G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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DBIBB
CAS:1569309-92-7
DBIBB: non-lipid LPA2 receptor agonist, treats acute radiation syndrome, aids in organic synthesis/drug research.
Formula:
C23H20N2O6S
Purity:
97.18% - 97.26%
Color and Shape:
Solid
Molecular weight:
452.48
Ref: TM-T22070
| 1mg | 41.00 € | ||
| 5mg | 92.00 € | ||
| 10mg | 131.00 € | ||
| 25mg | 258.00 € | ||
| 50mg | 370.00 € | ||
| 100mg | 543.00 € | ||
| 500mg | 1,089.00 € | ||
| 1mL*10mM (DMSO) | 92.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
AVN-322
CAS:1194574-68-9
AVN-322 is a 5-HT6 receptor antagonist. 5-HT6R antagonists improves cognition in animal models of cognitive …
Formula:
C17H20ClN5O2S
Purity:
98.83%
Color and Shape:
Solid
Molecular weight:
393.89
Ref: TM-T26691
| 1mg | 276.00 € | ||
| 5mg | 679.00 € | ||
| 10mg | 928.00 € | ||
| 25mg | 1,410.00 € | ||
| 50mg | 1,852.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
SB-215505
CAS:162100-15-4
SB215505: potent 5-HT2B/2C blocker, enhances rat wakefulness/motor activity. (pKi: 5-HT2B - 8.3, 5-HT2C - 7.66, …
Formula:
C19H16ClN3O
Purity:
98.33%
Color and Shape:
Solid
Molecular weight:
337.8
Ref: TM-T28680
| 1mg | 209.00 € | ||
| 5mg | 521.00 € | ||
| 10mg | 726.00 € | ||
| 25mg | 1,081.00 € | ||
| 50mg | 1,493.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Oxyfedrine L-form HCl
CAS:16777-42-7
Oxyfedrine L-form HCl (Ildamen) is a partial agonist at beta-adrenergic receptors and acts as a …
Formula:
C19H24ClNO3
Purity:
98.66%
Color and Shape:
Solid
Molecular weight:
349.85
Ref: TM-T24579
| 1mg | 95.00 € | ||
| 5mg | 184.00 € | ||
| 10mg | 322.00 € | ||
| 25mg | 500.00 € | ||
| 50mg | 722.00 € | ||
| 100mg | 922.00 € | ||
| 1mL*10mM (DMSO) | 226.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
WAY-260022
CAS:850692-43-2
WAY-260022 is the norepinephrine transporter inhibitor.
Formula:
C21H31F3N2O2
Purity:
98.65% - 99.06%
Color and Shape:
Solid
Molecular weight:
400.48
Ref: TM-T23711
| 1mg | 273.00 € | ||
| 2mg | 407.00 € | ||
| 5mg | 673.00 € | ||
| 10mg | 920.00 € | ||
| 25mg | 1,415.00 € | ||
| 50mg | 1,832.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
MK 1903
CAS:1268882-43-4
MK 1903 is a strong, selective HCA2/GPR109A agonist, reducing cAMP in CHO cells with EC50 …
Formula:
C8H8N2O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
164.16
Ref: TM-T22986
| 1mg | 49.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 142.00 € | ||
| 25mg | 244.00 € | ||
| 50mg | 342.00 € | ||
| 100mg | 481.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Opigolix
CAS:912587-25-8
Opigolix is a Gonadotropin-releasing hormone receptor antagonist.
Formula:
C25H19F3N4O5S
Purity:
98.07% - 99.54%
Color and Shape:
Solid
Molecular weight:
544.5
Ref: TM-T17301
| 1mg | 273.00 € | ||
| 5mg | 673.00 € | ||
| 10mg | 930.00 € | ||
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,599.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
MrgprX2 antagonist-8
CAS:2768216-96-0
MrgprX2 antagonist-8 is an MrgprX2 antagonist that can be used to study inflammatory diseases.
Formula:
C24H24ClF3N4O3S
Purity:
98.87%
Color and Shape:
Liquid
Molecular weight:
540.99
Ref: TM-T63812
| 1mg | 100.00 € | ||
| 5mg | 240.00 € | ||
| 10mg | 344.00 € | ||
| 25mg | 564.00 € | ||
| 50mg | 745.00 € | ||
| 100mg | 992.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
LY2881835
CAS:1292290-38-0
LY2881835 is a potent and selective GPR40 agonist.
