G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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TAK-875 Hemihydrate
CAS:1374598-80-7
TAK-875 Hemihydrate (Fasiglifam) is a selective GPR40 agonist with EC50 of 14 nM, 400-fold more …
Formula:
C29H32O7SH2O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
533.63
Ref: TM-T2351L
| 25mg | 621.00 € | ||
| 50mg | 810.00 € | ||
| 1mL*10mM (DMSO) | 304.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
AZD1940
CAS:881413-29-2
AZD1940 (UNII-0J0035E9FT) is a high affinity CB(1)/CB(2) receptor agonist of the cannabinoid with oral activity. …
Formula:
C20H29F2N3O2S
Purity:
99.43%
Color and Shape:
Solid
Molecular weight:
413.52
Ref: TM-T30252
| 1mg | 128.00 € | ||
| 5mg | 305.00 € | ||
| 10mg | 525.00 € | ||
| 25mg | 828.00 € | ||
| 50mg | 1,143.00 € | ||
| 100mg | 1,550.00 € | ||
| 1mL*10mM (DMSO) | 343.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
MM 77 dihydrochloride
CAS:159187-70-9
MM 77 dihydrochloride is an effecitve 5-HT1A receptor postsynaptic antagonist with anxiolytic-like activity.
Formula:
C19H29Cl2N3O3
Purity:
100.00%
Color and Shape:
Solid
Molecular weight:
418.36
Ref: TM-T23007
| 1mg | 85.00 € | ||
| 2mg | 67.00 € | ||
| 5mg | 155.00 € | ||
| 10mg | 212.00 € | ||
| 25mg | 467.00 € | ||
| 50mg | 678.00 € | ||
| 100mg | 926.00 € | ||
| 200mg | 717.00 € | ||
| 500mg | 1,850.00 € | ||
| 1mL*10mM (DMSO) | 278.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
Methiothepin maleate
CAS:19728-88-2
Methiothepin maleate (Metitepine) is a 5-HT1, 5-HT6, 5-HT7 serotonin receptor antagonist, which blocks serotonin autoreceptors.
Formula:
C24H28N2O4S2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
472.62
Ref: TM-T4375
| 10mg | 86.00 € | ||
| 25mg | 172.00 € | ||
| 50mg | 238.00 € | ||
| 100mg | 437.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
DBIBB
CAS:1569309-92-7
DBIBB: non-lipid LPA2 receptor agonist, treats acute radiation syndrome, aids in organic synthesis/drug research.
Formula:
C23H20N2O6S
Purity:
97.18% - 97.26%
Color and Shape:
Solid
Molecular weight:
452.48
Ref: TM-T22070
| 1mg | 41.00 € | ||
| 5mg | 92.00 € | ||
| 10mg | 131.00 € | ||
| 25mg | 258.00 € | ||
| 50mg | 370.00 € | ||
| 100mg | 543.00 € | ||
| 500mg | 1,089.00 € | ||
| 1mL*10mM (DMSO) | 92.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
Alniditan
CAS:152317-89-0
Alniditan is a receptors agonist of 5-HT1B/1D in HEK 293 cells (IC50: 1.7 and 1.3 …
Formula:
C17H26N4O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
302.41
Ref: TM-T14190
| 25mg | 1,410.00 € | ||
| 50mg | 1,852.00 € | ||
| 100mg | 2,338.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
L748337
CAS:244192-94-7
L748337 is a β3-adrenoceptor antagonist that inhibits β3-, β2-, and β1-adrenoceptors and inhibits the protective …
Formula:
C26H31N3O5S
Purity:
99.67% - 99.67%
Color and Shape:
Solid
Molecular weight:
497.61
Ref: TM-T22905
| 1mg | 68.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
Sergliflozin etabonate
CAS:408504-26-7
Sergliflozin etabonate (KGT-1251) is an inhibitor of SGLT2 and can be used in studies about …
Formula:
C23H28O9
Purity:
95.59%
Color and Shape:
Solid
Molecular weight:
448.46
Ref: TM-T28757
| 1mg | 182.00 € | ||
| 2mg | 272.00 € | ||
| 5mg | 418.00 € | ||
| 10mg | 612.00 € | ||
| 25mg | 922.00 € | ||
| 50mg | 1,281.00 € | ||
| 100mg | 1,762.00 € | ||
| 1mL*10mM (DMSO) | 486.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
Oxyfedrine L-form HCl
CAS:16777-42-7
Oxyfedrine L-form HCl (Ildamen) is a partial agonist at beta-adrenergic receptors and acts as a …
Formula:
C19H24ClNO3
Purity:
98.66%
Color and Shape:
Solid
Molecular weight:
349.85
Ref: TM-T24579
| 1mg | 95.00 € | ||
| 5mg | 184.00 € | ||
| 10mg | 322.00 € | ||
| 25mg | 500.00 € | ||
| 50mg | 722.00 € | ||
| 100mg | 922.00 € | ||
| 1mL*10mM (DMSO) | 226.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
MJ 15
CAS:944154-76-1
MJ 15 is a CB1 receptor antagonist with specificity for the study of obesity-induced diseases.
