G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Clozapine N-oxide
CAS:34233-69-7
Activates muscarinic GPCR DREADDs, which are unaffected by the endogenous ligand acetycholamine of the parent …
Formula:
C18H19ClN4O
Purity:
Min. 99 Area-%
Color and Shape:
Yellow Powder
Ref: 3D-FC20527
| 10mg | 238.00 € | ||
| 50mg | 697.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
Famotidine
CAS:76824-35-6
Famotidine is a selective histamine H2-receptor antagonist used in the treatment of gastric hypersecretory disorders. …
Formula:
C8H15N7O2S3
Purity:
Min. 98 Area-%
Color and Shape:
White Powder
Molecular weight:
337.45 g/mol
Ref: 3D-FF23221
| 100g | 186.00 € | ||
| 250g | 363.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
Leuprolide acetate
CAS:74381-53-6
Agonist of GnRH receptors
Formula:
C61H88N16O14
Purity:
Min. 95%
Color and Shape:
Powder
Molecular weight:
1,269.47 g/mol
Ref: 3D-FL24877
| 10mg | 172.00 € | ||
| 25mg | 232.00 € | ||
| 50mg | 349.00 € | ||
| 100mg | 491.00 € | ||
| 250mg | 925.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
Triptorelin acetate
CAS:140194-24-7
Gonadotropin-releasing hormone agonist
Formula:
C64H82N18O13•C2H4O2
Purity:
Min. 95 Area-%
Color and Shape:
Powder
Molecular weight:
1,371.5 g/mol
Ref: 3D-FT28582
| 10mg | 196.00 € | ||
| 25mg | 319.00 € | ||
| 50mg | 387.00 € | ||
| 100mg | 626.00 € | ||
| 250mg | 895.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
Etrasimod
CAS:1206123-37-6
Modulator of S1P receptor
Formula:
C26H26F3NO3
Purity:
Min. 98%
Color and Shape:
Off-White Powder
Molecular weight:
457.49 g/mol
Ref: 3D-FC158571
| 1mg | 172.00 € | ||
| 5mg | 364.00 € | ||
| 10mg | 453.00 € | ||
| 25mg | 647.00 € | ||
| 50mg | 770.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
Tolvaptan - Bio-X ™
Controlled ProductCAS:150683-30-0
Tolvaptan is a vasopressin receptor antagonist. It binds to the V2 receptor in the cytosol …
Formula:
C26H25ClN2O3
Purity:
Min. 95%
Color and Shape:
Powder
Molecular weight:
448.94 g/mol
Ref: 3D-BT164486
| 10mg | 142.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
Brimonidine-D-tartrate
CAS:70359-46-5
Brimonidine-D-tartrate is a synthetic, selective alpha 2-adrenergic receptor agonist that has been developed for use …
Formula:
C15H16BrN5O6
Color and Shape:
White Powder
Molecular weight:
442.22 g/mol
Ref: 3D-FB32174
| 1g | 310.00 € | ||
| 5g | 801.00 € | ||
| 10g | 1,160.00 € | ||
| 250mg | 155.00 € | ||
| 500mg | 225.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
Fingolimod - Bio-X ™
CAS:162359-55-9
Fingolimod is a sphingosine 1-phosphate receptor modulator that is used in the treatment of relapsing-remitting …
Formula:
C19H33NO2
Purity:
Min. 95%
Color and Shape:
Powder
Molecular weight:
307.47 g/mol
Ref: 3D-BF164460
| 100mg | 137.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
PD 149163 tetrahydrochloride hydrate
CAS:169528-11-4
Neurotensin 1 (NT1) receptor agonist
Formula:
C42H71N9O6·4HCl·xH2O
Purity:
Min. 95%
Color and Shape:
White To Light Brown Solid
Molecular weight:
943.91 g/mol
Ref: 3D-FP26774
| 10mg | 588.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
Nafarelin acetate
CAS:76932-56-4
Agonist of hypothalamic decapeptide GnRH; increases LH and FSH release
Formula:
C66H83N17O13·C2H4O2
Purity:
Min. 95%
Color and Shape:
White/Off-White Solid
Molecular weight:
1,382.52 g/mol
Ref: 3D-FN65097
| 10mg | 180.00 € | ||
| 50mg | 477.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
PTH hmn TFA-90%
CAS:68893-82-3
