29-2
AZD1940 (UNII-0J0035E9FT) is a high affinity CB(1)/CB(2) receptor agonist of the cannabinoid with oral activity. …
Formula:
C20H29F2N3O2S
Purity:
99.43%
Color and Shape:
Solid
Molecular weight:
413.52
Ref: TM-T30252
| 1mg | 128.00 € | ||
| 1ml | 343.00 € | ||
| 5mg | 305.00 € | ||
| 10mg | 525.00 € | ||
| 25mg | 828.00 € | ||
| 50mg | 1,143.00 € | ||
| 100mg | 1,550.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
MRS1220
CAS:183721-15-5
MRS1220, a selective and potent antagonist for the human A3 adenosine receptor (hA3AR) with a …
Formula:
C21H14ClN5O2
Purity:
96.59%
Color and Shape:
Solid
Molecular weight:
403.82
Ref: TM-T23016
| 1mg | 49.00 € | ||
| 5mg | 114.00 € | ||
| 10mg | 174.00 € | ||
| 25mg | 297.00 € | ||
| 50mg | 428.00 € | ||
| 100mg | 603.00 € | ||
| 500mg | To inquire |
Estimated delivery in United States, on Tuesday 26 Nov 2024
PD 144418
CAS:154130-99-1
PD 144418 displays potential antipsychotic activity.
Formula:
C18H22N2O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
282.38
Ref: TM-T16445
| 25mg | 682.00 € | ||
| 50mg | 887.00 € | ||
| 100mg | 1,338.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