Formula:
C23H17Cl3N4O
Purity:
99.63%
Color and Shape:
Solid
Molecular weight:
471.77
Ref: TM-T22984
| 1mg | 37.00 € | ||
| 5mg | 110.00 € | ||
| 10mg | 171.00 € | ||
| 25mg | 349.00 € | ||
| 50mg | 559.00 € | ||
| 100mg | 900.00 € | ||
| 500mg | 1,801.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
MK 1903
CAS:1268882-43-4
MK 1903 is a strong, selective HCA2/GPR109A agonist, reducing cAMP in CHO cells with EC50 …
Formula:
C8H8N2O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
164.16
Ref: TM-T22986
| 1mg | 49.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 142.00 € | ||
| 25mg | 244.00 € | ||
| 50mg | 342.00 € | ||
| 100mg | 481.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
Tildacerfont
CAS:1014983-00-6
Tildacerfont inhibits CRF1, lowers ACTH/adrenal androgens, and aids in congenital adrenal hyperplasia research.
Formula:
C20H26ClN5OS
Purity:
100.00%
Color and Shape:
Solid
Molecular weight:
419.97
Ref: TM-T26278
| 5mg | 35.00 € | ||
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 14 Jan 2025
AM404
CAS:183718-77-6
AM404 is a cannabinoid reuptake inhibitor and a TRPV (1) activator with neuroprotective and anticancer …
Formula:
C26H37NO2
Color and Shape:
Solid
Molecular weight:
395.58
Ref: TM-T39281
| 5mg | 68.00 € | ||
| 10mg | 109.00 € | ||
| 50mg | 434.00 € | ||
| 100mg | 740.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
YL-365
YL-365 is a highly potent and selective GPR34 antagonist that exhibits excellent activity in neuropathic …
Ref: TM-T80753
| 1mg | 75.00 € | ||
| 5mg | 167.00 € | ||
| 10mg | 261.00 € | ||
| 25mg | 527.00 € | ||
| 50mg | 838.00 € | ||
| 100mg | 1,332.00 € | ||
| 200mg | 1,801.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
CB2 modulator 1
CAS:666261-80-9
CB2 modulator 1 is a potent CB2 modulator. It can be used for the research …
Formula:
C18H19F3N4O2
Purity:
99.02%
Color and Shape:
Solid
Molecular weight:
380.36
Ref: TM-T10696
| 1mg | 35.00 € | ||
| 5mg | 55.00 € | ||
| 10mg | 78.00 € | ||
| 25mg | 112.00 € | ||
| 50mg | 164.00 € | ||
| 100mg | To inquire | ||
| 1mL*10mM (DMSO) | 64.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
Ticalopride
CAS:202590-69-0
Ticalopride: 5-HT3 agonist for digestive, orofacial, ENT disorders, and bulimia, GERD, IBS research.
Formula:
C14H20ClN3O3
Purity:
100%
Color and Shape:
Liquid
Molecular weight:
313.78
Ref: TM-T69984
| 1mg | 92.00 € | ||
| 5mg | 196.00 € | ||
| 10mg | 289.00 € | ||
| 25mg | 544.00 € | ||
| 50mg | 724.00 € | ||
| 100mg | 1,013.00 € | ||
| 500mg | 2,025.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
Repinotan HCl
CAS:144980-77-8
Repinotan HCl (Bay-x-3702) is a 5-HT1A receptor agonist with potent neuroprotective effects for the study …
Formula:
C21H25ClN2O4S
Purity:
99.57%
Color and Shape:
Solid
Molecular weight:
436.95
Ref: TM-T28518
| 1mg | 380.00 € | ||
| 5mg | 820.00 € | ||
| 10mg | 1,168.00 € | ||
| 25mg | 1,564.00 € | ||
| 50mg | 1,899.00 € | ||
| 100mg | 2,396.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
Irdabisant
CAS:1005402-19-6
Irdabisant (CEP-26401) is an H3R antagonist/inverse agonist, BBB permeable, with cognition-enhancing effects for schizophrenia/cognitive research.
Formula:
C18H23N3O2
Purity:
99.77%
Color and Shape:
Solid
Molecular weight:
313.39
Ref: TM-T32191
| 1mg | 57.00 € | ||
| 5mg | 131.00 € | ||
| 10mg | 184.00 € | ||
| 25mg | 328.00 € | ||
| 50mg | 460.00 € | ||
| 100mg | 647.00 € | ||
| 500mg | 1,291.00 € | ||
| 1mL*10mM (DMSO) | 92.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
CAY10786
CAS:1239987-91-7
CAY10786 (GPR52 antagonist-1) is an antagonist of G protein-coupled receptor 52 (GPR52, IC50 = 0.63 …
Formula:
C15H14OS
Purity:
99.84%
Color and Shape:
Solid
Molecular weight:
242.34
Ref: TM-T36036
| 2mg | 40.00 € | ||
| 5mg | 60.00 € | ||
| 10mg | 96.00 € | ||
| 25mg | 184.00 € | ||
| 50mg | 291.00 € | ||
| 100mg | 458.00 € | ||
| 1mL*10mM (DMSO) | 67.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
MRE3008F20
CAS:252979-43-4
MRE3008F20 is an AA3R antagonist that inhibits Cl-IB-MECA-induced cAMP production and can be used to …
Formula:
C21H20N8O3
Purity:
97.66%
Color and Shape:
Solid
Molecular weight:
432.44
Ref: TM-T16132
| 1mg | 69.00 € | ||
| 2mg | 91.00 € | ||
| 5mg | 149.00 € | ||
| 10mg | 212.00 € | ||
| 25mg | 360.00 € | ||
| 50mg | 536.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
