G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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NDT 9513727
CAS:439571-48-9
Complement C5a receptor (C5aR) antagonist
Formula:
C36H35N3O4
Purity:
Min. 95%
Molecular weight:
573.68 g/mol
Ref: 3D-BN162458
| 1mg | 213.00 € | ||
| 2mg | 341.00 € | ||
| 5mg | 498.00 € | ||
| 10mg | 746.00 € | ||
| 25mg | 1,276.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
SB 218795
CAS:174635-53-1
SB 218795 is an effective and selective antagonist of NK3 with a Ki 13 nM …
Formula:
C25H20N2O3
Purity:
99.71%
Color and Shape:
Solid
Molecular weight:
396.44
Ref: TM-T23316
| 1mg | 52.00 € | ||
| 2mg | 67.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 167.00 € | ||
| 25mg | 325.00 € | ||
| 50mg | 530.00 € | ||
| 100mg | 737.00 € | ||
| 500mg | 1,560.00 € | ||
| 1mL*10mM (DMSO) | 115.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
SLF1081851
CAS:2763730-97-6
SLF1081851 is a Spns2 inhibitor. SLF1081851 inhibits S1P release with IC50 of 1.93 μM.
Formula:
C21H33N3O
Purity:
98.57%
Color and Shape:
Liquid
Molecular weight:
343.51
Ref: TM-T61112
| 1mg | 55.00 € | ||
| 5mg | 118.00 € | ||
| 10mg | 183.00 € | ||
| 25mg | 392.00 € | ||
| 50mg | 586.00 € | ||
| 100mg | 835.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
Bedoradrine
CAS:194785-19-8
Bedoradrine (MN-221) free base is a novel, highly selective β2-adrenoceptor agonist.Cost-effective and quality-assured.
Formula:
C24H32N2O5
Purity:
100%
Color and Shape:
Liquid
Molecular weight:
428.52
Ref: TM-T70047
| 1mg | 724.00 € | ||
| 5mg | 1,477.00 € | ||
| 25mg | 2,556.00 € | ||
| 50mg | 3,139.00 € | ||
| 100mg | 4,272.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
PF-03654764
CAS:935840-35-0
PF-03654764, an oral H3 receptor blocker, Ki: human 1.2 nM, rat 7.9 nM, used with …
Formula:
C20H28F2N2O
Purity:
100%
Color and Shape:
Liquid
Molecular weight:
350.45
Ref: TM-T61213
| 1mg | 305.00 € | ||
| 5mg | 736.00 € | ||
| 25mg | 1,483.00 € | ||
| 50mg | 2,009.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
Sergliflozin etabonate
CAS:408504-26-7
Sergliflozin etabonate (KGT-1251) is an inhibitor of SGLT2 and can be used in studies about …
Formula:
C23H28O9
Purity:
95.59%
Color and Shape:
Solid
Molecular weight:
448.46
Ref: TM-T28757
| 1mg | 182.00 € | ||
| 2mg | 272.00 € | ||
| 5mg | 418.00 € | ||
| 10mg | 612.00 € | ||
| 25mg | 922.00 € | ||
| 50mg | 1,281.00 € | ||
| 100mg | 1,762.00 € | ||
| 1mL*10mM (DMSO) | 486.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
5-HT6/7 antagonist 1
CAS:131999-28-5
5-HT6/7 antagonist 1 is a dual 5-HT6/7/2A and D2 receptor antagonist for the study of …
Formula:
C22H20FN3O3
Purity:
98.55% - 98.78%
Color and Shape:
Liquid
Molecular weight:
393.41
Ref: TM-T61807
| 1mg | 650.00 € | ||
| 5mg | 1,671.00 € | ||
| 25mg | 3,336.00 € | ||
| 50mg | 4,529.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
Alniditan
CAS:152317-89-0
Alniditan is a receptors agonist of 5-HT1B/1D in HEK 293 cells (IC50: 1.7 and 1.3 …
Formula:
C17H26N4O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
302.41
Ref: TM-T14190
| 25mg | 1,410.00 € | ||
| 50mg | 1,852.00 € | ||
| 100mg | 2,338.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
Napitane
CAS:148152-63-0
napitane (A 75200) is a novel catecholamine uptake inhibitor with inhibitory effects on α-adrenergic receptors …
Formula:
C22H25NO2
Purity:
100% - 99.91%
Color and Shape:
Solid
Molecular weight:
335.44
Ref: TM-T26363L
| 1mg | 313.00 € | ||
| 5mg | 741.00 € | ||
| 10mg | 1,074.00 € | ||
| 25mg | 1,644.00 € | ||
| 50mg | 2,210.00 € | ||
| 100mg | 2,878.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
PD 144418
CAS:154130-99-1
PD 144418 displays potential antipsychotic activity.
Formula:
C18H22N2O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
282.38
Ref: TM-T16445
| 25mg | 682.00 € | ||
| 50mg | 887.00 € | ||
| 100mg | 1,338.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
H2L5186303
CAS:139262-76-3
H2L5186303 is an LPA2 antagonist and can be used in studies about asthma treatment.
