G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Ampreloxetine
CAS:1227056-84-9
Ampreloxetine (TD-9855) is a norepinephrine reuptake inhibitor used to study neurological diseases.
Formula:
C18H18F3NO
Purity:
98%
Color and Shape:
Solid
Molecular weight:
321.34
Ref: TM-T26622
| 25mg | 1,410.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
EMDT
CAS:263744-72-5
EMDT oxalate is a selective 5-HT6 agonist, and has antidepressant effects.
Formula:
C15H22N2O
Purity:
98.33% - 98.46%
Color and Shape:
Solid
Molecular weight:
246.35
Ref: TM-T11183
| 1mg | 91.00 € | ||
| 2mg | 123.00 € | ||
| 5mg | 168.00 € | ||
| 10mg | 211.00 € | ||
| 25mg | 467.00 € | ||
| 50mg | 680.00 € | ||
| 100mg | 926.00 € | ||
| 200mg | 717.00 € | ||
| 500mg | 1,838.00 € | ||
| 1mL*10mM (DMSO) | 167.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
EP1-antagonist-1
CAS:851204-35-8
EP1-antagonist-1 (EP1 antagonist 1) is an EP1 antagonist (pKi: 7.54; pIC50: 8.5).
Formula:
C19H15BrCl2N2O3
Purity:
98.51%
Color and Shape:
Solid
Molecular weight:
470.14
Ref: TM-T10031
| 1mg | 183.00 € | ||
| 5mg | 372.00 € | ||
| 10mg | 543.00 € | ||
| 25mg | 856.00 € | ||
| 50mg | 1,144.00 € | ||
| 100mg | 1,548.00 € | ||
| 1mL*10mM (DMSO) | 422.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
5HT6-ligand-1
CAS:1038988-11-2
5HT6-ligand-1 is an orally active ligand of 5-HT6 receptor (Ki = 1.43 nM).
Formula:
C20H22BrN3O2S
Purity:
98.48% - 98.95%
Color and Shape:
Solid
Molecular weight:
448.38
Ref: TM-T10053
| 1mg | 184.00 € | ||
| 5mg | 445.00 € | ||
| 10mg | 609.00 € | ||
| 25mg | 922.00 € | ||
| 50mg | 1,238.00 € | ||
| 100mg | 1,629.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
2-Methyl-5-HT maleate
CAS:78263-91-9
2-Methyl-5-HT maleate, a selective 5-HT3 agonist, shows anti-depressive effects.
Formula:
C15H18N2O5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
306.31
Ref: TM-T10075L
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
MRS1220
CAS:183721-15-5
MRS1220, a selective and potent antagonist for the human A3 adenosine receptor (hA3AR) with a …
Formula:
C21H14ClN5O2
Purity:
96.59%
Color and Shape:
Solid
Molecular weight:
403.82
Ref: TM-T23016
| 1mg | 49.00 € | ||
| 5mg | 114.00 € | ||
| 10mg | 174.00 € | ||
| 25mg | 297.00 € | ||
| 50mg | 428.00 € | ||
| 100mg | 603.00 € | ||
| 500mg | To inquire |
Estimated delivery in United States, on Tuesday 14 Jan 2025
SK609 HCl
CAS:1092797-77-7
SK609 HCl is a selective dopamine D3 receptor agonist. It also has atypical signaling properties.
Formula:
C10H15Cl2N
Purity:
99.02%
Color and Shape:
Solid
Molecular weight:
220.14
Ref: TM-T24797
| 1mg | 87.00 € | ||
| 5mg | 183.00 € | ||
| 10mg | 269.00 € | ||
| 25mg | 459.00 € | ||
| 50mg | 641.00 € | ||
| 100mg | 907.00 € | ||
| 500mg | 1,800.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
2-Arachidonoylglycerol
CAS:53847-30-6
In the central nervous system, 2-Arachidonoylglycerol is a second endogenous cannabinoid ligand
Formula:
C23H38O4
Purity:
95%
Color and Shape:
Liquid
Molecular weight:
378.55
Ref: TM-T14011
| 1mg (26.4mM*100μL in Acetonitrile) | 113.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
SB-269970
CAS:201038-74-6
SB-269970 is a antagonist of 5-HT7 receptor(pKi of 8.3).