Formula:
C33H33NO3
Purity:
97.65% - 97.65%
Color and Shape:
Solid
Molecular weight:
491.62
Ref: TM-T27937
| 1mg | 274.00 € | ||
| 5mg | 673.00 € | ||
| 10mg | 920.00 € | ||
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Indanidine
CAS:85392-79-6
Indanidine is a highly selective and potent α-adrenergic agonist with antihypertensive activity.Indanidine is an α-adrenergic …
Formula:
C11H13N5
Purity:
100%
Color and Shape:
Solid
Molecular weight:
215.25
Ref: TM-T11651
| 1mg | 650.00 € | ||
| 5mg | 1,671.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
CB2 modulator 1
CAS:666261-80-9
CB2 modulator 1 is a potent CB2 modulator. It can be used for the research …
Formula:
C18H19F3N4O2
Purity:
99.02%
Color and Shape:
Solid
Molecular weight:
380.36
Ref: TM-T10696
| 1mg | 35.00 € | ||
| 5mg | 55.00 € | ||
| 10mg | 78.00 € | ||
| 25mg | 112.00 € | ||
| 50mg | 164.00 € | ||
| 100mg | To inquire | ||
| 1mL*10mM (DMSO) | 64.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
L 651896
CAS:99134-29-9
L 651896 is an inhibitor of 5-lipoxygenase.
Formula:
C18H18O3
Purity:
95.87% - 99.70%
Color and Shape:
Solid
Molecular weight:
282.33
Ref: TM-T24306
| 1mg | 311.00 € | ||
| 5mg | 747.00 € | ||
| 10mg | 1,059.00 € | ||
| 25mg | 1,549.00 € | ||
| 50mg | 2,127.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
CP-66948
CAS:101189-47-3
CP-66948 is a potent histamine H2 receptor antagonist with inhibitory effect on gastric acid secretion …
Formula:
C13H20N6S
Purity:
99.14%
Color and Shape:
Solid
Molecular weight:
292.4
Ref: TM-T15005
| 1mg | 654.00 € | ||
| 5mg | 1,672.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
![N-[(4-Aminophenyl)methyl]adenosine](https://static.cymitquimica.com/products/TM/thumb/T16166.jpg)
N-[(4-Aminophenyl)methyl]adenosine
CAS:95523-13-0
N-[(4-Aminophenyl)methyl]adenosine is an adenosine receptor inhibitor (Ki: 29 nM for Rat ecto-5′-Nucleotidase).
Formula:
C17H20N6O4
Purity:
98.75%
Color and Shape:
Solid
Molecular weight:
372.38
Ref: TM-T16166
| 1mg | 90.00 € | ||
| 5mg | 184.00 € | ||
| 10mg | 276.00 € | ||
| 25mg | 546.00 € | ||
| 50mg | 865.00 € | ||
| 100mg | 1,395.00 € | ||
| 1mL*10mM (DMSO) | 235.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Fananserin
CAS:127625-29-0
Fananserin: Oral 5-HT2A antagonist (Ki=0.37 nM, rat), blocks human D4 receptor (Ki=2.93 nM).
Formula:
C23H24FN3O2S
Purity:
99.78%
Color and Shape:
Solid
Molecular weight:
425.52
Ref: TM-T15270
| 2mg | 41.00 € | ||
| 5mg | 55.00 € | ||
| 10mg | 79.00 € | ||
| 25mg | 113.00 € | ||
| 50mg | 171.00 € | ||
| 100mg | 243.00 € | ||
| 200mg | 359.00 € | ||
| 1mL*10mM (DMSO) | 60.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
AMG-009
CAS:1027847-67-1
AMG-009 is a prostaglandin D2 antagonist. For CRTH2 and DP receptors, the IC50s are 3 …
Formula:
C26H26Cl2N2O7S
Purity:
97.88%
Color and Shape:
Solid
Molecular weight:
581.47
Ref: TM-T14211
| 1mg | 48.00 € | ||
| 5mg | 89.00 € | ||
| 10mg | 129.00 € | ||
| 25mg | 208.00 € | ||
| 50mg | 366.00 € | ||
| 100mg | 623.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Neurokinin antagonist 1
CAS:214487-45-3
Neurokinin antagonist 1 is a potent is a neuropeptide antagonist that can be used to …
Formula:
C38H40N4O3
Purity:
100%
Color and Shape:
Solid
Molecular weight:
600.75
Ref: TM-T10056
| 1mg | 650.00 € | ||
| 5mg | 1,678.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
RS-601
CAS:207987-59-5
RS-601 is a potent dual leukotriene D4/thromboxane A2 inhibitor that inhibits antigen-induced airway hyperresponsiveness (AHR) …
Formula:
C22H23F6NO4S
Purity:
99.31%
Color and Shape:
Solid
Molecular weight:
511.48
Ref: TM-T12771
| 1mg | 650.00 € | ||
| 5mg | 1,682.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
PAF-AN-1
CAS:115621-84-6
PAF-AN-1 is a novel potent platelet-activating factor receptor (PAF) antagonist involved in the study of …
Formula:
C28H28N2O3
Purity:
98.06%
Color and Shape:
Solid
Molecular weight:
440.53
Ref: TM-T14007
| 1mg | 650.00 € | ||
| 5mg | 1,678.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
GSK1521498 free base
CAS:1007573-18-3
GSK1521498 free base is a potent and selective antagonist of the μ-opioid receptor.
Formula:
C24H20F2N4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
402.44
Ref: TM-T11478L
| 25mg | 1,178.00 € | ||
| 50mg | 1,537.00 € | ||
| 100mg | 2,329.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