Formula:
C26H20N2O8
Purity:
97.23%
Color and Shape:
Solid
Molecular weight:
488.45
Ref: TM-T22835
| 1mg | 35.00 € | ||
| 5mg | 63.00 € | ||
| 10mg | 102.00 € | ||
| 25mg | 221.00 € | ||
| 50mg | 328.00 € | ||
| 100mg | 460.00 € | ||
| 500mg | 917.00 € | ||
| 1mL*10mM (DMSO) | 76.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
TD-5471 hydrochloride
CAS:530084-35-6
TD-5471 hydrochloride is a selective and potent long-acting human β2-adrenergic receptor agonist for the treatment …
Formula:
C32H32ClN3O4
Purity:
99.57%
Color and Shape:
Solid
Molecular weight:
558.07
Ref: TM-T13106
| 1mg | 650.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
5-HT3 antagonist 2
CAS:128199-93-9
5-HT3 antagonist 2 is an antagonist of 5-HT3 receptor.
Formula:
C18H21N3O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
295.38
Ref: TM-T12988
| 25mg | 1,410.00 € | ||
| 50mg | 1,852.00 € | ||
| 100mg | 2,338.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
GSK299115A
CAS:864082-35-9
GSK299115A (GSK-299115A) is a selective ROCK1 Inhibitor. GSK299115A exhibits IC50 of 8nM, 620nM, 560nM for …
Formula:
C20H16Cl2N4O2
Purity:
98.99%
Color and Shape:
Solid
Molecular weight:
415.27
Ref: TM-T27471
| 1mg | 319.00 € | ||
| 5mg | 772.00 € | ||
| 10mg | 1,072.00 € | ||
| 25mg | 1,594.00 € | ||
| 50mg | 2,144.00 € | ||
| 100mg | 2,817.00 € | ||
| 1mL*10mM (DMSO) | 944.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
GPR40/FFAR1 modulator 1
CAS:874755-26-7
GPR40/FFAR1 modulator 1 is a Gq-coupled free fatty acid receptor 1 (GPR40/FFAR1) agonist and allosteric …
Formula:
C21H19N5O3
Purity:
99.72%
Color and Shape:
Solid
Molecular weight:
389.41
Ref: TM-T11458
| 10mg | 51.00 € | ||
| 25mg | 84.00 € | ||
| 50mg | 124.00 € | ||
| 100mg | 182.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
CRTh2 antagonist 2
CAS:780763-95-3
CRTh2 antagonist 2 is a selective and potent CRTH2 antagonist, IC50≤10 nM. CRTh2 antagonist 2 …
Formula:
C26H23ClN4O3
Purity:
99.53%
Color and Shape:
Solid
Molecular weight:
474.94
Ref: TM-T10889
| 1mg | 106.00 € | ||
| 5mg | 202.00 € | ||
| 10mg | 328.00 € | ||
| 25mg | 524.00 € | ||
| 50mg | 716.00 € | ||
| 100mg | 920.00 € | ||
| 500mg | 1,845.00 € | ||
| 1mL*10mM (DMSO) | 273.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
TAK-875 Hemihydrate
CAS:1374598-80-7
TAK-875 Hemihydrate (Fasiglifam) is a selective GPR40 agonist with EC50 of 14 nM, 400-fold more …
Formula:
C29H32O7SH2O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
533.63
Ref: TM-T2351L
| 25mg | 621.00 € | ||
| 50mg | 810.00 € | ||
| 1mL*10mM (DMSO) | 304.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
CL 316243
CAS:138908-40-4
CL316243 is a highly potent selective agonist of β3-adrenoceptor.Cost-effective and quality-assured.
Formula:
C20H18ClNNa2O7
Purity:
98.00% - 99.68%
Color and Shape:
Solid
Molecular weight:
465.79
Ref: TM-T10830
| 1mg | 52.00 € | ||
| 5mg | 109.00 € | ||
| 10mg | 167.00 € | ||
| 25mg | 322.00 € | ||
| 50mg | 516.00 € | ||
| 100mg | 824.00 € | ||
| 500mg | 1,654.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
MM 77 dihydrochloride
CAS:159187-70-9
MM 77 dihydrochloride is an effecitve 5-HT1A receptor postsynaptic antagonist with anxiolytic-like activity.
Formula:
C19H29Cl2N3O3
Purity:
100.00%
Color and Shape:
Solid
Molecular weight:
418.36
Ref: TM-T23007
| 1mg | 85.00 € | ||
| 5mg | 155.00 € | ||
| 10mg | 212.00 € | ||
| 25mg | 467.00 € | ||
| 50mg | 678.00 € | ||
| 100mg | 926.00 € | ||
| 500mg | 1,850.00 € | ||
| 1mL*10mM (DMSO) | 278.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
Methiothepin maleate
CAS:19728-88-2
Methiothepin maleate (Metitepine) is a 5-HT1, 5-HT6, 5-HT7 serotonin receptor antagonist, which blocks serotonin autoreceptors.
Formula:
C24H28N2O4S2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
472.62
Ref: TM-T4375
| 10mg | 86.00 € | ||
| 25mg | 172.00 € | ||
| 50mg | 238.00 € | ||
| 100mg | 437.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