Formula:
C18H28N2O3S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
352.49
Ref: TM-T12842
| 25mg | 1,406.00 € | ||
| 50mg | 1,845.00 € | ||
| 100mg | 2,329.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
CP-226269
CAS:220941-93-5
CP-226269 is a potent dopamine D4 receptor agonist that regulates calcium flux and has an …
Formula:
C18H19FN4
Purity:
99.08%
Color and Shape:
Solid
Molecular weight:
310.37
Ref: TM-T27060
| 1mg | 95.00 € | ||
| 5mg | 229.00 € | ||
| 10mg | 335.00 € | ||
| 25mg | 538.00 € | ||
| 50mg | 765.00 € | ||
| 100mg | 1,040.00 € | ||
| 500mg | 2,070.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
ONO-8713
CAS:459411-08-6
ONO-8713 is a selective prostaglandin E receptor subtype EP1 antagonist that can be used to …
Formula:
C25H24F3NO6S
Purity:
100.00%
Color and Shape:
Solid
Molecular weight:
523.52
Ref: TM-T63667
| 1mg | 378.00 € | ||
| 5mg | 900.00 € | ||
| 10mg | 1,122.00 € | ||
| 25mg | 1,502.00 € | ||
| 50mg | 1,838.00 € | ||
| 100mg | 2,320.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
Olorinab
CAS:1268881-20-4
Olorinab (APD 371) (APD 371) is a highly potent, selective and fully efficacious cannabinoid receptor …
Formula:
C18H23N5O3
Purity:
97.13%
Color and Shape:
Solid
Molecular weight:
357.41
Ref: TM-T14302
| 1mg | 55.00 € | ||
| 5mg | 118.00 € | ||
| 10mg | 184.00 € | ||
| 25mg | 369.00 € | ||
| 50mg | 550.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
L-161982
CAS:147776-06-5
L-161982 is a selective EP4 receptor antagonist that inhibits PGE2-induced ERK phosphorylation and cell proliferation …
Formula:
C32H29F3N4O4S2
Purity:
99.44% - 99.91%
Color and Shape:
Solid
Molecular weight:
654.72
Ref: TM-T15681
| 1mg | 78.00 € | ||
| 5mg | 184.00 € | ||
| 10mg | 299.00 € | ||
| 25mg | 531.00 € | ||
| 50mg | 757.00 € | ||
| 100mg | 1,006.00 € | ||
| 1mL*10mM (DMSO) | 279.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
ANR 94
CAS:634924-89-3
ANR94 is a potent hAA2AR antagonist (Ki 46 nM) with potential for Parkinson's research.
Formula:
C9H13N5O
Purity:
98.21%
Color and Shape:
Solid
Molecular weight:
207.23
Ref: TM-T22031
| 2mg | 41.00 € | ||
| 5mg | 62.00 € | ||
| 10mg | 93.00 € | ||
| 25mg | 182.00 € | ||
| 50mg | 318.00 € | ||
| 100mg | 449.00 € | ||
| 200mg | 631.00 € | ||
| 1mL*10mM (DMSO) | 61.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
Arbutamine
CAS:128470-16-6
Arbutamine (GP 21213) is a β-adrenoceptor agonist with alpha-1-sympathomimetic activity that can be used to …
Formula:
C18H23NO4
Purity:
95.06%
Color and Shape:
Solid
Molecular weight:
317.38
Ref: TM-T10364
| 1mg | 378.00 € | ||
| 5mg | 905.00 € | ||
| 10mg | 1,122.00 € | ||
| 25mg | 1,502.00 € | ||
| 50mg | 1,846.00 € | ||
| 100mg | 2,331.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
PGD2-IN-1
CAS:885066-67-1
PGD2-IN-1 (PGD2-inhibitor) is an effective DP receptor antagonist (IC50:0.3 nM), a compound that can inhibit …
Formula:
C23H23Cl2N3O3
Purity:
99%
Color and Shape:
Solid
Molecular weight:
460.35
Ref: TM-T4624
| 1mg | 69.00 € | ||
| 5mg | 156.00 € | ||
| 10mg | 255.00 € | ||
| 25mg | 428.00 € | ||
| 50mg | 631.00 € | ||
| 100mg | 895.00 € | ||
| 500mg | 1,791.00 € | ||
| 1mL*10mM (DMSO) | 167.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
L-168049
CAS:191034-25-0
L-168049: Human glucagon receptor antagonist, IC50 - 3.7 nM human, 63 nM murine, 60 nM …
Formula:
C24H20BrClN2O
Purity:
100%
Color and Shape:
Solid
Molecular weight:
467.79
Ref: TM-T22893
| 1mg | 52.00 € | ||
| 5mg | 110.00 € | ||
| 10mg | 176.00 € | ||
| 25mg | 369.00 € | ||
| 50mg | 551.00 € | ||
| 100mg | 783.00 € | ||
| 500mg | 1,613.00 € | ||
| 1mL*10mM (DMSO) | 123.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
Impromidine hydrochloride
CAS:65573-02-6
Impromidine hydrochloride is a very potent and specific histamine H2 receptor agonist for conducting cardiovascular …
Formula:
C14H26Cl3N7S
Purity:
99.50%
Color and Shape:
Solid
Molecular weight:
430.83
Ref: TM-T68921
| 1mg | 240.00 € | ||
| 5mg | 599.00 € | ||
| 10mg | 853.00 € | ||
| 25mg | 1,280.00 € | ||
| 50mg | 1,729.00 € | ||
| 100mg | 2,331.00 € | ||
| 500mg | 4,577.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
Medifoxamine
CAS:32359-34-5
Medifoxamine (LG 152) is a selective non-monoamine oxidase inhibitor that exhibits antidepressant activity through inhibition …
Formula:
C16H19NO2
Purity:
98.35%
Color and Shape:
Solid
Molecular weight:
257.33
Ref: TM-T24444
| 1mg | 96.00 € | ||
| 5mg | 229.00 € | ||
| 10mg | 344.00 € | ||
| 25mg | 618.00 € | ||
| 50mg | 868.00 € | ||
| 100mg | 1,128.00 € | ||
| 1mL*10mM (DMSO) | 252.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
Opioid receptor modulator 1
CAS:77514-44-4
Opioid receptor modulator 1 is a modulator of opioid receptor.
Formula:
C18H23NO2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
285.38
Ref: TM-T12314
| 25mg | 1,406.00 € | ||
| 50mg | 1,847.00 € | ||
| 100mg | 2,331.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