Parathyroid hormone receptor agonist
Formula:
C408H674N126O126S2•(C2HF3O2)x
Purity:
Min. 95%
Color and Shape:
Powder
Molecular weight:
9,424.62 g/mol
Ref: 3D-BP168671
| 1mg | 1,403.00 € | ||
| 5mg | 2,245.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
GLP-1 (9-36) amide trifluoroacetate
CAS:161748-29-4
GLP-1 (9-36) amide trifluoroacetate is a peptide that is cleaved from the larger molecule GLP-1. …
Formula:
C140H214N36O43
Purity:
Min. 95%
Color and Shape:
Powder
Molecular weight:
3,089.41 g/mol
Ref: 3D-FG109155
| 1mg | 542.00 € | ||
| 2mg | 827.00 € | ||
| 5mg | 1,167.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
Acipimox - Bio-X ™
CAS:51037-30-0
Acipimox is a niacin derivative that is used as a hypolipidemic agent. Acipimox prevents the …
Formula:
C6H6N2O3
Purity:
Min. 95%
Color and Shape:
Powder
Molecular weight:
154.12 g/mol
Ref: 3D-BA166874
| 100mg | 137.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
Ramelteon
Controlled ProductCAS:196597-26-9
Ramelteon is a melatonin receptor agonist that has been shown to be effective in the …
Formula:
C16H21NO2
Molecular weight:
259.34 g/mol
Ref: 3D-FR27673
| 5mg | 136.00 € | ||
| 10mg | 180.00 € | ||
| 50mg | 458.00 € | ||
| 100mg | 723.00 € | ||
| 250mg | 1,160.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
Exenatide acetate
CAS:141732-76-5
Agonist of glucagon-like peptide GLP1 which is used for treatment of type 2 diabetes mellitus. …
Formula:
C184H282N50O60S·C2H4O2
Purity:
Min. 95%
Color and Shape:
White Powder
Molecular weight:
4246.63
Ref: 3D-FE23212
| 5mg | 138.00 € | ||
| 10mg | 206.00 € | ||
| 25mg | 400.00 € | ||
| 50mg | 602.00 € | ||
| 100mg | 813.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
BNP-32 (human)
CAS:124584-08-3
Natriuretic; vasodilatory;diuretic; treats decompensated congestive hear failure
Formula:
C143H244N50O42S4
Purity:
Min. 95%
Color and Shape:
Powder
Molecular weight:
3,464.04 g/mol
Ref: 3D-FB110377
| 1mg | 645.00 € | ||
| 2mg | 934.00 € | ||
| 100µg | 367.00 € | ||
| 250µg | 487.00 € | ||
| 500µg | 544.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
FEMA 4774
CAS:1359963-68-0
Positive allosteric modulator of taste receptors T1R2 and T1R3 and enhancer of sucrose sweetness. In …
Formula:
C19H25N3O4
Purity:
Min. 95%
Color and Shape:
Slightly Yellow Powder
Molecular weight:
359.42 g/mol
Ref: 3D-BF168573
| 10mg | 329.00 € | ||
| 50mg | 922.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
Desmopressin acetate
CAS:62288-83-9
Synthetic analog of vasopressin; anti-diuretic; hemostatic
Formula:
C48H68N14O14S2
Purity:
Min. 95%
Color and Shape:
Powder
Molecular weight:
1128.44809
Ref: 3D-FD21366
| 25mg | 136.00 € | ||
| 50mg | 167.00 € | ||
| 100mg | 236.00 € | ||
| 250mg | 353.00 € | ||
| 500mg | 550.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
Mianserin HCl - Bio-X ™
Controlled ProductCAS:21535-47-7
Mianserin is a tetracyclic antidepressant drug that has antihistaminic and hypnosedative properties. It is used …
Formula:
C18H20N2•HCl
Purity:
Min. 95%
Color and Shape:
Powder
Molecular weight:
300.83 g/mol
Ref: 3D-BM166416
| 100mg | 137.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
Pranlukast
CAS:103177-37-3
Cysteinyl leukotriene receptor antagonist
Formula:
C27H23N5O4
Purity:
Min. 95%
Molecular weight:
481.5 g/mol
Ref: 3D-FP27120
| 25mg | 136.00 € | ||
| 50mg | 180.00 € | ||
| 100mg | 236.00 € | ||
| 250mg | 356.00 € | ||
| 500mg | 497.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
